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1. 发明授权

US06420423B1 Pesticides 失效
标题翻译：农药
公开(公告)号：US06420423B1
公开(公告)日：2002-07-16
申请号：US09343662
申请日：1999-06-29
申请人： Saleem Farooq , Stephan Trah , Hugo Ziegler , René Zurflüh , Alfons Pascual , Henry Szczepanski , Roger Graham Hall
发明人： Saleem Farooq , Stephan Trah , Hugo Ziegler , René Zurflüh , Alfons Pascual , Henry Szczepanski , Roger Graham Hall
IPC分类号： A61K3124
CPC分类号： C07D213/53 , A01N37/36 , A01N37/38 , A01N37/50 , A01N43/10 , A01N43/40 , A01N43/54 , A01N43/60 , A01N55/00 , C07C249/12 , C07C251/48 , C07C251/60 , C07C255/54 , C07C323/20 , C07C323/47 , C07C2601/02 , C07C2601/08 , C07D239/26 , C07D241/12 , C07D275/03 , C07D317/64 , C07D333/22 , C07F7/081
摘要： Compounds of the formula: in which n, q, A, X, G, Y, Z, R, R2, R3, R4, R5, R7 and R9 are as defined in claim 1, and, where appropriate, E/Z isomers, E/Z isomer mixtures and/or tautomers thereof, in each case in the free form or in an agrochemically suitable salt form, can be used as agrochemical active compounds and can be prepared in a manner known per se.
摘要翻译：下式的化合物：其中n，q，A，X，G，Y，Z，R，R 2，R 3，R 4，R 5，R 7和R 9如权利要求1中所定义，并且在适当的情况下，E / ，在各种情况下以游离形式或农业化学合适的盐形式的E / Z异构体混合物和/或互变异构体可以用作农业化学活性化合物，并且可以以本身已知的方式制备。

2. 发明授权

US06313344B1 Organic compounds 失效
标题翻译：有机化合物
公开(公告)号：US06313344B1
公开(公告)日：2001-11-06
申请号：US09085283
申请日：1998-05-27
申请人： Stephan Trah , Henry Szczepanski , Ottmar Franz Hüter , Roger Graham Hall , Saleem Farooq , Alfons Pascual
发明人： Stephan Trah , Henry Szczepanski , Ottmar Franz Hüter , Roger Graham Hall , Saleem Farooq , Alfons Pascual
IPC分类号： C07C32700
CPC分类号： C07D261/20 , A01N37/38 , A01N37/50 , A01N43/80 , C07C251/60 , C07C323/12 , C07D261/08 , C07F9/4021
摘要： Compounds of formula (I), wherein either X is CH or N, Y is OR1 and Z is O, or X is N, Y is NHR8 and Z is O, S or S(═O); R1, R2 and R3 are as defined according to the specification; m is 0, 1 or 2; R5 is, for example, halogen, C1-C6alkyl, halo-C1-C6alkyl or C3-C6cycloalkyl; n is 0, 1, 2, 3 or 4; R9 is methyl, fluoromethyl or difluoromethyl; A and R7 are as defined according to the specification; D is O, S, —S(═O) or S(═O)2; G is C1-C6aalkylene; T—R6 is R6, —C(═N—O—A1—R77)—R6; —SiR14(R15)—R6; —C(═O)—R6; —C(R16)═C(R17)—R6, —C≡C—R6 or —D—R6; R6 is C1-C4alkyl or unsubstituted or substituted aryl or heteroaryl; A1 and R77 are as defined above for A and R7; L is U—R18, P(OR)vR11R12, P(S)wR11R12 or N(aryl)R13; v and w are 0 or 1; U—R18 is —C(═O)—C(═O)—R18; —C(OH)—C(OH)—R18; —C(═N—O—A1—R7)—R18; a is 0 or 1; b is 0 or 1; R11, R12 and R13 are, for example, C1-C6alkyl, halo-C1-C6alkyl or C3-C6cycloalkyl; R14 and R15 are each independently of the other C1-C4alkyl; R16 and R17 are each independently of the other hydrogen, C1-C4alkyl or halogen and R18 is R5; and, where applicable, their possible E/Z isomers, mixtures of E/Z isomers and/or tautomers, in each case in free form or in salt form, a method of controlling pests, a process for the preparation of those compounds and their use are described.
摘要翻译：式（I）化合物，其中X是CH或N，Y是OR 1，Z是O，或X是N，Y是NHR 8，Z是O，S或S（= O）; R 1，R 2和R 3如上定义根据规范; m为0,1或2; R 5为例如卤素，C 1 -C 6烷基，卤代-C 1 -C 6烷基或C 3 -C 6环烷基; n为0,1,2,3或4; R9是甲基，氟甲基或二氟甲基; A和R7如本说明书所定义; D是O，S，-S（= O）或S（= O）2; G是C1-C6亚烷基; T-R6是R6，-C（= N-O-A1-R77）-R6; -SiR14（R15）-R6; -C（= O）-R6; -C（R 16）= C（R 17）-R 6，-C = C-R6或-D-R6; R6是C1-C4烷基或未取代或取代的芳基或杂芳基; A1和R77如对于A和R7所定义; L是U-R18，P（OR）vR11R12，P（S）wR11R12或N（芳基）R13; v和w为0或1; U-R 18为-C（= O）-C（= O）-R 18; -C（OH）-C（OH）-R 18; -C（= N-O-Al-R 7）-R 18; a为0或1; b为0或1; R 11，R 12和R 13为例如C 1 -C 6烷基，卤代-C 1 -C 6烷基或C 3 -C 6环烷基; R 14和R 15各自独立地为C 1 -C 4烷基; R 16和R 17各自独立地为另一个氢，C 1 -C 4烷基或卤素，R 18是R 5;并且在适用的情况下，它们可能的E / Z异构体，E / Z异构体和/或互变异构体的混合物，在每种情况下以游离形式或盐形式，控制害虫，制备这些化合物的方法及其用途。

3. 发明授权

US5985921A 2-Phenyl-2-methoxyimino acetic acid esters 失效
标题翻译： 2-苯基-2-甲氧基亚氨基乙酸酯
公开(公告)号：US5985921A
公开(公告)日：1999-11-16
申请号：US761675
申请日：1996-12-06
申请人： Saleem Farooq , Stephen Trah , Hugo Ziegler , Rene Zurfluh , Alfons Pascual , Henry Szczepanski , Roger Graham Hall
发明人： Saleem Farooq , Stephen Trah , Hugo Ziegler , Rene Zurfluh , Alfons Pascual , Henry Szczepanski , Roger Graham Hall
IPC分类号： A01N37/36 , A01N37/38 , A01N37/50 , A01N43/10 , A01N43/30 , A01N43/40 , A01N43/54 , A01N43/60 , A01N55/00 , C07C239/02 , C07C249/02 , C07C249/12 , C07C251/24 , C07C251/40 , C07C251/48 , C07C251/60 , C07C255/54 , C07C255/64 , C07C323/20 , C07C323/47 , C07D213/02 , C07D213/53 , C07D215/00 , C07D215/12 , C07D239/26 , C07D241/12 , C07D263/14 , C07D275/02 , C07D275/03 , C07D317/64 , C07D333/22 , C07D521/00 , C07F7/08 , C07F7/10 , A61K31/24 , A61K31/16 , C07C229/00 , C07C327/00
CPC分类号： C07D213/53 , A01N37/36 , A01N37/38 , A01N37/50 , A01N43/10 , A01N43/40 , A01N43/54 , A01N43/60 , A01N55/00 , C07C249/12 , C07C251/48 , C07C251/60 , C07C255/54 , C07C323/20 , C07C323/47 , C07D239/26 , C07D241/12 , C07D275/03 , C07D317/64 , C07D333/22 , C07F7/0818 , C07C2101/02 , C07C2101/08
摘要： Compounds of the formula ##STR1## in which n, q, A, X, G, Y, Z, R, R.sub.2, R.sub.3, R.sub.4, R.sub.5, R.sub.7 and R.sub.9 are as defined in claim 1, and, where appropriate, E/Z isomers, E/Z isomer mixtures and/or tautomers thereof, in each case in the free form or in an agrochemically suitable salt form, can be used as agrochemical active compounds and can be prepared in a manner known per se.
摘要翻译：其中n，q，A，X，G，Y，Z，R，R 2，R 3，R 4，R 5，R 7和R 9如权利要求1中所定义，并且在适当的情况下，E / 在各种情况下，E / Z异构体混合物和/或互变异构体以游离形式或农业化学合适的盐形式可以用作农业化学活性化合物，并且可以以本身已知的方式制备。

4. 发明授权

US5935908A Pesticidal indazole derivatives 失效
标题翻译：杀虫吲唑衍生物
公开(公告)号：US5935908A
公开(公告)日：1999-08-10
申请号：US11916
申请日：1998-02-17
申请人： Saleem Farooq , Rene Zurfluh , Henry Szczepanski , Roger Graham Hall
发明人： Saleem Farooq , Rene Zurfluh , Henry Szczepanski , Roger Graham Hall
IPC分类号： A01N43/56 , A01N55/00 , C07C69/734 , C07C251/42 , C07C251/48 , C07C255/54 , C07C255/64 , C07D231/56 , C07F7/08
CPC分类号： C07F7/0812 , A01N43/56 , A01N55/00 , C07C251/40 , C07C251/42 , C07C251/48 , C07C255/54 , C07C255/64 , C07C69/734 , C07D231/56 , C07C2101/02
摘要： Compounds of formula (1), wherein X, Y, Z R.sub.2, R.sub.3, R.sub.4, R.sub.5, R.sub.7, R.sub.9 and n are as defined in claim 1 and, where appropriate, E/Z isomers, mixtures of E/Z isomers and/or tautomers thereof, in each case in free form or in agrochemically suitable salt form, can be used as agrochemical active ingredients and can be prepared in a manner known per se. ##STR1##
摘要翻译： PCT No.PCT / EP96 / 03452 Sec。 371日期1998年2月17日 102（e）日期1998年2月17日PCT提交1996年8月5日PCT公布。公开号WO97 / 07103 日期1997年2月27日，式（1）的化合物，其中X，Y，Z R2，R3，R4，R5，R7，R9和n如权利要求1所定义，并且在适当的情况下，E / Z异构体，E / Z异构体和/或互变异构体，以游离形式或农业化学合适的盐形式，可以用作农业化学活性成分，并且可以以本身已知的方式制备。

5. 发明授权

US07795442B2 Preparation of thiazoles 失效
标题翻译：噻唑的制备
公开(公告)号：US07795442B2
公开(公告)日：2010-09-14
申请号：US12424594
申请日：2009-04-16
申请人： Thomas Pitterna , Henry Szczepanski , Peter Mainenfisch , Ottmar Franz Huter , Thomas Rapold , Marcel Senn , Thomas Gobel , Anthony Cornelius O'Sullivan
发明人： Thomas Pitterna , Henry Szczepanski , Peter Mainenfisch , Ottmar Franz Huter , Thomas Rapold , Marcel Senn , Thomas Gobel , Anthony Cornelius O'Sullivan
IPC分类号： C07D277/32
CPC分类号： C07D277/32 , C07D277/16 , C07D277/36 , C07D277/70 , C07D277/74
摘要： A process is provided for preparing compounds having the general formula I wherein R is a range of organic groups and X is a leaving group. The process comprises reacting a compound of formula II with a water-removing reagent. When X is halogen or a sulfonate, the compound of formula I may be prepared by reacting a compound of the formula III with a halogenating agent or a sulfonylating agent. Alternatively, when X is halogen, the compound of formula I can be prepared by reacting a compound of the formula IV where R2 and R2 are defined organic groups, with a compound of the formula halogen-C(—O)—O—C1-C8alkyl, halogen-C(—O)—O-aryl or halogen-C(—O)—O-benzyl.
摘要翻译：提供了一种制备具有通式I的化合物的方法，其中R是有机基团的范围，X是离去基团。该方法包括使式II化合物与除水试剂反应。当X是卤素或磺酸盐时，式I化合物可以通过使式III化合物与卤化剂或磺酰化剂反应来制备。或者，当X是卤素时，式I化合物可以通过其中R2和R2定义为有机基团的式IV化合物与式卤化-C（ - ） - O-C1- C8烷基，卤素-C（ - ） - O-芳基或卤素-C（ - ） - O-苄基。

7. 发明授权

US06864392B2 α-Sulfin and α-Sulfonamino amide derivatives 失效
标题翻译： α-亚砜和α-磺酰氨基酰胺衍生物
公开(公告)号：US06864392B2
公开(公告)日：2005-03-08
申请号：US10257085
申请日：2001-04-11
申请人： Martin Zeller , Clemens Lamberth , Henry Szczepanski , Alain De Mesmaeker
发明人： Martin Zeller , Clemens Lamberth , Henry Szczepanski , Alain De Mesmaeker
IPC分类号： C07D295/22 , A01N41/06 , A01N43/10 , A01N43/36 , A01N43/40 , A01N43/42 , A01N43/60 , C07C303/34 , C07C303/38 , C07C307/06 , C07C311/06 , C07C313/06 , C07D213/30 , C07D213/61 , C07D215/14 , C07D241/12 , C07D333/16 , C07D333/28 , C07C311/03
CPC分类号： A01N41/06 , C07C307/06 , C07C311/06 , C07C313/06
摘要： The invention relates to novel pesticidally active α-sulfin- and α-sulfonamino acid amides of the general formula (I) including the optical isomers thereof and mixtures of such isomers, wherein n is a number zero or one, R1-R7 have the meanings given in the specification. R8 is either hydrogen, (a), (b), (c), (d) or (e) wherein R11, R12, R14, R15 and R17 are each independently hydrogen or C1-C4alkyl, R13 is C4-C12alkyl; C1-C12 halogenalkyl; C3-C8 cycloalkyl; optionally substituted aryl or optionally substituted heteroaryl, R16 is optionally substituted aryl or optionally substituted heteroaryl; and Z is oxygen, sulfur —CR18R19— or —NR20—, wherein R18, R19, R20 independently of each other are hydrogen or C1-C4alkyl. The novel compounds possess plant-protecting properties and are suitable for protecting plants against infestation by phytopathogenic microorganisms
摘要翻译：本发明涉及通式（I）的新型农药活性α-亚磺酸和α-磺氨基酰胺，其包括其旋光异构体和这些异构体的混合物，其中n为数个零或一个，R 1 -R 7具有在规范中给出。 R8是氢，（a），（b），（c），（d）或（e）其中R11，R12，R14，R15和R17各自独立地是氢或C1-C4烷基，R13是C4-C12烷基; C1-C12卤代烷基; C3-C8环烷基; 任选取代的芳基或任选取代的杂芳基，R 16是任选取代的芳基或任选取代的杂芳基; Z为氧，硫-CR 18 R 19 - 或-NR 20 - ，其中R 18，R 19，R 20彼此独立地为氢或C 1 -C 4烷基。新型化合物具有植物保护性质，适用于保护植物免受植物病原微生物侵扰

8. 发明授权

US06310096B1 Cyclohexadiene-derivatives as pesticides 失效
标题翻译：环己二烯衍生物作为农药
公开(公告)号：US06310096B1
公开(公告)日：2001-10-30
申请号：US09555613
申请日：2000-06-01
申请人： Henry Szczepanski
发明人： Henry Szczepanski
IPC分类号： A01N3712
CPC分类号： C07D213/643 , A01N37/50 , C07C69/734 , C07C69/738 , C07C251/40 , C07C251/42 , C07C2601/16 , C07F7/081
摘要： Certain cyclohexadiene derivatives are useful as pesticides. The derivatives are of the formula: wherein X is N; Y is O; S, S═O or NR5; Z is OR2, SR2, N(R3)R4; V is a direct bond or a 1 to 4 membered, saturated or unsaturated carbon chain which is unsubstituted or substituted by C1-C3alkyl, halogen, hydroxy, C1-C4alkoxy, halo-C1-C4alkoxy or oxo; W is hydrogen or C1-C6 alkyl or a group of the formula: wherein n is an integer of from 0 to 5 and each D is identical or different and represents a moiety selected from the group consisting of halogen, cyano, nitro, C1 to C12 alkyl, halo-C1 to C12 alkyl, C2 to C12 alkenyl, halo-C2 to C12 alkenyl, C2 to C12 alkynyl, halo-C2 to C12 alkynyl, C3 to C6 cycloalkyl, halo-C3 to C6 cycloalkyl, C3 to C6 cycloalkylmethyl, halo-C3 to C6 cycoloalkylmethyl, etc.
摘要翻译：某些环己二烯衍生物可用作杀虫剂。衍生物具有下式：其中X是N; Y是O; S，S = O或NR 5; Z是OR 2，SR 2，N（R 3）R 4; V是直接键或1至4元饱和或不饱和的碳链，其未被取代或被C 1 -C 3烷基，卤素，羟基，C 1 -C 4烷氧基，卤代-C 1 -C 4烷氧基或氧代; W是氢或C 1 -C 6烷基或下式的基团：其中n是0至5的整数，并且每个D相同或不同，并且表示选出的部分由卤素，氰基，硝基，C1至C12烷基，卤代-C1至C12烷基，C2至C12烯基，卤代-C2至C12烯基，C2至C12炔基，卤代-C2至C12炔基，C3至C6组成的组环烷基，卤代-C 3至C 6环烷基，C 3至C 6环烷基甲基，卤代-C 3至C 6环烷基甲基等。

9. 发明授权

US4898607A Herbicidal imidazole derivatives 失效
标题翻译：除草咪唑衍生物
公开(公告)号：US4898607A
公开(公告)日：1990-02-06
申请号：US234240
申请日：1988-08-18
申请人： Henry Szczepanski , Lourens Wals
发明人： Henry Szczepanski , Lourens Wals
IPC分类号： A01N43/56 , A01N43/50 , A01N43/836 , C07D233/90 , C07D403/04 , C07D405/04
CPC分类号： C07D405/04 , A01N43/50 , C07D233/90
摘要： 1,5-substituted imidazole derivatives of formula I ##STR1## the stereochemically isomeric forms thereof, and the salts thereof, have useful herbicidal properties. The substituents R.sup.1, R.sup.2, R.sup.3, R.sup.4, X.sup.1, X.sup.2, X.sup.3, A, L and m have the meanings defined herein.
摘要翻译：式I的1,5-取代咪唑衍生物其中（I）其立体化学异构形式及其盐具有有用的除草性质。取代基R 1，R 2，R 3，R 4，X 1，X 2，X 3，A，L和m具有本文定义的含义。

10. 发明授权

US4600428A N-(cyclopropyl-pyrimidinyl-N'-(aryl-sulfonyl) ureas having herbicidal activity 失效
标题翻译：具有除草活性的N-（环丙基 - 嘧啶基-N' - （芳基 - 磺酰基）脲）
公开(公告)号：US4600428A
公开(公告)日：1986-07-15
申请号：US693655
申请日：1985-01-22
申请人： Henry Szczepanski
发明人： Henry Szczepanski
IPC分类号： C07D249/16 , A01N47/36 , C07C45/00 , C07C45/45 , C07C49/15 , C07C67/00 , C07D239/42 , C07D239/47 , C07D251/16 , C07D251/18 , C07D251/20 , C07D251/22 , C07D251/24 , C07D251/42 , C07D521/00 , A01N43/54
CPC分类号： C07D239/42 , A01N47/36 , C07C45/455 , C07D251/16 , C07D251/18 , C07D251/20 , C07D251/22 , C07D251/24 , C07D521/00
摘要： N-(Cyclopropyl-pyrimidinyl)-N'-aryl-sulfonyl ureas of the formula ##STR1## wherein Ar is a phenyl group ##STR2## or a naphthyl group andQ is a group X-A or R.sub.3,A is alkynyl, alkyl which is unsubstituted or substituted by halogen, alkoxy, alkylthio, alkylsulfinyl, alkylsulfonyl, haloalkoxy, haloalkylthio, haloalkylsulfinyl or haloalkylsulfonyl, or alkenyl which is unsubstituted or substituted by the substituents given above for alkyl, or A is a phenyl or benzyl group,E is methine,X is oxygen, sulfur, or a sulfinyl or sulfonyl bridge,Z is oxygen or sulfur,R.sub.1 is hydrogen, alkyl or alkoxy,R.sub.2 is halogen, alkyl, haloalkyl, alkoxy, haloalkoxy, amino, alkylamino, di-alkylamino, cycloalkyl or alkoxyalkyl, R.sub.3 is hydrogen, halogen, alkyl, alkenyl, haloalkyl, --CO--NR.sub.8 R.sub.9, --CN, --COR.sub.10, --NR.sub.1 R.sub.7 or --NR.sub.1 --COR.sub.12,R.sub.4 is hydrogen, alkyl, alkoxy, alkylthio, haloalkyl, haloalkoxy, halogen, or alkoxyalkyl,R.sub.5 is independently selected from the same groups as R.sub.3 or --X--R.sub.6,R.sub.6 and R.sub.7 are each alkyl, alkenyl or alkynyl,R.sub.8 and R.sub.9 independently of one another are each hydrogen, alkyl, alkenyl or alkynyl,R.sub.10 is hydrogen, alkyl or haloalkyl,R.sub.11 is hydrogen, alkyl, haloalkyl, alkenyl, alkynyl, phenyl or benzyl, andR.sub.12 is the same as R.sub.1 but independent thereof, and the salts of these compounds with amines, metal bases, or quaternary ammonium bases, have good herbicidal and plant-growth-regulating properties.
摘要翻译：式（I）的N-（环丙基 - 嘧啶基）-N'-芳基磺酰基脲其中Ar是苯基或萘基，Q是基团XA或R3，A是炔基，未取代或被卤素，烷氧基，烷硫基，烷基亚磺酰基，烷基磺酰基，卤代烷氧基，卤代烷硫基，卤代烷基亚磺酰基或卤代烷基磺酰基取代的烷基，或未取代或被上述烷基取代的取代基的烯基，或A是苯基或苄基，E 是次甲基，X是氧，硫或亚磺酰基或磺酰基桥，Z是氧或硫，R1是氢，烷基或烷氧基，R2是卤素，烷基，卤代烷基，烷氧基，卤代烷氧基，氨基，烷基氨基，二烷基氨基，环烷基或烷氧基烷基，R3是氢，卤素，烷基，烯基，卤代烷基，-CO-NR8R9，-CN，-COR10，-NR1R7或-NR1-COR12，R4是氢，烷基，烷氧基，烷硫基，卤代烷基，卤代烷氧基，或烷氧基烷基，R 5独立地选自与R 3或-X-R 6相同的基团，R 6和R 7各自为烷基，烯基 1或炔基，R 8和R 9彼此独立地各自为氢，烷基，烯基或炔基，R 10为氢，烷基或卤代烷基，R 11为氢，烷基，卤代烷基，烯基，炔基，苯基或苄基，R 12为作为R1但不相关，并且这些化合物与胺，金属碱或季铵碱的盐具有良好的除草和植物生长调节性质。

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