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1. 发明授权

US4243660A Composite insect attractant for male cabbage moths and a process for preparing its active agents 失效
标题翻译：用于大白菜蛾的复合昆虫引诱剂及其活性剂的制备方法
公开(公告)号：US4243660A
公开(公告)日：1981-01-06
申请号：US31583
申请日：1979-04-19
申请人： Csaba Szantay , Lajos Novak , Miklos Toth , Jozsef Balla , Bela Stefko , Attila Kis-Tamas
发明人： Csaba Szantay , Lajos Novak , Miklos Toth , Jozsef Balla , Bela Stefko , Attila Kis-Tamas
IPC分类号： A01N37/02 , A01N49/00 , C07C29/10 , C07C41/30 , C07C43/15 , C07C43/17 , C07C69/145 , C07D309/12 , C07F9/54 , A01N25/00 , A01N37/06
CPC分类号： C07D309/12 , A01N37/02 , C07C29/10 , C07C41/30 , C07C43/15 , C07C43/17 , C07C67/08 , C07C67/293 , C07C69/145 , C07F9/5407
摘要： The invention relates to a composite insect attractant for male cabbage moths (Mamestra brassicae) containing (Z)-11-hexadecenyl acetate and (Z)-11-heptadecenyl acetate as active agents in a weight ratio of 70 to 90:80 to 1, optionally along with a liquid or solid adjuvant. An insect trap can contain the composition which is used for attracting and trapping cabbage moth. Their mating is disrupted by air permeation techniques. (Z)-11-heptadecenyl acetate is a synergistically active new compound. The composition according to the invention produces a significantly stronger stimulating reaction on male cabbage moths than the known sex lure compositions.
摘要翻译：本发明涉及含有（Z）-11-十六碳烯基乙酸酯和（Z）-11-十七碳烯酸乙酯作为活性剂的重量比为70至90:80至1的男性白菜蛾（Mamestra brassicae）的复合昆虫引诱剂，任选地与液体或固体佐剂一起。昆虫陷阱可以包含用于吸引和捕获白菜蛾的组合物。它们的交配被空气渗透技术所破坏。（Z）-11-十七碳烯酸乙酯是协同活性的新化合物。根据本发明的组合物比已知的性诱剂组合物对雄性白菜蛾产生显着更强的刺激反应。

2. 发明授权

US4364931A Composite insect attractant for male white-line dart moths and a process for preparing the active ingredients thereof 失效
标题翻译：用于雄性白线飞蛾的复合昆虫引诱剂及其活性成分的制备方法
公开(公告)号：US4364931A
公开(公告)日：1982-12-21
申请号：US220113
申请日：1980-12-24
申请人： Csaba Szantay , Lajos Novak , Miklos Toth , Jozsef Jakab , Attila Kis-Tamas , Istvan Ujvari
发明人： Csaba Szantay , Lajos Novak , Miklos Toth , Jozsef Jakab , Attila Kis-Tamas , Istvan Ujvari
IPC分类号： C07D471/04 , A01N37/02 , A61K31/519 , A61P29/00 , C07C29/147 , C07C69/145 , C07D303/42 , A01N17/14
CPC分类号： A01N37/02 , C07C29/147 , C07C67/08 , C07C67/293 , C07C67/343 , C07D303/42
摘要： The invention relates to a composite insect attractant for male white-line dart moths [Scotia segetum] containing 7[Z]-dodecen-l-ol acetate of the formula [I] ##STR1## and 9[Z]-tetradecen-l-ol acetate of the formula [II] ##STR2## as active agents in a weight ratio of I to II of [50-99]:[50-1], optionally along with a liquid or solid adjuvant.Another object of the invention is an insect trap containing said composition and a process for attracting and trapping male white-line dart moths as well as a process for disrupting their mating by air permeation technique. The invention relates further to a novel process for the preparation of the active ingredients of the composition.
摘要翻译：本发明涉及含有式[I]图7（I）的7 [Z] - 十一碳烯-1-醇乙酸酯和9 [Z]十四碳烯的男性白线镖飞蛾（Scotia segetum）的复合昆虫引诱剂（II）的1-乙酸乙酯作为活性剂，其重量比为[50-99]的I至II：[50-1]，任选与液体或固体佐剂一起使用。本发明的另一个目的是含有所述组合物的昆虫陷阱和用于吸引和捕获雄性白线飞镖的方法以及通过空气渗透技术破坏它们的交配的方法。本发明进一步涉及用于制备组合物的活性成分的新方法。

3. 发明授权

US4344959A Terpene derivatives and insecticidal compositions containing terpenes 失效
标题翻译：含有萜烯的萜烯衍生物和杀虫组合物
公开(公告)号：US4344959A
公开(公告)日：1982-08-17
申请号：US251043
申请日：1981-04-06
申请人： Lajos Novak , Csaba Szantay , Janos Rohaly , Attila Kis-Tamas , Laszlo Varjas , Janos Csutak
发明人： Lajos Novak , Csaba Szantay , Janos Rohaly , Attila Kis-Tamas , Laszlo Varjas , Janos Csutak
IPC分类号： C07C69/003 , A01N37/42 , A01N43/08 , A01N49/00 , C07D307/33 , C07D307/58 , A61K31/365 , A61K31/23 , C07D307/20
CPC分类号： C07D307/33 , A01N49/00 , C07D307/58
摘要： The invention relates to new compounds of the general formula (I), ##STR1## wherein R.sup.1 is hydrogen or a lower alkoxy group andZ.sup.1 is hydrogen, orR.sup.1 and Z.sup.1 form together a double bond,Z.sup.2 is hydrogen andB is hydroxy, orZ.sup.2 and B form together a double bond,Z.sup.3 and Z.sup.4 each stand for hydrogen or they form together an ethylene group, orZ.sup.4 and D form together a double bond,C is oxygen atom or a lower alkoxy group,D is a valence bond if C stands for oxygen, or otherwise D forms a double bond together with Z.sup.4 or Z.sup.5,Z.sup.5 forms a double bond together with D or represents hydrogen, andR.sup.2 is a group of the general formula --COOR.sup.3, wherein R.sup.3 is lower alkyl, orZ.sup.5 and R.sup.2 form together a 1-oxo-2-oxa-tetramethylene group, with the proviso that if Z.sup.3 and Z.sup.4 form together an ethylene group, R.sup.2 may stand only for a --COOR.sup.3 group,insecticidal compositions containing them, as well as to a process for their preparation.
摘要翻译：本发明涉及通式（I）的新化合物，其中R1是氢或低级烷氧基，Z1是氢，或R1和Z1一起形成双键，Z2是氢，B是羟基或Z 2和B一起形成双键，Z 3和Z 4各自代表氢或它们一起形成亚乙基，或Z 4和D一起形成双键，C是氧原子或低级烷氧基，D是如果C代表氧，则键合键，否则D与Z4或Z5一起形成双键，Z5与D一起形成双键或代表氢，R2是通式-COOR3的基团，其中R3是低级烷基，或Z5和R2一起形成1-氧代-2-氧杂 - 四亚甲基，条件是如果Z 3和Z 4一起形成亚乙基，则R2可以仅为-COOR 3基团，还含有它们的杀虫组合物关于他们的准备过程。

4. 发明授权

US6162923A Process for the preparation of imidazolones 有权
标题翻译：咪唑啉酮的制备方法
公开(公告)号：US6162923A
公开(公告)日：2000-12-19
申请号：US463433
申请日：2000-04-26
申请人： Csaba Huszar , Attila Kis-Tamas , Attila Nemeth , Antal Gajary , Lajosne Pali
发明人： Csaba Huszar , Attila Kis-Tamas , Attila Nemeth , Antal Gajary , Lajosne Pali
IPC分类号： C07D235/02
CPC分类号： C07D235/02
摘要： The present invention relates to a process for the preparation of a compound of general formula (I), ##STR1## wherein R.sup.1 represents a hydrogen atom or an alkyl group of 1-6 carbon atoms, and their salts, wherein the compound of formula (II): ##STR2## is reacted with a compound of formula (III): ##STR3## wherein R represents an alkyl group of 1-4 carbon atoms and R.sup.1 is the same as defined above, by heating their neutral pH mixtures at the boiling temperature of the mixture, and the resulting compound of general formula (IV): ##STR4## wherein R and R.sup.1 are the same as defined above, is cyclized into the compound of general formula (I) by further elevating the temperature of the neutral mixture, and if desired, the compounds of general formula (I) are transformed into their salts, or the compounds of general formula (I) are liberated from their salts.
摘要翻译： PCT No.PCT / HU98 / 00065 Sec。 371日期：2000年04月26日 102（e）日期2000年4月26日PCT提交1998年7月22日PCT公布。出版物WO99 / 05118 日期1999年2月4日本发明涉及制备通式（I）化合物的方法，其中R1表示氢原子或1-6个碳原子的烷基，及其盐，其中化合物式（II）：与式（III）化合物反应：其中R表示1-4个碳原子的烷基且R1与上述定义相同，通过在混合物的沸点温度下加热其中性pH混合物，并且通过进一步提高中性混合物的温度将所得到的通式（IV）化合物（其中R和R 1与上述定义相同）环化成通式（I）的化合物，如果需要，化合物通式（I）的化合物转化为它们的盐，或者通式（I）的化合物从其盐中释放出来。

5. 发明授权

US4740228A Plant growth regulating compounds and compositions and a process for the preparation thereof 失效
标题翻译：植物生长调节化合物和组合物及其制备方法
公开(公告)号：US4740228A
公开(公告)日：1988-04-26
申请号：US569594
申请日：1984-01-10
申请人： Attila Kis-Tamas , Ferenc Jurak , Zoltan Vig , Pal Fekete , Judit Kulcsar
发明人： Attila Kis-Tamas , Ferenc Jurak , Zoltan Vig , Pal Fekete , Judit Kulcsar
IPC分类号： A01N37/18 , A01N37/34 , A01N43/46 , A01P21/00 , A47B13/04 , C07C67/00 , C07C253/00 , C07C255/32 , C07C255/35 , C07C255/41 , C07C255/56 , C07C255/58 , C07D295/10 , C07D295/16 , C07D295/18 , A01N37/22 , A01N37/20
CPC分类号： C07C255/00 , A01N37/34
摘要： The invention relates to new plant growth regulating compositions, which contain as active agent 0.001 to 95% by weight of one or more compound(s) of the general formula (I), ##STR1## wherein R.sup.1 and R.sup.2 each represent hydrogen atom, a C.sub.1-5 alkyl group, a C.sub.5-7 cycloalkyl group, an aryl group, a halogen-substituted aryl group, an aralkyl group, a C.sub.2-5 alkenyl group or a C.sub.2-5 alkynyl group, orR.sup.1 and R.sup.2 form, together with the adjacent nitrogen atom, a morpholino, pyrrolidino, piperidino or perhydroazepinyl group, andR.sup.3 stands for hydrogen or a C.sub.1-5 alkyl group,together with an inert, solid, liquid and/or gaseous carrier or diluent, and optionally one or more additives, such as surfactants or other substances of plant biological activity.The compounds of the general formula (I) in which R.sup.1 is hydrogen and R.sup.2 stands for hydrogen, C.sub.1-3 alkyl, aralkyl or C.sub.3-5 alkenyl group, furthermore in which R.sup.1 and R.sup.3 are hydrogen and R.sup.2 is an aryl group have already been described in the literature, whereas the remaining derivatives of the general formula (I) are new. These compounds can be prepared by reacting a compound of the general formula (II) ##STR2## with an amine of the general formula (III), ##STR3## or by alkylating a compound of the general formula (IV). ##STR4## In the above formulae X stands for halogen, hydroxy or C.sub.1-4 alkoxy, whereas R.sup.1, R.sup.2 and R.sup.3 have the meanings as defined above.
摘要翻译：本发明涉及新的植物生长调节组合物，其含有0.001至95重量％的一种或多种通式（I）化合物，其中R 1和R 2各自表示氢的活性剂原子，C1-5烷基，C5-7环烷基，芳基，卤素取代的芳基，芳烷基，C2-5烯基或C2-5炔基，或R1和R2形式与相邻的氮原子一起形成吗啉代，吡咯烷子基，哌啶子基或全氢氮杂基，R3代表氢或C1-5烷基，与惰性，固体，液体和/或气态载体或稀释剂一起使用，或更多的添加剂，例如表面活性剂或植物生物活性的其它物质。其中R1是氢并且R2代表氢，C1-3烷基，芳烷基或C3-5烯基的通式（Ⅰ）化合物，此外R1和R3是氢，R2是芳基，文献中描述的，而通式（I）的剩余衍生物是新的。这些化合物可以通过使通式（II）的化合物（II）与通式（III）的胺，（IMAGE）（III）反应或通过烷基化通式（IV）的化合物）。（IV）在上式中，X表示卤素，羟基或C 1-4烷氧基，而R 1，R 2和R 3具有如上定义的含义。

6. 发明授权

US4425158A Bicyclo(2.2.1)heptane oximes used for plant growth regulating 失效
标题翻译：用于植物生长调节的双环（2.2.1）庚烷肟
公开(公告)号：US4425158A
公开(公告)日：1984-01-10
申请号：US322675
申请日：1981-11-18
申请人： Zoltan Budai , Attila Kis-Tamas , Tibor Mezei , Aranka Lay nee Konya , Zoltan Vigh , Agnes Sokorai nee Janki
发明人： Zoltan Budai , Attila Kis-Tamas , Tibor Mezei , Aranka Lay nee Konya , Zoltan Vigh , Agnes Sokorai nee Janki
IPC分类号： A01N33/24 , A01N33/04 , A01N35/10 , A01P21/00 , C07C251/44 , C07C251/50
CPC分类号： A01N35/10
摘要： The invention relates to new bicyclo(2.2.1)heptane derivatives of the general formula I ##STR1## wherein R represents a C.sub.1-12 alkyl group optionally substituted by a lower alkoxy group, a C.sub.2-4 alkenyl group or a phenyl-(lower alkyl) group optionally substituted on the phenyl ring by one or more lower alkoxy groups or halogen atoms.The invention relates further to plant growth regulating compositions comprising as active agent 0.001 to 95% by weight of a racemic and/or optically active compound of the general formula I, wherein R has the above defined meanings, along with a conventional organic or inorganic, solid and/or liquid carrier and/or filler and/or diluent and/or surfactant.The invention encompasses also the preparation of the compounds of the general formula I which comprises reacting a racemic or optically active compound of the general formula II ##STR2## wherein Y is an oxygen or sulfur atom or an oxim group, with a compund of the general formula IIIR - XwhereinR is as defined above, andX represents a leaving group, preferably a halogen atom, a sulfonyloxy or an aminooxy group, with the proviso that when using a compound of the general formula II, in which Y is an oxim group, X is other than aminooxy group,in the presence of a basic condensing agent, and optionally resolving the racemic compound of the general formula I obtained into its optically active antipodes.
摘要翻译：本发明涉及通式I的新的双环（2.2.1）庚烷衍生物，其中R表示任选被低级烷氧基，C 2-4链烯基或苯基 - （低级烷基）基团，其任选在苯环上被一个或多个低级烷氧基或卤素原子取代。本发明进一步涉及植物生长调节组合物，其包含作为活性剂0.001至95重量％的通式I的外消旋和/或旋光活性化合物，其中R具有上述定义的含义，以及常规的有机或无机，固体和/或液体载体和/或填料和/或稀释剂和/或表面活性剂。本发明还包括通式I的化合物的制备，其包括使通式II的外消旋或旋光活性化合物其中Y是氧或硫原子或肟基，与下列化合物反应：通式III R-X其中R如上定义，X表示离去基团，优选卤素原子，磺酰氧基或氨基氧基，条件是当使用通式II的化合物时，其中Y为肟基，X不是氨基氧基，在碱性缩合剂的存在下，并且任选地将所得通式I的外消旋化合物拆分成其光学活性对映体。

7. 发明授权

US4469703A Nitroalkanol derivatives and plant protecting agents containing the same 失效
标题翻译：硝基链烷醇衍生物和含有它们的植物保护剂
公开(公告)号：US4469703A
公开(公告)日：1984-09-04
申请号：US350570
申请日：1982-02-22
申请人： Attila Kis-Tamas , Gyula Mikite , Erzsebet Csutak nee Jakucs , Laszlo Kocsis
发明人： Attila Kis-Tamas , Gyula Mikite , Erzsebet Csutak nee Jakucs , Laszlo Kocsis
IPC分类号： C07D317/52 , A01N37/02 , A01N37/10 , A01N37/12 , A01N43/06 , A01N43/08 , A01N43/30 , C07C67/00 , C07C201/00 , C07C205/40 , C07C205/42 , C07C205/45 , C07D307/42 , C07D307/45 , C07D307/70 , C07D317/32 , C07D317/54 , A01N37/06 , A01N43/16 , C07C67/02
CPC分类号： C07C205/42 , C07C205/40
摘要： The invention relates to nitroalkanol derivatives of the general formula (I), ##STR1## wherein R.sub.1 is a C.sub.2-12 alkenyl or alkadienyl group, a C.sub.4-12 alkoxyalkyl or alkoxyalkenyl group having one or more C.sub.1-3 alkyl substituents, a C.sub.3-6 cycloalkyl or cycloalkenyl group, a furyl group, a nitrofuryl group, or a phenyl group having optionally one or more identical or different substituents selected from the group consisting of hydroxy, C.sub.1-4 alkoxy, halogen, nitro, C.sub.1-4 alkylenedioxy and C.sub.1-4 alkenoyloxy groups,R.sub.2 and R.sub.4 each represent hydrogen or they form together a valence bond,R.sub.3 is a C.sub.1-12 alkanoyloxy group, a benzoyloxy group having optionally one or more halogen substituents or hydrogen atom, andR.sub.5 is a C.sub.1-12 alkyl group or a phenyl group having optionally one or more halogen substituents,with the proviso that if R.sub.2 and R.sub.4 each stand for hydrogen, R.sub.1 is other than unsubstituted phenyl and R.sub.3 may represent only a C.sub.1-4 alkanoyloxy group or a benzoyloxy group having optionally one or more halogen substituents, and with the further proviso that if R.sub.2 and R.sub.4 form together a valence bond and R.sub.5 is methyl, R.sub.1 is other than unsubstituted phenyl.The nitroalkenol derivatives defined above as well as the known 1-phenyl-2-nitro-3-acetoxy-propane-1 possess valuable pesticidal effects, primarily fungicidal activities, and can be applied to advantage in the agriculture as plant protecting agents.
摘要翻译：本发明涉及通式（I）的硝基链烷醇衍生物，其中R1是C2-12链烯基或链二烯基，具有一个或多个C 1-3烷基取代基的C 4-12烷氧基烷基或烷氧基烯基， C 3-6环烷基或环烯基，呋喃基，硝基呋喃基或具有任选一个或多个相同或不同取代基的苯基，所述取代基选自羟基，C 1-4烷氧基，卤素，硝基，C 1-4 亚烷基二氧基和C 1-4烯酰氧基，R 2和R 4各自表示氢或它们一起形成价键，R 3是C 1-12烷酰氧基，具有任选一个或多个卤素取代基或氢原子的苯甲酰氧基，R 5是C 1 -12烷基或具有任选一个或多个卤素取代基的苯基，条件是如果R 2和R 4各自代表氢，则R 1不是未取代的苯基，并且R 3可以仅表示C 1-4烷酰氧基或苯甲酰氧基任选地一个或更多的卤素取代基，进一步的条件是如果R 2和R 4一起形成一个价键，R 5是甲基，则R 1不是未取代的苯基。上述硝基烯醇衍生物以及已知的1-苯基-2-硝基-3-乙酰氧基 - 丙烷-1具有有价值的杀虫作用，主要是杀真菌活性，可作为植物保护剂在农业中有利地应用。

8. 发明授权

US4244888A Plant growth regulating and insecticidal compositions 失效
标题翻译：植物生长调节和杀虫组合物
公开(公告)号：US4244888A
公开(公告)日：1981-01-13
申请号：US65156
申请日：1979-08-09
申请人： Zoltan Budai , Ferenc Jurak , Attila Kis-Tamas , Aranka Lay nee Konya , Tibor Mezei , Zoltan Vig , Terez Zubovits nee Kristof
发明人： Zoltan Budai , Ferenc Jurak , Attila Kis-Tamas , Aranka Lay nee Konya , Tibor Mezei , Zoltan Vig , Terez Zubovits nee Kristof
IPC分类号： A01N33/24 , A01N35/10 , C07C249/04 , C07C251/44 , C07C131/02
CPC分类号： A01N35/10
摘要： Racemic or optically active 2-(propargyloxyimino)-1,7,7-trimethyl-bicyclo[2,2,1]heptane of the formula (I) ##STR1## or a mixture of these isomers is prepared by reacting a racemic or optically active 1,7,7-trimethyl-bicyclo[2,2,1]heptane derivative of the general formula (II), ##STR2## wherein Y stands for oxygen atom, sulfur atom or oxime group, with a propyne derivative of the general formula (III),R--CH.sub.2 --C.tbd.CH (III) whereinR stands for halogen atom or aminooxy group, with the proviso that if Y represents oxime group, R may stand only for halogen, and if R represents aminooxy group, Y may stand only for oxygen or sulfur atom.The resulting product is new and possesses strong plant growth promoting and insecticidal effects.
摘要翻译：式（I）的外消旋或光学活性的2-（炔丙氧基亚氨基）-1,7,7-三甲基 - 双环[2,2,1]庚烷或其混合物可以通过使外消旋或光学活性的通式（II）的17,7-三甲基 - 双环[2,2,1]庚烷衍生物，其中Y代表氧原子，硫原子或肟基，其中通式（III）的丙炔衍生物，其中R代表卤素原子或氨基氧基的R-CH 2 -C 3 CHCH（III），条件是如果Y表示肟基，则R可以仅为卤素，如果 R表示氨基氧基，Y可以仅为氧或硫原子。产生的产品是新的，具有很强的植物生长促进和杀虫作用。

9. 发明授权

US4588435A N-substituted amino propane sulfonic acid derivatives and plant growth regulating use 失效
标题翻译： N-取代氨基丙磺酸衍生物和植物生长调节用途
公开(公告)号：US4588435A
公开(公告)日：1986-05-13
申请号：US696658
申请日：1985-01-31
申请人： Zoltan Budai , Attila Kis-Tamas , Aranka Lay nee Konya , Zoltan Vig , Viktor Andriska , Tibor Mezei
发明人： Zoltan Budai , Attila Kis-Tamas , Aranka Lay nee Konya , Zoltan Vig , Viktor Andriska , Tibor Mezei
IPC分类号： A01N37/18 , A01N41/04 , A01N43/08 , A01P21/00 , C07C67/00 , C07C301/00 , C07C303/22 , C07C303/32 , C07C309/15 , C07D307/68 , A01N37/22 , C07C143/63
CPC分类号： A01N41/04 , A01N43/08
摘要： The invention relates to new N-substituted amino propane sulfonic acid derivatives of the Formula I ##STR1## and salts and hydrates thereof, a process for the preparation thereof and plant growth regulating agents comprising the same whereinR.sup.1 and R.sup.2 may be identical or different and stand for hydrogen, halogen, lower alkyl or lower alkoxy andR stands for furyl; or lower alkyl or phenyl the two latter groups being optionally substituted by one or more halogeno atom(s).
摘要翻译：本发明涉及式I的新的N-取代氨基丙磺酸衍生物及其盐及其水合物，其制备方法和包含其的植物生长调节剂，其中R1和R2可以相同或不同代表氢，卤素，低级烷基或低级烷氧基，R代表呋喃基; 或低级烷基或苯基，后两个基团任选被一个或多个卤素原子取代。

10. 发明授权

US4511737A Bicyclo(2.2.1)heptane oximes 失效
标题翻译：双环（2.2.1）庚烷肟
公开(公告)号：US4511737A
公开(公告)日：1985-04-16
申请号：US551941
申请日：1983-11-15
申请人： Zoltan Budai , Attila Kis-Tamas , Tibor Mezei , Aranka Lay , Zoltan Vigh , Agnes Sokorai
发明人： Zoltan Budai , Attila Kis-Tamas , Tibor Mezei , Aranka Lay , Zoltan Vigh , Agnes Sokorai
IPC分类号： A01N33/24 , A01N33/04 , A01N35/10 , A01P21/00 , C07C251/44 , C07C251/50 , C07C131/02
CPC分类号： A01N35/10
摘要： The invention relates to new bicyclo(2.2.1)heptane derivatives of the general formula I ##STR1## wherein R represents a C.sub.1-12 alkyl group optionally substituted by a lower alkoxy group, a C.sub.2-4 alkenyl group or a phenyl-(lower alkyl) group optionally substituted on (I), phenyl ring by one or more lower alkoxy groups or halogen atoms.The invention relates further to plant growth regulating compositions comprising as active agent 0.001 to 95% by weight of a racemic and/or optically active compound of the general formula I, wherein R has the above defined meanings, along with a conventional organic or inorganic, solid and/or liquid carrier and/or filler and/or diluent and/or surfactant.The invention encompasses also the preparation of the compounds of the general formula (I) which comprises reacting a racemic or optically active compound of the general formula (II) ##STR2## wherein Y is an oxygen or sulfur atom or an oxim group, with a compound of the general formula (III)R--XwhereinR is as defined above, andX represents a leaving group, preferably a halogen atom, a sulfonyloxy or an aminooxy group, with the proviso that when using a compound of the general formula (II), in which Y is an oxim group, X is other than aminooxy group,in the presence of a basic condensing agent, and optionally resolving the racemic compound of the general formula (I) obtained into its optically active antipodes.
摘要翻译：本发明涉及通式I（I）的新型双环（2.2.1）庚烷衍生物，其中R表示任选被低级烷氧基取代的C 1-12烷基，C 2-4链烯基或苯基 - （低级烷基）基团，其任选地在（I）上取代，苯基环由一个或多个低级烷氧基或卤素原子取代。本发明进一步涉及植物生长调节组合物，其包含作为活性剂0.001至95重量％的通式I的外消旋和/或旋光活性化合物，其中R具有上述定义的含义，以及常规的有机或无机，固体和/或液体载体和/或填料和/或稀释剂和/或表面活性剂。本发明还包括通式（I）的化合物的制备，其包括使通式（II）的外消旋或光学活性化合物其中Y是氧或硫原子或肟基的（II）与通式（III）RX的化合物，其中R如上定义，X表示离去基团，优选卤素原子，磺酰氧基或氨基氧基，条件是当使用通式（II），其中Y是肟基，X不是氨基氧基，在碱性缩合剂的存在下，并且任选地将通式（I）的外消旋化合物拆分成其光学活性对映体。

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