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1. 发明申请

WO2011042804A3 AN IMPROVED PROCESS FOR THE PREPARATION OF CLOPIDOGREL HYDROGEN SULFATE FORM I 审中-公开
公开(公告)号：WO2011042804A3
公开(公告)日：2011-04-14
申请号：PCT/IB2010/002553
申请日：2010-10-08
申请人： JUBLIANT LIFE SCIENCES LIMITED , ACHARYA, Hrishikesh, Dilip , SRIVASTAVA, Jayant , KUMAR, Satish , AWASTHI, Arun, Kumar , KUMAR, Pramod , VIR, Dharam
发明人： ACHARYA, Hrishikesh, Dilip , SRIVASTAVA, Jayant , KUMAR, Satish , AWASTHI, Arun, Kumar , KUMAR, Pramod , VIR, Dharam
IPC分类号： C07D495/04
摘要： Disclosed herein an improved process for the preparation of polymorphic Form I of clopidogrel hydrogen sulfate.

2. 发明申请

WO2011030213A8 IMPROVED PROCESS FOR THE PREPARATION OF 7-(4-BROMOBUTOXY) 3,4-DIHYDROCARBOSTYRIL, A PRECURSOR OF ARIPIPRAZOLE 审中-公开
标题翻译：改进的制备7-（4-溴代丁氧基）3,4-二氢苯并硅酮，一种阿立哌唑前体的方法
公开(公告)号：WO2011030213A8
公开(公告)日：2011-03-17
申请号：PCT/IB2010/002276
申请日：2010-09-14
申请人： JUBILANT LIFE SCIENCES LIMITED , SRIVASTAVA, Jayant , GUPTA, Vijay, Shankar , VARU, Bharat, Vithalbhai , KUMAR, Pramod , VIR, Dharam
发明人： SRIVASTAVA, Jayant , GUPTA, Vijay, Shankar , VARU, Bharat, Vithalbhai , KUMAR, Pramod , VIR, Dharam
IPC分类号： C07D215/227
摘要： Disclosed herein is an improved process for the preparation of 7-(4-bromobutoxy) 3,4-dihydrocarbostyril, a key intermediate used in the preparation of Aripiprazole.
摘要翻译：本文公开了制备用于制备阿立哌唑的关键中间体7-（4-溴丁氧基）3,4-二氢喹诺酮的改进方法。

3. 发明申请

WO2012063115A2 PROCESS FOR THE PREPARATION OF ROSUVASTATIN CALCIUM VIA NOVEL AMINE INTERMEDIATE 审中-公开
标题翻译：通过新型胺中间体制备罗苏伐他汀钙的方法
公开(公告)号：WO2012063115A2
公开(公告)日：2012-05-18
申请号：PCT/IB2011/002633
申请日：2011-11-09
申请人： JUBILANT LIFE SCIENCES LTD. , SINGH, Khushwant , SINGH, Anand, Kumar , SRIVASTAVA, Rahul , KUMAR, Pramod , VIR, Dharam , AGARWAL, Ashutosh
发明人： SINGH, Khushwant , SINGH, Anand, Kumar , SRIVASTAVA, Rahul , KUMAR, Pramod , VIR, Dharam , AGARWAL, Ashutosh
IPC分类号： C07D239/42
CPC分类号： C07D239/42
摘要： The present invention, relates to novel amine salts of rosuvastatin and its process for the preparation. Moreover, the present invention also relates to improved process for the preparation of rosuvastatin calcium, employing novel amine salts as an intermediate.
摘要翻译：本发明涉及瑞舒伐他汀的新型胺盐及其制备方法。此外，本发明还涉及使用新型胺盐作为中间体制备瑞舒伐他汀钙的改进方法。

4. 发明申请

WO2012131451A1 PROCESS FOR PRODUCING ARIPIPRAZOLE IN ANHYDROUS TYPE I CRYSTALS 审中-公开
标题翻译：在异型I型晶体中生产阿哌唑的方法
公开(公告)号：WO2012131451A1
公开(公告)日：2012-10-04
申请号：PCT/IB2012/000403
申请日：2012-03-05
申请人： JUBILANT LIFE SCIENCES LIMITED , GUPTA, Vijay Shankar , KUMAR, Pramod , VIR, Dharam
发明人： GUPTA, Vijay Shankar , KUMAR, Pramod , VIR, Dharam
IPC分类号： C07D215/227
CPC分类号： C07D215/227
摘要： Disclosed herein is an improved process for the preparation of anpiprazole in anhydrous Type I crystals, substantially free of other polymorphic forms of aripiprazole via improved drying technique.
摘要翻译：本文公开了一种通过改进的干燥技术制备无水I型晶体中的阿哌唑的改进方法，其基本上不含阿立哌唑的其它多晶型物。

5. 发明申请

WO2011140645A1 LIFTER BAR ASSEMBLY AND GRINDING MILL INCLUDING SAME 审中-公开
标题翻译： LIFTER BAR装配和研磨机，包括它们
公开(公告)号：WO2011140645A1
公开(公告)日：2011-11-17
申请号：PCT/CA2011/000554
申请日：2011-05-13
申请人： POLYCORP LTD. , KUMAR, Pramod , RAJAMANI, Raj K. , PAGE, David J. , MEPHAM, Robert
发明人： KUMAR, Pramod , RAJAMANI, Raj K. , PAGE, David J. , MEPHAM, Robert
IPC分类号： B02C17/22 , B02C17/04
CPC分类号： B02C17/1825 , B02C17/10
摘要： A grinding mill including one or more lifter bar assemblies mounted on a shell rotatable around a central axis thereof. Each lifter bar assembly is for lifting at least a lifted portion of a charge including ore, and includes a main portion for lifting and directing a main part of the lifted portion in a main part direction substantially orthogonal to the central axis of the shell. The lifter bar assembly also includes one or more terminal lifter bars located proximal to one or both of feed and discharge ends of the shell, for lifting and directing terminal part(s) of the lifted portion of the charge. The terminal lifter bar is positioned for directing the terminal part of the lifted portion of the charge at least partially in a terminal part direction which is substantially non-aligned with the main part direction.
摘要翻译：一种研磨机，包括安装在可围绕其中心轴线旋转的壳体上的一个或多个升降杆组件。每个升降杆组件用于至少提升包括矿石的电荷的提升部分，并且包括用于在与壳体的中心轴线基本正交的主要部分方向上提升和引导提升部分的主要部分的主要部分。提升杆组件还包括位于壳体的进料和排出端的一个或两个附近的一个或多个末端升降杆，用于提升和引导装料的提升部分的末端部分。端子升降杆被定位成用于将电荷的提升部分的端子部分至少部分地沿着与主要部分方向基本上不对准的端子部分方向引导。

6. 发明申请

WO2007141798A1 PROCESS FOR PRODUCING OXCARBAZEPINE VIA AN 11-ALKOXY-10-HALO-DIHYDROIMINOSTILBENE INTERMEDIATE 审中-公开
标题翻译：通过11-羟基-10-二羟基二氨基苯基中间体生产氧化萘的方法
公开(公告)号：WO2007141798A1
公开(公告)日：2007-12-13
申请号：PCT/IN2006/000190
申请日：2006-06-07
申请人： JUBILANT ORGANOSYS LIMITED , GUPTA, Nitin , SINGH, Harnam , KUMAR, Pramod , DUBEY, Sushil, Kumar
发明人： GUPTA, Nitin , SINGH, Harnam , KUMAR, Pramod , DUBEY, Sushil, Kumar
IPC分类号： C07D223/22
CPC分类号： C07D223/22 , C07D223/26
摘要： Disclosed herein is an economically viable and cost effective process for preparation of oxcarbazepine of formula (I) via a novel intermediate of formula (XVIII).
摘要翻译：本文公开了通过式（XVIII）的新型中间体制备式（I）的奥卡西平的经济可行且成本有效的方法。

7. 发明申请

WO2005092886A1 PROCESS FOR THE PREPARATION OF AMORPHOUS FORM OF TIAGABINE 审中-公开
标题翻译：制备不规则形式的方法
公开(公告)号：WO2005092886A1
公开(公告)日：2005-10-06
申请号：PCT/IB2005/000809
申请日：2005-03-29
申请人： RANBAXY LABORATORIES LIMITED , BOSE, Prosenjit , KUMAR, Pramod , SACHDEVA, Yoginder Pal , MITTAL, Shilpi , KUMAR, Yatendra
发明人： BOSE, Prosenjit , KUMAR, Pramod , SACHDEVA, Yoginder Pal , MITTAL, Shilpi , KUMAR, Yatendra
IPC分类号： C07D409/14
CPC分类号： C07D409/14
摘要： The present invention relates to processes for the preparation of amorphous form of tiagabine hydrochloride. The invention also relates to pharmaceutical compositions that include the amorphous form of tiagabine hydrochloride, and use of said compositions for the treatment of epilepsy and other diseases related to gamma-amino butyric acid uptake (GABA uptake).
摘要翻译：本发明涉及制备盐酸噻加滨的无定形形式的方法。本发明还涉及包含盐酸噻加滨的无定形形式的药物组合物，以及所述组合物用于治疗与γ-氨基丁酸摄取（GABA摄取）有关的癫痫和其它疾病的用途。

8. 发明申请

WO2011001212A1 IMIDAZO [4,5-C]QUINOLINE DERIVATIVES AND THEIR USE IN THE TREATMENT OF TUMORS AND/OR INFLAMMATION 审中-公开
标题翻译：咪唑并[4,5-C]喹啉衍生物及其在治疗肿瘤和/或炎症中的应用
公开(公告)号：WO2011001212A1
公开(公告)日：2011-01-06
申请号：PCT/IB2009/052819
申请日：2009-06-30
申请人： PIRAMAL LIFE SCIENCES LIMITED , KUMAR, Sanjay , VISHWAKARMA, Ram , MUNDADA, Ramswaroop , DEORE, Vijaykumar , KUMAR, Pramod , SHARMA, Somesh
发明人： KUMAR, Sanjay , VISHWAKARMA, Ram , MUNDADA, Ramswaroop , DEORE, Vijaykumar , KUMAR, Pramod , SHARMA, Somesh
IPC分类号： C07D471/04 , A61K31/437 , A61P17/06 , A61P35/00
CPC分类号： C07D471/04
摘要： The present invention provides the compounds of formula (I): (I) The present invention relates to imidazo[4,5-c]quinoline derivatives of formula (I), process for their preparation, pharmaceutical compositions containing them and their use in the treatment of diseases mediated by phosphatidylinositol-3-kinase (PBK) and/or mammalian target of rapamycin (mTOR) and/or tumor necrosis factor-α (TNF-oc) and/or interleukin-6 (IL-6), particularly in the treatment of cancer and inflammation.
摘要翻译：本发明提供式（I）化合物：（I）本发明涉及式（I）的咪唑并[4,5-c]喹啉衍生物，其制备方法，含有它们的药物组合物及其在治疗由磷脂酰肌醇-3-激酶（PBK）和/或哺乳动物雷帕霉素靶（mTOR）和/或肿瘤坏死因子-α（TNF-α）和/或白细胞介素-6（IL-6）介导的疾病，特别是在治疗癌症和炎症。

9. 发明申请

WO2005066120A2 PROCESS FOR ASYMMETRIC SYNTHESIS OF HYDROXY-ALKYL SUBSTITUTED AZETIDINONE DERIVATIVES OF INTERMEDIATES THEREOF 审中-公开
标题翻译：其中间体羟基烷基取代的三唑酮衍生物的不对称合成方法
公开(公告)号：WO2005066120A2
公开(公告)日：2005-07-21
申请号：PCT/IB2004/004281
申请日：2004-12-23
申请人： RANBAXY LABORATORIES LIMITED , KUMAR, Yatendra , MEERAN, Hashim, Nizar, Poovanathi, Nagoor , SINGH, Shailendra, Kumar , RATHOD, Parendu, Dhirajlal , GANAGAKHEDKAR, Kiran, Kumar , BOSE, Prosenjit , KUMAR, Pramod
发明人： KUMAR, Yatendra , MEERAN, Hashim, Nizar, Poovanathi, Nagoor , SINGH, Shailendra, Kumar , RATHOD, Parendu, Dhirajlal , GANAGAKHEDKAR, Kiran, Kumar , BOSE, Prosenjit , KUMAR, Pramod
IPC分类号： C07D205/00
CPC分类号： C07D205/08 , C07C67/31 , C07D263/22 , C07C69/732
摘要： Provided herein are processes for asymmetric synthesis of hydroxyalkyl-substituted azetidinone derivatives or intermediates thereof via stereoselective reduction of benzylic ketone using (-)-B-chlorodiisopinocampheylborane. Also provided herein are processes for preparing ezetimibe.
摘要翻译：本文提供了通过使用（ - ） - B-氯二氧杂环己烷硼烷通过苄基酮的立体选择性还原来不对称合成羟烷基取代的氮杂环丁酮衍生物或其中间体的方法。本文还提供了制备依泽替米贝的方法。

10. 发明申请

WO2011060540A1 LIFTER BAR 审中-公开
标题翻译：酒吧
公开(公告)号：WO2011060540A1
公开(公告)日：2011-05-26
申请号：PCT/CA2010/001836
申请日：2010-11-19
申请人： POLYCORP LTD. , PAGE, David, J. , KUMAR, Pramod , RAJAMANI, Raj K.
发明人： PAGE, David, J. , KUMAR, Pramod , RAJAMANI, Raj K.
IPC分类号： B02C17/18 , B02C17/00
CPC分类号： B02C17/1825
摘要： A lifter bar for lifting an engaged portion of a load comprising a number of ore pieces above a disengaged portion of the load in a grinding mill having a shell rotatable about an axis thereof. The lifter bar includes a leading face having one or more leading surfaces, and a trailing face. The lifter bar is mountable on the shell located at a predetermined distance from a trailing face of a preceding lifter bar. When the lifter bar and the preceding lifter bar are mounted on the shell, the leading face and the trailing face of the preceding lifter bar at least partially define a pocket therebetween in which a part of the engaged portion of the load is at least partially retainable, until the leading surface is located in a predetermined release position, at which the part has substantially exited the pocket under the influence of gravity.
摘要翻译：一种提升杆，用于在具有可围绕其轴线旋转的外壳的研磨机中提升包括多个矿石片的脱模部分上方的多个矿石片的接合部分。升降杆包括具有一个或多个前表面的引导面和后表面。升降杆安装在位于与前一升降杆的后表面预定距离处的外壳上。当升降杆和前一升降杆安装在壳体上时，前一提升杆的前表面和后表面至少部分地限定了一个凹槽，在该凹槽中，该载荷的啮合部分的一部分至少部分保持直到前导表面位于预定的释放位置，在预定的释放位置处，该部分在重力的作用下基本上离开了该口袋。

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