会员体验
专利管家(专利管理)
工作空间(专利管理)
风险监控(情报监控)
数据分析(专利分析)
侵权分析(诉讼无效)
联系我们
交流群
官方交流:
QQ群: 891211   
微信请扫码    >>>
现在联系顾问~
热词
    • 1. 发明申请
    • Piperazine Compounds Having Herbicidal Action
    • 具有除草作用的哌嗪化合物
    • US20100173777A1
    • 2010-07-08
    • US12663781
    • 2008-06-11
    • Eike HupeThomas SeitzMatthias WitschelDschun SongWilliam Karl MobergLiliana Parra RapadoFrank StelzerAndrea VescoviTrevor William NewtonRobert ReinhardBernd SievernichKlaus GrossmannThomas EhrhardtMichael RackElmar Kibler
    • Eike HupeThomas SeitzMatthias WitschelDschun SongWilliam Karl MobergLiliana Parra RapadoFrank StelzerAndrea VescoviTrevor William NewtonRobert ReinhardBernd SievernichKlaus GrossmannThomas EhrhardtMichael RackElmar Kibler
    • A01N43/60C07D241/04A01P13/00
    • C07D241/08A01N43/60
    • The present invention relates to piperazine compounds of the general formula I defined below and to their use as herbicides. Moreover, the invention relates to compositions for crop protection and to a method for controlling unwanted vegetation. R1 is selected from the group consisting of halogen, cyano, nitro, Z—C(═O)—R12, phenyl and a 5- or 6-membered heterocyclic radical which has 1, 2, 3 or 4 heteroatoms selected from the group consisting of O, N and S as ring atoms, where phenyl and the heterocyclic radical are unsubstituted or may have 1, 2, 3 or 4 substituents R1a; Z is a covalent bond or a CH2 group; R12 is hydrogen, C1-C6-alkyl, C3-C6-cycloalkyl, C2-C6-alkenyl, C5-C6-cycloalkenyl, C2-C6-alkynyl and the like; R2 is hydrogen, halogen, nitro, cyano, C1-C4-alkyl, C1-C4-haloalkyl, C2-C4-alkenyl, C1-C4-alkoxy, C1-C4-haloalkoxy, benzyl or a group S(O)nR21 in which R21 is C1-C4-alkyl or C1-C4-haloalkyl and n is 0, 1 or 2; R3 is hydrogen or halogen; R4 is C1-C4-alkyl, C3-C4-alkenyl or C3-C4-alkynyl; R5 is hydrogen, C1-C4-alkyl, C3-C4-alkenyl, C3-C4-alkynyl or a group C(═O)R51 in which R51 is hydrogen, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy or C1-C4-haloalkoxy; R6 is C1-C4-alkyl, C1-C4-hydroxyalkyl or C1-C4-haloalkyl; R7, R8 independently of one another are hydrogen, OH, C1-C4-alkoxy, C1-C4-haloalkyloxy, C1-C4-alkyl or C1-C4-haloalkyl; R9, R10 independently of one another are selected from the group consisting of hydrogen, halogen, CN, NO2, C1-C4-alkyl, C1-C4-haloalkyl, C2-C4-alkenyl, C1-C4-alkoxy and C1-C4-haloalkoxy; and R11 is hydrogen or C1-C4-alkyl; and the agriculturally useful salts of these compounds.
    • 本发明涉及下面定义的通式I的哌嗪化合物及其作为除草剂的用途。 此外,本发明涉及用于作物保护的组合物和用于防治不想要的植物的方法。 R 1选自卤素,氰基,硝基,Z-C(= O)-R 12,苯基和具有1,2,3或4个杂原子的5或6元杂环基,所述杂原子选自 的O,N和S作为环原子,其中苯基和杂环基是未取代的或可以具有1,2,3或4个取代基R 1a; Z是共价键或CH2基; R12是氢,C1-C6-烷基,C3-C6-环烷基,C2-C6-烯基,C5-C6-环烯基,C2-C6-炔基等; R2是氢,卤素,硝基,氰基,C1-C4-烷基,C1-C4卤代烷基,C2-C4-烯基,C1-C4-烷氧基,C1-C4-卤代烷氧基,苄基或基团S(O) 其中R 21为C 1 -C 4烷基或C 1 -C 4卤代烷基,n为0,1或2; R3是氢或卤素; R4是C1-C4-烷基,C3-C4-烯基或C3-C4-炔基; R 5为氢,C 1 -C 4 - 烷基,C 3 -C 4 - 烯基,C 3 -C 4 - 炔基或C(= O)R 51,其中R 51为氢,C 1 -C 4 - 烷基,C 1 -C 4 - 卤代烷基, C 4 - 烷氧基或C 1 -C 4 - 卤代烷氧基; R 6是C 1 -C 4烷基,C 1 -C 4羟基烷基或C 1 -C 4卤代烷基; R 7,R 8彼此独立地是氢,OH,C 1 -C 4 - 烷氧基,C 1 -C 4卤代烷氧基,C 1 -C 4 - 烷基或C 1 -C 4卤代烷基; R 9,R 10彼此独立地选自氢,卤素,CN,NO 2,C 1 -C 4 - 烷基,C 1 -C 4 - 卤代烷基,C 2 -C 4 - 烯基,C 1 -C 4 - 烷氧基和C 1 -C 4 - 卤代烷氧基 和R 11是氢或C 1 -C 4 - 烷基; 和这些化合物的农业上有用的盐。
    • 3. 发明申请
    • Piperazine Compounds Whith a Herbicidal Action
    • 哌嗪化合物具有除草作用
    • US20100152047A1
    • 2010-06-17
    • US12663784
    • 2008-06-11
    • Eike HupeThomas SeitzMatthias WitschelDschun SongWilliam Karl MobergLiliana Parra RapadoFrank StelzerAndrea VescoviTrevor William NewtonRobert ReinhardBernd SievernichKlaus GrossmannThomas EhrhardtMichael RackElmar Kibler
    • Eike HupeThomas SeitzMatthias WitschelDschun SongWilliam Karl MobergLiliana Parra RapadoFrank StelzerAndrea VescoviTrevor William NewtonRobert ReinhardBernd SievernichKlaus GrossmannThomas EhrhardtMichael RackElmar Kibler
    • A01N43/58C07D403/10C07D401/10C07D241/02C07D413/10A01N43/54A01N43/60A01P13/00
    • C07D241/08C07D403/10C07D407/10C07D409/10C07D413/10C07D417/10
    • The present invention relates to piperazine compounds of the general formula I defined below and to their use as herbicides. Moreover, the invention relates to compositions for crop protection and to a method for controlling unwanted vegetation. In formula I, the variables have the following meanings: R1 is selected from the group consisting of halogen, cyano, nitro, Z—C(═O)—R11, phenyl and a 5- or 6-membered heterocyclic radical which has 1, 2, 3 or 4 heteroatoms selected from the group consisting of O, N and S as ring atoms, where phenyl and the heterocyclic radical are unsubstituted or may have 1, 2, 3 or 4 substituents R1a; Z is a covalent bond or a CH2 group; R11 is hydrogen, C1-C6-alkyl, C3-C6-cycloalkyl, C2-C6-alkenyl, C5-C6-cycloalkenyl, C2-C6-alkynyl and the like; R2 is hydrogen, halogen, nitro, cyano, C1-C4-alkyl, C1-C4-haloalkyl, C2-C4-alkenyl, C1-C4-alkoxy, C1-C4-haloalkoxy, benzyl or a group S(O)nR21 in which R21 is C1-C4-alkyl or C1-C4-haloalkyl and n is 0, 1 or 2; R3 is hydrogen or halogen; R4 is C1-C4-alkyl, C3-C4-alkenyl or C3-C4-alkynyl; R5 is hydrogen, C1-C4-alkyl, C3-C4-alkenyl, C3-C4-alkynyl or a group C(═O)R51 in which R51 is hydrogen, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy or C1-C4-haloalkoxy; R6 is C1-C4-alkyl, C1-C4-hydroxyalkyl or C1-C4-haloalkyl; R7, R8 independently of one another are hydrogen, OH, C1-C4-alkoxy, C1-C4-haloalkyloxy, C1-C4-alkyl or C1-C4-haloalkyl; and R9, R10 independently of one another are selected from the group consisting of hydrogen, halogen, CN, NO2, C1-C4-alkyl, C1-C4-haloalkyl, C2-C4-alkenyl, C1-C4-alkoxy and C1-C4-haloalkoxy.
    • 本发明涉及下面定义的通式I的哌嗪化合物及其作为除草剂的用途。 此外,本发明涉及用于作物保护的组合物和用于防治不想要的植物的方法。 在式I中,变量具有以下含义:R 1选自卤素,氰基,硝基,Z-C(= O)-R 11,苯基和具有1, 2,3或4个选自O,N和S作为环原子的杂原子,其中苯基和杂环基是未取代的或可以具有1,2,3或4个取代基R 1a; Z是共价键或CH2基; R11是氢,C1-C6-烷基,C3-C6-环烷基,C2-C6-烯基,C5-C6-环烯基,C2-C6-炔基等; R2是氢,卤素,硝基,氰基,C1-C4-烷基,C1-C4卤代烷基,C2-C4-烯基,C1-C4-烷氧基,C1-C4-卤代烷氧基,苄基或基团S(O) 其中R 21为C 1 -C 4烷基或C 1 -C 4卤代烷基,n为0,1或2; R3是氢或卤素; R4是C1-C4-烷基,C3-C4-烯基或C3-C4-炔基; R 5为氢,C 1 -C 4 - 烷基,C 3 -C 4 - 烯基,C 3 -C 4 - 炔基或C(= O)R 51,其中R 51为氢,C 1 -C 4 - 烷基,C 1 -C 4 - 卤代烷基, C 4 - 烷氧基或C 1 -C 4 - 卤代烷氧基; R 6是C 1 -C 4烷基,C 1 -C 4羟基烷基或C 1 -C 4卤代烷基; R 7,R 8彼此独立地是氢,OH,C 1 -C 4 - 烷氧基,C 1 -C 4卤代烷氧基,C 1 -C 4 - 烷基或C 1 -C 4卤代烷基; R 9,R 10彼此独立地选自氢,卤素,CN,NO 2,C 1 -C 4 - 烷基,C 1 -C 4 - 卤代烷基,C 2 -C 4 - 烯基,C 1 -C 4 - 烷氧基和C 1 -C 4 卤代烷氧基。
    • 4. 发明申请
    • Herbicidally Active Composition
    • 除草活性成分
    • US20100190794A1
    • 2010-07-29
    • US12663795
    • 2008-06-11
    • Eike HupeWilliam Karl MobergRobert ReinhardBernd SievernichElmar Kibler
    • Eike HupeWilliam Karl MobergRobert ReinhardBernd SievernichElmar Kibler
    • A01N43/60A01N43/70A01P13/02
    • A01N37/46A01N43/60A01N33/18A01N43/10A01N43/40A01N43/42A01N43/50A01N43/54A01N43/70A01N43/80A01N43/82A01N47/12A01N47/30A01N2300/00
    • The present invention relates to herbicidally active compositions comprising at least one piperazinedione compound of the formula I in which: Rx, Ry are each hydrogen or together are a chemical bond; R1 is cyano or nitro; R2 is hydrogen, fluorine, chlorine, C1-C2-alkyl, ethenyl or C1-C2-alkoxy; R3 is fluorine or hydrogen; R4 is methyl; R5 is hydrogen, methyl or ethyl; R6 is hydrogen, methyl or ethyl; and R7 is hydrogen or halogen; and at least one further active compound selected from the group consisting of b1) lipid biosynthesis inhibitors; b2) acetolactate synthase inhibitors (ALS inhibitors); b3) photosynthesis inhibitors; b4) protoporphyrinogen-IX oxidase inhibitors, b5) bleacher herbicides; b6) enolpyruvyl shikimate 3-phosphate synthase inhibitors (EPSP inhibitors); b7) glutamine synthetase inhibitors; b8) 7,8-dihydropteroate synthase inhibitors (DHP inhibitors); b9) mitose inhibitors; b10) inhibitors of the synthesis of very long chain fatty acids (VLCFA inhibitors); b11) cellulose biosynthesis inhibitors; b12) decoupler herbicides; b13) auxin herbicides; b14) auxin transport inhibitors; b15) other herbicides, and C) safeners.
    • 本发明涉及包含至少一种式I的哌嗪二酮化合物的除草活性组合物,其中:Rx,Ry各自为氢或一起为化学键; R1是氰基或硝基; R2是氢,氟,氯,C1-C2-烷基,乙烯基或C1-C2-烷氧基; R3是氟或氢; R4是甲基; R5是氢,甲基或乙基; R6是氢,甲基或乙基; 并且R 7是氢或卤素; 和至少一种选自b1)脂质生物合成抑制剂的其它活性化合物; b2)乙酰乳酸合酶抑制剂(ALS抑制剂); b3)光合作用抑制剂; b4)原卟啉原-Ⅸ氧化酶抑制剂,b5)漂白剂除草剂; b6)烯醇丙酮酸莽沙鱼磷酸合酶抑制剂(EPSP抑制剂); b7)谷氨酰胺合成酶抑制剂; b8)7,8-二氢叶酸合酶抑制剂(DHP抑制剂); b9)丝裂抑制剂; b10)非常长链脂肪酸(VLCFA抑制剂)的合成抑制剂; b11)纤维素生物合成抑制剂; b12)除草剂除草剂; b13)生长素除草剂; b14)生长素运输抑制剂; b15)其他除草剂,和C)安全剂。
    • 6. 发明授权
    • Herbicidal mixture containing a 3-heterocyclyl-substituted benzoyl derivative and an adjuvant
    • 含有3-杂环基取代的苯甲酰基衍生物和佐剂的除草混合物
    • US06514910B1
    • 2003-02-04
    • US09914873
    • 2001-09-05
    • Matthias BratzRainer BerghausMartina OttenBernd SievernichElmar KiblerHerve Vantieghem
    • Matthias BratzRainer BerghausMartina OttenBernd SievernichElmar KiblerHerve Vantieghem
    • A01N4378
    • A01N43/78A01N43/80A01N37/06A01N37/02A01N25/30A01N2300/00
    • A herbicidal mixture, comprising a) a herbicidally effective amount of a benzoyl compound of formula I  where: R1, R2 are halogen, C1-C6-alkyl, C1-C6-alkylthio, C1-C6-alkyl-sulfinyl or C1-C6-alkylsulfonyl; R3 is hydrogen, halogen, C1-C6-alkyl; X is 4,5-dihydroisoxazolyl which is unsubstituted or mono- or polysubstituted by halogen, C1-C6-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylthio; R4 is a pyrazole of the formula II  which is attached in the 4-position and where R5 is hydrogen, R6 is methyl, or an environmentally compatible salt thereof; b) an adjuvant comprising i) a C1-C5-alkyl C5-C22-alkanoate, ii) a C10-C20-carboxylic acid, iii) a partial phosphoric ester or a partial sulfuric ester of a monohydroxy-functional polyalkyl ether and iv) optionally an alkyl polyoxyalkylene polyether, wherein the compound of formula I and the adjuvat are present in synergistically effective amounts.
    • 一种除草混合物,其包含a)除草有效量的式I的苯甲酰基化合物,其中:R 1,R 2是卤素,C 1 -C 6烷基,C 1 -C 6烷硫基,C 1 -C 6烷基亚磺酰基或C 1 -C 6烷基磺酰基 R 3是氢,卤素,C 1 -C 6 - 烷基; X是未被取代或被卤素,C 1 -C 6烷基,C 1 -C 4 - 烷氧基,C 1 -C 4 - 卤代烷基,C 1 -C 6 - 烷氧基取代或被单取代或多取代的4,5-二氢异恶唑基 -C 4 - 卤代烷氧基,C 1 -C 4 - 烷硫基; R 4是连接在4-位的式II的吡唑,其中R 5是氢,R 6是甲基或其环境相容的盐; b)佐剂,其包含:i) C1-C5烷基C5-C22-链烷酸酯,ii)C10-C20羧酸,iii)部分磷酸酯或单羟基官能聚烷基醚的部分硫酸酯,和/或任选的烷基聚氧化烯聚醚,其中化合物 并且佐剂以协同有效量存在。
    • 9. 发明申请
    • Synergistically acting herbicidal mixtures
    • 协同作用的除草混合物
    • US20050239653A1
    • 2005-10-27
    • US11079431
    • 2005-03-14
    • Bernd SievernichMax LandesElmar KiblerWolfgang DeynHelmut WalterMartina OttenKarl-Otto WestphalenHerve Vantieghem
    • Bernd SievernichMax LandesElmar KiblerWolfgang DeynHelmut WalterMartina OttenKarl-Otto WestphalenHerve Vantieghem
    • A01N43/40A01N43/72A01N43/78A01N43/80A01N57/00A01N61/00
    • A01N43/78A01N43/80A01N61/00A01N57/20A01N47/36A01N47/30A01N47/12A01N47/06A01N43/90A01N43/88A01N43/82A01N43/76A01N43/707A01N43/70A01N43/653A01N43/58A01N43/54A01N43/50A01N43/42A01N43/40A01N43/18A01N39/04A01N41/10A01N37/48A01N37/46A01N37/40A01N37/26A01N37/22A01N37/18A01N37/12A01N2300/00
    • A synergistic herbicidal mixture comprising A) at least one 3-heterocyclyl-substituted benzoyl derivative of the formula I in which the variables have the following meanings: R1, R3 are hydrogen, halogen, alkyl, halogenalkyl, alkoxy, halogenalkoxy, alkylthio, alkylsulfinyl or alkylsulfonyl; R2 is a heterocyclic radical selected from the group: thiazol-2-yl, thiazol-4-yl, thiazol-5-yl, isoxazol-3-yl, isoxazol-4-yl, isoxazol-5-yl, 4,5-dihydroisoxazol-3-yl, 4,5-dihydroisoxazol-4-yl and 4,5-dihydroisoxazol-5-yl, it being possible for these to be unsubstituted or mono- or polysubstituted by halogen, alkyl, alkoxy, haloalkyl, haloalkoxy or alkylthio; R4 is hydrogen, halogen or alkyl; R5 is alkyl; R6 is hydrogen or alkyl; or one of its environmentally compatible salts; and B) a synergistically effective amount of at least one herbicidal compound from the group of the acetyl-CoA carboxylase inhibitors (ACC), acetolactate synthase inhibitors (ALS), amides, auxin herbicides, auxin transport inhibitors, carotenoid biosynthesis inhibitors, enolpyruvylshikimate-3-phosphate synthase inhibitors (ESPS), glutamine synthetase inhibitors, lipid biosynthesis inhibitors, mitosis inhibitors, protophorphyrinogen [sic ] IX oxidase inhibitors, photosynthesis inhibitors, synergists, growth substances, cell wall biosynthesis inhibitors and a variety of other herbicides. Compositions comprising these mixtures, processes for the preparation of these compositions, and their use for controlling undesired plants.
    • 一种协同除草混合物,其包含A)至少一种式I的3-杂环基取代的苯甲酰基衍生物,其中变量具有以下含义:R 1,R 3, 氢,卤素,烷基,卤代烷基,烷氧基,卤代烷氧基,烷硫基,烷基亚磺酰基或烷基磺酰基; R 2是选自以下的杂环基:噻唑-2-基,噻唑-4-基,噻唑-5-基,异恶唑-3-基,异恶唑-4-基,异恶唑-4-基, 5,5-二氢异恶唑-3-基,4,5-二氢异恶唑-4-基和4,5-二氢异恶唑-5-基,这些可能是未被取代的或被卤素单取代或多取代, 烷基,烷氧基,卤代烷基,卤代烷氧基或烷硫基; R 4是氢,卤素或烷基; R 5是烷基; R 6是氢或烷基; 或其环境相容的盐之一; 乙酰辅酶A羧化酶抑制剂(ACC),乙酰乳酸合酶抑制剂(ALS),酰胺,生长素除草剂,生长素转运抑制剂,类胡萝卜素生物合成抑制剂,烯醇丙酮酸莽草酸-3(3)的协同有效量的至少一种除草化合物 磷酸合成酶抑制剂(ESPS),谷氨酰胺合成酶抑制剂,脂质生物合成抑制剂,有丝分裂抑制剂,原卟啉原IX氧化酶抑制剂,光合作用抑制剂,增效剂,生长物质,细胞壁生物合成抑制剂和各种其它除草剂。 包含这些混合物的组合物,这些组合物的制备方法以及它们用于控制不期望的植物的用途。