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1. 发明公开

KR1020080017405A 살진균성 5-히드록시피라졸린, 이들의 제조 방법 및 이들을포함하는 제제 无效
标题翻译：杀真菌剂5-羟基吡唑啉酮，其生产方法及其同类物质
公开(公告)号：KR1020080017405A
公开(公告)日：2008-02-26
申请号：KR1020077030692
申请日：2006-05-24
申请人： 바스프 에스이
发明人： 게베르,마르쿠스 , 디에쯔,요헨 , 그로테,토마스 , 귀프세르,안드레아스 , 니에덴브뤼크,마티아스
IPC分类号： C07D231/08 , A01N43/56
CPC分类号： A01N43/56 , C07D231/06
摘要： The invention relates to novel 5-hydroxypyrazolines of formula (I) wherein the substituents have the following designations: B represents phenyl, naphthyl or 5-membered or 6-membered hetaryl containing between one and four heteroatoms from the group comprising O, N or S; A represents C=O, C=S or SO2; W represents CX1X2; X1, X2 represent hydrogen, fluorine, chlorine, or bromine; R1 represents alkyl, halogenalkyl, alkenyl, halogenalkenyl, alkinyl or halogenalkinyl, cycloalkyl, cycloalkenyl, cycloalkinyl, phenyl, 5-membered or 6-membered heterocyclyl or hetaryl containing between one and four heteroatoms from the group comprising O, N or S; R2 represents hydrogen or alkyl; R3 represents hydrogen, nitro, cyano, alkyl, halogenalkyl, alkoxy, halogenalkoxy, alkenyl, halogenalkenyl, alkinyl, halogenalkinyl or NR'2, wherein R' represents hydrogen or alkyl; and R4 represents hydrogen, halogen, nitro, cyano, NR'2, alkyl, halogenalkyl, COOR' or 5-membered or 6-membered hetaryl or heterocyclyl. The pre-cited variables can be substituted according to the description. The invention also relates to methods for the production of said components, to the use thereof for controlling pathogenic fungi, and to agents containing the same.
摘要翻译：本发明涉及式（I）的新型5-羟基吡唑啉，其中取代基具有以下指定：B代表苯基，萘基或含有一个至四个包含O，N或S的杂原子的5元或6元杂芳基 ; A表示C = O，C = S或SO 2; W代表CX1X2; X1，X2表示氢，氟，氯或溴; R1代表烷基，卤代烷基，烯基，卤代烯基，炔基或卤代烯基，环烷基，环烯基，环烯基，苯基，含有一个至四个包含O，N或S的杂原子的5元或6元杂环基或杂芳基; R2代表氢或烷基; R 3表示氢，硝基，氰基，烷基，卤代烷基，烷氧基，卤代烷氧基，烯基，卤素链烯基，炔基，卤代炔基或NR'2，其中R'表示氢或烷基; R 4代表氢，卤素，硝基，氰基，NR'2，烷基，卤代烷基，COOR'或5元或6元杂芳基或杂环基。引用前的变量可以根据描述进行替代。本发明还涉及生产所述组分的方法，其用于控制致病真菌的用途，以及含有它们的试剂。

2. 发明公开

KR1020080016693A 살진균성 5-히드록시피라졸린, 이들의 제조 방법 및 이들을포함하는 제제 无效
标题翻译：杀真菌剂5-羟基吡唑啉酮及其制备方法和包含其的药剂
公开(公告)号：KR1020080016693A
公开(公告)日：2008-02-21
申请号：KR1020077030691
申请日：2006-05-24
申请人： 바스프 에스이
发明人： 게베르,마르쿠스 , 디에쯔,요헨 , 그로테,토마스 , 귀프세르,안드레아스 , 니에덴브뤼크,마티아스
IPC分类号： C07D231/08 , A01N43/56 , A61P3/00
CPC分类号： A01N43/56
摘要： The invention relates to the novel 5-hydroxypyrazolines of formula (I), wherein the substituents are defined as follows: B represents phenyl, naphthyl or 5-or 6-membered hetaryl having one to four hetero atoms from the group including O, N or S; A represents C=O, C=S or SO2; R1 represents alkyl, alkyl halide, alkenyl, alkenyl halide, alkinyl or alkinyl halide, cycloalkyl, cycloalkenyl, cycloalkinyl, phenyl, 5-or 6-membered heterocyclyl or hetaryl, having one to four hetero atoms from the group including O, N or S; R2 represents alkyl, alkyl halide, alkenyl, alkyl halide, alkinyl, alkinyl halide, cycloalkyl, cycloalkenyl, cycloalkinyl, phenyl, 5-or 6-membered hetaryl or heterocyclyl having one to four hetero atoms from the group including O, N or S; R3 represents hydrogen, nitro, cyano, alkyl, alkyl halide, alkoxy, halogenalkoxy, alkenyl, alkenyl halide, alkinyl, alkinyl halide or NR'2, wherein R' independently represents hydrogen or alkyl; R4 represents hydrogen, halogen, nitro, cyano, NR'2, alkyl, alkyl halide, COOR' or 5-or 6-membered hetaryl or heterocyclyl; wherein the aforementioned variables may be substituted as defined in the description. The invention also relates to a method for producing the inventive compounds, to their use for controlling parasitic fungi and to agents comprising the same.
摘要翻译：本发明涉及式（I）的新型5-羟基吡唑啉，其中取代基定义如下：B代表苯基，萘基或5-或6-元杂芳基，其具有一个至四个杂原子，包括O，N或 S; A表示C = O，C = S或SO 2; R1代表烷基，烷基卤，烯基，烯基卤，炔基或炔基卤化物，环烷基，环烯基，环烯基，苯基，5-或6-元杂环基或杂芳基，具有一个至四个包括O，N或S ; R2代表烷基，烷基卤，烯基，烷基卤，炔基，炔基卤，环烷基，环烯基，环烯基，苯基，5-或6-元杂芳基或具有1-4个杂原子的杂环基，包括O，N或S; R3表示氢，硝基，氰基，烷基，烷基卤，烷氧基，卤代烷氧基，烯基，烯基卤，链炔基，炔基卤或NR'2，其中R'独立地表示氢或烷基; R4表示氢，卤素，硝基，氰基，NR'2，烷基，烷基卤，COOR'或5-或6-元杂芳基或杂环基; 其中上述变量可以如说明书中定义的那样被替代。本发明还涉及用于制备本发明化合物的方法，其用于控制寄生真菌和包含其的试剂。

3. 发明公开

KR1020080017406A 살진균성 Ｎ-벤질-5-히드록시-5-페닐피라졸린, 이들의 제조방법 및 이들을 포함하는 제제 无效
标题翻译：杀真菌N-苄基-5-羟基-5-苯基吡唑啉，其生产方法及其同类物质
公开(公告)号：KR1020080017406A
公开(公告)日：2008-02-26
申请号：KR1020077030694
申请日：2006-05-24
申请人： 바스프 에스이
发明人： 게베르,마르쿠스 , 디에쯔,요헨 , 그로테,토마스 , 귀프세르,안드레아스 , 니에덴브뤼크,마티아스
IPC分类号： C07D231/20 , A01N43/56
CPC分类号： C07D231/08 , A01N43/56
摘要： The invention relates to N-benzoyl-5-hydroxy-5-phenylpyrazolines of formula (I) wherein the substituents have the following designations: L 1, L2 represent hydrogen, halogen, halogenalkyl, alkenyl, halogenalkenyl, alkinyl or haIogenalkinyl; L3, L4, L5 represent alkyl or one of the groups cited for L1 and L2; X represents oxygen or sulphur; R1 represents halogen, nitro, cyano, NR'2, alkyl, halogenalkyl, alkoxy, alkenyl, halogenalkyl, alkinyl, halogenalkinyl, cycloalkyl, cycloalkenyl, cycloalkinyl, phenyl, or 5-membered or 6-membered heterocycle or hetaryl containing between one and four heteroatoms from the group comprising O, N or S; R' represents hydrogen or alkyl; m represents 1, 2, 3, 4 or 5; R2 represents hydrogen or alkyl; R3 represents hydrogen, nitro, cyano, alkyl, halogenalkyl, alkoxy, halogenalkoxy, alkenyl, halogenalkenyl, alkinyl, halogenalkinyl or NR'2; and R4 represents hydrogen, halogen, nitro, cyano, NR'2, alkyl, halogenalkyl, COOR' or 5-membered or 6-membered heterocyclyl or hetaryl containing between one and four heteroatoms from the group comprising O, N or S. The pre-cited variables can be substituted according to the description. The invention also relates to methods for the production of said compounds, to the use thereof for controlling pathogenic fungi, and to agents containing the same.
摘要翻译：本发明涉及式（I）的N-苯甲酰基-5-羟基-5-苯基吡唑啉，其中取代基具有以下指定：L 1，L 2代表氢，卤素，卤代烷基，烯基，卤素链烯基，炔基或卤素基; L3，L4，L5表示烷基或对L1和L2引用的基团之一; X表示氧或硫; R1代表卤素，硝基，氰基，NR'2，烷基，卤代烷基，烷氧基，烯基，卤代烷基，炔基，卤代烯基，环烷基，环烯基，环烯基，苯基或含1至4个的5-元或6-元杂环或杂芳基包含O，N或S的基团的杂原子; R'表示氢或烷基; m表示1,2,3,4或5; R2代表氢或烷基; R 3表示氢，硝基，氰基，烷基，卤代烷基，烷氧基，卤代烷氧基，烯基，卤代烯基，炔基，卤代炔基或NR'2; R4代表氢，卤素，硝基，氰基，NR'2，烷基，卤代烷基，COOR'或含有一个至四个来自O，N或S的杂原子的五元或六元杂环基或杂芳基。所引用的变量可以根据描述进行替换。本发明还涉及生产所述化合物的方法，其用于控制致病真菌的用途，以及含有它们的药剂的方法。

4. 发明公开

KR1020080018916A 비시클릭 5-히드록시피라졸린, 이들의 제조 방법 및 이들을포함하는 제제 无效
标题翻译：双羟基-5-羟基吡唑啉酮及其制备方法和包含其的试剂
公开(公告)号：KR1020080018916A
公开(公告)日：2008-02-28
申请号：KR1020077030695
申请日：2006-05-24
申请人： 바스프 에스이
发明人： 게베르,마르쿠스 , 디에쯔,요헨 , 그로테,토마스 , 귀프세르,안드레아스 , 니에덴브뤼크,마티아스
IPC分类号： A01N43/56 , C07D231/54 , C07D401/06 , A01P3/00
CPC分类号： C07D401/12 , A01N43/56 , C07D231/56
摘要： The invention relates to the novel 5-hydroxypyrazolines of formula (I), wherein the substituents are defined as follows: B represents phenyl, naphthyl or 5-or 6-membered hetaryl having one to four hetero atoms from the group including O, N or S; A represents C=O, C=S or SO2; R1 represents alkyl, alkyl halide, alkenyl, alkenyl halide, alkinyl or alkinyl halide, cycloalkyl, cycloalkenyl, cycloalkinyl, phenyl, 5-or 6-membered heterocyclyl or hetaryl, having one to four hetero atoms from the group including O, N or S; R2 together with R1 or R4 represents C3-C4 alkyls or C3-C4 alkenyls, which groups can be defined as in the description; R3 represents hydrogen, nitro, cyano, NR''2, alkyl, alkyl halide, alkoxy, halogenalkoxy, alkenyl, alkenyl halide, alkinyl or alkinyl halide, wherein R'' independently represents hydrogen or alkyl; R4 represents hydrogen, halogen, nitro, cyano, NR''2, alkyl, alkyl halide, COOR'' or 5-or 6-membered hetaryl or heterocyclyl; wherein the aforementioned variables may be substituted as defined in the description. The invention also relates to a method for producing the inventive compounds, to their use for controlling parasitic fungi and to agents comprising the same.
摘要翻译：本发明涉及式（I）的新型5-羟基吡唑啉，其中取代基定义如下：B代表苯基，萘基或5-或6-元杂芳基，其具有一个至四个杂原子，包括O，N或 S; A表示C = O，C = S或SO 2; R1代表烷基，烷基卤，烯基，烯基卤，炔基或炔基卤化物，环烷基，环烯基，环烯基，苯基，5-或6-元杂环基或杂芳基，具有一个至四个包括O，N或S ; R2与R1或R4一起代表C3-C4烷基或C3-C4烯基，这些基团可以在描述中定义; R3表示氢，硝基，氰基，NR'2，烷基，烷基卤，烷氧基，卤代烷氧基，烯基，烯基卤，炔基或炔基卤，其中R“独立地表示氢或烷基; R4表示氢，卤素，硝基，氰基，NR'2，烷基，烷基卤，COOR“或5-或6-元杂芳基或杂环基; 其中上述变量可以如说明书中定义的那样被替代。本发明还涉及用于制备本发明化合物的方法，其用于控制寄生真菌和包含其的试剂。

5. 发明公开

KR1020070047819A 트리아졸로피리미딘 유도체로부터 제조된 살진균성상승작용적 혼합물 无效
标题翻译：三唑并嘧啶衍生物的杀真菌混合物
公开(公告)号：KR1020070047819A
公开(公告)日：2007-05-07
申请号：KR1020077005086
申请日：2005-07-28
申请人： 바스프 에스이
发明人： 블레트너,카르스텐 , 디에츠,요헨 , 그라메노스,바실리오스 , 그로테,토마스 , 휜거,우도 , 뮐러,베른트 , 니에덴브뤼크,마티아스 , 라인하이머,요아힘 , 섀퍼,피터 , 쉬베크,프란크 , 쉬뵈글러,안야 , 네이브,바바라 , 쉐레르,마리아 , 스트라트만,지그프리트 , 쉐플,울리히 , 스티를,라인하르트
IPC分类号： A01N43/90 , A01P3/00
CPC分类号： A01N43/90 , A01N43/653 , A01N47/14 , A01N43/50 , A01N57/12 , A01N47/04 , A01N37/34 , A01N43/40 , A01N37/50 , A01N37/46 , A01N43/84 , A01N37/38 , A01N43/28 , A01N47/38 , A01N43/54 , A01N43/32 , A01N59/20 , A01N2300/00
摘要： 본 발명은 활성 성분으로서, 1) 하기 화학식 I의 5-클로르-6-페닐-7-헤테로시클릴아미노트리아졸로피리미딘, 및 2) 하기 군 A) 내지 R)로부터 선택되는 1종 이상의 활성 화합물 II를 상승작용적 활성량으로 함유하는 살진균성 혼합물에 관한 것이다.

상기 식 중,
D는 비치환되거나 또는 하나 또는 2개의 메틸기로 또는 에틸, 프로필 또는 부틸기로 치환된, 질소 원자와 함께 피롤리딘, 피페리딘 또는 아제핀 고리를 형성하며,
L은 메틸, 불소 또는 염소이다.
A) 아졸, B) 스트로빌루린, C) 아실알라닌, D) 아민 유도체, E) 아닐리노피리미딘, F) 디카르복시미드, G) 신남산 아미드 및 유사 화합물, H) 항생제, K) 디티오카르바메이트, L) 명세서에서 언급된 헤테로시클릭 화합물, M) 황 및 구리 살진균제, N) 니트로페닐 유도체, O) 페닐피롤, P) 술펜산 유도체, Q) 명세서에서 언급된 기타 살진균제, 또는 R) 성장 억제제.
본 발명은 또한 신규한 트리아졸로피리미딘, 화학식 I의 화합물 또는 화학식 I의 화합물과 군 A) 내지 R)의 활성 성분의 혼합물을 사용하여 유해 진균류를 방제하는 방법 및 상기 화합물 또는 혼합물 함유하는 상기 유형의 혼합물 및 수단을 제조하기 위한 화학식 I의 화합물과 군 A) 내지 R)의 활성 화합물의 용도에 관한 것이다.
5-클로로-6-페닐-7-헤테로시클릴아미노트리아졸로피리미딘, 아졸, 스트로빌루린, 아실알라닌, 살진균성 혼합물.

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