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1. 发明授权

US3970752A Coccidiocidal compositions utilizing 1-phenyl-substituted 1,3,5-triazine 失效
标题翻译：使用1-苯基取代的1,3,5-三嗪的杀微生物剂组合物
公开(公告)号：US3970752A
公开(公告)日：1976-07-20
申请号：US532221
申请日：1974-12-12
申请人： Gerd Aichinger , Axel Haberkorn , Heinrich Kolling , Eckart Kranz , Josef Reisdorff
发明人： Gerd Aichinger , Axel Haberkorn , Heinrich Kolling , Eckart Kranz , Josef Reisdorff
IPC分类号： A23K1/16 , C07C317/42 , C07C323/66 , A61K31/53
CPC分类号： C07C323/66 , A23K20/116 , C07C317/42
摘要： 1-Phenyl-substituted 1,3,5-triazines of the formula: ##SPC1##And pharmaceutically acceptable nontoxic salts thereofWherein R.sub.1, R.sub.2, R.sub.3, R.sub.4, R.sub.5, R.sub.6, R.sub.7, R.sub.8 and R.sub. 9 are the same or different and each is selected from the group consisting of hydrogen, straight or branched chain alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio, haloalkylthio, halogen, nitro, cyano, amino, acylamino, alkoxycarbonylamino, carboxy, alkoxycarbonyl, carbamoyl, acyl, haloacyl, alkylsulphinyl, alkylsulphonyl, haloalkylsulphonyl and sulphamoyl;R.sub.10 is hydrogen, straight or branched chain alkyl, cycloalkyl, haloalkyl, alkoxy, alkoxyalkyl, haloalkoxyalkyl, alkylthioalkyl, haloalkylthioalkyl, alkenyl, alkynyl, alkoxycarbonyl, (alkylthio)carbonyl, (alkylthio)thiocarbonyl, acylamino, diacylamino, amino, dialkylamino, polymethyleneimino, polymethyleneimino interrupted by a heteroatom in the chain, or unsubstituted or substituted benzyl or aryl;R.sub.11 is hydrogen, or alkyl;X is sulphur, sulphinyl, or sulphonyl; andY is oxygen or sulphur,Are useful for their activity against coccidiosis in humans and animals.
摘要翻译：具有下式的1-苯基取代的1,3,5-三嗪：

2. 发明授权

US3966725A 1-(4-Phenoxy-phenyl)-1,3,5-triazines 失效
标题翻译： 1-（4-苯氧基 - 苯基）-1,3,5-三嗪
公开(公告)号：US3966725A
公开(公告)日：1976-06-29
申请号：US559562
申请日：1975-03-18
申请人： Josef Helmut Reisdorff , Gerd Aichinger , Axel Haberkorn , Heinrich Kolling , Eckart Kranz
发明人： Josef Helmut Reisdorff , Gerd Aichinger , Axel Haberkorn , Heinrich Kolling , Eckart Kranz
IPC分类号： C07D251/34 , A23K1/16 , A61K31/53 , A61P33/02 , C07C273/18 , C07C275/36 , C07C319/20 , C07C323/20 , C07D251/38
CPC分类号： C07D251/26 , A23K20/116 , C07C273/1827 , C07C319/20
摘要： 1-(4-Phenoxy-phenyl)-1,3,5-triazine derivatives of the formula ##SPC1##And pharmaceutically-acceptable, nontoxic salts thereof whereinR.sub.1 to R.sub.9 are the same or different and each is hydrogen, alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio, haloalkylthio, halo, nitro, cyano, amino, acylamino, alkoxycarbonylamino, carboxy, alkoxycarbonyl, carbamoyl, acyl, haloacyl, alkylsulphinyl, alkylsulphonyl, haloalkylsulphinyl, haloalkylsulphonyl or sulphamoyl; provided that at least one of R.sub.1 to R.sub.9 is haloalkyl, haloalkylthio, haloalkylsulphinyl or haloalkylsulphonyl;R.sub.10 is hydrogen, alkyl, cycloalkyl, haloalkyl, alkoxy, alkoxyalkyl, haloalkoxyalkyl, alkylthioalkyl, haloalkylthioalkyl, alkenyl, alkinyl, alkoxycarbonyl, alkylthiocarbonyl, alkylthiothiocarbonyl, acylamino, diacylamino, dialkylamino, polymethylene-imino, polymethylene-imino interrupted by a heteroatom, unsubstituted or substituted benzyl or unsubstituted or substituted aryl;R.sub.11 is hydrogen or alkyl; andY is oxygen or sulphur;Are useful in treating coccidiosis in humans and animals.
摘要翻译： 1-（4-苯氧基 - 苯基）-1,3,5-三嗪衍生物及其药学上可接受的，其中R 1至R 9相同或不同并且各自为氢，烷基，卤代烷基，烷氧基，卤代烷氧基的非对映体烷硫基，卤代烷硫基，卤素，硝基，氰基，氨基，酰氨基，烷氧基羰基氨基，羧基，烷氧基羰基，氨基甲酰基，酰基，卤代酰基，烷基亚磺酰基，烷基磺酰基，卤代烷基亚磺酰基，卤代烷基磺酰基或氨磺酰基。条件是R 1至R 9中的至少一个为卤代烷基，卤代烷硫基，卤代烷基亚磺酰基或卤代烷基磺酰基; R 10为氢，烷基，环烷基，卤代烷基，烷氧基，烷氧基烷基，卤代烷氧基烷基，烷硫基烷基，卤代烷硫基烷基，烯基，炔基，烷氧基羰基，烷硫基羰基，烷基硫代羰基，酰氨基，二酰基氨基，二烷基氨基，聚亚甲基亚氨基，被杂原子中断的聚亚甲基亚氨基，取代的苄基或未取代或取代的芳基; R11是氢或烷基; Y为氧或硫; 有用于治疗人类和动物的结核病。

3. 发明授权

US5416209A 5,6-dihydro-dibenz[b,e]azepine-6,11-dione-11-oximes 失效
标题翻译： 5,6-二氢 - 二苯并[b，e]吖庚因-6,11-二酮-11-肟
公开(公告)号：US5416209A
公开(公告)日：1995-05-16
申请号：US978001
申请日：1992-11-18
申请人： Hanno Wild , Wolfgang Roeben , Gerd Aichinger , Arnold Paessens , Jorg Peters n-von Gehr
发明人： Hanno Wild , Wolfgang Roeben , Gerd Aichinger , Arnold Paessens , Jorg Peters n-von Gehr
IPC分类号： A61K31/00 , A61K31/55 , A61P31/12 , A61P43/00 , C07D223/20 , C07D405/12 , C12N9/99
CPC分类号： C07D405/12 , C07D223/20
摘要： The invention relates to 5,6-dihydro-dibenz[b,e]azepine-6,11-dione-11-oximes, to processes for their preparation and to their use as inhibitors of reverse transcriptase and in particular as antiretroviral agents.
摘要翻译：本发明涉及5,6-二氢 - 二苯并[b，e]吖庚因-6,11-二酮-11-肟，用于其制备及其作为逆转录酶抑制剂，特别是抗逆转录病毒剂的用途。

4. 发明授权

US3948893A 1-Phenyl-substituted 1,3,5-triazines 失效
标题翻译： 1-苯基取代的1,3,5-三嗪
公开(公告)号：US3948893A
公开(公告)日：1976-04-06
申请号：US452140
申请日：1974-03-18
申请人： Gerd Aichinger , Axel Haberkorn , Heinrich Kolling , Eckart Kranz , Josef Reisdorff
发明人： Gerd Aichinger , Axel Haberkorn , Heinrich Kolling , Eckart Kranz , Josef Reisdorff
IPC分类号： C07D251/34 , A23K1/16 , A61K31/53 , C07C317/42 , C07C323/44 , C07C323/66 , C07D209/48 , C07D251/04 , C07D251/38 , C07D51/26
CPC分类号： C07D209/48 , A23K20/116 , C07C317/42 , C07C323/44 , C07C323/66
摘要： 1-Phenyl-substituted 1,3,5-triazines of the formula: ##SPC1##And pharmaceutically acceptable nontoxic salts thereof whereinR.sub.1, r.sub.2, r.sub.3, r.sub.4, r.sub.5, r.sub.6, r.sub.7, r.sub.8 and R.sub.9 are the same or different and each is selected from the group consisting of hydrogen, straight or branched chain alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio, haloalkylthio, halogen, nitro, cyano, amino, acylamino, alkoxycarbonylamino, carboxy, alkoxycarbonyl, carbamoyl, acyl, haloacyl, alkylsulphinyl, alkylsulphonyl, haloalkylsulphonyl and sulphamoyl;R.sub.10 is hydrogen, straight or branched chain alkyl, cycloalkyl, haloalkyl, alkoxy, alkoxyalkyl, haloalkoxyalkyl, alkylthioalkyl, haloalkylthioalkyl, alkenyl, alkynyl, alkoxycarbonyl, (alkylthio)carbonyl, (alkylthio)thiocarbonyl, acylamino, diacylamino, amino, dialkylamino, polymethyleneimino, polymethyleneimino interrupted by a heteroatom in the chain, or unsubstituted or substituted benzyl or aryl;R.sub.11 is hydrogen, or alkyl;X is sulphur, sulphinyl, or sulphonyl; andY is oxygen or sulphur,Are useful for their activity against coccidiosis in humans and animals.
摘要翻译：具有下式的1-苯基取代的1,3,5-三嗪：

5. 发明授权

US5385899A Aminoalkyl-substituted 5,6-dihydro-dibenz[b,e]azepine-6,11-dione-11-oximes 失效
标题翻译：氨基烷基取代的5,6-二氢 - 二苯并[b，e]吖庚因-6,11-二酮-11-肟
公开(公告)号：US5385899A
公开(公告)日：1995-01-31
申请号：US977379
申请日：1992-11-17
申请人： Hanno Wild , Wolfgang Roeben , Gerd Aichinger , Arnold Paessens , Jorg Petersen-von Gehr
发明人： Hanno Wild , Wolfgang Roeben , Gerd Aichinger , Arnold Paessens , Jorg Petersen-von Gehr
IPC分类号： A61K31/00 , A61K31/55 , A61P31/12 , A61P43/00 , C07D223/20 , C07D413/12 , C12N9/99 , C07D223/16
CPC分类号： C07D223/20
摘要： The invention relates to aminoalkyl-substituted 5,6-dihydro-dibenz[b,e]azepine-6,11-dione-11-oximes, to processes for their preparation and to their use as antiretroviral agents.
摘要翻译：本发明涉及氨基烷基取代的5,6-二氢 - 二苯并[b，e]吖庚因-6,11-二酮-11-肟，用于其制备及其作为抗逆转录病毒剂的用途。

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