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1. 发明授权

US07829580B2 Cyclic amine derivative having heteroaryl ring 失效
标题翻译：具有杂芳基环的环胺衍生物
公开(公告)号：US07829580B2
公开(公告)日：2010-11-09
申请号：US11442429
申请日：2006-05-26
申请人： Tomio Kimura , Naoki Tanaka , Atsuhiro Sugidachi , Toshiyuki Konosu
发明人： Tomio Kimura , Naoki Tanaka , Atsuhiro Sugidachi , Toshiyuki Konosu
IPC分类号： A61K31/445 , C07D211/54
CPC分类号： C07D211/72 , C07D401/06 , C07D401/14 , C07D405/06 , C07D409/06 , C07D413/06 , C07D417/06
摘要： A compound having the general formula (I) wherein R1 represents C1-C6 alkyl, etc., R2 represents hydrogen, C2-C7 alkanoyl, C7-C11 arylcarbonyl, the formula R4—(CH2)l—, etc., R3 represents C6-C10 aryl, etc., X1, X2, X3, X4 and X5 each independently represents hydrogen, halogen, etc., and n represents an integer of 0 to 2, pharmacologically acceptable salts thereof or prodrugs thereof. They have excellent inhibition of platelet activation, etc. and are useful as a prophylactic or therapeutic agents for diseases related to thrombus or embolus formation.
摘要翻译：具有通式（I）的化合物，其中R1表示C1-C6烷基等，R2表示氢，C2-C7烷酰基，C7-C11芳基羰基，式R4-（CH2）-1-等，R3表示C6 -C 10芳基等，X 1，X 2，X 3，X 4和X 5各自独立地表示氢，卤素等，n表示0〜2的整数，其药理学上可接受的盐或其前药。它们具有优异的血小板活化抑制等，并且可用作与血栓或栓塞形成有关的疾病的预防或治疗剂。

2. 发明申请

US20100201810A1 IMAGE DISPLAY APPARATUS AND IMAGE DISPLAY METHOD 审中-公开
标题翻译：图像显示装置和图像显示方法
公开(公告)号：US20100201810A1
公开(公告)日：2010-08-12
申请号：US12676063
申请日：2008-10-06
申请人： Kazunori Shimazaki , Tomio Kimura , Yutaka Nakashima , Masami Tomioka
发明人： Kazunori Shimazaki , Tomio Kimura , Yutaka Nakashima , Masami Tomioka
IPC分类号： H04N7/18
CPC分类号： B60R1/00 , B60R11/04 , B60R2300/30 , B60R2300/301 , B60R2300/303 , B60R2300/607 , B60R2300/806 , G06T7/73 , G06T2207/30204 , G06T2207/30264
摘要： Images are taken by a fixed camera and a moving camera, and a relative position calculation unit recognizes a current position and orientation of the moving object based on a detection signal that is input from a sensor for obtaining positional information of a moving object and calculates a relative positional relationship of the moving camera with respect to the fixed camera by comparing the current position and orientation of the moving object with a given position at which the fixed camera is installed. Based on the relative positional relationship, the image taken by the fixed camera and the image taken by the moving camera are synthesized into one image by an image composition unit, and a composite image viewed from a virtual viewpoint is displayed on a monitor.
摘要翻译：图像由固定摄像机和移动摄像机拍摄，相对位置计算单元基于从用于获取移动物体的位置信息的传感器输入的检测信号来识别移动物体的当前位置和姿态，并且计算出通过将移动物体的当前位置和姿态与安装固定照相机的给定位置进行比较，移动摄像机相对于固定照相机的相对位置关系。基于相对位置关系，通过图像合成单元将由固定摄像机拍摄的图像和由移动摄像机拍摄的图像合成为一个图像，并且将从虚拟视点观看的合成图像显示在监视器上。

3. 再颁专利

USRE39420E1 1,2-Diphenylpyrrole derivatives, their preparation and their therapeutic uses 有权
标题翻译： 1,2-二苯基吡咯衍生物及其制备方法及其治疗用途
公开(公告)号：USRE39420E1
公开(公告)日：2006-12-05
申请号：US09678218
申请日：2000-09-29
申请人： Tomio Kimura , Yasuo Noguchi , Akira Nakao , Keisuke Suzuki , Shigeru Ushiyama , Akihiro Kawara , Masaaki Miyamoto
发明人： Tomio Kimura , Yasuo Noguchi , Akira Nakao , Keisuke Suzuki , Shigeru Ushiyama , Akihiro Kawara , Masaaki Miyamoto
IPC分类号： A61K31/40 , C07D207/333 , C07D207/335 , C07D207/337
CPC分类号： C07D207/333 , C07D207/335 , C07D207/337
摘要： Compounds of formula (I) and (II): [wherein R is hydrogen, halogen or alkyl; R1 is alkyl, amino or substituted amino; R2 is optionally substituted phenyl; R3 is hydrogen, halogen or optionally substituted alkyl; R4 is hydrogen, optionally substituted alkyl, cycloalkyl, aryl, or aralkyl] have valuable analgesic, anti-inflammatory, anti-pyretic and anti-allergic activities and have the ability to inhibit the production of leukotrienes and to inhibit bone resorption. They are relatively free from the side effects which generally result from the administration of compounds having these kinds of activities.
摘要翻译：式（I）和（II）的化合物：[其中R是氢，卤素或烷基; R 1是烷基，氨基或取代的氨基; R 2是任选取代的苯基; R 3是氢，卤素或任选取代的烷基; R 4是氢，任选取代的烷基，环烷基，芳基或芳烷基]具有有价值的镇痛，抗炎，抗裂解和抗过敏活性，并且具有抑制白三烯生产的能力和以抑制骨吸收。它们相对没有通常由施用具有这些活性的化合物引起的副作用。

4. 发明授权

US07091352B2 Compounds substituted with bicyclic amino groups 失效
标题翻译：被双环氨基取代的化合物
公开(公告)号：US07091352B2
公开(公告)日：2006-08-15
申请号：US10625024
申请日：2003-07-22
申请人： Tomio Kimura , Akira Nakao
发明人： Tomio Kimura , Akira Nakao
IPC分类号： C07D221/02
CPC分类号： C07D471/04 , C07D455/02 , C07D487/04
摘要： Compounds of the formula (I) below, or pharmacologically acceptable salts, esters or other derivatives thereof: wherein A is furan, thiophene, pyrazole, imidazole, isoxazole or isothiazole; R1 is a substituted or unsubstituted aryl or a substituted or unsubstituted heteroaryl; R2 is a substituted or unsubstituted heteroaryl; and R3 is a bicyclic amino group; provided that the substituents R1 and R2 are bonded to the two atoms of the cyclic group A which are adjacent to the atom of the cyclic group A to which the substituent R2 is bonded. The compounds inhibit the production of inflammatory cytokines.
摘要翻译：式（I）的化合物或其药理学上可接受的盐，酯或其衍生物：其中A为呋喃，噻吩，吡唑，咪唑，异恶唑或异噻唑; R 1是取代或未取代的芳基或取代或未取代的杂芳基; R 2是取代或未取代的杂芳基; R 3是双环氨基; 条件是取代基R 1和R 2与键合在与环状基团A的原子相邻的环状基团A的两个原子上，取代基R ^{2 键合。这些化合物抑制炎性细胞因子的产生。}

5. 发明授权

US07000586B2 Control device for compression ignition operation of internal combustion engine 失效
标题翻译：内燃机压缩点火运行控制装置
公开(公告)号：US07000586B2
公开(公告)日：2006-02-21
申请号：US10851648
申请日：2004-05-24
申请人： Akira Kato , Toru Kitamura , Tomio Kimura , Shohei Okazaki , Toshihiro Yamaki , Katsura Okubo
发明人： Akira Kato , Toru Kitamura , Tomio Kimura , Shohei Okazaki , Toshihiro Yamaki , Katsura Okubo
IPC分类号： F02B5/00 , F02M25/07 , F02D41/04
CPC分类号： F01N3/0842 , F01N3/0807 , F01N2430/085 , F02B1/12 , F02D41/006 , F02D41/3035 , F02D41/401 , F02D2200/703 , Y02T10/44
摘要： A controller for an internal combustion engine capable of performing a compression ignition operation. The internal combustion engine includes a combustion chamber, and a fuel injector for injecting fuel directly in the combustion chamber. The controller includes: an air pressure detecting unit configured to detect at least one of an air pressure and an exhaust air pressure; and a fuel injection control unit configured to actuate the fuel injector to control a fuel injection timing according to a detected result by the air pressure detecting unit. The fuel injection control unit puts the fuel injection timing forward as the detected result by the air pressure detecting unit is lowered.
摘要翻译：一种用于执行压缩点火操作的内燃机的控制器。内燃机包括燃烧室和用于直接在燃烧室中喷射燃料的燃料喷射器。控制器包括：气压检测单元，被配置为检测空气压力和排气压力中的至少一个; 以及燃料喷射控制单元，其构造成根据气压检测单元的检测结果致动燃料喷射器以控制燃料喷射正时。燃料喷射控制单元随着气压检测单元的检测结果降低而将燃料喷射正时向前。

6. 发明授权

US06711473B2 Parking assisting device 失效
标题翻译：停车辅助装置
公开(公告)号：US06711473B2
公开(公告)日：2004-03-23
申请号：US10176459
申请日：2002-06-21
申请人： Kazunori Shimazaki , Tomio Kimura , Satoshi Yamada
发明人： Kazunori Shimazaki , Tomio Kimura , Satoshi Yamada
IPC分类号： G06F700
CPC分类号： B62D15/028 , B60T2201/10
摘要： A parking assisting device is provided with: a yaw rate sensor for detecting a yaw angle of a vehicle; a controller having a navigation function control unit and a parking assisting function control unit; a function selecting switch for determining switching to a parking assisting mode from a navigation mode; a monitor for providing navigation information, as well as for setting the reference position of the yaw angle and selecting a parking mode; and a speaker for providing parking assisting information to a driver in accordance with a vehicle position specified on the basis of the yaw angle.
摘要翻译：一种停车辅助装置设置有用于检测车辆的偏航角的偏航率传感器; 控制器，具有导航功能控制单元和停车辅助功能控制单元; 功能选择开关，用于确定从导航模式切换到驻车辅助模式; 用于提供导航信息的监视器，以及用于设置偏航角的参考位置并选择停车模式; 以及扬声器，用于根据基于偏航角指定的车辆位置向驾驶员提供停车辅助信息。

7. 发明授权

US4997943A Quinoline-3-carboxylic acid derivatives 失效
标题翻译：喹啉-3-羧酸衍生物
公开(公告)号：US4997943A
公开(公告)日：1991-03-05
申请号：US33066
申请日：1987-03-31
申请人： Masayuki Iwata , Tomio Kimura , Yoshimi Fujihara , Tetsushi Katsube
发明人： Masayuki Iwata , Tomio Kimura , Yoshimi Fujihara , Tetsushi Katsube
IPC分类号： A61K31/47 , A61K31/495 , A61K31/535 , A61K31/54 , A61P31/04 , C07D215/56 , C07D215/58 , C07D401/04 , C07D521/00
CPC分类号： C07D215/56 , C07D215/58 , C07D231/12 , C07D233/56 , C07D249/08 , C07D401/04
摘要： Compounds of formula (I): ##STR1## (in which R.sup.1 is alkoxy, R is alkyl, haloalkyl, alkylamino, cycloalkyl or optionally substituted phenyl, X is chlorine or fluorine and Y is selected from certain specific heterocycles) have excellent antibacterial activity. They may be prepared by introducing the group represented by Y into the corresponding compound in which Y is replaced by a halogen atom.
摘要翻译：式（I）化合物：其中R 1为烷氧基，R为烷基，卤代烷基，烷基氨基，环烷基或任意取代的苯基，X为氯或氟，Y为某些特定杂环）抗菌活性。它们可以通过将由Y表示的基团引入到其中Y被卤素原子代替的相应化合物中来制备。

8. 发明申请

US20110298926A1 PARKING ASSISTANCE APPARATUS AND PARKING ASSISTANCE METHOD 审中-公开
标题翻译：停车辅助设备和停车辅助方法
公开(公告)号：US20110298926A1
公开(公告)日：2011-12-08
申请号：US13202004
申请日：2010-02-25
申请人： Hiroshi Katsunaga , Kazunori Shimazaki , Tomio Kimura , Yutaka Nakashima , Koji Hika , Keisuke Inoue
发明人： Hiroshi Katsunaga , Kazunori Shimazaki , Tomio Kimura , Yutaka Nakashima , Koji Hika , Keisuke Inoue
IPC分类号： H04N7/18
CPC分类号： B62D15/027 , G06K9/00798 , G06K9/00912 , G06T7/73 , G06T2207/30208 , G06T2207/30264 , G08G1/16 , G08G1/168
摘要： Provided is a parking assistance apparatus utilizing a fixed target by taking an image thereof, the parking assistance apparatus being capable of recognizing the fixed target with high recognition accuracy while using simple image recognition processing. A mark (M) includes a plurality of illuminators (1). Sets of the plurality of illuminators (1) form characteristic points C1 to C4. Turn-ON request generation means (36) of a vehicle-side device (20) sequentially generates turn-ON requests for each characteristic point and transmits the generated turn-ON requests to a parking-lot-side device (10). A display control unit (11) of the parking-lot-side device (10) turns ON the characteristic points based on the turn-ON requests. An image recognition unit (31) of the vehicle-side device (20) performs image recognition for the characteristic points sequentially. Using the recognition result, positional parameter calculation means (34) of the vehicle-side device (20) calculates positional parameters of a camera with respect to the mark (M).
摘要翻译：提供一种通过拍摄图像来利用固定目标的停车辅助装置，在使用简单的图像识别处理的同时，能够以高识别精度识别固定目标的停车辅助装置。标记（M）包括多个照明器（1）。多个照明器（1）的组合形成特征点C1〜C4。车辆侧设备（20）的接通请求产生装置（36）顺序地产生每个特征点的接通请求，并将生成的接通请求发送到停车场侧设备（10）。停车场侧装置（10）的显示控制单元（11）基于接通请求接通特征点。车辆侧装置（20）的图像识别单元（31）依次对特征点进行图像识别。使用识别结果，车辆侧装置（20）的位置参数计算装置（34）计算相机相对于标记（M）的位置参数。

9. 发明申请

US20100060486A1 PARKING ASSIST APPARATUS 审中-公开
标题翻译：停车辅助装置
公开(公告)号：US20100060486A1
公开(公告)日：2010-03-11
申请号：US12556157
申请日：2009-09-09
申请人： Yutaka NAKASHIMA , Kazunori SHIMAZAKI , Tomio KIMURA , Koji HIKA
发明人： Yutaka NAKASHIMA , Kazunori SHIMAZAKI , Tomio KIMURA , Koji HIKA
IPC分类号： G08G1/14
CPC分类号： B62D15/027 , B60W2420/42 , B62D15/029 , G08G1/168
摘要： A parking assist apparatus has a camera for capturing an image of a mark from a vehicle, wherein the mark is fixed to a parking area with a predetermined positional relation to the parking area and has a predetermined figure, and the vehicle is supposed to park in the parking area. The parking assist apparatus further has a vehicle-position detecting device for detecting a position of the vehicle based on the image of the mark captured by the camera and outputting a position data of the vehicle, a vehicle position data-storing device for storing the position data of the vehicle, a data acquisition device for acquiring attribute data of the parking area and the vicinities of the parking area; and a vehicle guide device for guiding the vehicle in moving out of the parking area, based on the position data of the vehicle in the parking area stored in the vehicle position data-storing device and the attribute data of the parking area and the vicinities of the parking area given by the data acquisition device.
摘要翻译：停车辅助装置具有用于从车辆捕获标记的图像的照相机，其中，标记以与停车区域的预定位置关系固定到停车区域并具有预定的数字，并且车辆应该停放在停车场。停车辅助装置还具有车辆位置检测装置，其基于由照相机拍摄的标记的图像来检测车辆的位置，并输出车辆的位置数据，用于存储位置的车辆位置数据存储装置车辆的数据，用于获取停车区域的属性数据和停车区域附近的数据获取装置; 以及车辆引导装置，其基于车辆位置数据存储装置中存储的停车区域中的车辆的位置数据和停车区域的附近的属性数据，引导车辆离开停车区域由数据采集装置给出的停车区域。

10. 发明申请

US20090306059A1 CYCLIC AMINE DERIVATIVE HAVING SUBSTITUTED ALKYL GROUP 审中-公开
标题翻译：具有取代的烷基的环胺衍生物
公开(公告)号：US20090306059A1
公开(公告)日：2009-12-10
申请号：US11915522
申请日：2006-05-26
申请人： Tomio Kimura , Naoki Tanaka , Hiroyuki Kobayashi , Atsuhiro Sugidachi
发明人： Tomio Kimura , Naoki Tanaka , Hiroyuki Kobayashi , Atsuhiro Sugidachi
IPC分类号： A61K31/541 , C07D413/06 , A61K31/5377 , C07D417/06 , C07D401/06 , A61K31/4545 , A61P7/02
CPC分类号： F16D3/2233 , F16D2003/22309 , Y10T403/32655
摘要： A compound having the general formula (I), pharmacologically acceptable salts thereof or prodrugs thereof: [wherein R1 represents a hydrogen atom, a C1-C6 alkyl group which may be substituted, a C3-C6 cycloalkyl group which may be substituted, a C1-C6 alkoxy group which may be substituted or a C6-C10 aryl group which may be substituted; R2 represents a hydrogen atom, a halogen atom, a carboxy group, a C2-C7 alkoxycarbonyl group, a carbamoyl group, a cyano group, a C1-C6 alkyl group, a halogeno C1-C6 alkyl group, a C1-C6 alkyl group substituted by a heteroaryl group, a C1-C6 alkoxy group, a halogeno C1-C6 alkoxy group, a hydroxy C1-C6 alkyl group, a C2-C12 alkoxyalkyl group, a formyl group, a C2-C7 alkanoyl group, a C4-C7 cycloalkylcarbonyl group, a C2-C7 alkylcarbamoyl group, a di(C1-C6 alkyl)carbamoyl group, a group of formula R4—CO—CR5R6—(CH2)m—, a group of formula R7—CO—(CH2)l—N(R8)— or a sulfamoyl C1-C6 alkyl group; R3 represents a substituted C1-C6 alkyl group, a heterocyclyl group or a heterocyclyl group substituted with 1 to 5 substituents; X1, X2, X3, X4 and X5 each independently represents a hydrogen atom, a halogen atom, an amino group, a carboxy group, a carbamoyl group, a cyano group, a nitro group, a C1-C6 alkyl group, a halogeno C1-C6 alkyl group, a C1-C6 alkoxy group, or a halogeno C1-C6 alkoxy group; and n represents an integer of 0 to 2].
摘要翻译：具有通式（I）的化合物，其药学上可接受的盐或其前药：其中R1表示氢原子，可被取代的C1-C6烷基，可被取代的C3-C6环烷基，C1 可被取代的-C6烷氧基或可被取代的C6-C10芳基; R2表示氢原子，卤素原子，羧基，C2-C7烷氧基羰基，氨基甲酰基，氰基，C1-C6烷基，卤代C1-C6烷基，C1-C6烷基被杂芳基，C 1 -C 6烷氧基，卤代C 1 -C 6烷氧基，羟基C 1 -C 6烷基，C 2 -C 12烷氧基烷基，甲酰基，C 2 -C 7烷酰基， C7环烷基羰基，C2-C7烷基氨基甲酰基，二（C1-C6烷基）氨基甲酰基，式R4-CO-CR5R6-（CH2）m-的基团，式R7-CO-（CH2）（R8） - 或氨磺酰基C1-C6烷基; R 3表示取代的C 1 -C 6烷基，杂环基或被1至5个取代基取代的杂环基; X1，X2，X3，X4和X5各自独立地表示氢原子，卤素原子，氨基，羧基，氨基甲酰基，氰基，硝基，C1-C6烷基，卤代C1 C 1-6烷基，C 1 -C 6烷氧基或卤代C 1 -C 6烷氧基; n表示0〜2的整数]。

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