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61. 发明授权

US4518415A 1-(Tetrahydrofurylmethyl)azoles 失效
标题翻译： 1-（四氢呋喃基甲基）唑
公开(公告)号：US4518415A
公开(公告)日：1985-05-21
申请号：US459966
申请日：1983-01-21
申请人： Anthony F. Marchington , Timothy Lewis , John M. Clough , Paul A. Worthington , John Dalziel
发明人： Anthony F. Marchington , Timothy Lewis , John M. Clough , Paul A. Worthington , John Dalziel
IPC分类号： C07C29/14 , C07C29/147 , C07C29/36 , C07C29/40 , C07C45/29 , C07C45/60 , C07C45/68 , C07C47/24 , C07C51/347 , C07C59/88 , C07D233/60 , C07D249/08 , C07D303/40 , C07D307/10 , C07D319/06 , C07D521/00 , A01N43/50 , A01N43/64 , C07D405/06 , C07F1/00
CPC分类号： C07D307/10 , C07C29/14 , C07C29/147 , C07C29/36 , C07C29/40 , C07C45/292 , C07C45/60 , C07C45/68 , C07C47/24 , C07C51/347 , C07C59/88 , C07D231/12 , C07D233/56 , C07D249/08 , C07D303/40 , C07D319/06
摘要： Compounds useful as plant growth regulators and fungicides and having the formula ##STR1## and stereoisomers thereof, wherein W is --CH.dbd. or .dbd.N--; Q is optionally substituted aryl, especially optionally substituted phenyl, or optionally substituted aralkyl or alkyl; R.sup.1, R.sup.2, R.sup.3, R.sup.4, R.sup.5 and R.sup.6, which may be the same or different, are H, optionally substituted alkyl, cycloalkyl, aralkyl or phenyl; R.sup.7 and R.sup.8 are H, alkyl or optionally substituted phenyl; and acid addition salts and metal complexes thereof, and processes and intermediates for their preparation.
摘要翻译：可用作植物生长调节剂和杀真菌剂并具有式（I）的式（I）及其立体异构体的化合物，其中W为-CH =或= N-; Q是任选取代的芳基，特别是任选取代的苯基，或任选取代的芳烷基或烷基; R 1，R 2，R 3，R 4，R 5和R 6可以相同或不同，为H，任选取代的烷基，环烷基，芳烷基或苯基; R 7和R 8是H，烷基或任选取代的苯基; 及其加成盐及其金属络合物，以及其制备方法和中间体。

62. 发明授权

US5229391A Pyrimidine derivatives and their use as fungicidal agents 失效
标题翻译：嘧啶衍生物及其作为杀真菌剂的用途
公开(公告)号：US5229391A
公开(公告)日：1993-07-20
申请号：US739468
申请日：1991-08-02
申请人： John M. Clough , Christopher R. A. Godfrey , Ian T. Streeting
发明人： John M. Clough , Christopher R. A. Godfrey , Ian T. Streeting
IPC分类号： A01N43/54 , C07D401/12
CPC分类号： C07D401/12 , A01N43/54
摘要： Fungicidal compounds having the formula (I): ##STR1## in which any two of K, L and M are nitrogen and the other is CE; X and Y are independently hydrogen, halogen, C.sub.1-4 alkyl, C.sub.3-6 cycloalkyl, C.sub.2-4 alkenyl, C.sub.2-4 alkynyl, C.sub.2-4 alkenyloxy, C.sub.2-4 alkynyloxy, phenyl, benzyloxy, cyano, isocyano, isothiocyanato, nitro, NR.sup.1 R.sup.2, NR.sup.1 OR.sup.2, N.sub.3, NHCOR.sup.1, NR.sup.1 CO.sub.2 R.sup.2, NHCONR.sup.1 R.sup.2, N.dbd.CHNR.sup.1 R.sup.2, NHSO.sub.2 R.sup.1, OR.sup.1, OCOR.sup.1, OSO.sub.2 R.sup.1, SR.sup.1, SOR.sup.1, SO.sub.2 R.sup.1, SO.sub.2 OR.sup.1, SO.sub.2 NR.sup.1 R.sup.2, COR.sup.1, CR.sup.1 .dbd.NOR.sup.2, CHR.sup.1 CO.sub.2 R.sup.2, CO.sub.2 R.sup.1, CONR.sup.1 R.sup.2, CSNR.sup.1 R.sup.2, CH.sub.3 O.sub.2 C.C:CH.OCH.sub.3, 1-(imidazol-1-yl)vinyl, a 5-membered heterocyclic ring containing one, two or three nitrogen heteroatoms, or a 5- or 6-membered heterocyclic ring containing one or two oxygen or sulphur heteroatoms, optionally a nitrogen heteroatom and optionally one or two oxo or thioxo substituents; or X and Y, when ortho to one another, join to form a 5- or 6-membered aliphatic or aromatic ring optionally containing one or two oxygen, sulphur or nitrogen atoms or one, two or three nitrogen or sulphur atoms; A, B, E, G and U are independently hydrogen, halogen, C.sub.1-4 alkyl, C.sub.1-4 alkoxy, cyano, nitro or trifluoromethyl; and R.sup.1 and R.sup.2 are independently hydrogen, C.sub.1-4 alkyl, C.sub.2-4 alkenyl or phenyl; the aliphatic moieties of any of the foregoing being optionally substituted with one or more of halogen, cyano, OR.sup.1, SR.sup.1, NR.sup.1 R.sup.2, SiR.sup.1.sub.3 or OCOR.sup.1 and the phenyl moieties of any of the foregoing being optionally substituted with one or more of halogen, C.sub.1-4 alkyl, C.sub.1-4 alkoxy, nitro or cyano; and their pyridine N-oxides and N-alkyl pyridinium salts.
摘要翻译：具有式（I）的杀真菌化合物：其中K，L和M中的任一个为氮，另一个为CE; X和Y独立地是氢，卤素，C 1-4烷基，C 3-6环烷基，C 2-4烯基，C 2-4炔基，C 2-4链烯氧基，C 2-4炔氧基，苯基，苄氧基，氰基，异氰基，异硫氰酸根合，硝基，NR1R2，NR1OR2，N3，NHCOR1，NR1CO2R2，NHCONR1R2，N = CHNR1R2，NHSO2R1，OR1，OCOR1，OSO2R1，SR1，SOR1，SO2R1，SO2OR1，SO2NR1R2，COR1，CR1 = NOR2，CHR1CO2R2，CO2R1，CONR1R2，CSNR1R2，CH3O2C C：CH.OCH 3，1-（咪唑-1-基）乙烯基，含有一个，两个或三个氮杂原子的5元杂环，或含有一个或两个氧或硫的5-或6-元杂环杂原子，任选的氮杂原子和任选的一个或两个氧代或硫代取代基; 或X和Y，当彼此邻接时，连接形成任选地含有一个或两个氧，硫或氮原子或一个，两个或三个氮或硫原子的5-或6-元脂族或芳族环; A，B，E，G和U独立地为氢，卤素，C 1-4烷基，C 1-4烷氧基，氰基，硝基或三氟甲基; 并且R 1和R 2独立地是氢，C 1-4烷基，C 2-4链烯基或苯基; 前述任何一个的脂肪族部分任选被一个或多个卤素，氰基，OR 1，SR 1，NR 1 R 2，SiR 13或OCOR 1取代，并且前述任何一个的苯基部分任选被一个或多个卤素， 4烷基，C 1-4烷氧基，硝基或氰基; 和它们的吡啶N-氧化物和N-烷基吡啶鎓盐。

63. 发明授权

US5221691A Fungicides aromatic oxime amides 失效
标题翻译： FUNGICIDES AROMATIC OXIME AMIDES
公开(公告)号：US5221691A
公开(公告)日：1993-06-22
申请号：US827236
申请日：1992-01-29
申请人： John M. Clough , Christopher R. A. Godfrey , Paul J. de Fraine , Ian R. Matthews
发明人： John M. Clough , Christopher R. A. Godfrey , Paul J. de Fraine , Ian R. Matthews
IPC分类号： A01N37/18 , A01N37/50 , A01N43/06 , A01N43/36 , A01N43/40 , A01N43/54 , A01N43/56 , A01N43/60 , A01N43/74 , C07C251/60 , C07C255/62 , C07C317/28 , C07C323/47 , C07D207/06 , C07D207/32 , C07D207/335 , C07D213/26 , C07D213/53 , C07D213/61 , C07D213/63 , C07D213/64 , C07D213/84 , C07D215/18 , C07D215/50 , C07D231/20 , C07D231/22 , C07D233/54 , C07D237/14 , C07D239/26 , C07D239/34 , C07D239/38 , C07D239/42 , C07D239/52 , C07D241/12 , C07D241/18 , C07D241/24 , C07D249/08 , C07D251/02 , C07D263/14 , C07D277/28 , C07D277/54 , C07D277/64 , C07D307/52 , C07D307/81 , C07D307/82 , C07D333/20 , C07D333/22 , C07D333/28 , C07D333/38 , C07D333/58 , C07D521/00 , C07F9/40
CPC分类号： C07D207/335 , A01N37/50 , A01N43/06 , A01N43/36 , A01N43/40 , A01N43/54 , A01N43/56 , A01N43/60 , A01N43/74 , C07C251/60 , C07D213/26 , C07D213/53 , C07D213/61 , C07D213/63 , C07D213/64 , C07D213/84 , C07D231/22 , C07D239/26 , C07D239/34 , C07D239/38 , C07D239/42 , C07D239/52 , C07D241/12 , C07D241/18 , C07D241/24 , C07D277/54 , C07D307/52 , C07D307/82 , C07D333/22 , C07D333/28 , C07D333/58 , C07C2101/14
摘要： Fungicidal compounds having the formula (I): ##STR1## and stereoisomers thereof, wherein A is hydrogen, halo, hydroxy, C.sub.1-4 alkyl, C.sub.1-4 alkoxy, C.sub.1-4 haloalkyl, C.sub.1-4 haloalkoxy, C.sub.1-4 alkylcarbonyl, C.sub.1-4 alkoxycarbonyl, phenoxy, nitro or cyano; R.sup.1 and R.sup.2, which may be the same or different, are hydrogen, optionally substituted alkyl, optionally substituted cycloalkyl, optionally substituted heterocyclylalkyl, optionally substituted cycloalkylalkyl, optionally substituted aralkyl, optionally substituted aryloxyalkyl, optionally substituted heterocyclyloxyalkyl, optionally substituted alkenyl, optionally substituted alkynyl, optionally substituted alkoxy, optionally substituted aryl, optionally substituted heterocyclyl, optionally substituted aryloxy, optionally substituted heterocyclyloxy, nitro, halo, cyano, --NR.sup.3 R.sup.4, --CO.sub.2 R.sup.3, --CONR.sup.3 R.sup.4, --COR.sup.3, --S(O).sub.n R.sup.3 wherein n is 0, 1 or 2, (CH.sub.2).sub.m PO(OR.sup.3).sub.2 wherein m is 0 or 1, or R.sup.1 and R.sup.2 join to form a carbocyclic or heterocyclic ring system; R.sup.3 and R.sup.4, which are the same or different, are hydrogen, optionally substituted alkyl, optionally substituted aralkyl, optionally substituted alkenyl, optionally substituted alkynyl, optionally substituted aryl or optionally substituted heteroaryl, or R.sup.3 and R.sup.4 join to form an optionally substituted heterocyclic ring; and R.sup.5 and R.sup.6 are independently hydrogen or C.sub.1-4 alkyl.
摘要翻译：具有式（I）的杀真菌化合物及其立体异构体，其中A为氢，卤素，羟基，C 1-4烷基，C 1-4烷氧基，C 1-4卤代烷基，C 1-4卤代烷氧基， 4-烷基羰基，C 1-4烷氧基羰基，苯氧基，硝基或氰基; R 1和R 2可以相同或不同，为氢，任选取代的烷基，任选取代的环烷基，任选取代的杂环基烷基，任选取代的环烷基烷基，任选取代的芳烷基，任选取代的芳氧基烷基，任选取代的杂环基烷基，任选取代的烯基，任选取代的炔基，任选取代的烷氧基，任选取代的芳基，任选取代的杂环基，任选取代的芳氧基，任选取代的杂环氧基，硝基，卤素，氰基，-NR 3 R 4，-CO 2 R 3，-CONR 3 R 4，-COR 3，-S（O）n R 3，其中n为0， 1或2，（CH 2）m PO（OR 3）2，其中m为0或1，或R 1和R 2连接形成碳环或杂环系; R 3和R 4相同或不同，为氢，任选取代的烷基，任选取代的芳烷基，任选取代的烯基，任选取代的炔基，任选取代的芳基或任选取代的杂芳基，或R 3和R 4连接形成任选取代的杂环 ; 并且R 5和R 6独立地是氢或C 1-4烷基。

64. 发明授权

US5206245A Fungicidal aromatic pyrimidinyl oxime ethers 失效
标题翻译：杀真菌抗真菌药
公开(公告)号：US5206245A
公开(公告)日：1993-04-27
申请号：US736168
申请日：1991-07-26
申请人： John M. Clough , Christopher R. A. Godfrey , Ian T. Streeting , Rex Cheetham , Paul J. de Fraine
发明人： John M. Clough , Christopher R. A. Godfrey , Ian T. Streeting , Rex Cheetham , Paul J. de Fraine
IPC分类号： A01N43/54 , C07D239/52 , C07D401/12 , C07D403/12 , C07D405/12 , C07D409/12 , C07D413/12 , C07D417/12
CPC分类号： C07D401/12 , A01N43/54 , C07D239/52 , C07D403/12 , C07D405/12 , C07D409/12 , C07D413/10 , C07D417/12
摘要： Fungicidal compounds having the formula (I): ##STR1## in which any two of K, L and M are nitrogen and the other is CE; X and Y are independently hydrogen, halogen, C.sub.1-4 alkyl, C.sub.3-6 cycloalkyl, C.sub.2-4 alkenyl, C.sub.2-4 alkynyl, C.sub.2-4 alkynyloxy, phenyl, benzyloxy, cyano, isocyano, thiocyanato, isothiocyanato, nitro, NR.sup.1 R.sup.2, NR.sup.1 OR.sup.2, N.sub.3, NHCOR.sup.1, NR.sup.1 CO.sub.2 R.sup.2, NHCONR.sup.1 R.sup.2, N.dbd.CHNR.sup.1 R.sup.2, NHSO.sub.2 R.sup.1, OR.sup.1, OCOR.sup.1, OSO.sub.2 R.sup.1, SR.sup.1, SOR.sup.1, SO.sub.2 R.sup.1, SO.sub.2 OR.sup.1,SO.sub.2 NR.sup.1 R.sup.2, COR.sup.1, CR.sup.1 .dbd.NOR.sup.2, CHR.sup.1 CO.sub.2 R.sup.2, CO.sub.2 R.sup.1, CONR.sup.1 R.sup.2, CSNR.sup.1 R.sup.2, CH.sub.3 O.sub.2 C.C:CH.OCH.sub.3, 1-(imidazol-1-yl)vinyl, a 5-membered heterocyclic ring containing one, two or three nitrogen heteroatoms, or a 5- or 6-membered heterocyclic ring containing one or two oxygen or sulphur heteroatoms, optionally a nitrogen heteroatom and optionally one or two oxo or thioxo substituents; or X and Y, when ortho to one another, join to form a 5- or 6-membered aliphatic or aromatic ring optionally containing one or two oxygen, sulphur or nitrogen atoms or one, two or three nitrogen atoms; A, Q, D, E, G, U and V are independently hydrogen, halogen (especially fluorine and chlorine), C.sub.1-4 alkyl (especially methyl), C.sub.1-4 alkoxy (especially methoxy), cyano, nitro or trifluoromethyl; and R.sup.1 and R.sup.2 are independently hydrogen, C.sub.1-4 alkyl, C.sub.2-4 alkenyl or phenyl; the aliphatic moieties of any of the foregoing being optionally substituted with one of more of halogen, cyano, OR.sup.1, SR.sup.1, NR.sup.1 R.sup.2, SiR.sup.1.sub.3 or OCOR.sup.1 and the phenyl moieties of any of the foregoing being optionally substituted with one or more of halogen, C.sub.1-4 alkyl, C.sub.1-4 alkoxy, nitro or cyano.

65. 发明授权

US5198444A Methyl .alpha.-(2-substituted)pyrid-3-yl-.beta.-methoxyacrylates, compositions containing them and their use as fungicides 失效
标题翻译：甲基α-（2-取代）吡啶-3-基-β-甲氧基丙烯酸酯，含有它们的组合物及其作为杀真菌剂的用途
公开(公告)号：US5198444A
公开(公告)日：1993-03-30
申请号：US597398
申请日：1990-10-15
申请人： John M. Clough , Christopher R. A. Godfrey , Stephen P. Heaney , Kenneth Anderton
发明人： John M. Clough , Christopher R. A. Godfrey , Stephen P. Heaney , Kenneth Anderton
IPC分类号： A01N43/40 , A01N43/54 , A01N43/78 , C07D213/64 , C07D213/643 , C07D213/65 , C07D213/68 , C07D213/70 , C07D213/71 , C07D213/74 , C07D213/79 , C07D213/80 , C07D213/81 , C07D213/84 , C07D213/85 , C07D213/89 , C07D401/12 , C07D405/12 , C07D409/12 , C07D413/12 , C07D417/12 , C07D473/30 , C07D473/34 , C07D473/38
CPC分类号： C07D213/643 , A01N43/40 , A01N43/54 , A01N43/78 , C07D213/65 , C07D213/68 , C07D213/70 , C07D213/71 , C07D213/74 , C07D213/79 , C07D213/80 , C07D213/81 , C07D213/84 , C07D213/85 , C07D213/89 , C07D401/12 , C07D405/12 , C07D409/12 , C07D413/12 , C07D417/12 , C07D473/30 , C07D473/34 , C07D473/38
摘要： Fungicidal compounds of the formula (I): ##STR1## and stereoisomers thereof, wherein K is oxygen or sulphur; Z is optionally substituted aryl or optionally substituted heteroaryl; X is O, S(O).sub.n, NR.sup.4, CR.sup.1 R.sup.2, CHR.sup.5, CO, CR.sup.1 (OR.sup.2), C.dbd.CR.sup.1 R.sup.2, CHR.sup.1 CHR.sup.2, CR.sup.1 .dbd.CR.sup.2, CHR.sup.1 CR.sup.2 .dbd.CH, C.dbd.C, OCHR.sup.1, CHR.sup.1 O, OCHR.sup.1 O, S(O).sub.n CHR.sup.1, S(O).sub.n CHR.sup.1 O, CHR.sup.1 S(O).sub.n, CHR.sup.1 OSO.sub.2, NR.sup.4 CHR.sup.1, CHR.sup.1 NR.sup.4, CO.sub.2, O.sub.2 C, SO.sub.2 O, OSO.sub.2, CO.CO, COCHR.sup.1, COCHR.sup.1 O, CHR.sup.1 CO, CHOH.CHR.sup.1, CHR.sup.1.CHOH, ##STR2## CONR.sup.4, OCONR.sup.4, NR.sup.4 CO, CSNR.sup.4, OCS.NR.sup.4, SCO.NR.sup.4, NR.sup.4 CO.sub.2, NR.sup.4 CS, NR.sup.4 CSO, NR.sup.4 COS, NR.sup.4 CONR.sup.4, S(O).sub.n NR.sup.4, NR.sup.4 S(O).sub.n, CS.sub.2, S.sub.2 C, CO.S, SCO, N.dbd.N, N.dbd.CR.sup.1, CR.sup.1 .dbd.N, CHR.sup.1 CHR.sup.2 CH(OH), CHR.sup.1 OCO, CHR.sup.1 SCO, CHR.sup.1 NR.sup.4 CO, CHR.sup.1 NR.sup.4 COR.sup.4, CHR.sup.1 CHR.sup.2 CO, O.N.dbd.CR.sup.1, CHR.sup.1 O.N.dbd.CR.sup.2, CO.OCR.sup.1 R.sup.2, CHR.sup.1 CHR.sup.2 CHR.sup.3, OCHR.sup.1 CHR.sup.2, (CH.sub.2).sub.m O, CHR.sup.1 OCHR.sup.2, CHR.sup.1 CHR.sup.2 O, OCHR.sup.1 CHR.sup.2 O, S(O).sub.n CHR.sup.1 CHR.sup.2, CHR.sup.1 S(O).sub.n CHR.sup.2, CHR.sup.1 CHR.sup.2 S(O).sub.n, CR.sup.1 .dbd.NNR.sup.4, NR.sup.4 N.dbd.CR.sup.1, CHR.sup.1 CONR.sup.2, CHR.sup.1 OCO.NR.sup.2, CH.dbd.CHCH.sub.2 O, COCHR.sup.1 CHR.sup.2 O or (R.sup.5).sub.2 P.sup. + CHR.sup.2 Q.sup.- ; A, B and E, which may be the same or different, are H, hydroxy, halo, C.sub.1-4 alkyl, C.sub.1-4 alkoxy, C.sub.1-4 haloalkyl, C.sub.1-4 haloalkoxy, C.sub.1-4 alkylcarbonyl, C.sub.1-4 alkoxycarbonyl, phenoxy, nitro or cyano; R.sup.1, R.sup.2 and R.sup.3, which may be the same or different, are H, C.sub.1-4 alkyl or phenyl; R.sup.4 is H, C.sub.1-4 alkyl or COR.sup.1 ; R.sup.5 is optionally substituted phenyl; Q.sup.- is a halide anion; n is 0, 1, or 2 and m is a 3, 4 or 5.
摘要翻译：式（I）的杀真菌化合物：其中K为氧或硫; Z是任选取代的芳基或任选取代的杂芳基; X是O，S（O）n，NR4，CR1R2，CHR5，CO，CR1（OR2），C = CR1R2，CHR1CHR2，CR1 = CR2，CHR1CR2 = CH，C = C，OCHR1，CHR1O，OCHR1O，）nCHR1，S（O）nCHR1O，CHR1S（O）n，CHR1OSO2，NR4CHR1，CHR1NR4，CO2，O2C，SO2O，OSO2，CO.CO，COCHR1，COCHR1O，CHR1CO，CHOH.CHR1，CHR1.CHOH， CONR4，OCONR4，NR4CO，CSNR4，OCS.NR4，SCO.NR4，NR4CO2，NR4CS，NR4CSO，NR4COS，NR4CONR4，S（O）nNR4，NR4S（O）n，CS2，S2C，CO.S，SCO，N = N = CR1，CR1 = N，CHR1CHR2CH（OH），CHR1OCO，CHR1SCO，CHR1NR4CO，CHR1NR4COR4，CHR1CHR2CO，ON = CR1，CHR1O.N = CR2，CO.OCR1R2，CHR1CHR2CHR3，OCHR1CHR2，（CH2）mO，CHR1OCHR2， CHR1CHR2O，OCHR1CHR2O，S（O）nCHR1CHR2，CHR1S（O）nCHR2，CHR1CHR2S（O）n，CR1 = NNR4，NR4N = CR1，CHR1CONR2，CHR1OCO.NR2，CH = CHCH2O，COCHR1CHR2O或（R5）2P + CHR2Q-; A，B和E可以相同或不同，是H，羟基，卤素，C 1-4烷基，C 1-4烷氧基，C 1-4卤代烷基，C 1-4卤代烷氧基，C 1-4烷基羰基，C 1-4烷氧基羰基，苯氧基，硝基或氰基; R 1，R 2和R 3可以相同或不同，为H，C 1-4烷基或苯基; R4是H，C1-4烷基或COR1; R5是任选取代的苯基; Q-是卤素阴离子; n为0,1或2，m为3,4或5。

66. 发明授权

US5179098A Fungicides 失效
标题翻译：杀真菌剂
公开(公告)号：US5179098A
公开(公告)日：1993-01-12
申请号：US616454
申请日：1990-11-20
申请人： John M. Clough , Christopher R. A. Godfrey , Ian T. Streeting , David P. Bacon
发明人： John M. Clough , Christopher R. A. Godfrey , Ian T. Streeting , David P. Bacon
IPC分类号： C07D239/47 , A01N43/54 , A01N43/647 , A01N43/653 , C07D239/36 , C07D239/54 , C07D401/04 , C07D403/04 , C07D413/04 , C07D521/00
CPC分类号： C07D239/36 , A01N43/54 , A01N43/647 , A01N43/653 , C07D231/12 , C07D233/56 , C07D249/08 , C07D401/04 , C07D403/04 , C07D413/04
摘要： Fungicidal compounds having the formula (I): ##STR1## in which any two of K, L and M are nitrogen and the other is CH; and X is an optionally substituted 3- to 6-membered heterocyclic ring containing at least one trivalent nitrogen atom by which it is attached to the central pyrimidine ring.

67. 发明授权

US5124353A Fungicidal alpha-substituted acrylates 失效
标题翻译：杀真菌α-取代丙烯酸酯
公开(公告)号：US5124353A
公开(公告)日：1992-06-23
申请号：US416609
申请日：1989-10-03
申请人： John M. Clough , Christopher R. A. Godfrey
发明人： John M. Clough , Christopher R. A. Godfrey
IPC分类号： C07C253/00 , A01N37/34 , A01N37/36 , A01N37/38 , A01N37/42 , A01N37/44 , A01N37/46 , A01N37/48 , A01N39/00 , A01N39/02 , A01N43/40 , C07C67/00 , C07C69/618 , C07C69/734 , C07C229/30 , C07C229/44 , C07C233/15 , C07C233/25 , C07C233/43 , C07C233/54 , C07C235/42 , C07C237/30 , C07C255/54 , C07C255/57 , C07C313/00 , C07C323/54 , C07C323/62 , C07C323/63 , C07C325/00 , C07D207/323 , C07D213/30 , C07D213/64 , C07D307/38 , C07D307/54 , C07D333/14 , C07D333/24 , C07D333/54
CPC分类号： C07C321/00 , A01N37/36 , A01N37/44 , A01N39/00 , A01N39/02 , A01N43/40 , C07C323/00
摘要： Compounds of formula (I): ##STR1## and stereoisomers thereof, wherein V is an oxygen or a sulphur atom; X and Y, which may be the same or different, are hydrogen or halogen atoms, or optionally substituted alkyl, optionally substituted alkenyl, optionally substituted aryl, optionally substituted heteroaryl, optionally substituted alkynyl, haloalkyl, alkoxy, haloalkoxy, optionally substituted aryloxy, optionally substituted arylalkoxy, optionally substituted acyloxy, optionally substituted amino, acylamino, nitro, nitrile, --CO.sub.2 R.sup.3, --CONR.sup.4 R.sup.5, or --COR.sup.6 groups; or the groups X and Y, when they are in adjacent positions on the phenyl ring, may join to form a fused ring, either aromatic or aliphatic, optionally containing one or more heteroatoms; and Z is optionally substituted methylene, optionally substituted amino, oxygen or sulphur and when Z is a substituted methylene group, the substituent may join the 2-position of the phenyl ring to form a non-aromatic fused ring; R.sup.1 and R.sup.2 are alkyl groups containing from one to four carbon atoms, optionally substituted with one or more halogen atoms; and R.sup.3, R.sup.4, R.sup.5, and R.sup.6, which may be the same or different, are hydrogen atoms or optionally substituted alkyl, cycloalkyl, alkenyl, alkynyl, optionally substituted aryl, optionally substituted aralkyl, or cycloalkylalkyl groups: and metal complexes thereof.
摘要翻译：式（I）化合物：其中V是氧或硫原子; X和Y可以相同或不同，是氢或卤素原子，或任选取代的烷基，任选取代的烯基，任选取代的芳基，任选取代的杂芳基，任选取代的炔基，卤代烷基，烷氧基，卤代烷氧基，任选取代的芳氧基，取代的芳基烷氧基，任选取代的酰氧基，任选取代的氨基，酰氨基，硝基，腈，-CO 2 R 3，-CONR 4 R 5或-COR 6基团; 或基团X和Y当它们在苯环上的相邻位置时，可以连接形成任选含有一个或多个杂原子的芳族或脂族稠合的稠环; Z是任选取代的亚甲基，任选取代的氨基，氧或硫，当Z是取代的亚甲基时，取代基可以连接苯环的2-位，形成非芳香稠环; R1和R2是含有1-4个碳原子的烷基，任选地被一个或多个卤素原子取代; 和可以相同或不同的R 3，R 4，R 5和R 6是氢原子或任选取代的烷基，环烷基，烯基，炔基，任选取代的芳基，任选取代的芳烷基或环烷基烷基：及其金属络合物。

68. 发明授权

US5008276A Methyl .alpha.-(2-substituted)pyrid-3-yl-.beta.-methoxyacrylates, compositions containing them and their use as fungicides 失效
标题翻译：甲基α-（2-取代）吡啶-3-基-β-甲氧基丙烯酸酯，含有它们的组合物及其作为杀真菌剂的用途
公开(公告)号：US5008276A
公开(公告)日：1991-04-16
申请号：US258742
申请日：1988-10-17
申请人： John M. Clough , Christopher R. A. Godfrey , Stephen P. Heaney , Kenneth Anderton
发明人： John M. Clough , Christopher R. A. Godfrey , Stephen P. Heaney , Kenneth Anderton
IPC分类号： A01N43/40 , A01N43/42 , A01N43/52 , A01N43/54 , A01N43/58 , A01N43/60 , A01N43/64 , A01N43/647 , A01N43/653 , A01N43/66 , A01N43/76 , A01N43/78 , A01N43/824 , A01N43/836 , A01N43/90 , A01N47/20 , A01N47/22 , A01N47/30 , A01P3/00 , C07D213/64 , C07D213/643 , C07D213/65 , C07D213/68 , C07D213/70 , C07D213/71 , C07D213/74 , C07D213/79 , C07D213/80 , C07D213/81 , C07D213/84 , C07D213/85 , C07D213/89 , C07D401/12 , C07D405/12 , C07D409/12 , C07D413/12 , C07D417/12 , C07D473/30 , C07D473/34 , C07D473/38
CPC分类号： C07D213/643 , A01N43/40 , A01N43/54 , A01N43/78 , C07D213/65 , C07D213/68 , C07D213/70 , C07D213/71 , C07D213/74 , C07D213/79 , C07D213/80 , C07D213/81 , C07D213/84 , C07D213/85 , C07D213/89 , C07D401/12 , C07D405/12 , C07D409/12 , C07D413/12 , C07D417/12 , C07D473/30 , C07D473/34 , C07D473/38
摘要： Fungicidal compounds of the formula (I): ##STR1## and stereoisomers thereof, wherein K is oxygen or sulphur; Z is optionally substituted aryl or optionally substituted heteroaryl; X is O, S(O).sub.n, NR.sup.4, CR.sup.1 R.sup.2, CHR.sup.5, CO, CR.sup.1 (OR.sup.2), C.dbd.CR.sup.1 R.sup.2, CHR.sup.1 CHR.sup.2, CR.sup.1 .dbd.CR.sup.2, CHR.sup.1 CR.sup.2 .dbd.CH, C.dbd.C, OCHR.sup.1, CHR.sup.1 O, OCHR.sup.1 O, S(O).sub.n CHR.sup.1, S(O).sub.n CHR.sup.1 O, CHR.sup.1 S(O).sub.n, CHR.sup.1 OSO.sub.2, NR.sup.4 CHR.sup.1, CHR.sup.1 NR.sup.4, CO.sub.2, O.sub.2 C, SO.sub.2 O, OSO.sub.2, CO.CO, COCHR.sup.1, COCHR.sup.1 O, CHR.sup.1 CO, CHOH.CHR.sup.1, CHR.sup.1.CHOH, ##STR2## CONR.sup.4, OCONR.sup.4, NR.sup.4 CO, CSNR.sup.4, OCS.NR.sup.4, SCO.NR.sup.4, NR.sup.4 CO.sub.2, NR.sup.4 CS, NR.sup.4 CSO, NR.sup.4 COS, NR.sup.4 CONR.sup.4, S(O).sub.n NR.sup.4, NR.sup.4 S(O).sub.n, CS.sub.2, S.sub.2 C, CO.S, SCO, N.dbd.N, N.dbd.CR.sup.1, CR.sup.1 .dbd.N, CHR.sup.1 CHR.sup.2 CH(OH), CHR.sup.1 OCO, CHR.sup.1 SCO, CHR.sup.1 NR.sup.4 CO, CHR.sup.1 NR.sup.4 COR.sup.4, CHR.sup.1 CHR.sup.2 CO, O.N.dbd.CR.sup.1, CHR.sup.1 O.N.dbd.CR.sup.2, CO.OCR.sup.1 R.sup.2, CHR.sup.1 CHR.sup.2 CHR.sup.3, OCHR.sup.1 CHR.sup.2, (CH.sub.2).sub.m O, CHR.sup.1 OCHR.sup.2, CHR.sup.1 CHR.sup.2 O, OCHR.sup.1 CHR.sup.2 O, S(O).sub.n CHR.sup.1 CHR.sup.2, CHR.sup.1 S(O).sub.n CHR.sup.2, CHR.sup.1 CHR.sup.2 S(O).sub.n, CR.sup.1 .dbd.NNR.sup.4, NR.sup.4 N.dbd.CR.sup.1, CHR.sup.1 CONR.sup.2, CHR.sup.1 OCO.NR.sup.2, CH.dbd.CHCH.sub.2 O, COCHR.sup.1 CHR.sup.2 O or (R.sup.5).sub.2 P.sup. + CHR.sup.2 Q.sup.- ; A, B and E, which may be the same or different, are H, hydroxy, halo, C.sub.1-4 alkyl, C.sub.1-4 alkoxy, C.sub.1-4 haloalkyl, C.sub.1-4 haloalkoxy, C.sub.1-4 alkylcarbonyl, C.sub.1-4 alkoxycarbonyl, phenoxy, nitro or cyano; R.sup.1, R.sup.2 and R.sup.3, which may be the same or different, are H, C.sub.1-4 alkyl or phenyl; R.sup.4 is H, C.sub.1-4 alkyl or COR.sup.1 ; R.sup.5 is optionally substituted phenyl; Q.sup.- is a halide anion; n is 0, 1 or 2 and m is a 3, 4 or 5.

69. 发明授权

US4913721A Fungicides 失效
公开(公告)号：US4913721A
公开(公告)日：1990-04-03
申请号：US264874
申请日：1988-10-31
申请人： John M. Clough , Christopher R. A. Godfrey
发明人： John M. Clough , Christopher R. A. Godfrey
IPC分类号： C07C253/00 , A01N37/34 , A01N37/36 , A01N37/38 , A01N37/42 , A01N37/44 , A01N37/46 , A01N37/48 , A01N39/00 , A01N39/02 , A01N43/40 , C07C67/00 , C07C69/618 , C07C69/734 , C07C229/30 , C07C229/44 , C07C233/15 , C07C233/25 , C07C233/43 , C07C233/54 , C07C235/42 , C07C237/30 , C07C255/54 , C07C255/57 , C07C313/00 , C07C323/54 , C07C323/62 , C07C323/63 , C07C325/00 , C07D207/323 , C07D213/30 , C07D213/64 , C07D307/38 , C07D307/54 , C07D333/14 , C07D333/24 , C07D333/54
CPC分类号： C07C321/00 , A01N37/36 , A01N37/44 , A01N39/00 , A01N39/02 , A01N43/40 , C07C323/00
摘要： Compounds of formula (I): ##STR1## and stereoisomers thereof, wherein V is an oxygen or a sulphur atom; X and Y, which may be the same or different, are hydrogen or halogen atoms, or optionally substituted alkyl, optionally substituted alkenyl, optionally substituted aryl, optionally substituted heteroaryl, optionally substituted alkynyl, haloalkyl, alkoxy, haloalkoxy, optionally substituted aryloxy, optionally substituted arylalkoxy, optionally substituted acyloxy, optionally substituted amino, acylamino, nitro, nitrile, --CO.sub.2 R.sup.3, --CONR.sup.4 R.sup.5, or --COR.sup.6 groups; or the groups X and Y, when they are in adjacent positions on the phenyl ring, may join to form a fused ring, either aromatic or aliphatic, optionally containing one or more heteroatoms; and Z is optionally substituted methylene, optionally substituted amino, oxygen or sulphur and when Z is a substituted methylene group, the substituent may join the 2-position of the phenyl ring to form a non-aromatic fused ring; R.sup.1 and R.sup.2 are alkyl groups containing from one to four carbon atoms, optionally substituted with one or more halogen atoms; and R.sup.3, R.sup.4, R.sup.5 and R.sup.6, which may be the same or different, are hydrogen atoms or optionally substituted alkyl, cycloalkyl, alkenyl, alkynyl, optionally substituted aryl, optionally substituted aralkyl, or cycloalkylalkyl groups; and metal complexes thereof.

70. 发明授权

US4870075A Fungicides 失效
标题翻译：杀菌剂
公开(公告)号：US4870075A
公开(公告)日：1989-09-26
申请号：US85412
申请日：1987-08-14
申请人： John M. Clough , Christopher R. A. Godfrey
发明人： John M. Clough , Christopher R. A. Godfrey
IPC分类号： A01N43/58 , A01N43/60 , A01N43/66 , A01N43/707 , A01N43/713 , C07D237/14 , C07D237/18 , C07D237/28 , C07D241/18 , C07D241/44 , C07D251/20 , C07D251/22 , C07D251/26 , C07D251/30 , C07D251/38 , C07D253/02 , C07D253/04 , C07D253/06 , C07D253/07 , C07D253/08 , C07D253/10 , C07D257/08
CPC分类号： C07D257/08 , A01N43/58 , A01N43/60 , A01N43/66 , A01N43/707 , A01N43/713 , C07D237/14 , C07D237/18 , C07D237/28 , C07D241/18 , C07D241/44 , C07D251/20 , C07D251/22 , C07D251/26 , C07D253/02 , C07D253/07 , C07D253/10
摘要： This invention relates to derivatives of acrylic acid of the formula: ##STR1## useful as fungicides, to processes for preparing them, to fungicidal compositions containing them, and to methods of using them to combat fungi, especially fungal infections in plants. The values of the variables are provided herein.
摘要翻译：本发明涉及下式的丙烯酸衍生物：可用作杀真菌剂的“IMAGE”，其制备方法，含有它们的杀真菌组合物，以及使用它们来对抗真菌，特别是植物真菌感染的方法。变量的值在这里提供。

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