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1. 发明授权

US4521339A Ansatrienols 失效
标题翻译：安息托龙
公开(公告)号：US4521339A
公开(公告)日：1985-06-04
申请号：US444474
申请日：1982-11-24
申请人： Noboru Otake , Haruo Seto , Tetsuo Sasaki , Masanori Sugita , Yohei Natori , Noriyoshi Sueda
发明人： Noboru Otake , Haruo Seto , Tetsuo Sasaki , Masanori Sugita , Yohei Natori , Noriyoshi Sueda
IPC分类号： C07D225/06 , C12P17/10
CPC分类号： C12R1/465 , C07D225/06 , C12P17/10
摘要： The disclosure describes a microbiological process for the preparation of mycotrien-related compounds.The compounds are isolated and characterized by structural formula and other identifying data.The compounds are useful in the treatment of tumors.
摘要翻译：本公开描述了用于制备微生物相关化合物的微生物过程。通过结构式和其他识别数据分离和表征化合物。这些化合物可用于治疗肿瘤。

2. 发明授权

US4649135A Mycotrienin-related compounds 失效
标题翻译：生长霉素相关化合物
公开(公告)号：US4649135A
公开(公告)日：1987-03-10
申请号：US852441
申请日：1986-04-15
申请人： Noboru Otake , Haruo Seto , Tetsuo Sasaki , Masanori Sugita , Shigeru Hiramoto
发明人： Noboru Otake , Haruo Seto , Tetsuo Sasaki , Masanori Sugita , Shigeru Hiramoto
IPC分类号： C07D225/06 , C12P17/10 , A61K31/395
CPC分类号： C12R1/465 , C07D225/06 , C12P17/10
摘要： Mycotrienin-related compounds called the T-23-X, -XI, -XII, -XIII and -XIV. These compounds are isolated and characterized by structural formula and other identifying data. They are useful in the treatment of tumors.
摘要翻译：称为T-23-X，-XI，-XII，-XIII和-XIV的类霉素相关化合物。这些化合物被分离并通过结构式和其他鉴定数据表征。它们可用于治疗肿瘤。

3. 发明授权

US4587237A Mycotrienin-related compounds 失效
标题翻译：生长霉素相关化合物
公开(公告)号：US4587237A
公开(公告)日：1986-05-06
申请号：US773445
申请日：1985-09-06
申请人： Noboru Otake , Haruo Seto , Tetsuo Sasaki , Masanori Sugita , Shigeru Hiramoto
发明人： Noboru Otake , Haruo Seto , Tetsuo Sasaki , Masanori Sugita , Shigeru Hiramoto
IPC分类号： C07D225/06 , A61K31/395 , C12P17/10
CPC分类号： C07D225/06
摘要： Mycotrienin-related compounds called the T-23-VIII and T-23-IX substances. These substances are isolated and characterized by structural formula and other identifying data. These substances are useful in the treatment of tumors.
摘要翻译：称为T-23-VIII和T-23-IX物质的类霉素相关化合物。这些物质被隔离并用结构式和其他识别数据表征。这些物质可用于治疗肿瘤。

4. 发明授权

US5252580A Indole derivatives and anti-ulcer compositions thereof 失效
标题翻译：吲哚衍生物及其抗溃疡组合物
公开(公告)号：US5252580A
公开(公告)日：1993-10-12
申请号：US947169
申请日：1992-09-18
申请人： Toshihiro Takahashi , Hitoshi Inoue , Masato Horigome , Kenichi Momose , Masanori Sugita , Kouichi Katsuyama , Chikako Suzuki , Shinji Nagai , Masao Nagase , Koichi Nakamaru
发明人： Toshihiro Takahashi , Hitoshi Inoue , Masato Horigome , Kenichi Momose , Masanori Sugita , Kouichi Katsuyama , Chikako Suzuki , Shinji Nagai , Masao Nagase , Koichi Nakamaru
IPC分类号： A61K31/395 , A61K31/435 , A61K31/437 , A61P1/04 , C07D471/04 , C07D471/14 , C07D487/04 , C07D519/00 , A61K31/445 , C07D401/06
CPC分类号： C07D471/04
摘要： Disclosed are indole derivatives of formula (I) ##STR1## wherein Y represents H, C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.6 alkoxy or halogen;Z represents --CH.sub.2 N(R.sub.5)--;R represents H or --CH.sub.2 CH.sub.2 X where X represents pyridyl, aralkyloxy or substituted amino of NR.sub.6 R.sub.7 where R.sub.6 represents H, C.sub.1 -C.sub.6 alkyl, aralkyl, C.sub.1 -C.sub.6 alkoxycarbonyl, aralkyloxycarbonyl or halogenated C.sub.1 -C.sub.6 alkoxycarbonyl and R.sub.7 represents H, C.sub.1 -C.sub.6 alkyl or aralkyl, or together with R.sub.2 may form a ring of --(CH.sub.2).sub.n -- (n is 1-4) or ##STR2## R.sub.1 represents H, C.sub.1 -C.sub.6 alkyl, aralkyl or arylsulfonyl; R.sub.2 represents C.sub.1 -C.sub.6 alkyl, hydroxy, C.sub.1 -C.sub.6 alkoxy or aralkyloxy;R.sub.3 represents H, C.sub.1 -C.sub.6 alkyl, aralkyl or halogenated C.sub.1 -C.sub.6 alkyl;R.sub.4 and R.sub.5 may be the same or different and each represents H, C.sub.1 -C.sub.6 alkyl or aralkyl or both may together form a ring of --(CH.sub.2).sub.m -- (m is 3 or 4);or pharmaceutically acceptable acid addition salts thereof. They are useful as an antiulcer agent.

5. 发明授权

US4892164A Frame and body construction for small snowmobile 失效
标题翻译：小型雪地车的框架和车身构造
公开(公告)号：US4892164A
公开(公告)日：1990-01-09
申请号：US163389
申请日：1988-03-02
申请人： Toshihiro Yasui , Masanori Sugita , Tsuneo Isobe
发明人： Toshihiro Yasui , Masanori Sugita , Tsuneo Isobe
IPC分类号： B60K13/02 , B62M27/02 , F02M15/00 , F02M19/00
CPC分类号： B62M27/02 , B60K13/02 , F02M15/00 , F02M19/00 , B62M2027/021
摘要： A frame and body construction for a small snowmobile comprised of a generally open tubular frame to which a light weight generally inverted cup shape body is detachably connected. To prevent carburetor icing, an insulating box encircles the carburetor and cooperates with the body, when the body is in place.
摘要翻译：一种用于小型雪地车的框架和车身构造，其由大体上敞开的管状框架组成，轻量级大体上倒置的杯形体可拆卸地连接到该框架上。为了防止化油器结冰，绝缘箱环绕化油器，并在机体就位时与机身配合。

6. 发明授权

US5380723A Indole derivatives 失效
标题翻译：吲哚衍生物
公开(公告)号：US5380723A
公开(公告)日：1995-01-10
申请号：US228505
申请日：1994-04-15
申请人： Toshihiro Takahashi , Hitoshi Inoue , Masato Horigome , Kenichi Momose , Masanori Sugita , Kouichi Katsuyama , Chikako Suzuki , Shinji Nagai , Masao Nagase , Koichi Nakamaru
发明人： Toshihiro Takahashi , Hitoshi Inoue , Masato Horigome , Kenichi Momose , Masanori Sugita , Kouichi Katsuyama , Chikako Suzuki , Shinji Nagai , Masao Nagase , Koichi Nakamaru
IPC分类号： A61K31/40 , A61K31/403 , A61K31/404 , A61K31/4045 , A61K31/44 , A61K31/4427 , A61K31/4439 , A61K31/445 , A61K31/454 , A61K31/47 , A61K31/4725 , A61K31/5377 , A61P1/04 , C07D209/14 , C07D209/16 , C07D401/04 , C07D401/14 , C07D413/04 , C07D403/14 , C07D413/14
CPC分类号： C07D401/14 , C07D209/16
摘要： Disclosed are indole derivatives of formula (I) ##STR1## wherein X and Y each independently represent H or --CH.sub.2 CH.sub.2 R; R represents pyridyl or substituted amino of NR.sub.1 R.sub.2 ;R.sub.1 represents H or C.sub.1 -C.sub.6 alkyl;R.sub.2 represents 2-(3-indolyl)ethyl or aralkyl; orR.sub.1 and R.sub.2 together with the nitrogen atom to which they are attached may form an N-containing 5 to 6 membered hetero ring, an N, O-containing hetero ring, which hetero ring may be fused with benzene;n is an integer of 4 to 8;with the proviso that X and Y both do not represent H or piperizinoethyl when n is 4, or pharmaceuticaly acceptable acid addition salts thereof. They are useful as an antiulcer agent.
摘要翻译：公开了式（I）的吲哚衍生物其中X和Y各自独立地表示H或-CH 2 CH 2 R; R代表NR1R2的吡啶基或取代氨基; R1代表H或C1-C6烷基; R2代表2-（3-吲哚基）乙基或芳烷基; 或R 1和R 2与它们所连接的氮原子一起可以形成含N的5至6元杂环，含N，O的杂环，该杂环可以与苯稠合; n为4〜8的整数，条件是当n为4时X和Y都不表示H或哌嗪子基，或其药学上可接受的酸加成盐。它们作为抗溃疡剂是有用的。

7. 发明授权

US5326879A Indole derivatives 失效
标题翻译：吲哚衍生物
公开(公告)号：US5326879A
公开(公告)日：1994-07-05
申请号：US949028
申请日：1992-09-22
申请人： Toshihiro Takahashi , Hitoshi Inoue , Masato Horigome , Kenichi Momose , Masanori Sugita , Kouichi Katsuyama , Chikako Suzuki , Shinji Nagai , Masao Nagase , Koichi Nakamaru
发明人： Toshihiro Takahashi , Hitoshi Inoue , Masato Horigome , Kenichi Momose , Masanori Sugita , Kouichi Katsuyama , Chikako Suzuki , Shinji Nagai , Masao Nagase , Koichi Nakamaru
IPC分类号： A61K31/40 , A61K31/403 , A61K31/404 , A61K31/4045 , A61K31/44 , A61K31/4427 , A61K31/4439 , A61K31/445 , A61K31/454 , A61K31/47 , A61K31/4725 , A61K31/5377 , A61P1/04 , C07D209/14 , C07D209/16 , C07D401/04 , C07D401/14 , C07D413/04 , C07D403/06
CPC分类号： C07D401/14 , C07D209/16
摘要： Disclosed are indole derivatives of formula (I) ##STR1## wherein X and Y each independently represent H or --CH.sub.2 CH.sub.2 R;R represents pyridyl or substituted amino of NR.sub.1 R.sub.2 ;R.sub.1 represents H or C.sub.1 -C.sub.6 alkyl;R.sub.2 represents 2-(3-indolyl)ethyl or aralkyl; orR.sub.1 and R.sub.2 together with the nitrogen atom to which they are attached may form an N-containing 5 to 6 membered hetero ring, an N, O-containing hetero ring, which hetero ring may be fused with benzene;n is an integer of 4 to 8;with the proviso that X and Y both do not represent H or piperizinoethyl when n is 4, or pharmaceuticaly acceptable acid addition salts thereof. They are useful as an antiulcer agent.
摘要翻译：公开了式（I）的吲哚衍生物代表H或-CH 2 CH 2 R; R代表NR1R2的吡啶基或取代氨基; R1代表H或C1-C6烷基; R2代表2-（3-吲哚基）乙基或芳烷基; 或R 1和R 2与它们所连接的氮原子一起可以形成含N的5至6元杂环，含N，O的杂环，该杂环可以与苯稠合; n为4〜8的整数，条件是当n为4时X和Y都不表示H或哌嗪子基，或其药学上可接受的酸加成盐。它们作为抗溃疡剂是有用的。

8. 发明授权

US5182267A Anti-cancer activity potentiator 失效
标题翻译：抗癌活性增强剂
公开(公告)号：US5182267A
公开(公告)日：1993-01-26
申请号：US626302
申请日：1990-12-12
申请人： Osamu Ogawa , Ikuo Kishi , Yoshiyuki Tahara , Masanori Sugita
发明人： Osamu Ogawa , Ikuo Kishi , Yoshiyuki Tahara , Masanori Sugita
IPC分类号： A61K9/107 , A61K31/135
CPC分类号： A61K9/1075 , A61K31/135
摘要： A pharmaceutical oil-in-water type microemulsion having an action of potentiating the activities of anti-cancer agents, said micro-emulsion comprisesfine particles of a vegetable oil or a triglyceride of a medium-chain fatty acid having 8 to 12 carbon atoms containing 0.1 to 10% (w/v) of N-solanesyl-N,N'-bis(3,4-dimethoxybenzyl)ethylenediamine malate of formula (I) below, ##STR1## an aqueous medium, and 0.05 to 25% (w/v) of a physiologically acceptable phospholipid for dispersing said fine particles in said aqueous medium.
摘要翻译：具有增强抗癌剂活性的作用的药用油包水型微乳液，所述微乳液包含具有8至12个碳原子的中链脂肪酸的植物油或甘油三酸酯的细颗粒，其含有 0.1至10％（w / v）下式（I）的N-茄酰基-N，N'-双（3,4-二甲氧基苄基）乙二胺苹果酸盐，水性介质，和用于将所述细颗粒分散在所述水性介质中的生理学上可接受的磷脂的0.05至25％（w / v）。

9. 发明授权

US5217398A Pedal operated catamaran 失效
标题翻译：脚踏双体船
公开(公告)号：US5217398A
公开(公告)日：1993-06-08
申请号：US868225
申请日：1992-04-14
申请人： Abraham Meron , Masanori Sugita
发明人： Abraham Meron , Masanori Sugita
IPC分类号： B63H16/18 , B63H16/20
CPC分类号： B63H16/14 , B63H2016/202
摘要： A pedal operated catamaran includes a pair of side-by-side buoyant hulls, and a rigid frame releasably mounted to the hulls in one of two alternative positions, to maintain the hulls parallel to one another. The catamaran includes a propeller mounted for rotation with an elongated, longitudinal propeller drive shaft. A gear train drivably associates the propeller drive shaft and a crankshaft, for propeller rotation responsive to rotation of the crankshaft. The propeller drive shaft further is pivotally mounted to allow selective alternative latching of the propeller in a retracted position and in one of several operating positions, as controlled by a hand-operated lever. The latching mechanism allows on-the-fly adjustment of the propeller position. In the retracted position, the propeller is automatically angularly locked above the hulls, to facilitate car top carrying of the craft without disassembly.
摘要翻译：踏板操作的双体船包括一对并排浮力船体，以及刚性框架，其可拆卸地安装在两个替代位置之一的船体上，以保持船体彼此平行。双体船包括螺旋桨，其安装成与细长的纵向螺旋桨传动轴一起旋转。齿轮系可驱动地将螺旋桨驱动轴和曲轴相关联，用于响应于曲轴的旋转的螺旋桨旋转。螺旋桨驱动轴进一步枢转地安装，以允许螺旋桨在缩回位置和由手动操作杆控制的多个操作位置中的一个中选择性地替换。闩锁机构允许螺旋桨位置的即时调节。在缩回位置，螺旋桨自动地角度地锁定在船体上方，以方便车顶运送而不拆卸。

10. 发明授权

US5060745A Engine mounting arrangement and drive mechanism for small snowmobiles 失效
标题翻译：小型雪车的发动机安装布置和驱动机构
公开(公告)号：US5060745A
公开(公告)日：1991-10-29
申请号：US480532
申请日：1990-02-15
申请人： Toshihiro Yasui , Masanori Sugita , Tsuneo Isobe , Haruhiko Nakanosono
发明人： Toshihiro Yasui , Masanori Sugita , Tsuneo Isobe , Haruhiko Nakanosono
IPC分类号： B62M27/02
CPC分类号： B62M27/02 , B62M2027/021 , B62M2027/023 , B62M2027/026
摘要： An improved drive unit and suspension arrangement therefor for a small snowmobile having an open tubular frame. The drive unit includes an internal combustion engine and a pulley type transmission. The pulley type transmission is supported within a transmission casing and is affixed to the frame for rigidifying the frame. The suspension permits more vertical compliance than for and aft compliance for vibration dampening without adversely effecting the rigidity.

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