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91. 发明授权

US4925832A Silver halide photographic light-sensitive systems 失效
标题翻译：卤化银照相感光系统
公开(公告)号：US4925832A
公开(公告)日：1990-05-15
申请号：US264988
申请日：1988-10-31
申请人： Kevin P. Hall , Andrew W. Mott
发明人： Kevin P. Hall , Andrew W. Mott
IPC分类号： G03C1/485 , C07C243/32 , C07C243/34 , C07C243/38 , G03C1/06
CPC分类号： G03C1/061 , C07C243/32 , C07C243/34 , C07C243/38 , Y10S430/15
摘要： A silver halide photographic light sensitive emulsion containing a hydrazine of the general formulaR.sup.3 -NR.sup.4 -NR.sup.5 -G-X (I)in whichR.sup.3 represents an aryl group,one of R.sup.4 and R.sup.5 is a hydrogen and the other is selected from hydrogen, aryl sulphonyl and trifluoroacetyl,G represents carbonyl, sulphonyl, sulphoxy, phosphoryl or an N-substituted or unsubstituted imino group and X is a moiety such that at a pH in the range of 9.5 to 12.5 in the presence of an oxidized hydroquinone a cyclization reaction takes place cleaving the moiety -G-X from the remainder of the molecule and forming a cyclic structure comprising atoms of the moiety -G-X.

92. 发明授权

US4859233A 2,3,6-trichlorobenzohydroxamic acid derivatives 失效
标题翻译： 2,3,6-三氯苯肟酸衍生物
公开(公告)号：US4859233A
公开(公告)日：1989-08-22
申请号：US147409
申请日：1988-01-25
申请人： John W. Williams
发明人： John W. Williams
IPC分类号： C07C259/10 , A01N37/36 , A01N37/40 , A01N37/44 , C07C243/38
CPC分类号： A01N37/36 , A01N37/40 , A01N37/44
摘要： Disclosed are herbicidal compounds of the general formula I; ##STR1## wherein A is O-alkylene of 1 to 5 carbon atoms, O-alkenylene of 3 to 6 carbon atoms in which the unsaturation is non-adjacent the oxygen atom thereof or NH-alkylene in which the alkylene is of 1 to 5 carbon atoms, and --COZR is an acid function or forms certain ester or thioester functions, and the mono- and di-salt forms thereof.
摘要翻译：公开了通式I的除草化合物; 其中A是1至5个碳原子的O-亚烷基，3至6个碳原子的O-亚烯基，其中不饱和度不与其氧原子相邻或其中亚烷基的亚烷基为1〜 5个碳原子，-COZR是酸官能团或形成某些酯或硫酯官能团，以及它们的单盐和二盐形式。

93. 发明授权

US4814349A Insecticidal substituted and unsubstituted benzoic acid 1-alkyl, 2 alkyl and 2-cycloalkylhydrazides 失效
标题翻译：杀虫取代和未取代的苯甲酸1-烷基，2-烷基和2-环烷基酰肼
公开(公告)号：US4814349A
公开(公告)日：1989-03-21
申请号：US926780
申请日：1986-11-12
申请人： Roger W. Addor , David G. Kuhn , Donald P. Wright, Jr.
发明人： Roger W. Addor , David G. Kuhn , Donald P. Wright, Jr.
IPC分类号： A01N37/28 , A01N37/34 , A01N37/40 , A01N37/48 , A01N41/10 , A01N43/30 , C07C243/38 , C07D317/68 , A01N33/26
CPC分类号： A01N37/48 , A01N37/28 , A01N37/34 , A01N37/40 , A01N41/10 , A01N43/30 , C07C243/38 , C07D317/68 , C07C2101/08 , C07C2101/14
摘要： The present invention relates to methods for controlling insect populations and for protecting living plants from insect attack by applying to said plants or to the soil in which they are growin an insecticidally-effective amount of a substituted benzoic acid 1 or 2-alkyl or 2-cycloalkylhydrazide.Novel substituted benzoic acid 1 and 2-alkyl and 2-cycloalkylhydrazides effective as insecticides or intermediates for the preparation of insecticidal diacylhydrazides also are presented.
摘要翻译：本发明涉及通过向所述植物或其生长的土壤中施用杀虫有效量的取代的苯甲酸1或2-烷基或2-烷基或2-烷基的方法来控制昆虫种群和保护活植物免受昆虫侵袭的方法，环烷基酰肼。还提供了有效用作杀虫剂二酰肼的杀虫剂或中间体的新型取代的苯甲酸1和2-烷基和2-环烷基酰肼。

94. 发明授权

US4727084A Novel 4H-1,2,4-triazole derivatives 失效
标题翻译：新型4H-1,2,4-三唑衍生物
公开(公告)号：US4727084A
公开(公告)日：1988-02-23
申请号：US896858
申请日：1986-08-14
申请人： Jean Meier , Francois Clemence
发明人： Jean Meier , Francois Clemence
IPC分类号： A61K31/41 , A61P25/04 , C07C243/38 , C07D249/08 , C07D317/46 , C07D405/04
CPC分类号： C07D249/08 , C07C243/38 , C07D317/46 , Y10S514/886
摘要： Compounds selected from the group consisting of 4H-1,2,4-triazoles of the formula ##STR1## wherein R.sub.1, R.sub.2, R.sub.3 and R.sub.4 may be in different positions of the benzene ring, R.sub.1, R.sub.3 and R.sub.4 are individually selected from the group consisting of hydrogen, --OH, alkyl of 1 to 4 carbon atoms, alkoxy of 1 to 4 carbon atoms, halogen, --CH.sub.3, --NO.sub.2, --NH.sub.2 and NH--AlK and ##STR2## R.sub.2 is selected from the group consisting of hydrogen, --OH, alkyl of 1 to 4 carbon atoms, halogen, --CF.sub.3, --NO.sub.2, --NH.sub.2, --NH--AlK and ##STR3## and AlK, AlK.sub.1 and AlK.sub.2 are alkyl of 1 to 4 carbon atoms or R.sub.1 and R.sub.2 together and/or R.sub.3 and R.sub.4 together are methylenedioxy, R is selected from the group consisting of ethyl, --CH.sub.2 --COOH and CH.sub.2 --COOAlK.sub.3 and AlK.sub.3 is alkyl of 1 to 4 carbon atoms and their non-toxic, pharmaceutically acceptable acid addition salts, with the proviso that R.sub.1, R.sub.2, R.sub.3 and R.sub.4 are not all hydrogen having a remarkable analgesic activity and a novel method for their preparation.
摘要翻译：选自下列化合物的化合物的化合物其中R 1，R 2，R 3和R 4可以位于苯环，R 1，R 3和R 4的不同位置的式Ia，由氢，-OH，1至4个碳原子的烷基，1至4个碳原子的烷氧基，卤素，-CH 3，-NO 2，-NH 2和NH-AlK和R 2选自下组：的氢，-OH，1至4个碳原子的烷基，卤素，-CF 3，-NO 2，-NH 2，-NH-AlK和AlGaN，AlK，AlK1和AlK2是1至4个碳原子的烷基或R1和 R 2一起和/或R 3和R 4一起是亚甲二氧基，R选自乙基，-CH 2 -COOH和CH 2 -COOAlK 3，AlK 3是1至4个碳原子的烷基及其无毒的药学上可接受的酸加成盐，条件是R1，R2，R3和R4不都是具有显着镇痛活性的氢和它们制备的新方法。

95. 发明授权

US4655785A Process for photochemical stabilization of polyamide and polyurethane fiber materials with metal complex compounds 失效
标题翻译：用金属络合物进行聚酰胺和聚氨酯纤维材料的光化学稳定化工艺
公开(公告)号：US4655785A
公开(公告)日：1987-04-07
申请号：US736927
申请日：1985-05-21
申请人： Gerhard Reinert , Gerhard Back , Helmut Huber-Emden
发明人： Gerhard Reinert , Gerhard Back , Helmut Huber-Emden
IPC分类号： C07F1/08 , C07C243/38 , C07C309/49 , C07F13/00 , C07F15/04 , C09B55/00 , D06M13/02 , D06M13/322 , D06M13/50 , D06M13/503 , D06M101/00 , D06M101/16 , D06M101/30 , D06M101/34 , D06M101/36 , D06P1/62 , D06P1/642 , D06P3/24 , D06P3/26 , D06P5/00 , D06P5/06 , D06P5/10 , D06P1/64
CPC分类号： D06P3/26 , C07C243/38 , C09B55/007 , D06M13/503 , D06P1/6423 , D06P3/241 , Y10S8/924 , Y10S8/926
摘要： A process for the photochemical stabilization of undyed and dyed polyamide or polyurethane fibre material that is characterized in that the fibre material is treated with a water soluble, organic copper, manganese or nickel complex that displays an affinity for the fibres. The polyamide or polyurethane fibre material, e.g., textile, that has been so treated retains its stretch characteristics and elasticity even after prolonged periods of illumination. In addition, in the case of dyed material, treatment with the metal complex results in a marked improvement in light-fastness.
摘要翻译：一种用于未染色和染色的聚酰胺或聚氨酯纤维材料的光化学稳定的方法，其特征在于纤维材料用对纤维显示亲和力的水溶性有机铜，锰或镍络合物处理。已经如此处理的聚酰胺或聚氨酯纤维材料，例如纺织品即使在长时间的照明之后也保持其拉伸特性和弹性。此外，在染色材料的情况下，用金属络合物的处理导致耐光性显着提高。

96. 发明授权

US4629812A Method for producing N,N'-bis-salicyloyl hydrazine 失效
标题翻译：制备N，N'-双 - 水杨酰肼的方法
公开(公告)号：US4629812A
公开(公告)日：1986-12-16
申请号：US294032
申请日：1981-08-18
申请人： Wolfgang von Gentzkow
发明人： Wolfgang von Gentzkow
IPC分类号： C07C243/22 , B01J21/02 , B01J21/04 , B01J23/06 , B01J27/08 , B01J27/125 , B01J27/138 , C07C67/00 , C07C241/00 , C07C243/38 , C08K5/25 , H01B3/18 , H01B7/28 , C07C103/20
CPC分类号： C07C241/04 , C08K5/25 , H01B3/18 , H01B7/2806
摘要： The invention relates to a method for the production of N,N'-bis-salicyloyl hydrazine by a catalytic reaction of salicylic-acid alkyl esters with hydrazine or salicylic-acid hydrazide and has the object to develop such a method in such a manner that not only an N,N'-bis-salicyloyl hydrazine with reduced eye irritation is obtained, but wherein the product is also produced with a high yield and purity. For this purpose, the invention provides that hydrazine or salicylic-acid hydrazide is heated with a 1-to-10 times excess of salicylic-acid alkyl ester in the presence of a halogenide, hydroxide or oxide of boron, aluminum or zinc to temperatures of up to 150.degree. C. The N,N'-bis-salicyloyl hydrazine prepared by the method according to the invention is suitable particularly as an additive to polymers for cable and wire insulation in power and communication engineering.
摘要翻译：本发明涉及通过水杨酸烷基酯与肼或水杨酸酰肼的催化反应生产N，N'-双 - 水杨酰肼的方法，目的是开发这样一种方法，使得不仅得到具有减轻眼睛刺激性的N，N'-双 - 水杨酰肼，而且其产物也以高产率和纯度生产。为此，本发明提供了在卤化物，硼，铝或锌的卤化物，氢氧化物或氧化物存在下，将肼或水杨酸酰肼与水杨酸 - 酸烷基酯的1至10倍过量加热至通过根据本发明的方法制备的N，N'-双 - 水杨酰肼特别适用于电力和通信工程中用于电缆和电线绝缘的聚合物的添加剂。

97. 发明授权

US4495185A 1,2,4-Triazin-3(2H) ones 失效
标题翻译： 1,2,4-三嗪-3（2H）酮
公开(公告)号：US4495185A
公开(公告)日：1985-01-22
申请号：US436801
申请日：1982-10-26
申请人： David Brown , Rodney B. Hargreaves , Bernard J. McLoughlin , Stuart D. Mills
发明人： David Brown , Rodney B. Hargreaves , Bernard J. McLoughlin , Stuart D. Mills
IPC分类号： A61K31/535 , A61K31/5375 , A61K31/54 , A61P9/04 , A61P9/12 , C07C45/00 , C07C45/64 , C07C49/82 , C07C67/00 , C07C239/00 , C07C243/38 , C07C281/04 , C07D253/06 , C07D273/04 , C07D285/16 , C07D295/18 , C07D295/21 , A61K31/53
CPC分类号： C07D253/06 , C07C243/38 , C07C45/64 , C07D273/04 , C07D285/16 , C07D295/21
摘要： Heterocyclic compounds of the formula ##STR1## wherein either X is --CR.sup.1 R.sup.2 and Y is --O--, --S-- or --NR.sup.3 --, wherein R.sup.1, R.sup.2 and R.sup.3, which may be the same or different, each is hydrogen or alkyl of up to 4 carbon atoms;or X is --O--, --S-- or --NH-- and Y is --CR.sup.1 R.sup.2 -- wherein R.sup.1 and R.sup.2 have the meanings stated above;wherein either R.sup.4 is hydrogen, fluoro or chloro, or alkyl, alkenyl, halogenoalkyl, aminoalkyl, hydroxyalkyl, alkoxyalkyl or alkoxy each of up to 6 carbon atoms, and R.sup.5, R.sup.6 and R.sup.7, which may be the same or different, each is hydrogen, fluoro, chloro, bromo or iodo, or alkyl, alkenyl, halogenoalkyl, aminoalkyl, hydroxyalkyl, alkoxyalkyl or alkoxy each of up to 6 carbon atoms, provided that R.sup.4, R.sup.5, R.sup.6 and R.sup.7 are not all hydrogen;or R.sup.4 is bromo and R.sup.5, R.sup.6 and R.sup.7 have the meanings stated above, provided that R.sup.5, R.sup.6 and R.sup.7 are not all hydrogen;or R.sup.4 and R.sup.5 together, or R.sup.5 and R.sup.6 together, or R.sup.4 and R.sup.7 together, form the --CH.dbd.CH--CH.dbd.CH-- group and the other two or R.sup.4, R.sup.5, R.sup.6 and R.sup.7 have the meanings stated above; processes for their manufacture and pharmaceutical compositions containing them. The compounds possess cardiotonic and/or antihypertensive activity.
摘要翻译：其中X是-CR 1 R 2和Y的杂环化合物是其中R 1，R 2和R 3可以相同或不同，各自为氢或烷基，最多4个碳原子; 或X是-O - ， - S-或-NH-，Y是-CR 1 R 2 - ，其中R 1和R 2具有上述含义; 其中R 4是氢，氟或氯，或至多6个碳原子的烷基，烯基，卤代烷基，氨基烷基，羟基烷基，烷氧基烷基或烷氧基，以及可以相同或不同的R 5，R 6和R 7各自为氢，氟，氯，溴或碘，或各自具有至多6个碳原子的烷基，烯基，卤代烷基，氨基烷基，羟基烷基，烷氧基烷基或烷氧基，条件是R4，R5，R6和R7不全部为氢; 或R 4为溴，R 5，R 6和R 7具有上述含义，条件是R 5，R 6和R 7不全为氢; 或R 4和R 5一起，或R 5和R 6一起，或者R 4和R 7一起形成-CH = CH-CH = CH-基，而另外两个或者R 4，R 5，R 6和R 7具有上述含义; 其制造方法和含有它们的药物组合物。该化合物具有强心剂和/或抗高血压活性。

98. 发明授权

US4175184A Manufacture of 2,1,3-thiadiazin-4-one-2,2-dioxide derivatives 失效
标题翻译：制备2,1,3-噻二嗪-4-酮-2,2-二氧化物衍生物
公开(公告)号：US4175184A
公开(公告)日：1979-11-20
申请号：US879722
申请日：1978-02-21
申请人： Hans Merkle , Albrecht Mueller , Karl Zoller
发明人： Hans Merkle , Albrecht Mueller , Karl Zoller
IPC分类号： C07C243/38 , C07D213/18 , C07D285/16 , C07D513/04 , C07D285/22
CPC分类号： C07D285/16 , C07C243/38 , C07D213/18 , C07D513/04
摘要： New and valuable process for the manufacture of 2,1,3-thiadiazin-4-one-2,2-dioxide derivatives by reaction of anthranilic acid amide or aminopyridine carboxamide derivatives with sulfur trioxide derivatives to give the sulfamic acid salts, followed by cyclization of these salts.
摘要翻译：通过邻氨基苯甲酰胺或氨基吡啶甲酰胺衍生物与三氧化硫衍生物的反应制备2,1,3-噻二嗪-4-酮-2,2-二氧化物衍生物的新的和有价值的方法得到氨基磺酸盐，随后环化的这些盐。

99. 发明授权

US4160862A 1-Acyl-3-(amino-lower-alkyl)indoles 失效
标题翻译： 1-酰基-3-（氨基 - 低级 - 烷基）吲哚
公开(公告)号：US4160862A
公开(公告)日：1979-07-10
申请号：US439279
申请日：1974-02-04
申请人： Bernard L. Zenitz
发明人： Bernard L. Zenitz
IPC分类号： C07C243/32 , C07C243/38 , C07D207/06 , C07D207/20 , C07D209/10 , C07D209/12 , C07D209/14 , C07D209/18 , C07D211/12 , C07D211/14 , C07D213/16 , C07D401/06
CPC分类号： C07D213/16 , C07C243/32 , C07C243/38 , C07D207/06 , C07D207/20 , C07D209/10 , C07D209/12 , C07D209/14 , C07D209/18 , C07D211/12 , C07D211/14
摘要： 1-Acyl-3-(amino-lower-alkyl)indoles, useful as anti-inflammatory agents, are prepared either by acylation of a 3-(amino-lower-alkyl)indole; by Fisher indole synthesis from an N'-acylphenylhydrazine and an amino-lower-alkanone; by alkylation of an amine with a 1-acyl-3-(halo-lower-alkyl)indole; or by reductive alkylation of a 1-acyl-3-indole-lower-alkylcarboxaldehyde.
摘要翻译：通过3-（氨基 - 低级 - 烷基）吲哚的酰化制备可用作抗炎剂的1-酰基-3-（氨基 - 低级 - 烷基）吲哚; 通过来自N'-酰基苯肼和氨基 - 低级烷酮的Fisher吲哚合成; 通过用1-酰基-3-（卤代 - 低级 - 烷基）吲哚烷基化胺; 或通过1-酰基-3-吲哚 - 低级 - 烷基甲醛的还原烷基化。

100. 发明授权

US4150235A Interphenylene 11,12-secoprostaglandins 失效
标题翻译：亚苯基11,12-前列腺素
公开(公告)号：US4150235A
公开(公告)日：1979-04-17
申请号：US751831
申请日：1976-12-17
申请人： Edward J. Cragoe, Jr. , John B. Bicking
发明人： Edward J. Cragoe, Jr. , John B. Bicking
IPC分类号： C07C69/66 , A61K31/16 , A61K31/165 , A61K31/19 , A61K31/215 , A61P7/10 , A61P9/08 , A61P9/12 , A61P37/06 , A61P43/00 , C07C45/46 , C07C51/00 , C07C51/08 , C07C51/29 , C07C59/125 , C07C59/48 , C07C59/68 , C07C59/70 , C07C59/84 , C07C59/90 , C07C63/04 , C07C65/01 , C07C65/32 , C07C65/40 , C07C67/00 , C07C69/612 , C07C69/76 , C07C231/00 , C07C235/10 , C07C235/20 , C07C235/34 , C07C235/42 , C07C235/78 , C07C235/84 , C07C241/00 , C07C243/32 , C07C243/38 , C07C255/32 , C07D309/12
CPC分类号： C07D309/12 , C07C243/38 , C07C255/00 , C07C403/20 , C07C45/46 , C07C51/08 , C07C59/90 , C07C65/01 , C07C65/40 , C07C2101/14
摘要： Novel interphenylene derivatives of 11,12-secoprostaglandins are prepared by the stepwise alkylation of the ethyl ester or the t-butyl ester of acetoacetic acid. One such method involves treatment of the t-butyl ester of acetoacetic acid with a strong base to form the anion followed by treatment with ethyl p-(3-bromopropyl)benzoate to produce ethyl 4-(4-tert-butoxycarbonyl-5-oxo-hexyl)benzoate, subsequently reacting the anion of the thus-formed benzoate with 1-chloro-4-acetoxynonane to produce ethyl 4-(4-acetyl-4-tert-butoxycarbonyl-8-acetoxytridecyl)benzoate followed by decarboxylation and alkaline hydrolysis to produce the desired product 4-(4-acetyl-8-hydroxytridecyl)benzoic acid which is useful as pharmaceutical in the treatment of patients with renal failure and in the prevention of transplant rejection.
摘要翻译：通过乙酸乙酯或乙酸乙酯的叔丁酯的逐步烷基化制备11,12-前列腺素的新型间苯二酚衍生物。一种这样的方法包括用强碱处理乙酰乙酸的叔丁酯以形成阴离子，然后用对 - （3-溴丙基）苯甲酸乙酯处理，得到4-（4-叔丁氧基羰基-5-氧代 - 己基）苯甲酸酯，随后将由此形成的苯甲酸酯的阴离子与1-氯-4-乙酰氧基壬烷反应，生成4-（4-乙酰基-4-叔丁氧基羰基-8-乙酰氧基十三烷基）苯甲酸乙酯，然后脱羧和碱水解以产生所需产物4-（4-乙酰基-8-羟基十三烷基）苯甲酸，其可用作治疗肾衰竭患者和预防移植排斥的药物。

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