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1. 发明授权

US06420423B1 Pesticides 失效
标题翻译：农药
公开(公告)号：US06420423B1
公开(公告)日：2002-07-16
申请号：US09343662
申请日：1999-06-29
申请人： Saleem Farooq , Stephan Trah , Hugo Ziegler , René Zurflüh , Alfons Pascual , Henry Szczepanski , Roger Graham Hall
发明人： Saleem Farooq , Stephan Trah , Hugo Ziegler , René Zurflüh , Alfons Pascual , Henry Szczepanski , Roger Graham Hall
IPC分类号： A61K3124
CPC分类号： C07D213/53 , A01N37/36 , A01N37/38 , A01N37/50 , A01N43/10 , A01N43/40 , A01N43/54 , A01N43/60 , A01N55/00 , C07C249/12 , C07C251/48 , C07C251/60 , C07C255/54 , C07C323/20 , C07C323/47 , C07C2601/02 , C07C2601/08 , C07D239/26 , C07D241/12 , C07D275/03 , C07D317/64 , C07D333/22 , C07F7/081
摘要： Compounds of the formula: in which n, q, A, X, G, Y, Z, R, R2, R3, R4, R5, R7 and R9 are as defined in claim 1, and, where appropriate, E/Z isomers, E/Z isomer mixtures and/or tautomers thereof, in each case in the free form or in an agrochemically suitable salt form, can be used as agrochemical active compounds and can be prepared in a manner known per se.
摘要翻译：下式的化合物：其中n，q，A，X，G，Y，Z，R，R 2，R 3，R 4，R 5，R 7和R 9如权利要求1中所定义，并且在适当的情况下，E / ，在各种情况下以游离形式或农业化学合适的盐形式的E / Z异构体混合物和/或互变异构体可以用作农业化学活性化合物，并且可以以本身已知的方式制备。

2. 发明授权

US5985921A 2-Phenyl-2-methoxyimino acetic acid esters 失效
标题翻译： 2-苯基-2-甲氧基亚氨基乙酸酯
公开(公告)号：US5985921A
公开(公告)日：1999-11-16
申请号：US761675
申请日：1996-12-06
申请人： Saleem Farooq , Stephen Trah , Hugo Ziegler , Rene Zurfluh , Alfons Pascual , Henry Szczepanski , Roger Graham Hall
发明人： Saleem Farooq , Stephen Trah , Hugo Ziegler , Rene Zurfluh , Alfons Pascual , Henry Szczepanski , Roger Graham Hall
IPC分类号： A01N37/36 , A01N37/38 , A01N37/50 , A01N43/10 , A01N43/30 , A01N43/40 , A01N43/54 , A01N43/60 , A01N55/00 , C07C239/02 , C07C249/02 , C07C249/12 , C07C251/24 , C07C251/40 , C07C251/48 , C07C251/60 , C07C255/54 , C07C255/64 , C07C323/20 , C07C323/47 , C07D213/02 , C07D213/53 , C07D215/00 , C07D215/12 , C07D239/26 , C07D241/12 , C07D263/14 , C07D275/02 , C07D275/03 , C07D317/64 , C07D333/22 , C07D521/00 , C07F7/08 , C07F7/10 , A61K31/24 , A61K31/16 , C07C229/00 , C07C327/00
CPC分类号： C07D213/53 , A01N37/36 , A01N37/38 , A01N37/50 , A01N43/10 , A01N43/40 , A01N43/54 , A01N43/60 , A01N55/00 , C07C249/12 , C07C251/48 , C07C251/60 , C07C255/54 , C07C323/20 , C07C323/47 , C07D239/26 , C07D241/12 , C07D275/03 , C07D317/64 , C07D333/22 , C07F7/0818 , C07C2101/02 , C07C2101/08
摘要： Compounds of the formula ##STR1## in which n, q, A, X, G, Y, Z, R, R.sub.2, R.sub.3, R.sub.4, R.sub.5, R.sub.7 and R.sub.9 are as defined in claim 1, and, where appropriate, E/Z isomers, E/Z isomer mixtures and/or tautomers thereof, in each case in the free form or in an agrochemically suitable salt form, can be used as agrochemical active compounds and can be prepared in a manner known per se.
摘要翻译：其中n，q，A，X，G，Y，Z，R，R 2，R 3，R 4，R 5，R 7和R 9如权利要求1中所定义，并且在适当的情况下，E / 在各种情况下，E / Z异构体混合物和/或互变异构体以游离形式或农业化学合适的盐形式可以用作农业化学活性化合物，并且可以以本身已知的方式制备。

3. 发明授权

US06646151B1 Process for the preparation of pesticides 失效
标题翻译：农药制备工艺
公开(公告)号：US06646151B1
公开(公告)日：2003-11-11
申请号：US09670147
申请日：2000-09-26
申请人： Saleem Farooq , Stephan Trah , Hugo Ziegler , René Zurflüh
发明人： Saleem Farooq , Stephan Trah , Hugo Ziegler , René Zurflüh
IPC分类号： C07C24904
CPC分类号： C07C249/12 , C07C251/48 , C07C251/60
摘要： The invention relates to a process for the preparation of compounds of the formula or, if appropriate, a tautomer thereof, in each case in the free form or in salt form, in which A, X, Y, Z, R2, R3, R4, R5, R7, R9 and n are as defined in claim 1 and the C═N double bond marked with E has the E configuration, which comprises a1) reacting either a compound of the formula (II) mentioned above with a compound of the formula (III) mentioned above, in which X1 is a leaving group, or a2) a compound of the formula (IV) mentioned above, if appropriate in the presence of a base, with a compound of the formula (V) mentioned above, or b1) reacting a compound of the formula (VI) mentioned above with a compound of the formula R7—A—X2 (VII), in which X2 is a leaving group, and either further reacting the compound thus obtainable, of the formula (IV), for example according to method a2), or b2) reacting it with hydroxylamine or a salt thereof, if appropriate in the presence of a basic or acid catalyst, and further reacting the compound thus obtainable, of the formula (II), for example according to method a1), or c) reacting a compound of the formula (VIII), mentioned above with a C1-C6alkyl nitrite and further reacting the compound thus obtainable, of the formula (VI), for example according to method b), the E isomers of the compounds of the formulae (II), (IV) and (VI), a process for their preparation and their use for the preparation of compounds of the formula (I).
摘要翻译：本发明涉及一种制备式的化合物的方法，如果合适，其合适的是其互变异构体，其各自为游离形式或盐形式，其中A，X，Y，Z，R 2，R 3，R 4， R5，R7，R9和n如权利要求1中所定义，并且用E标记的C = N双键具有E构型，其包括a）使上述式（II）的化合物与式（II） III），其中X1是离去基团，ora2）如果合适的话，在碱的存在下，上述式（Ⅳ）的化合物与上述式（Ⅴ）的化合物相同，反应1）使上述式（Ⅵ）化合物与式R7-A-X2（Ⅶ）化合物反应，其中X 2为离去基团，并进一步使由此得到的式（Ⅳ）化合物与根据方法a2）的示例，orb2）如果合适，在碱性或酸性催化剂存在下，使其与羟胺或其盐反应，以及进一步使由式（II）得到的化合物，例如按照方法a1）进行反应，或者使上述式（Ⅷ）化合物与亚硝酸C 1 -C 6烷基酯反应，并进一步使由此得到的化合物，式（Ⅵ）化合物的方法，例如根据方法b），式（II），（Ⅳ）和（Ⅵ）化合物的E异构体，其制备方法及其制备方法式（I）。

4. 发明授权

US06313166B1 Phenyl acetic acid derivatives as pesticides 失效
标题翻译：苯乙酸衍生物作为农药
公开(公告)号：US06313166B1
公开(公告)日：2001-11-06
申请号：US09338236
申请日：1999-06-22
申请人： Hugo Ziegler , Stephan Trah , Saleem Farooq , René Zurflüh
发明人： Hugo Ziegler , Stephan Trah , Saleem Farooq , René Zurflüh
IPC分类号： A01N3734
CPC分类号： C07D213/77 , A01N37/36 , A01N37/50 , A01N43/28 , A01N43/30 , A01N43/36 , A01N43/40 , A01N43/46 , A01N43/653 , A01N43/84 , A01N55/00 , C07C251/60 , C07C251/76 , C07C251/80 , C07C255/54 , C07C255/61 , C07C2601/02 , C07D231/12 , C07D233/56 , C07D249/08 , C07D295/088 , C07D295/30 , C07D317/18 , C07D317/58 , C07D333/22
摘要： Compounds of the formula I and the isomers thereof, in which either a) X is an N atom and Y is OR11 or N(R12)R13, or b) X is CH and Y is OR11, and in which furthermore: R11 is C1-C4alkyl; R12 and R13, independenty, are hydrogen or C1-C4alkyl; A is an O atom or the group NR4; and wherein R1, R2 and R3 are as defined herein, are pesticidal active ingredients. They can be used for pest control, in particular as microbicides, insecticides and acaricides in agriculture, horticulture and in the hygiene sector.
摘要翻译：其中a）X是N原子，Y是OR 11或N（R 12）R 13，orb）X是CH，Y是OR 11，此外：R 11是C 1 -C 4烷基; R 12和 R 13独立地为氢或C 1 -C 4烷基; A为O原子或NR 4基团; 并且其中R1，R2和R3如本文所定义，是杀虫活性成分。它们可用于害虫防治，特别是农业，园艺和卫生领域的杀微生物剂，杀虫剂和杀螨剂。

5. 发明授权

US6156923A Process for the preparation of pesticides 失效
标题翻译：农药制备工艺
公开(公告)号：US6156923A
公开(公告)日：2000-12-05
申请号：US762217
申请日：1996-12-06
申请人： Saleem Farooq , Stephan Trah , Hugo Ziegler , Rene Zurfluh
发明人： Saleem Farooq , Stephan Trah , Hugo Ziegler , Rene Zurfluh
IPC分类号： C07C249/04 , C07C249/12 , C07C251/48 , C07C251/60
CPC分类号： C07C249/12 , C07C251/48 , C07C251/60
摘要： The invention relates to a process for the preparation of compounds of the formula ##STR1## or, if appropriate, a tautomer thereof, in each case in the free form or in salt form, in whichA, X, Y, Z, R.sub.2, R.sub.3, R.sub.4, R.sub.5, R.sub.7, R.sub.9 and n are as defined in claim 1 and the C.dbd.N double bond marked with E has the E configuration, which comprisesa1) reacting either a compound of the formula (II) mentioned above with a compound of the formula (III) mentioned above, in which X.sub.1 is a leaving group, ora2) a compound of the formula (IV) mentioned above, if appropriate in the presence of a base, with a compound of the formula (V) mentioned above, orb1) reacting a compound of the formula (VI) mentioned above with a compound of the formula R.sub.7 --A--X.sub.2 (VII), in which X.sub.2 is a leaving group, and either further reacting the compound thus obtainable, of the formula (IV), for example according to method a2), orb2) reacting it with hydroxylamine or a salt thereof, if appropriate in the presence of a basic or acid catalyst, and further reacting the compound thus obtainable, of the formula (II), for example according to method a1), orc) reacting a compound of the formula (VII), mentioned above with a C.sub.1 -C.sub.6 alkyl nitrite and further reacting the compound thus obtainable, of the formula (VI), for example according to method b), the E isomers of the compounds of the formulae (II), (IV) and (VI), a process for their preparation and their use for the preparation of compounds of the formula (I).
摘要翻译：本发明涉及一种制备下式的化合物或其合适的互变异构体的方法，其各自为游离形式或盐形式，其中A，X，Y，Z，R 2，R 3，R 4 ，R 5，R 7，R 9和n如权利要求1中所定义，并且用E标记的C = N双键具有E构型，其包括a1）使上述式（II）的化合物与上述式（III），其中X1是离去基团，或a2）上述式（Ⅳ）化合物，如果合适，在碱的存在下，与上述式（Ⅴ）化合物，或b1）使上述式（Ⅵ）化合物与式R7-A-X2（Ⅶ）化合物反应，其中X 2为离去基团，并进一步使由此得到的化合物（式（Ⅴ） IV），例如根据方法a2），或b2）如果合适，在碱性或酸性催化剂存在下，使其与羟胺或其盐反应，进一步使由式（II）得到的化合物，例如按照方法a1）进行反应，或c）使上述式（Ⅶ）化合物与亚硝酸C 1 -C 6烷基酯反应，然后进一步使化合物式（Ⅵ）化合物的E异构体，其制备方法及其制备方法（Ⅵ）的制备方法及其制备方法式（I）的化合物。

6. 发明授权

US5756426A Phenyl acetic acid derivatives as pesticides 失效
标题翻译：苯乙酸衍生物作为农药
公开(公告)号：US5756426A
公开(公告)日：1998-05-26
申请号：US526859
申请日：1995-09-11
申请人： Hugo Ziegler , Stephan Trah , Saleem Farooq , Rene Zurfluh
发明人： Hugo Ziegler , Stephan Trah , Saleem Farooq , Rene Zurfluh
IPC分类号： A01N37/34 , A01N37/36 , A01N37/44 , A01N37/50 , A01N43/28 , A01N43/30 , A01N43/36 , A01N43/40 , A01N43/46 , A01N43/653 , A01N43/84 , A01N55/00 , C07C229/00 , C07C251/60 , C07C251/76 , C07C251/80 , C07C255/00 , C07C255/54 , C07C255/61 , C07D213/77 , C07D295/088 , C07D295/30 , C07D317/18 , C07D317/58 , C07D333/22 , C07D521/00 , A61K31/275
CPC分类号： C07D213/77 , A01N37/36 , A01N37/50 , A01N43/28 , A01N43/30 , A01N43/36 , A01N43/40 , A01N43/46 , A01N43/653 , A01N43/84 , A01N55/00 , C07C251/60 , C07C251/76 , C07C251/80 , C07C255/54 , C07C255/61 , C07D231/12 , C07D233/56 , C07D249/08 , C07D295/088 , C07D295/30 , C07D317/18 , C07D317/58 , C07D333/22 , C07C2101/02
摘要： Described herein are compounds of the formula I ##STR1## and the isomers thereof, in which either a) X is an N atom and Y is OR.sub.11 or N(R.sub.12)R.sub.13, or b) X is CH and Y is OR.sub.11, and in which furthermore: R.sub.11 is C.sub.1 -C.sub.4 alkyl; R.sub.12 and R.sub.13, independently, are hydrogen or C.sub.1 -C.sub.4 alkyl; A is an O atom or the group NR.sub.4 ; and wherein R.sub.1, R.sub.2 and R.sub.3 are as defined herein, are pesticidal active ingredients. They can be used for pest control, in particular as microbicides, insecticides and acaricides in agriculture, horticulture and in the hygiene sector.
摘要翻译：本文描述的是式I的化合物及其异构体，其中a）X是N原子，Y是OR 11或N（R 12）R 13，或b）X是CH，Y是OR 11，以及其中R11为C1-C4烷基; R 12和R 13独立地是氢或C 1 -C 4烷基; A是O原子或NR4基团; 并且其中R1，R2和R3如本文所定义，是农药活性成分。它们可以用于害虫控制，特别是作为农业，园艺和卫生领域的杀菌剂，杀虫剂和杀螨剂。

7. 发明授权

US5981585A Phenyl acetic acid derivatives as pesticides 失效
标题翻译：苯乙酸衍生物作为农药
公开(公告)号：US5981585A
公开(公告)日：1999-11-09
申请号：US968143
申请日：1997-11-12
申请人： Hugo Ziegler , Stephan Trah , Saleem Farooq , Rene Zurfluh
发明人： Hugo Ziegler , Stephan Trah , Saleem Farooq , Rene Zurfluh
IPC分类号： A01N37/34 , A01N37/36 , A01N37/44 , A01N37/50 , A01N43/28 , A01N43/30 , A01N43/36 , A01N43/40 , A01N43/46 , A01N43/653 , A01N43/84 , A01N55/00 , C07C229/00 , C07C251/60 , C07C251/76 , C07C251/80 , C07C255/00 , C07C255/54 , C07C255/61 , C07D213/77 , C07D295/088 , C07D295/30 , C07D317/18 , C07D317/58 , C07D333/22 , C07D521/00 , A61K31/24 , A01N37/12
CPC分类号： C07D213/77 , A01N37/36 , A01N37/50 , A01N43/28 , A01N43/30 , A01N43/36 , A01N43/40 , A01N43/46 , A01N43/653 , A01N43/84 , A01N55/00 , C07C251/60 , C07C251/76 , C07C251/80 , C07C255/54 , C07C255/61 , C07D231/12 , C07D233/56 , C07D249/08 , C07D295/088 , C07D295/30 , C07D317/18 , C07D317/58 , C07D333/22 , C07C2101/02
摘要： Compounds of the formula I ##STR1## and the isomers thereof, in which either a) X is an N atom and Y is OR.sub.11 or N(R.sub.12)R.sub.13, orb) X is CH and Y is OR.sub.11,and in which furthermore:R.sub.11 is C.sub.1 -C.sub.4 alkyl;R.sub.12 and R.sub.13, independently, are hydrogen or C.sub.1 -C.sub.4 alkyl;A is an O atom or the group NR.sub.4 ; and whereinR.sub.1, R.sub.2 and R.sub.3 are as defined herein, are pesticidal active ingredients. They can be used for pest control, in particular as microbicides, insecticides and acaricides in agriculture, horticulture and in the hygiene sector.
摘要翻译：式Ⅰ化合物及其异构体，其中a）X为N原子，Y为OR 11或N（R 12）R 13，或b）X为CH，Y为OR 11，此外，R 11为Cl -C 1-4烷基; R 12和R 13独立地是氢或C 1 -C 4烷基; A是O原子或NR4基团; 并且其中R1，R2和R3如本文所定义，是农药活性成分。它们可以用于害虫控制，特别是作为农业，园艺和卫生领域的杀菌剂，杀虫剂和杀螨剂。

8. 发明授权

US06372787B1 Phenyl-methoxyimino-glyoxylic acid derivatives as pesticides 失效
标题翻译：苯甲氧基亚氨基 - 乙醛酸衍生物作为农药
公开(公告)号：US06372787B1
公开(公告)日：2002-04-16
申请号：US09671421
申请日：2000-09-27
申请人： Hugo Ziegler , René Zurflüh
发明人： Hugo Ziegler , René Zurflüh
IPC分类号： C07C22940
CPC分类号： C07C251/58 , A01N37/50 , C07C251/48 , C07C251/86 , C07C251/88 , C07C2601/02
摘要： Compounds of formula I wherein A is a group OCHR4 or N═CR4; Y is O or NH, R1 is C1-C6-alkyl; R2 is C1-C6-alkyl or C1-C6-alkyl substituted by 1 to 5 fluorine atoms; R3 is C1-C6-alkyl, C1-C6-alkoxy, C3-C6-cycloalkyl, C3-C6-cycloalkoxy, C2-C6-alkenyl, C2-C6-alkenyloxy, C2-C6-alkinyl, C2-C6-alkinyloxy, C1-C6-alkoxycarbonyl, CN or halogen, aryl, hetaryl, heterocyclyl, aryloxy, hetaryloxy or heterocyclyloxy, whereby the above-mentioned groups, with the exception of CN and halogen, may be substituted by the same or different substituents; R4 is methyl, ethyl or cyclopropyl; R6 is hydrogen or methyl; have microbicidal, insecticidal and acaricidal activity, and may be used to control plant-pathogenic fungi, acarids and insects in agriculture and in the field of hygiene.
摘要翻译：式I的化合物，其中A是基团OCHR 4或N = CR 4; Y是O或NH，R 1是C 1 -C 6烷基; R 2是被1至5个氟原子取代的C 1 -C 6烷基或C 1 -C 6烷基; R 3是 C 1 -C 6 - 烷基，C 1 -C 6 - 烷氧基，C 3 -C 6 - 环烷基，C 3 -C 6 - 环烷氧基，C 2 -C 6 - 烯基，C 2 -C 6 - 烯氧基，C 2 -C 6 - C 6 - 烷氧基羰基，CN或卤素，芳基，杂芳基，杂环基，芳氧基，杂芳氧基或杂环氧基，其中除CN和卤素以外的上述基团可以被相同或不同的取代基取代; R4是甲基，乙基或环丙基; R 6为氢或甲基;具有杀菌，杀虫和杀螨活性，可用于控制农业和卫生领域的植物病原真菌，螨虫和昆虫。

9. 发明授权

US06664422B1 Process for the preparation of strobilurin intermediates 失效
标题翻译：制备嗜球果伞素中间体的方法
公开(公告)号：US06664422B1
公开(公告)日：2003-12-16
申请号：US09857391
申请日：2001-08-13
申请人： Rudolf Waditschatka , René Zurflüh , Edward Kelsall , Hugo Ziegler , Linhua Wang
发明人： Rudolf Waditschatka , René Zurflüh , Edward Kelsall , Hugo Ziegler , Linhua Wang
IPC分类号： C07C24900
CPC分类号： C07C249/08 , C07C45/00 , C07C49/233 , C07C251/48
摘要： The present invention relates to a novel improved process and intermediates for the process of preparing the oxime intermediates of formula (II) wherein R1 is hydrogen, fluoro or chloro, and R2 is methyl, ethyl, methoxy, ethoxy, trifluoromethyl, trifluoromethoxy, cyano, fluoro, chloro or bromo. The novel process comprises diazotizing an aniline of formula (VI) reacting the resulting diazonium salt with isopropenylacetate of formula (X) and reacting the resulting ketone of formula (XI) with an organic nitrite in the presence of hydrogene chloride, and methylating the resulting ketooxime of formula (VIII) with a methylating agent and reacting the resulting O-methyl ketooxime of formula (IX) with hydroxylamine. The compounds of formula (II) are intermediates for highly active fungicides from the class of the strobilurins.
摘要翻译：本发明涉及制备式（II）的肟中间体的方法和中间体，其中R1是氢，氟或氯，R2是甲基，乙基，甲氧基，乙氧基，三氟甲基，三氟甲氧基，氰基，氟，氯或溴。该新方法包括使式（Ⅵ）的苯胺重氮化，使得到的重氮盐与式（X）的异丙烯基乙酸酯反应，并使所得的式（Ⅺ）酮与有机亚硝酸酯在氯化氢存在下反应，并使所得酮肟甲基化（VIII）与甲基化剂反应，并使所得的式（IX）的O-甲基酮肟与羟胺反应。式（II）化合物是来自嗜球果伞素类的高活性杀真菌剂的中间体。

10. 发明授权

US06525092B1 Pesticidal bis-oxime compounds 失效
标题翻译：杀虫双肟化合物
公开(公告)号：US06525092B1
公开(公告)日：2003-02-25
申请号：US09787481
申请日：2001-04-27
申请人： Hugo Ziegler , Stephan Trah
发明人： Hugo Ziegler , Stephan Trah
IPC分类号： A01N3734
CPC分类号： C07C251/48 , A01N37/50 , C07C251/60 , C07C255/61
摘要： Bis-oxime compounds of the general formula (I) are provided wherein X, Y, R1, R2 R3 and n are as defined in the specification. The bis-oxime compounds possess pesticidal activity, which may provide plants with protection from phytopathogenic microorganisms.
摘要翻译：提供通式（I）的双肟化合物，其中X，Y，R 1，R 2，R 3和n如说明书中所定义。双肟化合物具有杀虫活性，可为植物提供植物病原微生物的保护。

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