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1. 发明授权

US06812233B1 Therapeutic nucleosides 失效
标题翻译：治疗核苷
公开(公告)号：US06812233B1
公开(公告)日：2004-11-02
申请号：US09007502
申请日：1998-01-15
申请人： Dennis C. Liotta
发明人： Dennis C. Liotta
IPC分类号： A01N4354
CPC分类号： A61K31/505 , A61K31/70 , C07D327/04 , C07D405/04 , C07D411/04
摘要： The use of a 1,3-oxathiolane nucleoside analogue and pharmaceutically acceptable derivatives thereof for the treatment of hepatitis B virus infections is disclosed. Pharmaceutical formulations are also provided.
摘要翻译：公开了1,3-氧硫杂环戊烷核苷类似物及其药学上可接受的衍生物用于治疗乙型肝炎病毒感染的用途。还提供药物制剂。

2. 发明授权

US06790851B2 Fungicidal compositions 有权
标题翻译：杀真菌剂
公开(公告)号：US06790851B2
公开(公告)日：2004-09-14
申请号：US10258513
申请日：2003-03-11
申请人： Neil Leadbitter
发明人： Neil Leadbitter
IPC分类号： A01N4354
CPC分类号： A01N43/54 , A01N37/02 , A01N35/04 , A01N2300/00
摘要： The invention comprises a method of combating phytopathogenic diseases on crop plants which comprises applying to the crop plants or the locus thereof being infested with said phytopathogenic disease an effective amount of a combination of a) a benzophenone of formula I wherein R1 is methoxy, methyl, hydroxy, acetoxy or pivaloyloxy, R2 is C1-C4alkoxy or 2-halogenbenzyloxy, R3 is C1-C4alkoxy, R4 is C1-C4alkyl, halogen or trifluoromethyl, and R5 is hydrogen, halogen, C1-C4alkoxy, trifluoromethyl or nitro; in association with b) the strobilurin of formula II and a composition comprising fungicidally effective amounts of components I and II and a composition.
摘要翻译：本发明包括在作物植物上对抗植物病原性疾病的方法，其包括向作物植物或其受到所述植物病原性疾病侵袭的场所施用有效量的a）式I的二苯甲酮的组合，其中R1是甲氧基，甲基，羟基，乙酰氧基或新戊酰氧基，R 2是C 1 -C 4烷氧基或2-卤代苄氧基，R 3是C 1 -C 4烷氧基，R 4是C 1 -C 4烷基，卤素或三氟甲基，R 5是氢，卤素，C 1 -C 4烷氧基，三氟甲基或硝基; 与b）式II的嗜球果伞素和包含杀真菌有效量的组分I和II的组合物和组合物。

3. 发明授权

US06699874B2 Fungicidal mixtures 失效
标题翻译：杀菌混合物
公开(公告)号：US06699874B2
公开(公告)日：2004-03-02
申请号：US10314594
申请日：2002-12-10
申请人： Henry Van Tuyl Cotter , Leslie May , Gunter Reichert , Ewald Sieverding
发明人： Henry Van Tuyl Cotter , Leslie May , Gunter Reichert , Ewald Sieverding
IPC分类号： A01N4354
CPC分类号： A01N43/90 , A01N2300/00
摘要： Fungicidal compositions comprising an acceptable carrier and/or surface active agent and synergistically effective amounts of (a) at least one azolopyrimidine of formula I in which R1, R2, L1, L2 and L3 have the meaning given in claim 1; and (b) at least one fungicidal active ingredient selected from benomyl, carboxin, captan, chlorothalonil, copper oxychloride, cyprodinil, dimethomorph, dithianon, dodine, famoxadone, fenhexamid, fenpiclonil, fenpropimorph, fluazinam, mancozeb, metalaxyl, pyrimethanil, quinoxifen, sulfur, triforine, vinclozolin, a fungicidal triazole derivative, and a synthetic strobilurine derivative. The invention also provides a method of controlling the growth of phytopathogenic fungi at a locus by applying synergistically effective amounts of at least one azolopyrimidine of formula I and at least one fungicidal active ingredient (b) to the locus.
摘要翻译：包含可接受的载体和/或表面活性剂和协同有效量的（a）至少一种R 1，R 2，L 1，L 2和L 3的式Iin的偶氮嘧啶的杀真菌组合物 >具有权利要求1中给出的含义; 和（b）至少一种杀真菌活性成分，其选自苯菌灵，呋喃丹，克拉曼，百菌清，氯氧化铜，西酞替尼，烯酰吗啉，二噻吩，十二烷，恶唑酮，芬己酰，芬替尼，芬卡芬，氟啶胺，代森锰锌，甲霜灵，嘧霉胺，喹喔啉，，triperine，长春菌素，杀真菌三唑衍生物和合成次溴酸衍生物。本发明还提供了一种通过将协同有效量的至少一种式I的偶氮嘧啶和至少一种杀真菌活性成分（b）施用于该基因座来控制植物病原真菌在一个场所生长的方法。

4. 发明授权

US06511941B2 Herbicidal synergistic composition, and method of controlling weeds 失效
标题翻译：除草协同组合物及控制杂草的方法
公开(公告)号：US06511941B2
公开(公告)日：2003-01-28
申请号：US10058676
申请日：2002-01-29
申请人： Jean Louis Allard , Manfred Hudetz
发明人： Jean Louis Allard , Manfred Hudetz
IPC分类号： A01N4354
CPC分类号： A01N43/54 , A01N37/22 , A01N39/02 , A01N43/78 , A01N47/36 , A01N2300/00
摘要： A herbicidal synergistic composition, comprising, besides customary inert formulation auxiliaries, a compound of formula I and a synergistically active amount of at least one active ingredient selected from among the compounds of formula II in which A is a group X is —O—, —CH2— or —NH—; Y is OCH3; E is N; R1 is OC2H5, O(CH2)2OCH3
摘要翻译：一种除草协同组合物，除了常规惰性制剂助剂外，还包含式I化合物和协同活性量的至少一种活性成分，其选自式Ⅱ中其中A为基团X的至少一种活性成分是-O-，-CH 2 - 或 -NH-; Y是OCH 3; E是N; R 1是OC 2 H 5，O（CH 2）2 OCH 3

5. 发明授权

US06500836B1 Fungicidal active compound combinations 失效
标题翻译：杀真菌活性化合物组合
公开(公告)号：US06500836B1
公开(公告)日：2002-12-31
申请号：US10173409
申请日：2002-06-17
申请人： Klaus Stenzel , Wilhelm Brandes , Stefan Dutzmann , Bernd-Wieland Krüger , Karl-Heinz Kuck , Rolf Pontzen , Thomas Seitz , Atsumi Kamochi , Ikuya Saitoh
发明人： Klaus Stenzel , Wilhelm Brandes , Stefan Dutzmann , Bernd-Wieland Krüger , Karl-Heinz Kuck , Rolf Pontzen , Thomas Seitz , Atsumi Kamochi , Ikuya Saitoh
IPC分类号： A01N4354
CPC分类号： A01N37/24 , A01N61/00 , A01N47/44 , A01N47/12 , A01N43/90 , A01N43/653 , A01N43/54 , A01N43/40 , A01N43/36 , A01N43/30 , A01N41/02 , A01N37/50 , A01N2300/00
摘要： There are described new active compound combinations of a compound of the formula (I) with known fungicidal active compounds, and their use for combating phytopathogenic fungi.
摘要翻译：描述了式（I）化合物与已知的杀真菌活性化合物的新的活性化合物组合，以及它们用于对抗植物病原真菌的用途。

6. 发明授权

US06355645B2 Lipid-lowering quinazoline derivative 失效
标题翻译：降脂喹唑啉衍生物
公开(公告)号：US06355645B2
公开(公告)日：2002-03-12
申请号：US09756483
申请日：2001-01-08
申请人： Fatih M. Uckun , Vuong N. Trieu , Xing-Ping Liu
发明人： Fatih M. Uckun , Vuong N. Trieu , Xing-Ping Liu
IPC分类号： A01N4354
CPC分类号： C07D239/74
摘要： A novel carbonyl-substituted quinazoline, preferably 4-(3′-bromobenzoyl)-6,7-dimethoxyquinazoline (WHI-P164), and methods for lowering blood cholesterol, including reducing total cholesterol and LDL-cholesterol levels by administration of the carbonyl quinazolines and compositions thereof.

7. 发明授权

US06346535B1 Fungicidal mixtures 有权
公开(公告)号：US06346535B1
公开(公告)日：2002-02-12
申请号：US09240412
申请日：1999-01-29
申请人： Henry Van Tuyl Cotter , Gunther Reichert , Ewald Sieverding , Petrus Martinus Franciscus Emanuel Jegerings
发明人： Henry Van Tuyl Cotter , Gunther Reichert , Ewald Sieverding , Petrus Martinus Franciscus Emanuel Jegerings
IPC分类号： A01N4354
CPC分类号： A01N35/04 , A01N59/20 , A01N59/02 , A01N55/00 , A01N47/44 , A01N47/38 , A01N47/14 , A01N47/04 , A01N43/90 , A01N43/84 , A01N43/82 , A01N43/76 , A01N43/653 , A01N43/60 , A01N43/56 , A01N43/54 , A01N43/40 , A01N43/42 , A01N43/36 , A01N43/32 , A01N43/30 , A01N37/50 , A01N37/46 , A01N37/38 , A01N37/34 , A01N37/06 , A01N2300/00
摘要： The invention relates to a novel fungicidal composition comprising synergistically effective amounts of at least one benzophenone of formula I wherein R1 represents a halogen atom, an optionally substituted alkyl, alkanoyloxy or alkoxy group; or a hydroxy group, R2 represents a halogen atom or an optionally substituted alkyl group, R3 independently represents a halogen atom, an optionally substituted alkyl or alkoxy group or a nitro group; m is 0 or an integer of 1 to 3; R4 represents a halogen atom, a cyano, carboxy, hydroxy or nitro group or an optionally substituted alkyl, alkoxy, alkenyl, alkylthio, alkylsulphinyl, alkylsulphonyl or amino group; R5 represents an optionally substituted alkyl group; R6 represents a halogen atom or a nitro group, an optionally substituted alkyl, alkoxy, alkenyloxy, alkynyloxy, alkylthio, cycloalkyl, cycloalkyloxy, aryloxy group; R7 independently represents a halogen atom, an optionally substituted alkyl, alkenyl, alkynyl, alkoxy, alkenyloxy, alkynyloxy, cycloalkyl, cycloalkoxy group; n is 0 or 1; and at least one fungicidally active ingredient selected from the groups consisting of (A), (B), (C), (D) and (E) wherein: (A) is an ergosterol biosynthesis inhibitor; (B) is a strobilurine derivative, (C) is a melanin biosynthesis inhibitor; (D) is a compound selected from the group consisting of acibenzolar, benomyl, captan, carboxin, chlorothalonil, copper, cyprodinil, dinocap, dithianon, dimethomorph, dodine, ethirimol, famoxadone, fenpiclonil, fluazinam, mancozeb, metalaxyl, pyrifenox, sulfur, vinclozolin and (E) is an azolopyrimidine of formula II iwherein R8 and R9 each independently represent hydrogen or an optionally substituted alkyl, alkenyl, alkynyl, alkadienyl, aryl, heteroaryl, cycloalkyl, bicycloalkyl or heterocyclyl group, or R8 and R9 together with the interjacent nitrogen atom represent an optionally substituted heterocyclic ring, R10 represents hydrogen or an alkyl or aryl group, R11 represents a hydrogen or halogen atom or an alkyl or alkoxy group, L independently represents a halogen atom or an optionally substituted alkyl or alkoxy group, p is 0 or an integer from 1 to 5; and A represents N or CR2, wherein R12 has the meaning given for R10; together with a fungicidally acceptable carrier and/or surface active agent, and to a method of controlling the growth of phytopathogenic fungi which comprises applying synergistically effective amounts of the composition to the locus.

8. 发明授权

US06342499B1 Parasitic and saprophagous mite control in beneficial insects 失效
标题翻译：寄生虫和螨虫控制有益昆虫
公开(公告)号：US06342499B1
公开(公告)日：2002-01-29
申请号：US09352507
申请日：1999-07-12
申请人： Bruce Christian Black , William R. Baumbach , Michael P. Beluch
发明人： Bruce Christian Black , William R. Baumbach , Michael P. Beluch
IPC分类号： A01N4354
CPC分类号： A01N43/54 , A01K51/00
摘要： The present invention provides a method to control parasitic and saprophagous mites on beneficial insects such as honeybees via the application of a parasiticidally or saprophagouscidally effective amount of a mitochondrial electron transport inhibitor or a pyrimidine compound of formula I.
摘要翻译：本发明提供了一种通过施用杀虫剂或杀真菌有效量的线粒体电子传递抑制剂或式I的嘧啶化合物来控制有益昆虫例如蜜蜂的寄生虫和螨虫螨的方法。

9. 发明授权

US06316453B1 Aqueous pharmaceutical composition 有权
标题翻译：水性药物组合物
公开(公告)号：US06316453B1
公开(公告)日：2001-11-13
申请号：US09573504
申请日：2000-05-18
申请人： Peter Loeliger
发明人： Peter Loeliger
IPC分类号： A01N4354
CPC分类号： A61K31/506 , A61K9/0019 , A61K47/18 , Y10S514/97
摘要： Difficulties in preparing a stable pharmaceutical composition containing 5-Isopropyl-pyridine-2-sulfonic acid 6-(2-hydroxy-ethoxy)-5(2-methoxy-phenoxy)2-(2-1H-tetrazol-5-yl-pyridin-4yl)-pyrimidin-4-ylamide in form of the water soluble disodium salt, a buffer and preferably a metal complex forming agent, have been encountered. It was unexpectedly found that these difficulties can be overcome by adjusting the pH of the solution with an acid to over and above 8,2, preferably to 9,0, but not higher than 10.
摘要翻译：制备含有5-异丙基 - 吡啶-2-磺酸6-（2-羟基 - 乙氧基）-5（2-甲氧基 - 苯氧基）-2-（2-1H-四唑-5-基 - 吡啶）的稳定药物组合物困难 -4-基） - 嘧啶-4-基酰胺，其形式为水溶性二钠盐，缓冲剂，优选金属络合物形成剂。意外地发现，通过用酸调节溶液的pH超过和高于8,2，优选至9,0，但不高于10，可以克服这些困难。

10. 发明授权

US06281221B1 Substituted 1,3-dioxan-5-ylamino-hererocyclic compounds, processes for their preparation and their use as pest control compositions 失效
标题翻译：取代的1,3-二恶烷-5-基氨基 - 异环化合物，其制备方法及其作为害虫防治组合物的用途
公开(公告)号：US06281221B1
公开(公告)日：2001-08-28
申请号：US09161350
申请日：1998-09-25
申请人： Wolfgang Schaper , Werner Knauf , Ulrich Sanft , Manfred Kern , Heinz Ehrhardt , Adolf Heinz Linkies , Dieter Bernd Reuschling , Werner Bonin
发明人： Wolfgang Schaper , Werner Knauf , Ulrich Sanft , Manfred Kern , Heinz Ehrhardt , Adolf Heinz Linkies , Dieter Bernd Reuschling , Werner Bonin
IPC分类号： A01N4354
CPC分类号： C07D405/12 , A01N43/40 , A01N43/54 , C07F7/0812
摘要： The invention relates to novel substituted 1,3-dioxan-5-ylamino-heterocyclic compounds of the formula in which A is CH or N; X is NH, O or S(O)q, where q=0-2; Y is O or S(O)m, where m=0-2, and R1, R2, R3, R4, R4′ and R5 have the meanings given in the description, processes for their preparation and their use as pest control compositions and fungicides.
摘要翻译：本发明涉及A为CH或N的新型取代的1,3-二恶烷-5-基氨基 - 杂环化合物， X是NH，O或S（O）q，其中q = 0-2; Y是O或S（O）m，其中m = 0-2，并且R 1，R 2，R 3，R 4，R 4'和R 5具有本说明书中给出的含义，其制备方法及其作为害虫防治组合物的用途，杀菌剂。

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