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1. 发明授权

US4841091A Process for producing 16-substituted prostaglandin es. 失效
标题翻译：生产16-取代的前列腺素的方法。
公开(公告)号：US4841091A
公开(公告)日：1989-06-20
申请号：US913889
申请日：1986-09-29
申请人： Toshio Tanaka , Atsuo Hazato , Seizi Kurozumi , Masahiro Koga
发明人： Toshio Tanaka , Atsuo Hazato , Seizi Kurozumi , Masahiro Koga
IPC分类号： C07C405/00
CPC分类号： C07C405/0033 , C07C405/00
摘要： A novel process for manufacturing 16-substituted .DELTA..sup.7 -prostaglandin Es, which include compounds expressed by the following formula (I), their enanantiomers, or their mixtures of arbitray mixing ratio, ##STR1## wherein R.sup.1 indicates COOR.sup.2, CH.sub.2 OR.sup.3, in which R.sup.2 indicates a hydrogen atom, a dubstituted or unsubstituted C.sub.1 -C.sub.10 alkyl group, a substituted or unsubstituted C.sub.3 -C.sub.10 cycloalkyl group, or a substituted or unsubstituted phenyl group, and R.sup.3 indicates a hydrogen atom, a tri(C.sub.1 -C.sub.7) hydrocarbon silyl group, a group which forms an acetal bond together with the oxygen atom of a hydroxyl group, or a C.sub.2 -C.sub.7 acyl group; R.sup.4 and R.sup.5 are identical or different, each representing a hydrogen atom, a tri(C.sub.1 -C.sub.7 ) hydrocarbon silyl group, or a group which forms an acetal bond together with the oxygen atom of a hydroxyl group; R.sup.6 indicates a hydrogen atom, a C.sub.1 -C.sub.4 alkyl group, or a vinyl group; R.sup.7 indicates a linear or branched C.sub.3 -C.sub.8 alkyl group, an alkyenyl group, or an alkynyl group, which may contain an oxygen atom; a phenyl group, a phenoxy group, or a C.sub.3 -C.sub.10 cycloalkyl group, which may be substituted; or a linear or branched C.sub.1 -C.sub.5 alkyl group which is substituted by a C.sub.1 -C.sub.6 alkoxy group, a phenyl group a phenoxy group, or a C.sub.3 -C.sub.10 cycloalkyl group, which may be substituted; and Y indicates CH.sub.2 X or XCH.sub.2, in which X represents an ethylene group, a cis -or trans-vinylene group, or an ethynylene group.
摘要翻译： PCT No.PCT / JP86 / 00034 Sec。 371日期1986年9月29日第 102（e）1986年9月29日PCT PCT公布1986年1月28日PCT公布。出版物WO86 / 04330 日期：1986年7月31日。一种用于制备16取代的DELTA 7-前列腺素Es的新方法，其包括由下式（I）表示的化合物，其对映异构体或其混合比的混合物，其中R1表示COOR2，CH2OR3，其中R2表示氢原子，取代或未取代的C1-C10烷基，取代或未取代的C3-C10环烷基或取代或未取代的苯基，R3表示氢原子，三（C 1 -C 7）烃甲硅烷基，与羟基的氧原子一起形成缩醛键的基团或C 2 -C 7酰基; R4和R5相同或不同，各自表示氢原子，三（C1-C7）烃甲硅烷基，或与羟基的氧原子一起形成缩醛键的基团; R6表示氢原子，C1-C4烷基或乙烯基; R7表示可含有氧原子的直链或支链C 3 -C 8烷基，链烯基或炔基; 可被取代的苯基，苯氧基或C3-C10环烷基; 或被可被取代的C1-C6烷氧基，苯基苯氧基或C3-C10环烷基取代的直链或支链C1-C5烷基; Y表示CH2X或XCH2，其中X表示亚乙基，顺式或反式亚乙烯基或亚乙炔基。

2. 发明授权

US4921995A Process for producing 16-substituted prostaglandines 失效
标题翻译：生产16-取代的前列腺素的方法
公开(公告)号：US4921995A
公开(公告)日：1990-05-01
申请号：US153881
申请日：1988-02-09
申请人： Toshio Tanaka , Atsuo Hazato , Seizi Kurozumi , Masahiro Koga
发明人： Toshio Tanaka , Atsuo Hazato , Seizi Kurozumi , Masahiro Koga
IPC分类号： C07C405/00
CPC分类号： C07C405/0033 , C07C405/00
摘要： A novel process for manufacturing 16-substituted .DELTA..sup.7 -prostaglandin Es, which include compounds expressed by the following formula (I), their enanantiomers, or their mixtures of arbitrary mixing ratio, ##STR1## wherein R.sup.1 indicates COOR.sup.2, CH.sub.2 OR.sup.3, or COCH.sub.2 OR.sup.3, in which R.sup.2 indicates a hydrogen atom, a substituted or unsubstituted C.sub.1 -C.sub.10 alkyl group, a substituted or unsubstituted C.sub.3 -C.sub.10 cycloalkyl group, or a substituted or unsubstituted phenyl group, and R.sup.3 indicates a hydrogen atom, a tri(C.sub.1 -C.sub.7) hydrocarbon silyl group, a group which forms an acetal bond together with the oxygen atom of a hydroxyl group, or a C.sub.2 -C.sub.7 acyl group; R.sup.4 and R.sup.5 are identical or different, each representing a hydrogen atom, a tri(C.sub.1 -C.sub.7) hydrocarbon silyl group, or a group which forms an acetal bond together with the oxygen atom of a hydroxyl group; R.sup.6 indicates a hydrogen atom, a C.sub.1 -C.sub.4 alkyl group, or a vinyl group; R.sup.7 indicates a linear or branched C.sub.3 -C.sub.8 alkyl group, an alkyenyl group, or an alkynyl group, which may contain an oxygen atom; a phenyl group, a phenoxy group, or a C.sub.3 - C.sub.10 cycloalkyl group, which may be substituted; or a linear or branched C.sub.1 -C.sub.5 alkyl group which is substituted by a C.sub.1 -C.sub.6 alkoxy group, a phenyl group, a phenoxy group, or a C.sub.3 -C.sub.10 cycloalkyl group, which may be substituted; and Y indicates CH.sub.2 X or XCH.sub.2, in which X represents an ethylene group, a cis -or trans-vinylene group, or an ethynylene group.

3. 发明授权

US5532408A .alpha.-chain-modified isocarbacyclins and process for the production thereof 失效
标题翻译： α-链改性的异卡巴菌素及其制备方法
公开(公告)号：US5532408A
公开(公告)日：1996-07-02
申请号：US411649
申请日：1995-04-05
申请人： Masahiro Koga , Toshio Tanaka , Takao Fujii , Tsukio Masegi
发明人： Masahiro Koga , Toshio Tanaka , Takao Fujii , Tsukio Masegi
IPC分类号： C07C65/19 , C07C69/76 , C07C405/00 , C07C62/06 , C07C69/74 , C07C277/00 , C07F7/04
CPC分类号： C07C65/19 , C07C405/0083 , C07C69/76
摘要： Provided are .alpha.-chain-modified isocarbacyclins of which the .alpha.-chain is modified with a phenylene group, a cycloalkylene group or a thiophendiyl group, and these .alpha.-chain-modified isocarbacyclins show the activity for inhibiting the DNA synthesis of human smooth muscle cell and are expected to be capable of inhibiting the hypertrophy of a blood vessel.
摘要翻译： PCT No.pct / jp93 / 01407 Sec。 371日期1995年04月5日 102（e）日期1995年4月5日PCT提交1993年10月1日PCT公布。 No.WO94 / 07838 PCT出版物日期为1995年4月14日。提供了α-链改性的异卡巴环素，其中α-链用亚苯基，亚环烷基或噻吩二基修饰，并且这些α-链修饰的异卡巴菌素显示出抑制预期人平滑肌细胞的DNA合成能够抑制血管的肥大。

4. 发明申请

US20110148146A1 PICK-UP STYLE UTILITY VEHICLE WITH EXPANDABLE CARGO BED 有权
标题翻译：具有可扩展性的货架的拾起风格的实用车辆
公开(公告)号：US20110148146A1
公开(公告)日：2011-06-23
申请号：US12646041
申请日：2009-12-23
申请人： Satoshi TAKAYA , Masafumi Inoue , Shinichi Tanba , Daisuke Takagi , Masahiro Koga , Yoshitaka Nishikawa , Takao Kawabata , Dave Reinke
发明人： Satoshi TAKAYA , Masafumi Inoue , Shinichi Tanba , Daisuke Takagi , Masahiro Koga , Yoshitaka Nishikawa , Takao Kawabata , Dave Reinke
IPC分类号： B60N2/36 , B60N2/30
CPC分类号： B60N2/36 , B60N2/3011 , B60N2/3065 , B60N2002/363
摘要： The present invention is a pick-up style utility vehicle with an expandable cargo bed, including a front seat, a rear seat, a stationary bottom plate serving as a bottom face of the cargo bed, an expansion bottom plate for expanding the bottom face of the cargo bed, and a shared linkage mechanism for holding the rear seat at a use position where the rear seat is positioned on the upper side of the stationary bottom plate and a shunting position where the rear seat is shunted into a rear leg room provided on the front lower side of the stationary bottom plate, and also for holding the expansion bottom plate at a storage position where the expansion bottom plate is placed out of the upper side of the leg room and an expansion position where the expansion bottom plate is positioned on the upper side of the leg room.
摘要翻译：本发明是一种具有可膨胀货物床的拾取式多用途车，包括前排座椅，后座椅，用作货物底面的固定底板，膨胀底板，用于将底面扩张货舱，以及用于将后座椅保持在后座位于固定底板上侧的使用位置的共用连杆机构以及后排座椅分流到设置在其上的后腿房间的分流位置固定底板的前下侧，还用于将膨胀底板保持在扩张底板放置在腿部房间上侧的存放位置和膨胀底板位于其上的展开位置腿部房间的上侧。

5. 发明授权

US4167506A Diazaphenalene derivatives and resin containing color compositions 失效
标题翻译：二氮杂萘衍生物和含有颜色组合物的树脂
公开(公告)号：US4167506A
公开(公告)日：1979-09-11
申请号：US832914
申请日：1977-09-13
申请人： Keizo Shimada , Toshiaki Harada , Masahiro Koga , Shizuo Nagahama , Hiroyoshi Minematsu , Hidetsugu Yoshida
发明人： Keizo Shimada , Toshiaki Harada , Masahiro Koga , Shizuo Nagahama , Hiroyoshi Minematsu , Hidetsugu Yoshida
IPC分类号： C07D215/04 , C07D215/18 , C07D215/38 , C07D471/16 , C07D471/22 , C07D519/00 , C08K5/00 , C09B57/08 , C09B57/12 , C07D471/06
CPC分类号： C07D215/04 , C07D215/18 , C07D215/38 , C08K5/0041 , C09B57/08 , C09B57/12
摘要： A group of novel polynuclear heterocyclic compounds having a diazaphenalene skeleton. These compounds assume orange to reddish violet colors according to the types of substituents on the diazaphenalene skeleton, and have excellent thermal stability and weatherability and good dispersibility in polymeric materials. They are useful as orange to reddish violet pigments, especially for coloring polymeric materials.
摘要翻译：一组具有二氮杂萘骨架的新型多核杂环化合物。这些化合物根据二氮杂萘骨架上的取代基的类型，呈橙色至红紫色，并具有优异的热稳定性和耐候性以及在聚合物材料中的良好分散性。它们可用作橙色以使紫色颜料变红，特别是用于着色聚合物材料。

6. 发明申请

US20080305677A1 Electrical Connector for Flat Flexible Cable 审中-公开
标题翻译：扁平柔性电缆用电连接器
公开(公告)号：US20080305677A1
公开(公告)日：2008-12-11
申请号：US11666564
申请日：2005-11-01
申请人： Masahiro Koga
发明人： Masahiro Koga
IPC分类号： H01R12/24
CPC分类号： H01R12/79 , H01R12/88
摘要： An electric connector enabling multipolarization increasing the number of contact pieces by reducing a pressing force with which the contact pieces act on an actuator when the actuator is opened, including the actuator, the contact pieces, and a casing. The actuator includes an actuator body part and an actuator operation part. Each of the contact pieces comprises includes a top part beam, a contact beam, and a fixed base part beam. The contact beam and the top beam are formed in cantilever configurations. The contact beam opens the actuator so as to be pushed up when the actuator operation part touches near the free end of the contact beam to act a pressing force in one direction on the actuator operation part. The top part is pushed up when the actuator body part touches near the free end of the top beam to act a pressing force in the other direction facing the opposite direction of the pressing force to one direction of the contact beam on the actuator body part.
摘要翻译：一种能够实现多极化的电连接器，包括致动器，接触片和壳体，通过减小当致动器打开时接触片作用在致动器上的按压力来增加接触件的数量。致动器包括致动器主体部和致动器操作部。每个接触件包括顶部梁，接触梁和固定的基部梁。接触梁和顶梁以悬臂结构形成。接触梁打开致动器，以便当致动器操作部分接触接触梁的自由端附近以在致动器操作部分上沿一个方向施加按压力时被推动。当致动器主体部分靠近顶部梁的自由端接触时，顶部被向上推动，以在朝向与致动器主体部分上的接触梁的一个方向相反的按压力的另一方向上施加按压力。

7. 发明申请

US20060128198A1 Movable connector 失效
标题翻译：活动连接器
公开(公告)号：US20060128198A1
公开(公告)日：2006-06-15
申请号：US10540812
申请日：2003-12-26
申请人： Masahiro Koga
发明人： Masahiro Koga
IPC分类号： H01R13/64
CPC分类号： H01R12/724 , H01R13/639
摘要： A connector, being a connector whereof one portion of the housing protrudes, and wherefor an electrical connection and mechanical fixation is achieved by said protruding portion being housed within a recessed portion of an opposing connector, wherein the housing has a fixing portion for fixing to a board and a movable said protruding portion, and said protruding portion is supported by the fixing portion of the housing via contact portions, and said protruding portion has stoppers for stopping said protruding portion by coming into contact with the contact portions when inserting the connector, and said contact portions have stoppers for stopping said protruding portion by coming into contact with the housing when removing the connector.
摘要翻译：作为连接器的连接器，其中壳体的一部分突出，并且通过所述突出部分容纳在相对的连接器的凹部内而实现电连接和机械固定，其中所述壳体具有用于固定到并且所述突出部分通过接触部分由壳体的固定部分支撑，并且所述突出部分具有用于在插入连接器时通过与接触部分接触而停止所述突出部分的止动件，并且所述接触部分具有用于在移除连接器时通过与壳体接触来停止所述突出部分的止动件。

8. 发明授权

US06753435B1 Intermediates for vitamin D and processes for the preparation thereof 失效
标题翻译：维生素D的中间体及其制备方法
公开(公告)号：US06753435B1
公开(公告)日：2004-06-22
申请号：US10239778
申请日：2002-09-25
申请人： Masahiro Koga , Toru Minoshima
发明人： Masahiro Koga , Toru Minoshima
IPC分类号： C07C40100
CPC分类号： C07C401/00 , C07C309/65 , C07C2601/14 , C07C2601/16 , C07C2602/24 , C07F7/1804 , C07F7/1892
摘要： An object of the present invention is to provide intermediates for the synthesis of 1&agr;-hydroxyvitamin D derivatives useful as drugs and processes for the preparation thereof. Namely, the present invention is a process for the preparation of a compound represented by the formula (2), which comprises reacting a compound represented by the formula (1) with a compound represented by the formula (4) in the presence of a palladium catalyst, a process for the preparation of a compound represented by the formula (3), which comprises further catalytically reducing the resulting compound represented by the formula (2) in the presence of a Lindlar catalyst and hydrogen gas and heating the obtained product and a process for the preparation of a compound represented by the formula (5), which comprises further oxidizing the resulting compound represented by the formula (3) with an oxidizing agent and the compounds represented by the formulae (1) to (3):
摘要翻译：本发明的目的是提供用作合成作为药物的1α-羟基维生素D衍生物的中间体及其制备方法。本发明是制备式（2）表示的化合物的方法，其包括在钯催化剂存在下使式（1）表示的化合物与式（4）表示的化合物反应，制备由式（3）表示的化合物的方法，该方法还包括在Lindlar催化剂和氢气的存在下催化还原由式（2）表示的化合物，并加热得到的产物和制备由式（5）表示的化合物的方法，该方法包括进一步氧化所得由式（3）表示的化合物与氧化剂和由式（1）至（3）表示的化合物：

9. 发明授权

US4067870A 8-Benzimido substituted quinaphthalone derivatives 失效
标题翻译： 8-苯甲亚胺基取代的喹酞酮衍生物
公开(公告)号：US4067870A
公开(公告)日：1978-01-10
申请号：US718198
申请日：1976-08-26
申请人： Keizo Shimada , Toshiaki Harada , Masahiro Koga , Shizuo Nagahama
发明人： Keizo Shimada , Toshiaki Harada , Masahiro Koga , Shizuo Nagahama
IPC分类号： C09B25/00
CPC分类号： C09B25/00 , Y10S8/92
摘要： A compound of the following formula ##STR1## wherein R represents an alkyl group containing 1 to 4 carbon atoms or a phenyl group; X.sub.1 represents a chlorine or bromine atom; Y represents the group of the formula ##STR2## WHEREIN X.sub.2 and X.sub.3 each represent a chlorine or bromine atom, and n is an integer of 2 to 4; and ring A may be substituted by an alkyl group containing 1 to 4 carbon atoms and or a halogen atom.The compound of formula (I) can be easily produced by reacting a quinoline derivative of the formula ##STR3## wherein R, X.sub.1 and the ring A are the same as defined above, with an aryldicarboxylic acid or its reactive derivatives.The compounds of formula (I) are useful as yellow organic pigments.
摘要翻译：下式的化合物，其中R表示含有1至4个碳原子的烷基或苯基; X1表示氯或溴原子; Y表示式中的基团，其中X 1和X 2各自表示氯或溴原子，n表示2〜4的整数。并且环A可以被含有1至4个碳原子的烷基和/或卤素原子取代。

10. 发明申请

US20140051291A1 FPC SHIELDED CONNECTOR 审中-公开
标题翻译： FPC屏蔽连接器
公开(公告)号：US20140051291A1
公开(公告)日：2014-02-20
申请号：US13810732
申请日：2011-07-19
申请人： Michel Safir , Jean Razafiarivelo , Nicolas Hermeline , Jean-Francois Michel , Masahiro Koga
发明人： Michel Safir , Jean Razafiarivelo , Nicolas Hermeline , Jean-Francois Michel , Masahiro Koga
IPC分类号： H01R12/61
CPC分类号： H01R12/61 , H01R12/67 , H01R12/775 , H01R12/79 , H01R12/88
摘要： Connector (1) for flexible printed circuit (FPC) (3) comprising a connector housing (5) including an insertion slot (4) adapted to receive the FPC (3). The connector comprises a shield (18) adapted to be electrically connected to a ground path (2a) of a circuit substrate (2) on which the connector (1) is to be mounted. Said insertion slot (4) comprises a signal side corresponding to conductive tracks (29) of the FPC and a ground side (26a) opposite to said signal side. The shield comprises at least one electrically conductive tooth (25), movable from a retracted position outside the insertion slot (4), to a protruding position where said tooth (25) protrudes from the ground side (26a) to the inside of the insertion slot (4).
摘要翻译：一种用于柔性印刷电路（FPC）（3）的连接器（1），包括连接器壳体（5），该连接器壳体包括适于容纳FPC（3）的插槽（4）。连接器包括适于电连接到要安装连接器（1）的电路基板（2）的接地路径（2a）的屏蔽（18）。所述插槽（4）包括对应于FPC的导电轨道（29）的信号侧和与所述信号侧相对的接地侧（26a）。所述护罩包括至少一个导电齿（25），其可从所述插入槽（4）的外部的缩回位置移动到所述齿（25）从所述接地侧（26a）向所述插入件的内部突出的突出位置槽（4）。

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