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21. 发明申请

US20100247462A1 SYNTHESIS OF RESVERATROL-BASED NATURAL PRODUCTS 有权
标题翻译：基于RESPARATROL的天然产物的合成
公开(公告)号：US20100247462A1
公开(公告)日：2010-09-30
申请号：US12733750
申请日：2008-09-17
申请人： Scott Alan Snyder , Steven P. Breazzano , Audrey G. Ross , Yunqing Lin , Alexandros L. Zografos
发明人： Scott Alan Snyder , Steven P. Breazzano , Audrey G. Ross , Yunqing Lin , Alexandros L. Zografos
IPC分类号： A61K8/34 , C07C43/20 , A61K31/075 , A01N31/14 , C07F9/02 , A61K31/66 , A01N57/10 , C07C69/63 , A61K31/215 , A01N37/02 , C07C49/297 , A61K31/12 , A01N35/00 , C07C323/00 , A61K31/095 , A01N31/00 , C07C39/12 , A61K31/05 , A01N31/08 , A61K8/35 , A61K8/37 , A01P3/00 , A61P35/00 , A61Q17/04
CPC分类号： A01N31/16 , C07C37/00 , C07C37/055 , C07C41/18 , C07C41/22 , C07C41/24 , C07C41/26 , C07C41/30 , C07C49/755 , C07C67/04 , C07C67/11 , C07C319/14 , C07C2602/08 , C07C2603/32 , C07C2603/40 , C07C2603/86 , C07C2603/90 , C07C39/23 , C07C39/17 , C07C43/23 , C07C43/21 , C07C43/215 , C07C43/225 , C07C69/63 , C07C69/013 , C07C323/17 , C07C69/157
摘要： Processes for synthesizing resveratrol-based oligomers are provided. In addition, resveratrol-based oligomer compounds free of plant extract are provided.
摘要翻译：提供了合成基于白藜芦醇的低聚物的方法。此外，提供了不含植物提取物的白藜芦醇低聚物化合物。

22. 发明授权

US07728177B2 Optically active 3-methylcyclopentadecanone and method for producing intermediate thereof 有权
标题翻译：光学活性3-甲基环十五烷酮及其中间体的制备方法
公开(公告)号：US07728177B2
公开(公告)日：2010-06-01
申请号：US11920600
申请日：2006-05-17
申请人： Shigeru Tanaka , Kenya Ishida , Hiroyuki Matsuda
发明人： Shigeru Tanaka , Kenya Ishida , Hiroyuki Matsuda
IPC分类号： C07C45/00
CPC分类号： C07B53/00 , C07B2200/07 , C07C45/513 , C07C45/54 , C07C67/00 , C07C2601/18 , C07F9/657154 , C07C49/385 , C07C69/013 , C07C69/24
摘要： Disclosed is a method for producing an optically active 3-methylcyclopentadecan-1-one which is characterized in that 2-cyclopentadecen-1-one is subjected to a 1,4-conjugate addition reaction of a methyl group by using a methylated organic metal in the presence of a copper catalyst, an enol anion scavenger and a specific optically active phosphoramidite for obtaining an optically active 3-methyl-1-cyclopentadecene derivative, and then the thus-obtained 3-methyl-1-cyclopentadecene derivative is subjected to a solvolysis.
摘要翻译：公开了一种光学活性3-甲基环戊烷-1-酮的制备方法，其特征在于2-环戊烯-1-酮通过使用甲基化有机金属在甲基化有机金属中进行1,4-偶合物加成反应存在铜催化剂，烯醇阴离子清除剂和用于获得光学活性的3-甲基-1-环戊烯衍生物的特定光学活性亚磷酰胺，然后由此得到的3-甲基-1-环戊烯衍生物进行溶剂分解。

23. 发明授权

US07723255B2 Recyclable metathesis catalysts 有权
标题翻译：可回收复分解催化剂
公开(公告)号：US07723255B2
公开(公告)日：2010-05-25
申请号：US11178884
申请日：2005-07-11
申请人： Amir H. Hoveyda , Jason Kingsbury , Steven Garber , Brian Lawrence Gray , John T. Fourkas
发明人： Amir H. Hoveyda , Jason Kingsbury , Steven Garber , Brian Lawrence Gray , John T. Fourkas
IPC分类号： B01J31/18
CPC分类号： C07F15/0046 , B01J23/462 , B01J31/1625 , B01J31/1641 , B01J31/1666 , B01J31/1683 , B01J31/1805 , B01J31/2208 , B01J31/2273 , B01J31/2404 , B01J31/28 , B01J31/4038 , B01J2231/482 , B01J2231/543 , B01J2531/821 , C07B2200/11 , C07C6/02 , C07C29/00 , C07C67/293 , C07C2531/22 , C07C2601/08 , C07C2601/16 , C07D233/56 , C08F290/00 , C08G83/003 , C08L51/04 , C08L51/08 , Y02P20/584 , Y02P20/588 , C07C35/18 , C07C35/06 , C07C35/21 , C07C69/013 , C07C69/145
摘要： Highly active, recoverable and recyclable transition metal-based metathesis catalysts and their organometallic complexes including dendrimeric complexes are disclosed, including a Ru complex bearing a 1,3-dimesityl-4,5-dihydroimidazol-2-ylidene and styrenyl ether ligand. The heterocyclic ligand significantly enhances the catalytic activity, and the styrenyl ether allows for the easy recovery of the Ru complex. Derivatized catalysts capable of being immobilized on substrate surfaces are also disclosed. The present catalysts can be used to catalyze ring-closing metathesis (RCM), ring-opening (ROM) and cross metatheses (CM) reactions, and promote the efficient formation of various trisubstituted olefins at ambient temperature in high yield.
摘要翻译：公开了高活性，可回收和可回收的基于过渡金属的复分解催化剂及其有机金属配合物，包括树枝状复合物，包括带有1,3-二甲基-4,5-二氢咪唑-2-亚基和苯乙烯基醚配体的Ru络合物。杂环配体显着增强了催化活性，苯乙烯醚容易回收Ru络合物。还公开了能够固定在基材表面上的衍生化催化剂。本催化剂可用于催化闭环复分解（RCM），开环（ROM）和交叉元（CM）反应，促进各种三取代烯烃在环境温度下的高效率形成。

24. 发明申请

US20100041918A1 CYCLOPENTENE DIOL MONOACETATE DERIVATIVES 审中-公开
标题翻译：环戊二醇单酸酯衍生物
公开(公告)号：US20100041918A1
公开(公告)日：2010-02-18
申请号：US12312311
申请日：2007-11-05
申请人： Kurt Laumen
发明人： Kurt Laumen
IPC分类号： C07C61/06
CPC分类号： C07C45/59 , C07B2200/07 , C07C67/08 , C12P7/62 , C12P41/004 , C12Y301/01003 , C07C49/707 , C07C69/013 , C07C69/16
摘要： A process for the preparation of organic compounds of formula (I), wherein R1 is as described herein.
摘要翻译：制备式（I）的有机化合物的方法，其中R 1如本文所述。

25. 发明申请

US20100036153A1 Method for Producing Substituted Diamantanes 失效
标题翻译：生成取代的金刚烷的方法
公开(公告)号：US20100036153A1
公开(公告)日：2010-02-11
申请号：US12086058
申请日：2006-12-04
申请人： Peter R. Schreiner , Andrey A. Fokin
发明人： Peter R. Schreiner , Andrey A. Fokin
IPC分类号： C07C35/44 , C07C239/08 , C07C233/08 , C07C61/125 , C07C69/753
CPC分类号： C07C203/08 , C07C29/12 , C07C51/353 , C07C67/11 , C07C2603/90 , C07C35/44 , C07C61/135 , C07C69/013 , C07C69/14
摘要： The invention at hand provides at least dinitroxylated diamantanes. In addition, it provides methods for producing substituted diamantanes with high yields and selectivity.According to the invention, dinitroxylated diamantanes are suitable for being reacted with nucleophiles to form the corresponding disubstituted diamantanes. Surprisingly, it was discovered that at least dinitroxylated or hydroxylated diamantanes are rearranged in the presence of a strong acid, creating at least 4,9-nitroxylated or hydroxylated diamantanes. On the basis of this, 4,9-substituted diamantanes are able to be produced in a targeted manner by reaction with further nucleophiles.Thus, the invention at hand provides the following methods according to the present invention for producing at least disubstituted diamantanes: a) at least dinitroxylation, followed by the substitution of all nitroxy groups by a nucleophile or b) at least dinitroxylation, subsequent rearrangement in the presence of a strong acid, after realised rearrangement all nitroxy groups are replaced by a nucleophile or c) at least dinitroxylation, subsequent reaction with water (as nucleophile), rearrangement of the at least dihydroxylated compound in the presence of a strong acid, after realised rearrangement all hydroxy groups are replaced by another nucleophile.
摘要翻译：本发明至少提供二硝基甲酰化的二金刚烷。此外，它提供了以高产率和选择性生产取代的二金刚烷的方法。根据本发明，二硝基氧化的二金刚烷适于与亲核试剂反应以形成相应的二取代的二金刚烷。令人惊奇的是，发现在强酸存在下重新排列了二硝基氧化或羟基化的二金刚烷，产生了至少4,9-氨基氧化或羟基化的金刚烷。基于此，4,9-取代的二金刚烷可以通过与另外的亲核试剂反应而以目标方式制备。因此，本发明提供了根据本发明的用于生产至少二取代的二金刚烷的以下方法：a）至少二硝基甲酰化，然后用亲核试剂取代所有硝基，或b）至少二硝基甲酰化，随后在强酸的存在，在实现重排之后，所有的硝基都被亲核试剂取代，或c）至少二硝基甲酰化，随后与水（作为亲核试剂）反应，在强酸存在下重排至少二羟基化的化合物，重排所有羟基被另一个亲核试剂取代。

26. 发明申请

US20090275752A1 Novel Process for Statins and its Pharmaceutically Acceptable Salts Thereof 失效
标题翻译：他汀类药物及其药学上可接受的盐的新方法
公开(公告)号：US20090275752A1
公开(公告)日：2009-11-05
申请号：US12226932
申请日：2007-04-30
申请人： Manne Satyanarayana Reddy , Srinivasan Thirumalai Rajan , Maramreddy Sahadeva Reddy
发明人： Manne Satyanarayana Reddy , Srinivasan Thirumalai Rajan , Maramreddy Sahadeva Reddy
IPC分类号： C07D239/42 , C07D215/06 , C07D209/08 , C07D213/30 , C07D207/333 , C07C69/76
CPC分类号： C07D239/42 , C07C67/28 , C07C67/283 , C07C67/29 , C07C67/31 , C07C317/44 , C07C323/52 , C07C2602/10 , C07D207/34 , C07D209/24 , C07D213/55 , C07D215/14 , C07D319/06 , C07D403/12 , C07D405/06 , C07C69/013 , C07C69/734
摘要： Novel process for statins and its pharmaceutically acceptable salts thereof represented by general formula (I).
摘要翻译：由通式（I）表示的他汀类药物及其药学上可接受的盐的新方法。

27. 发明授权

US07459414B2 Herbicides 有权
标题翻译：除草剂
公开(公告)号：US07459414B2
公开(公告)日：2008-12-02
申请号：US11083465
申请日：2005-03-18
申请人： Thomas Maetzke , André Stoller , Sebastian Wendeborn , Henry Szczepanski
发明人： Thomas Maetzke , André Stoller , Sebastian Wendeborn , Henry Szczepanski
IPC分类号： A01N31/06 , C07C49/537
CPC分类号： C07D221/20 , A01N35/06 , A01N43/08 , A01N43/10 , A01N43/16 , A01N43/18 , A01N43/36 , A01N43/38 , A01N43/40 , A01N43/42 , A01N43/56 , A01N43/72 , A01N43/80 , A01N43/82 , A01N43/86 , A01N43/90 , A01N47/06 , A01N47/18 , C07C25/02 , C07C49/747 , C07C49/753 , C07C69/013 , C07C69/708 , C07C323/22 , C07D207/38 , C07D209/54 , C07D209/96 , C07D211/86 , C07D231/32 , C07D231/34 , C07D231/36 , C07D237/04 , C07D265/02 , C07D279/06 , C07D303/32 , C07D307/60 , C07D307/94 , C07D309/32 , C07D309/38 , C07D311/74 , C07D311/94 , C07D311/96 , C07D333/32 , C07D333/50 , C07D335/02 , C07D403/12 , C07D409/12 , C07D413/12 , C07D417/12 , C07D471/04 , C07D487/04 , C07D487/08 , C07D487/10 , C07D491/10 , C07D491/14 , C07D493/10 , A01N25/32 , A01N2300/00
摘要： Compounds of formula wherein the substituents have the meanings given in claim 1, and agronomically tolerable salts, isomers and enantiomers of those compounds, are suitable for use as herbicides.
摘要翻译：下式的化合物，其中取代基具有权利要求1中给出的含义，并且这些化合物的农学上可耐受的盐，异构体和对映异构体适合用作除草剂。

28. 发明授权

US07393985B2 Supported ruthenium nanoparticle catalyst for cis -dihydroxylation and oxidative cleavage of alkenes 有权
标题翻译：负载钌纳米颗粒催化剂用于顺式二羟基化和烯烃的氧化裂解
公开(公告)号：US07393985B2
公开(公告)日：2008-07-01
申请号：US11110317
申请日：2005-04-19
申请人： Chi-Ming Che , Wing-Yiu Yu , Chi-Ming Ho
发明人： Chi-Ming Che , Wing-Yiu Yu , Chi-Ming Ho
IPC分类号： C07C29/04 , C07C29/03
CPC分类号： C07C41/26 , C07B2200/07 , C07B2200/09 , C07C29/48 , C07C41/16 , C07C43/13 , C07C45/28 , C07C45/30 , C07C45/40 , C07C45/64 , C07C51/29 , C07C51/31 , C07C67/29 , C07C67/31 , C07C2601/06 , C07C2601/14 , C07C2603/26 , C07C33/26 , C07C31/202 , C07C35/42 , C07C47/54 , C07C47/544 , C07C47/30 , C07C49/78 , C07C47/12 , C07C49/497 , C07C63/06 , C07C55/02 , C07C59/185 , C07C69/003 , C07C69/013 , C07C69/675 , C07C69/732 , C07C69/70 , C07C69/14 , C07C43/1782
摘要： The present invention relates to the use of nanosized metal particles (e.g., ruthenium) grafted on inert solid support for oxidation of alkenes. The supported metal catalyst can effect cis-dihydroxylation and oxidative cleavage of alkenes to give the respective cis-diols and carbonyl products.
摘要翻译：本发明涉及接枝在惰性固体载体上用于氧化烯烃的纳米金属颗粒（例如钌）的用途。负载的金属催化剂可以进行顺式二羟基化和烯烃的氧化裂解，得到各自的顺式二醇和羰基产物。

29. 发明申请

US20080081807A1 Arylphenyl-substituted cyclic keto-enols 有权
标题翻译：芳基苯基取代的环状酮 - 烯醇
公开(公告)号：US20080081807A1
公开(公告)日：2008-04-03
申请号：US11901471
申请日：2007-09-17
申请人： Folker Lieb , Reiner Fischer , Alan Graff , Udo Schneider , Thomas Bretschneider , Christoph Erdelen , Wolfram Andersch , Mark-Wilhelm Drewes , Markus Dollinger , Ingo Wetcholowsky , Randy Myers
发明人： Folker Lieb , Reiner Fischer , Alan Graff , Udo Schneider , Thomas Bretschneider , Christoph Erdelen , Wolfram Andersch , Mark-Wilhelm Drewes , Markus Dollinger , Ingo Wetcholowsky , Randy Myers
IPC分类号： A01N43/38 , A01N31/06 , A01N43/08 , A01N43/10 , A01N43/56 , A01N43/86 , A01P7/02 , A61K31/365 , A61K31/381 , C07D209/54 , C07D207/24 , C07C49/573 , A61K31/54 , A61K31/50 , A61K31/4433 , A61K31/415 , A61K31/403 , A61K31/4015 , C07D487/04 , C07D405/04 , C07D333/32 , C07D309/38 , C07D307/94 , C07D307/60 , C07D279/06 , A61K31/366 , A61K31/122 , A01P13/00 , A01N43/58 , A01N43/40 , A01N43/16 , A01N43/36
CPC分类号： A01N43/36 , C07C45/673 , C07C45/68 , C07C49/747 , C07C57/58 , C07C57/72 , C07C57/76 , C07C59/88 , C07C62/38 , C07C69/013 , C07C69/24 , C07C69/65 , C07C69/67 , C07C69/738 , C07C69/757 , C07C69/96 , C07C211/47 , C07C233/51 , C07C233/52 , C07C255/29 , C07C323/61 , C07C2601/14 , C07C2601/16 , C07C2602/08 , C07C2602/50 , C07D207/38 , C07D209/96 , C07D307/60 , C07D307/94 , C07D311/74 , C07D333/50 , C07D401/12 , C07D405/04 , C07D491/10 , C07D493/10
摘要： The present invention relates to novel arylphenyl-substituted cyclic ketoenols of the formula (I) in which X represents halogen, alkyl, alkoxy, alkenyloxy, alkylthio, alkylsulphinyl, alkylsulphonyl, halogenoalkyl, halogenoalkoxy, halogenoalkenyloxy, nitro, cyano or in each case optionally substituted phenyl, phenoxy, phenylthio, phenylalkoxy or phenylalkylthio, Y represents in each case optionally substituted cycloalkyl, aryl or hetaryl, Z represents hydrogen, halogen, alkyl, alkoxy, alkenyloxy, halogenoalkyl, halogenoalkoxy, halogenoalkenyloxy, nitro or cyano, CKE represents one of the groups in which A, B, D, G and Q1 to Q6 are each as defined in the description, to a plurality of processes for their preparation and to their use as pesticides and herbicides.
摘要翻译：本发明涉及式（I）的新型芳基苯基取代的环酮酮，其中X表示卤素，烷基，烷氧基，烯氧基，烷硫基，烷基亚磺酰基，烷基磺酰基，卤代烷基，卤代烷氧基，卤代烯基氧基，硝基，氰基或在各种情况下任选取代苯基，苯氧基，苯硫基，苯基烷氧基或苯基烷硫基，Y代表各自为任选取代的环烷基，芳基或杂芳基，Z表示氢，卤素，烷基，烷氧基，烯氧基，卤代烷基，卤代烷氧基，卤代烯氧基，硝基或氰基，CKE代表其中A，B，D，G和Q 1至Q 6的基团各自如说明书中所定义，涉及多种制备方法及其用途作为农药和除草剂。

30. 发明授权

US07301045B2 Method for preparing ester condensate 失效
标题翻译：制备酯缩合物的方法
公开(公告)号：US07301045B2
公开(公告)日：2007-11-27
申请号：US10399233
申请日：2001-08-23
申请人： Kazuaki Ishihara , Hisashi Yamamoto
发明人： Kazuaki Ishihara , Hisashi Yamamoto
IPC分类号： C07C69/74 , C07C69/76 , C07C321/00
CPC分类号： B01J31/0212 , B01J27/135 , B01J31/2208 , B01J2231/40 , B01J2531/40 , C07C67/08 , C07C327/22 , C07D309/30 , C08G63/81 , C08G63/85 , C07C69/007 , C07C69/013 , C07C69/017 , C07C69/003 , C07C69/612 , C07C69/618 , C07C69/75 , C07C69/24 , C07C69/734 , C07C69/78
摘要： The present invention provides a method for preparing ester or thioester that can conduct catalytic esterification reaction with an equimolar amount of carboxylic acid and alcohol, or catalytic thioesterification reaction with carboxylic acid and an equimolar amount or small amount of thiol, and can be expected as an industrial method that needs an enormous amount of synthesis in the light of green chemistry. By using hafnium chloride (IV), especially tetravalent hafnium compounds represented by hafnium chloride (IV)·(THF)2 or hafnium (IV)t-butoxide as a (poly) condensation catalyst, direct condensation reaction is conducted from carboxylic acid and an equimolar amount of alcohol or a little smaller amount of thiol, in the nonpolar solvent such as toluene and the like, in a deoxidization atmosphere and under heating reflux, and the reaction synthesizes ester monomer or thioester monomer, polyester or polythioester. When heating reflux is conducted by using a nonpolar solvent, it is preferable to remove azeotropic water from the reaction system.
摘要翻译：本发明提供了一种制备可与等摩尔量的羧酸和醇进行催化酯化反应或与羧酸和等摩尔量或少量硫醇进行催化酯基酯化反应的酯或硫酯的方法，并且可以作为在绿色化学方面需要大量合成的工业方法。通过使用氯化铪（IV），特别是作为（多）缩合催化剂的氯化铪（IV）（THF）2 H 2或叔（叔丁醇）铪代表的四价铪化合物，直接缩合反应在脱氧气氛和加热回流下，在非极性溶剂如甲苯等中，从羧酸和等摩尔量的醇或少量的硫醇进行反应，合成酯单体或硫酯单体，聚酯或聚硫酯。当使用非极性溶剂进行加热回流时，优选从反应体系中除去共沸水。

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