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1. 发明授权

US06890932B2 Anthranilic acid derivative 失效
标题翻译：邻氨基苯甲酸衍生物
公开(公告)号：US06890932B2
公开(公告)日：2005-05-10
申请号：US10355125
申请日：2003-01-31
申请人： Naoki Tsuchiya , Susumu Takeuchi , Takumi Takeyasu , Naoki Hase , Takao Yamori , Takashi Tsuruo
发明人： Naoki Tsuchiya , Susumu Takeuchi , Takumi Takeyasu , Naoki Hase , Takao Yamori , Takashi Tsuruo
IPC分类号： C07C235/38 , C07C235/56 , C07C271/16 , C07C271/26 , C07C307/08 , C07C311/07 , C07C311/20 , C07C311/29 , C07C323/25 , C07C323/30 , C07C323/41 , C07C323/42 , C07C323/43 , C07C323/60 , C07C323/62 , C07C327/44 , C07D207/08 , C07D211/02 , C07D211/46 , C07D213/30 , C07D213/64 , C07D213/643 , C07D213/70 , C07D213/82 , C07D213/89 , C07D295/092 , C07D295/185 , C07D307/42 , C07D307/58 , C07D309/10 , C07D405/12 , A61K31/435 , A01N43/40 , C07D213/00 , C07D213/63
CPC分类号： C07D207/08 , C07C235/38 , C07C235/56 , C07C271/16 , C07C271/26 , C07C307/08 , C07C311/07 , C07C311/20 , C07C311/29 , C07C323/25 , C07C323/30 , C07C323/41 , C07C323/42 , C07C323/43 , C07C323/60 , C07C323/62 , C07C327/44 , C07C2601/08 , C07C2601/14 , C07C2601/18 , C07C2601/20 , C07C2602/28 , C07D211/02 , C07D211/46 , C07D213/30 , C07D213/64 , C07D213/643 , C07D213/70 , C07D213/82 , C07D213/89 , C07D295/088 , C07D295/185 , C07D307/42 , C07D307/58 , C07D309/10 , C07D405/12
摘要： The present invention relates to an anthranilic acid derivative expressed by the following formula (1) or the following formula (2), or its pharmacologically permissible salt or solvate.
摘要翻译：本发明涉及由下式（1）或下式（2）表示的邻氨基苯甲酸衍生物或其药理学上允许的盐或溶剂合物。

2. 发明授权

US06649656B1 Anthranilic acid derivatives 失效
标题翻译：邻氨基苯甲酸衍生物
公开(公告)号：US06649656B1
公开(公告)日：2003-11-18
申请号：US09744388
申请日：2001-04-04
申请人： Naoki Tsuchiya , Susumu Takeuchi , Takumi Takeyasu , Naoki Hase , Takao Yamori , Takashi Tsuruo
发明人： Naoki Tsuchiya , Susumu Takeuchi , Takumi Takeyasu , Naoki Hase , Takao Yamori , Takashi Tsuruo
IPC分类号： A61K31195
CPC分类号： C07D207/08 , C07C235/38 , C07C235/56 , C07C271/16 , C07C271/26 , C07C307/08 , C07C311/07 , C07C311/20 , C07C311/29 , C07C323/25 , C07C323/30 , C07C323/41 , C07C323/42 , C07C323/43 , C07C323/60 , C07C323/62 , C07C327/44 , C07C2601/08 , C07C2601/14 , C07C2601/18 , C07C2601/20 , C07C2602/28 , C07D211/02 , C07D211/46 , C07D213/30 , C07D213/64 , C07D213/643 , C07D213/70 , C07D213/82 , C07D213/89 , C07D295/088 , C07D295/185 , C07D307/42 , C07D307/58 , C07D309/10 , C07D405/12
摘要： The present invention relates to an anthranilic acid derivative expressed by the following formula (1) or the following formula (2), or its pharmacologically permissible salt or solvate.
摘要翻译：本发明涉及由下式（1）或下式（2）表示的邻氨基苯甲酸衍生物或其药理学上允许的盐或溶剂合物。

3. 发明申请

US20050267148A1 Benzimidazole derivative 审中-公开
标题翻译：苯并咪唑衍生物
公开(公告)号：US20050267148A1
公开(公告)日：2005-12-01
申请号：US11129508
申请日：2005-05-16
申请人： Naoki Tsuchiya , Tsuyoshi Mizuno , Hiroshi Saitou , Yoshiyuki Matsumoto , Susumu Takeuchi , Naoki Hase
发明人： Naoki Tsuchiya , Tsuyoshi Mizuno , Hiroshi Saitou , Yoshiyuki Matsumoto , Susumu Takeuchi , Naoki Hase
IPC分类号： A61K31/4184 , A61K31/4745 , C07D401/06 , C07D403/06 , C07D405/06 , C07D409/06 , C07D413/06 , C07D471/02
CPC分类号： C07D401/06 , C07D403/06 , C07D405/06 , C07D409/06 , C07D413/06
摘要： The present invention is a thiobenzimidazole derivative represented by the following formula (1) or a medically acceptable salt thereof wherein said thiobenzimidazole derivative and a medically acceptable salt thereof have a potent activity of inhibiting human chymase. Thus, they are potential preventive and/or therapeutic agents clinically applicable to various diseases in which human chymase is involved.
摘要翻译：本发明是由下式（1）表示的硫代苯并咪唑衍生物或其医学上可接受的盐，其中所述硫代苯并咪唑衍生物及其医学上可接受的盐具有抑制人胃促胰酶的有效活性。因此，它们是临床适用于涉及人胃促胰酶的各种疾病的潜在的预防和/或治疗剂。

4. 发明申请

US20070073064A1 Method for producing aminopyrrolidine derivatives and intermediate compounds 审中-公开
标题翻译：制备氨基吡咯烷衍生物和中间体化合物的方法
公开(公告)号：US20070073064A1
公开(公告)日：2007-03-29
申请号：US10574688
申请日：2004-10-07
申请人： Takumi Takeyasu , Yoshinori Sato , Minoru Imai , Mitsuru Sakai , Kenji Manabe , Yoshiyuki Matsumoto , Susumu Takeuchi , Asahi Kawana , Masahiro Koga , Mitsuharu Asahita
发明人： Takumi Takeyasu , Yoshinori Sato , Minoru Imai , Mitsuru Sakai , Kenji Manabe , Yoshiyuki Matsumoto , Susumu Takeuchi , Asahi Kawana , Masahiro Koga , Mitsuharu Asahita
IPC分类号： C07D403/02
CPC分类号： C07C237/44 , C07D403/06
摘要： There is provided an industrial production method of an aminopyrrolidine derivative having chemokine receptor antagonist activity represented by the following formula, a synthetic intermediate thereof and a production method thereof: wherein R11 is H, C1-C6 alkyl or C2-C7 alkanoyl; R12, R14, R15, R16 and R17 are H, halogen, optionally halogenated C1-C6 alkyl, optionally halogenated C1-C6 alkoxy, hydroxyl or C2-C7 alkoxycarbonyl; R23, R24, R25 and R26 are H, halogen, optionally halogenated C1-C6 alkyl, optionally halogenated C1-C6 alkoxy or hydroxyl; and R3 is H or C1-C6 alkyl.
摘要翻译：提供了具有下式表示的趋化因子受体拮抗剂活性的氨基吡咯烷衍生物及其合成中间体及其制备方法的工业生产方法：其中R 11是H，C 1 C 6 -C 6烷基或C 2 -C 7烷酰基; R 12，R 14，R 15，R 16和R 17均为 H，卤素，任选卤代C 1 -C 6烷基，任意卤代C 1 -C 6烷氧基，羟基或C 2 -C 7烷氧基羰基; R 23，R 24，R 25和R 26是H，卤素，任选卤代的C 1 -C 12烷基， C 1 -C 6烷基，任选卤代C 1 -C 6烷氧基或羟基; R 3是H或C 1 -C 6烷基。

5. 发明授权

US07268145B2 Thiobenzimidazole derivatives 失效
标题翻译：硫代苯并咪唑衍生物
公开(公告)号：US07268145B2
公开(公告)日：2007-09-11
申请号：US10963710
申请日：2004-10-14
申请人： Yoshiyuki Matsumoto , Susumu Takeuchi , Naoki Hase
发明人： Yoshiyuki Matsumoto , Susumu Takeuchi , Naoki Hase
IPC分类号： A01N43/42 , A01N43/52 , A61K31/44 , A61K31/415 , C07D513/02
CPC分类号： C07D401/12 , C07D235/28 , C07D405/12 , C07D409/12 , C07D413/12 , C07D417/12 , C07D471/04
摘要： The present invention is a thiobenzimidazole derivative represented by the following formula (1) or a medically acceptable salt thereof wherein said thiobenzimidazole derivative and a medically acceptable salt thereof have a potent activity of inhibiting human chymase. Thus, they are potential preventive and/or therapeutic agents clinically applicable to various diseases in which human chymase is involved.
摘要翻译：本发明是由下式（1）表示的硫代苯并咪唑衍生物或其医学上可接受的盐，其中所述硫代苯并咪唑衍生物及其医学上可接受的盐具有抑制人胃促胰酶的有效活性。因此，它们是临床适用于涉及人胃促胰酶的各种疾病的潜在的预防和/或治疗剂。

6. 发明申请

US20060040976A1 Thiobenzimidazole derivatives 失效
标题翻译：硫代苯并咪唑衍生物
公开(公告)号：US20060040976A1
公开(公告)日：2006-02-23
申请号：US10963710
申请日：2004-10-14
申请人： Yoshiyuki Matsumoto , Susumu Takeuchi , Naoki Hase
发明人： Yoshiyuki Matsumoto , Susumu Takeuchi , Naoki Hase
IPC分类号： C07D471/02 , A61K31/4745 , A61K31/4184
CPC分类号： C07D401/12 , C07D235/28 , C07D405/12 , C07D409/12 , C07D413/12 , C07D417/12 , C07D471/04
摘要： The present invention is a thiobenzimidazole derivative represented by the following formula (1) or a medically acceptable salt thereof wherein said thiobenzimidazole derivative and a medically acceptable salt thereof have a potent activity of inhibiting human chymase. Thus, they are potential preventive and/or therapeutic agents clinically applicable to various diseases in which human chymase is involved.
摘要翻译：本发明是由下式（1）表示的硫代苯并咪唑衍生物或其医学上可接受的盐，其中所述硫代苯并咪唑衍生物及其医学上可接受的盐具有抑制人胃促胰酶的有效活性。因此，它们是临床适用于涉及人胃促胰酶的各种疾病的潜在的预防和/或治疗剂。

7. 发明申请

US20070275995A1 Thiobenzimidazole derivatives 审中-公开
公开(公告)号：US20070275995A1
公开(公告)日：2007-11-29
申请号：US11797975
申请日：2007-05-09
申请人： Yoshiyuki Matsumoto , Susumu Takeuchi , Naoki Hase
发明人： Yoshiyuki Matsumoto , Susumu Takeuchi , Naoki Hase
IPC分类号： A61K31/4164 , A61K31/44 , A61P19/00 , A61P19/02 , A61P37/08 , A61P9/00
CPC分类号： C07D401/12 , C07D235/28 , C07D405/12 , C07D409/12 , C07D413/12 , C07D417/12 , C07D471/04
摘要： The present invention is a thiobenzimidazole derivative represented by the following formula (1) or a medically acceptable salt thereof wherein said thiobenzimidazole derivative and a medically acceptable salt thereof have a potent activity of inhibiting human chymase. Thus, they are potential preventive and/or therapeutic agents clinically applicable to various diseases in which human chymase is involved.

8. 发明授权

US07517875B2 Piperidine derivatives having CCR3 antagonism 失效
标题翻译：具有CCR3拮抗作用的哌啶衍生物
公开(公告)号：US07517875B2
公开(公告)日：2009-04-14
申请号：US10511174
申请日：2003-04-16
申请人： Yoshiyuki Matsumoto , Minoru Imai , Yoshiyuki Sawai , Susumu Takeuchi , Akinobu Nakanishi , Kunio Minamizono , Tomonori Yokoyama
发明人： Yoshiyuki Matsumoto , Minoru Imai , Yoshiyuki Sawai , Susumu Takeuchi , Akinobu Nakanishi , Kunio Minamizono , Tomonori Yokoyama
IPC分类号： C07D487/04 , C07D403/12 , C07D403/14 , A61K31/4523 , A61K31/454 , A61P11/06
CPC分类号： C07D401/12 , A61K31/454 , A61K31/4545 , A61K31/4709 , A61K31/517 , A61K31/5377 , A61K31/5415 , C07D401/14 , C07D405/14 , C07D409/14 , C07D413/14 , C07D417/14 , C07D487/04
摘要： The invention provides low molecular compounds having activity which inhibits binding of CCR3 ligands to CCR3 on target cells, i.e. CCR3 antagonists. The invention also provides compounds represented by formula (I) below, pharmaceutically acceptable acid adducts thereof, or pharmaceutically acceptable C1-C6 alkyl adducts thereof, as well as pharmaceutical compositions comprising them as effective ingredients, which are useful for treatment or prevention of diseases associated with CCR3, such as asthma and allergic rhinitis.
摘要翻译：本发明提供具有抑制靶细胞CCR3拮抗剂上CCR3配体与CCR3结合的活性的低分子化合物。本发明还提供由下式（I）表示的化合物，其药学上可接受的酸加合物或其药学上可接受的C1-C6烷基加合物，以及包含它们作为有效成分的药物组合物，其可用于治疗或预防相关疾病与CCR3，如哮喘和过敏性鼻炎。

9. 发明授权

US5132186A Mask for X-ray lithography and method of manufacturing the same 失效
标题翻译：掩蔽X射线光刻及其制造方法
公开(公告)号：US5132186A
公开(公告)日：1992-07-21
申请号：US678423
申请日：1991-04-01
申请人： Susumu Takeuchi , Nobuyuki Yoshioka
发明人： Susumu Takeuchi , Nobuyuki Yoshioka
IPC分类号： G03F1/00 , G03F1/22 , G03F1/84 , G03F1/86 , H01L21/027
CPC分类号： G03F1/22 , Y10S430/167
摘要： A mask for X-ray lithography includes a transparent thin film (1) of SiC, an X-ray absorbing pattern (2) of Au formed on the surface of the transparent thin film (1) and a support member (3) of Si formed on the back surface of the transparent thin film (1). The support member (3) has an opening (4) for exposing the back surface of the transparent thin film (1). A transparent conductive thin film (5) of In.sub.2 O.sub.3 is formed over the back surfaces of the exposed transparent thin film (1) and the support member (3).

10. 发明授权

US4794646A Charged beam pattern defect inspection apparatus 失效
标题翻译：充电光束图案缺陷检查装置
公开(公告)号：US4794646A
公开(公告)日：1988-12-27
申请号：US896213
申请日：1986-08-14
申请人： Susumu Takeuchi , Koichi Moriizumi
发明人： Susumu Takeuchi , Koichi Moriizumi
IPC分类号： H01L21/66 , G01N23/18 , G01Q10/06 , G06T7/00 , H01J37/28 , G06K9/00 , G06K9/62
CPC分类号： G06T7/001 , G01N23/18 , G06T2207/10061 , G06T2207/20036 , G06T2207/30148
摘要： A charged beam pattern defect inspection apparatus for inspecting pattern defects on materials such as masks or wafers comprising: a collecting charged beam irradiation apparatus including scanning deflection device for accelerating and focusing the scanning beam, and a detector for detecting phenomenon produced by incident particles such as reflected electrons, secondary electrons, cathodeluminescent light, X rays, or absorption currents; a scanning and synchronous signal generator for generating a scanning signal to be control the scanning deflection means and a synchronous signal to fed into an A/D converter; a two-dimensional video memory including an A/D converter and an address signal generator; a video signal operator for operating the video signal stored in the two-dimensional video memory; a stage driving apparatus for driving a stage for holding the material to be inspected, which includes a position detector for detecting the position of the stage; an auxiliary memory device for storing inspection data; and a control operation apparatus for controlling the scanning and synchronous signal generator, the two dimensional video memory, the video signal operator, the stage driving apparatus, and the auxiliary memory device, and for outputting the output of the video signal operator as the result of pattern defect inspection.
摘要翻译：一种用于检查诸如掩模或晶片的材料上的图案缺陷的带电束图案缺陷检查装置，包括：包括用于加速和聚焦扫描光束的扫描偏转装置的收集带电束照射装置，以及用于检测由诸如反射电子，二次电子，阴极发光，X射线或吸收电流; 用于产生要控制扫描偏转装置的扫描信号和馈送到A / D转换器的同步信号的扫描和同步信号发生器; 包括A / D转换器和地址信号发生器的二维视频存储器; 用于操作存储在二维视频存储器中的视频信号的视频信号操作器; 用于驱动用于保持待检查材料的台架的舞台驱动装置，其包括用于检测舞台位置的位置检测器; 用于存储检查数据的辅助存储装置; 以及用于控制扫描和同步信号发生器，二维视频存储器，视频信号操作器，平台驱动装置和辅助存储装置的控制操作装置，并且用于输出视频信号操作器的输出作为结果图案缺陷检查。

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