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21. 发明授权

US4291047A Combating fungi with .alpha.-azolyl-.beta.-hydroxy-ketones 失效
标题翻译：抗真菌与α-唑基-β-羟基酮
公开(公告)号：US4291047A
公开(公告)日：1981-09-22
申请号：US54061
申请日：1979-07-02
申请人： Eckart Kranz , Wolfgang Kramer , Karl H. Buchel , Wilhelm Brandes , Paul-Ernst Frohberger
发明人： Eckart Kranz , Wolfgang Kramer , Karl H. Buchel , Wilhelm Brandes , Paul-Ernst Frohberger
IPC分类号： A01N43/50 , A01N43/653 , C07D233/60 , C07D249/08 , C07D521/00 , A01N43/64
CPC分类号： C07D231/12 , A01N43/50 , A01N43/653 , C07D233/56 , C07D249/08
摘要： .alpha.-Azolyl-.beta.-hydroxy-ketones of the formula ##STR1## in which R.sup.1 represents optionally substituted alkyl or optionally substituted phenyl,R.sup.2 represents the grouping --CX.sup.1 X.sup.2 R.sup.3 or alkoxycarbonyl,R.sup.3 represents halogen, halogenoalkyl or optionally substituted phenyl,X.sup.1 and X.sup.2, which may be identical or different, each represents hydrogen or halogen, andY represents a nitrogen atom or the CH group, or physiologically acceptable acid-addition salts or metal-salt complexes thereof which possess fungicidal properties.
摘要翻译：其中R 1表示任选取代的烷基或任选取代的苯基，R 2表示基团-CX 1 X 2 R 3或烷氧基羰基，R 3表示卤素，卤代烷基或任选取代的苯基，X 1和X 2，其可以相同或不同，各自表示氢或卤素，Y表示具有杀真菌性质的氮原子或CH基团或其生理上可接受的酸加成盐或其金属盐络合物。

22. 发明授权

US3933814A 1-(4-Phenoxyphenyl)-1,3,5-triazines 失效
标题翻译： 1-（4-苯氧基苯基）-1,3,5-三嗪
公开(公告)号：US3933814A
公开(公告)日：1976-01-20
申请号：US397812
申请日：1973-09-17
申请人： Axel Haberkorn , Heinrich Kolling , Eckart Kranz , Jurgen Schramm
发明人： Axel Haberkorn , Heinrich Kolling , Eckart Kranz , Jurgen Schramm
IPC分类号： C07D251/30 , A01N43/64 , A23K1/16 , A61K31/53 , A61K31/535 , A61P33/02 , C07C275/36 , C07C275/60 , C07C275/64 , C07C335/18 , C07D251/26 , C07D251/34 , C07D251/38 , C07D495/04
CPC分类号： C07C275/36 , C07C275/60 , C07C275/64 , C07C335/18
摘要： 1-(4-Phenoxyphenyl)-1,3,5-triazines of the formula: ##SPC1##Or pharmaceutically acceptable nontoxic salts thereof are produced by reacting a urea or thiourea derivative of the formula: ##SPC2##With a carbonylisocyanate of the formula: ##EQU1## to produce a 1-(4-phenoxyphenyl)-1,3,5-triazine as above defined wherein R.sup.11 is hydrogen, and when a 1-(4-phenoxyphenyl)-1,3,5-triazine as above defined wherein R.sup.11 is alkyl is desired, reacting the triazine wherein R.sup.11 is hydrogen with a compound of the formula (alk).sub.n Y.The above defined triazines and their salts are useful as agents against protozoan infections and are particularly useful against coccidiosis.
摘要翻译： 1-（4-苯氧基苯基）-1,3,5-三嗪的下式：

23. 发明授权

US5010208A Novel alkylcycloalkyl triazolylmethyl ketones as fungicide intermediates 失效
标题翻译：新型烷基环烷基三唑甲基酮作为杀真菌剂中间体
公开(公告)号：US5010208A
公开(公告)日：1991-04-23
申请号：US482106
申请日：1990-02-16
申请人： Wolfgang Kramer , Manfred Jautelat , Eckart Kranz
发明人： Wolfgang Kramer , Manfred Jautelat , Eckart Kranz
IPC分类号： A01N43/653 , C07C17/26 , C07C43/225 , C07C45/51 , C07C49/327 , C07D249/08 , C07D521/00
CPC分类号： C07D249/08 , A01N43/653 , C07C17/269 , C07C43/225 , C07C45/513 , C07C49/327 , C07D231/12 , C07D233/56 , C07C2101/08
摘要： New alkylcycloalkyl triazolylmethyl ketones of the general formula ##STR1## in which R represents an alkyl group andn is 3, 4, 5, 6 and 7,are produced as described and find use as intermediate products for the preparation of cycloalkyl (.alpha.-triazolyl-.beta.-hydroxy)-ketones, which possess fungicidal and plant growth-regulating properties.

24. 发明授权

US4766144A 3-carbamoyl-4-hydroxy-coumarins for combating parasitic heiminths 失效
标题翻译： 3-氨基甲酰基-4-羟基香豆素，用于防治寄生性重锤
公开(公告)号：US4766144A
公开(公告)日：1988-08-23
申请号：US35543
申请日：1987-04-03
申请人： Nikolaus Muller , Eckart Kranz , Peter Andrews
发明人： Nikolaus Muller , Eckart Kranz , Peter Andrews
IPC分类号： A61K31/37 , A61K31/443 , A61K31/445 , A61P33/00 , C07D311/56 , C07D405/12 , C07D311/12
CPC分类号： C07D405/12 , C07D311/56
摘要： 3-carbamoyl-4-hydroxy-couramins for combating parasitic helminths of the formula ##STR1## in which R.sup.1 represents hydrogen, halogen, alkyl, NO.sub.2, CN or alkoxy,X represents O, S, SO or SO.sub.2R.sup.2 represents alkyl, halogenoalkyl, phenyl, naphthyl or pyridyl, which can optionally be substituted; or the radical -X-R.sup.2, together with the radical R.sup.3 can also form an alkylenedioxy (-O-alk-O), halogenoalkylenedioxy, oxyalkyleneoxyalkylene (-O-Alk-O-Alk-) or oxyhalogenoalkylene-oxyhalogenoalkylene bridge; andR.sup.3 and R.sup.4 independently of one another represent hydrogen, halogen, CN, OH, NO.sub.2, amino, mono- or dialklylamino, alkyl, halogenoalkyl, aralkyl or aryl, which can optionally be substituted,can be used for combating parasitic helminths.
摘要翻译： 3-氨基甲酰基-4-羟基维生素，用于对抗式为“IMAGE”的寄生蠕虫，其中R 1表示氢，卤素，烷基，NO 2，CN或烷氧基，X表示O，S，SO或SO 2 R 2表示烷基，卤代烷基，苯基，萘基或吡啶基，其可任选被取代; 或基团-X-R2与基团R3一起也可以形成亚烷基二氧基（-O-烷基-O），卤代亚烷基二氧基，氧亚烷基氧化烯（-O-Alk-O-Alk-）或氧卤代亚烷基 - 氧卤代亚烷基桥; 并且R 3和R 4彼此独立地表示氢，卤素，CN，OH，NO 2，氨基，单或二烷基氨基，烷基，卤代烷基，芳烷基或芳基，其可任选被取代，可用于对抗寄生蠕虫。

25. 发明授权

US4492795A Alkylcycloalkyl imidazolylmethyl ketones as fungicide intermediates 失效
标题翻译：烷基环烷基咪唑甲基酮作为杀真菌剂中间体
公开(公告)号：US4492795A
公开(公告)日：1985-01-08
申请号：US438087
申请日：1982-11-01
申请人： Wolfgang Kramer , Manfred Jautelat , Eckart Kranz
发明人： Wolfgang Kramer , Manfred Jautelat , Eckart Kranz
IPC分类号： A01N43/50 , C07C17/26 , C07C43/225 , C07C45/51 , C07C49/327 , C07D233/60 , C07D521/00
CPC分类号： C07D249/08 , C07C17/269 , C07C43/225 , C07C45/513 , C07C49/327 , C07D231/12 , C07D233/56
摘要： New alkylcycloalkyl imidazolylmethyl ketones of the general formula ##STR1## in which R represents an alkyl group andn is 3, 4, 5, 6 or 7,are produced as described and find use as intermediate products for the preparation of imidazolyl-vinyl-dithioacetals, which possess fungicidal properties.
摘要翻译：其中R表示烷基且n为3,4,5,6或7的通式为“IMAGE”的新的烷基环烷基咪唑基甲基酮如所述制备，可用作制备咪唑基 - 乙烯基 - 二硫代缩醛的中间产物，具有杀菌性。

26. 发明授权

US4229580A Preparation of 1-azolyl-3,3-dimethyl-1-phenoxy-butan-2-ones 失效
标题翻译： 1-噻唑基-3,3-二甲基-1-苯氧基 - 丁-2-酮的制备
公开(公告)号：US4229580A
公开(公告)日：1980-10-21
申请号：US885053
申请日：1978-03-09
申请人： Hermann Arold , Hans-Ludwig Elbe , Eckart Kranz , Wolfgang Kramer , Jorg Stetter , Claus Stolzer , Rudolf Thomas
发明人： Hermann Arold , Hans-Ludwig Elbe , Eckart Kranz , Wolfgang Kramer , Jorg Stetter , Claus Stolzer , Rudolf Thomas
IPC分类号： A01N43/50 , A01N43/836 , C07D233/60 , C07D249/08 , C07D521/00
CPC分类号： C07D231/12 , C07D233/56 , C07D249/08
摘要： In the reaction of 1-chloro-3,3-dimethylbutan-2-one with a phenol to form an ether-ketone, halogenating it to form a halogenoether-ketone and reacting it with imidazole or 1,2,4-triazole to form a 1-azolyl-3,3-dimethyl-1-phenoxybutan-2-one of the formula ##STR1## in which X is N or CH,n is an integer from 0 to 4, andY each independently is halogen, phenyl, phenoxy, nitro, alkyl, alkoxy or cycloalkyl,the improvement which comprises effecting all steps successively in an aromatic hydrocarbon or chlorinated aliphatic or aromatic hydrocarbon as solvent without intermediate isolation. The products are obtained in high yield.
摘要翻译：在1-氯-3,3-二甲基丁-2-酮与苯酚反应形成醚 - 酮的反应中，将其卤化形成卤代醚 - 酮并与咪唑或1,2,4-三唑反应形成其中X为N或CH，n为0至4的整数，并且Y各自独立地为卤素，苯基，环烷基，环烷基，苯氧基，硝基，烷基，烷氧基或环烷基，其改进包括在芳族烃或氯化脂族或芳族烃作为溶剂中连续进行所有步骤而不中间分离。以高产率获得产品。

27. 发明授权

US3970752A Coccidiocidal compositions utilizing 1-phenyl-substituted 1,3,5-triazine 失效
标题翻译：使用1-苯基取代的1,3,5-三嗪的杀微生物剂组合物
公开(公告)号：US3970752A
公开(公告)日：1976-07-20
申请号：US532221
申请日：1974-12-12
申请人： Gerd Aichinger , Axel Haberkorn , Heinrich Kolling , Eckart Kranz , Josef Reisdorff
发明人： Gerd Aichinger , Axel Haberkorn , Heinrich Kolling , Eckart Kranz , Josef Reisdorff
IPC分类号： A23K1/16 , C07C317/42 , C07C323/66 , A61K31/53
CPC分类号： C07C323/66 , A23K20/116 , C07C317/42
摘要： 1-Phenyl-substituted 1,3,5-triazines of the formula: ##SPC1##And pharmaceutically acceptable nontoxic salts thereofWherein R.sub.1, R.sub.2, R.sub.3, R.sub.4, R.sub.5, R.sub.6, R.sub.7, R.sub.8 and R.sub. 9 are the same or different and each is selected from the group consisting of hydrogen, straight or branched chain alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio, haloalkylthio, halogen, nitro, cyano, amino, acylamino, alkoxycarbonylamino, carboxy, alkoxycarbonyl, carbamoyl, acyl, haloacyl, alkylsulphinyl, alkylsulphonyl, haloalkylsulphonyl and sulphamoyl;R.sub.10 is hydrogen, straight or branched chain alkyl, cycloalkyl, haloalkyl, alkoxy, alkoxyalkyl, haloalkoxyalkyl, alkylthioalkyl, haloalkylthioalkyl, alkenyl, alkynyl, alkoxycarbonyl, (alkylthio)carbonyl, (alkylthio)thiocarbonyl, acylamino, diacylamino, amino, dialkylamino, polymethyleneimino, polymethyleneimino interrupted by a heteroatom in the chain, or unsubstituted or substituted benzyl or aryl;R.sub.11 is hydrogen, or alkyl;X is sulphur, sulphinyl, or sulphonyl; andY is oxygen or sulphur,Are useful for their activity against coccidiosis in humans and animals.
摘要翻译：具有下式的1-苯基取代的1,3,5-三嗪：

28. 发明授权

US3966725A 1-(4-Phenoxy-phenyl)-1,3,5-triazines 失效
标题翻译： 1-（4-苯氧基 - 苯基）-1,3,5-三嗪
公开(公告)号：US3966725A
公开(公告)日：1976-06-29
申请号：US559562
申请日：1975-03-18
申请人： Josef Helmut Reisdorff , Gerd Aichinger , Axel Haberkorn , Heinrich Kolling , Eckart Kranz
发明人： Josef Helmut Reisdorff , Gerd Aichinger , Axel Haberkorn , Heinrich Kolling , Eckart Kranz
IPC分类号： C07D251/34 , A23K1/16 , A61K31/53 , A61P33/02 , C07C273/18 , C07C275/36 , C07C319/20 , C07C323/20 , C07D251/38
CPC分类号： C07D251/26 , A23K20/116 , C07C273/1827 , C07C319/20
摘要： 1-(4-Phenoxy-phenyl)-1,3,5-triazine derivatives of the formula ##SPC1##And pharmaceutically-acceptable, nontoxic salts thereof whereinR.sub.1 to R.sub.9 are the same or different and each is hydrogen, alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio, haloalkylthio, halo, nitro, cyano, amino, acylamino, alkoxycarbonylamino, carboxy, alkoxycarbonyl, carbamoyl, acyl, haloacyl, alkylsulphinyl, alkylsulphonyl, haloalkylsulphinyl, haloalkylsulphonyl or sulphamoyl; provided that at least one of R.sub.1 to R.sub.9 is haloalkyl, haloalkylthio, haloalkylsulphinyl or haloalkylsulphonyl;R.sub.10 is hydrogen, alkyl, cycloalkyl, haloalkyl, alkoxy, alkoxyalkyl, haloalkoxyalkyl, alkylthioalkyl, haloalkylthioalkyl, alkenyl, alkinyl, alkoxycarbonyl, alkylthiocarbonyl, alkylthiothiocarbonyl, acylamino, diacylamino, dialkylamino, polymethylene-imino, polymethylene-imino interrupted by a heteroatom, unsubstituted or substituted benzyl or unsubstituted or substituted aryl;R.sub.11 is hydrogen or alkyl; andY is oxygen or sulphur;Are useful in treating coccidiosis in humans and animals.
摘要翻译： 1-（4-苯氧基 - 苯基）-1,3,5-三嗪衍生物及其药学上可接受的，其中R 1至R 9相同或不同并且各自为氢，烷基，卤代烷基，烷氧基，卤代烷氧基的非对映体烷硫基，卤代烷硫基，卤素，硝基，氰基，氨基，酰氨基，烷氧基羰基氨基，羧基，烷氧基羰基，氨基甲酰基，酰基，卤代酰基，烷基亚磺酰基，烷基磺酰基，卤代烷基亚磺酰基，卤代烷基磺酰基或氨磺酰基。条件是R 1至R 9中的至少一个为卤代烷基，卤代烷硫基，卤代烷基亚磺酰基或卤代烷基磺酰基; R 10为氢，烷基，环烷基，卤代烷基，烷氧基，烷氧基烷基，卤代烷氧基烷基，烷硫基烷基，卤代烷硫基烷基，烯基，炔基，烷氧基羰基，烷硫基羰基，烷基硫代羰基，酰氨基，二酰基氨基，二烷基氨基，聚亚甲基亚氨基，被杂原子中断的聚亚甲基亚氨基，取代的苄基或未取代或取代的芳基; R11是氢或烷基; Y为氧或硫; 有用于治疗人类和动物的结核病。

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