专利快速检索-快速检索全球专利，免费商用专利数据库-IPRDB

1. 发明申请

WO2003075875A1 UV ABSORBER COMPOSITIONS COMPRISING A HYDROXYPHENYLTRIAZINE COMPOUND 审中-公开
标题翻译：含有羟基苯乙烯化合物的紫外线吸收剂组合物
公开(公告)号：WO2003075875A1
公开(公告)日：2003-09-18
申请号：PCT/EP2003/002200
申请日：2003-03-04
申请人： CIBA SPECIALTY CHEMICALS HOLDING INC. , HAASE, Jürg , EHLIS, Thomas , BORSOS, Elek , HÜGLIN, Dietmar , HERZOG, Bernd
发明人： HAASE, Jürg , EHLIS, Thomas , BORSOS, Elek , HÜGLIN, Dietmar , HERZOG, Bernd
IPC分类号： A61K7/42
CPC分类号： A61K8/4966 , A61Q17/04
摘要： UV absorber compositions are described, comprising (a) from 1 to 99 % by weight of a hydroxyphenyltriazine compound of formula (I) wherein R 1 , R 2 and R 3 are each independently of the others C 1 -C 18 alkyl; C 2 -C 10 ,alkenyl; or phenyl-C,-C 4 alkyl; R 4 is hydrogen; or C 1 -C 5 alkyl; and (b) from 99 to 1 % by weight of a further UV absorber selected from the group of (b) hydroxyphenyltriazines that are different from component (a), (b 2 ) benzotriazoles, (b 3 ) dibenzoylmethane derivatives and (b 4 ) camphor derivatives. The compositions are suitable as UV filters in cosmetic compositions.
摘要翻译：描述了紫外线吸收剂组合物，其包含（a）1至99重量％的式（I）的羟基苯基三嗪化合物，其中R 1，R 2和R 3各自独立地为C 1 -C 18烷基; C2-C10烯基; 或苯基-C 1 -C 4烷基; R4是氢; 或C 1 -C 5烷基; 和（b）99重量％至1重量％的另外的紫外线吸收剂，其选自（b）不同于组分（a），（b 2）苯并三唑，（b3）二苯甲酰甲烷衍生物和（b4）樟脑）的羟苯基三嗪衍生物。该组合物适用于化妆品组合物中的UV过滤器。

2. 发明申请

WO2004052837A2 AMINO SUBSTITUTED HYDROXYPHENYL BENZOPHENONE DERIVATIVES 审中-公开
标题翻译：氨基取代的羟基苯并噻吩酮衍生物
公开(公告)号：WO2004052837A2
公开(公告)日：2004-06-24
申请号：PCT/EP2003/050937
申请日：2003-12-03
申请人： CIBA SPECIALTY CHEMICALS HOLDING INC. , HAASE, Jürg , EHLIS, Thomas , BORSOS, Elek , MÜLLER, Stefan
发明人： HAASE, Jürg , EHLIS, Thomas , BORSOS, Elek , MÜLLER, Stefan
IPC分类号： C07C229/52
CPC分类号： C07D295/192 , A61K8/42 , A61K8/44 , A61K8/49 , A61K8/4973 , A61Q17/04 , C07C229/52 , C07C237/32 , C07C237/34 , C07C237/40 , C07C237/42 , C07D277/46 , C07D277/66 , C07D313/12
摘要： Described are amino substituted hydroxyphenyl benzophenone derivatives of formula (I), wherein R 1 , and R 2 independently from each other are; C 1 ,-C 20 alkyl; C 2 -C 20 alkenyl; C 3 -C 10 ,cycloalkyl; C 3 -C 10 cycloalkenyl; or R 1 , and R 2 together with the linking nitogen atom form a 5- or 6-membered heterocyclic ring; n 1 is a number from 1 to 4; when n 1 =1, R 3 is a saturated or unsaturated heterocyclic radical; hydroxy-C 1 -C 5 alkyl; cyclohexyl optionally substituted with one or more C 1 ,-C 5 alkyl; phenyl optionally substituted with a heterocyclic radical, aminocarbonyl or C 1 -C 5 alkylcarboxy; wenn n 1 is 2, R 3 is an alkylene-, cycloalkylene- or alkenylene radical which is optionally substituted by a carbonyl- or carboxy group; o R 3 together with A forms a bivalent radical of the formula (Ia), wherein n 2 is a number from 1 to 3; when n 1 is 3, R 3 is an alkanetriyl radical; wenn n 1 is 4, R 3 is an alkanetetrayl radical; A is -O-; or -N(R 5 )-; and R 5 is hydrogen; C 1 -C 5 alkyl; or hydroxy-C 1 -C 5 alkyl. The compounds are useful as UV filters in sunscreen applications.
摘要翻译：描述了式（I）的氨基取代的羟基苯基二苯甲酮衍生物，其中R1和R2彼此独立地是; C1，-C20alkyl; C2-C20alkenyl; C3-C10，环烷基; C3-C10cycloalkenyl; 或R1和R2与连接的硝原子一起形成5-或6-元杂环; n1是从1到4的数字; 当n1 = 1时，R3是饱和或不饱和杂环基; 羟基C1-C5烷基; 任选被一个或多个C 1 -C 5烷基取代的环己基; 任选被杂环基取代的苯基，氨基羰基或C 1 -C 5烷基羧基; wn1是2，R3是任选被羰基或羧基取代的亚烷基，亚环烷基或亚烯基; O与A一起形成式（Ia）的二价基团，其中n2为1至3的数; 当n1为3时，R3为烷三基; wenn n1为4，R3为烷基四氢呋喃基; A为-O- 或-N（R 5） - ; R5是氢; C1-C5烷基; 或羟基-C 1 -C 5烷基。这些化合物可用作防晒霜中的紫外线过滤器。

3. 发明申请

WO2006003094A2 MEROCYANINE DERIVATIVES 审中-公开
公开(公告)号：WO2006003094A2
公开(公告)日：2006-01-12
申请号：PCT/EP2005/052850
申请日：2005-06-20
申请人： CIBA SPECIALTY CHEMICALS HOLDING INC. , WAGNER, Barbara , BIENEWALD, Frank , WOLLEB, Heinz , WALLQUIST, Olof , HERZOG, Bernd , EHLIS, Thomas , HAASE, Jürg
发明人： WAGNER, Barbara , BIENEWALD, Frank , WOLLEB, Heinz , WALLQUIST, Olof , HERZOG, Bernd , EHLIS, Thomas , HAASE, Jürg
IPC分类号： A61K7/42
CPC分类号： A61K8/498 , A61K8/4913 , A61K8/494 , A61Q17/04
摘要： Disclosed is the use of merocyanine derivatives of formula (I), wherein Q is hydrogen; C 1 -C 22 alkyl; -OH; -OR 7 ; -NR 7 R 8 ; or -N=R 9 ; R 1 is hydrogen; C 1 -C 22 alkyl; -OR 7 , -SR 7 ; -NR 7 R 8 ; C 1 -C 22 alkyl; C 2 -C 12 alkenyl; C 2 -C 12 alkinyl; C 3 -C 12 cycloalkyl; C 3 -C 12 cycloalkenyl; C 7 -C 12 aralkyl; C 1 -C 12 heteroalkyl, C 2 -C 11 heteroaralkyl; C 6 -C 10 aryl; or C 1 -C 9 heteroaryl; R 4 is cyano; COR 7 , COOR 7 ; CONR 7 R 8 ; SO 2 (C 6 -C 12 )aryl; C 2 -C 12 alk-1-enyl; C 3 -C 12 cycloalk-1-enyl; C 2 -C 12 alk-1-inyl; C 2 -C 12 heteroalkyl; C 3 -C 5 heterocycloalkyl; C 6 -C 10 aryl; or C 1 -C 9 heteroaryl; R 5 is -COR 7 ; -COOR 7 ; -OR 7 ; -SR 7 , -NHR 7 , -NR 7 R 8 ; C 1 -C 22 alkyl; C 2 -C 12 alkenyl; C 2 -C 12 alkinyl; C 3 -C 12 cycloalkyl; C 3 -C 12 cycloalkenyl; C 7 -C 12 aralkyl; C 1 -C 12 alkylphenyl; C 1 -C 12 alkoxy-C 6 -C 10 aryl; C 1 -C 12 heteroalkyl; C 2 -C 11 heteroaralkyl; C 3 -C 12 cycloheteroalkyl; C 6 -C 10 aryl; C 1 - C 12 alkoxy-C 6 -C 10 aryl; or C 1 -C 9 heteroaryl; R 6 is hydrogen; C 1 -C 22 alkyl; C 1 -C 22 alkoxy; or COR 7 ; R 7 and R 8 independently from each other are hydrogen; C 1 -C 22 alkyl; C 2 -C 12 alkenyl; C 2 -C 12 alkinyl; C 3 -C 12 cycloalkyl; C 3 -C 12 cycloalkenyl; -(CH 2 ) t COOH; C 7 -C 12 aralkyl; C 1 -C 12 heteroalkyl; C 2 -C 11 heteroaralkyl; C 6 -C 10 aryl; C 1 -C 9 heteroaryl; Si-R 10 R 11 R 12 ; Si(OR 10 )(OR 11 )(OR 12 ); SiR 10 (OR 11 )(OR 12 ); SiR 10 R 11 (OR 12 ); -(CH 2 ) u -O-(CH 2 ) v -SiR 10 R 11 R 12 ; or a radical X-Sil; t, u and v, independently from each other are a number from 1 to 5; R 9 is a (C 1 -C 6 )alkylidene radical; R 10 , R 11 , R 12 independently form each other are C 1 -C 22 alkyl; X is a linker; Sil is a silane-, oligosiloxane- or polysiloxane radical; R 1 and R 2 , R 1 and Q, R 1 and R 6 , R 1 and T, R 2 and R 3 , R 2 and R 4 , R 2 and R 6 , R 2 and Q, R 4 and R 6 , R 4 and T, R 6 and Q, T and Q, each independently, are linked together, so that 1, 2, 3 or 4 carbocyclic or N, O and/or S-heterocyclic rings are formed, wherein each of them, independently from each other, may be condensed with an aromatic or heteroaromatic ring, and/or more N-, O- and/or S-heterocyclic rings, and each N atom in a N-heterocyclic ring may be substituted by C 1 -C 22 alkyl; n is a number from 1 to 4; wherein at least one of the radicals R 1 , R 6 or Q is different from hydrogen; if n = 1 T is -COR 5 ; -CN; C 6 -C 10 aryl; -NHR 5 ; or -SO 2 -(C 6 -C 12 )aryl; R 2 and R 3 independently from each other are C 1 -C 22 alkyl; hydroxy-C 1 -C 22 alkyl; C 2 -C 12 alkenyl; C 2 -C 12 alkinyl; C 3 -C 12 cycloalkyl, C 3 -C 12 cycloalkenyl; C 7 -C 12 aralkyl; C 1 -C 12 heteroalkyl; C 3 -C 12 cycloheteroalkyl; C 6 -C 10 aryl; C 1 -C 9 heteroaryl; or a radical of formula (II); p is a number from 5 to 100; q is a number from 1 to 5; s is a number from 0 to 4; if n = 2 R 2 and R 3 are each C 1 -C 5 alkylene; and simultaneously T is defined as for n = 1; or T is a bivalent radical of formula -NR 7 -V-NR 7 -, wherin V is phenylene; or C 1 -C 5 alkylene; R 7 is hydrogen; or C 1 -C 5 alkyl; and R 2 and R 3 simultaneously are defined as for n = 1; if n = 3 one of R 2 , R 3 or T is a trivalent radical; if n = 4 one of R 2 , R 3 or T is a tetravalent radical; for protecting of human hair and skin against the damaging effect of UV radiation.

4. 发明申请

WO2007071584A2 USE OF TRANSMISSION DYES 审中-公开
标题翻译：使用传染性染色体
公开(公告)号：WO2007071584A2
公开(公告)日：2007-06-28
申请号：PCT/EP2006/069519
申请日：2006-12-11
申请人： CIBA SPECIALTY CHEMICALS HOLDING INC. , MÜLLER, Stefan , HAASE, Jürg , EHLIS, Thomas , KREYER, Gilbert , GIESINGER, Jochen , VOGT, Martin
发明人： MÜLLER, Stefan , HAASE, Jürg , EHLIS, Thomas , KREYER, Gilbert , GIESINGER, Jochen , VOGT, Martin
CPC分类号： C07D295/192 , A61K8/411 , A61K8/42 , A61K8/49 , A61K8/494 , A61K2800/43 , A61Q17/04
摘要： Disclosed is the use of an aqueous dispersion comprising (a) a micronized sparingly soluble organic compound which has a UV-Vis spectrum with a maximum from 380 to 420 nm; and (b) an anionic dispersing agent for protecting the human skin from browning and skin aging.
摘要翻译：公开了包含（a）微波化的微溶有机化合物的水分散体的使用，其具有最大值为380至420nm的UV-Vis光谱; 和（b）用于保护人体皮肤免于褐变和皮肤老化的阴离子分散剂。

5. 发明申请

WO2007090832A1 HYDROXYBENZOPHENONE DERIVATIVES 审中-公开
标题翻译：羟基苯并噻吩衍生物
公开(公告)号：WO2007090832A1
公开(公告)日：2007-08-16
申请号：PCT/EP2007/051117
申请日：2007-02-06
申请人： CIBA SPECIALTY CHEMICALS HOLDING INC. , HAASE, Jürg , MÜLLER, Stefan , EHLIS, Thomas
发明人： HAASE, Jürg , MÜLLER, Stefan , EHLIS, Thomas
IPC分类号： C07F7/08 , A61Q17/04 , A61K8/58
CPC分类号： C07F7/0854 , A61K8/585 , A61Q17/04
摘要： Disclosed are hydroxyphenylbenzophenone derivatives of formula (1), wherein R 1 and R 2 independently from each other are hydrogen; C 1 -C 20 alkenyl; C 3 - C 10 cycloalkyl; or R 1 and R 2 together with the linking nitrogen atom form a 5- 6-membered heterocyclic ring; R 3 , R 4 and R 5 independently from each other are C 1 -C 4 alkyl; C 1 -C 4 alkoxy; or a radical of formula (1a) R 6 is C 1 -C 6 alkyl; and A is a straight-chain or branched C 3 -C 6 alkylene, which is optionally interrupted by one or more *-O-*, or *-O-(CO)-* groups; and m is 0; or anumber from 1 to 5. The compounds are useful as cosmetic UV filters with outstanding solubility properties in cosmetic oils.
摘要翻译：公开了式（1）的羟基苯基二苯甲酮衍生物，其中R 1和R 2彼此独立地是氢; ç_{1 -C _{20 烯基; C 3 -C 10环烷基; 或R 1和R 2与连接氮原子一起形成5-6元杂环; R 3，R 4和R 5彼此独立地是C 1 -C 4烷基， / SUB>烷基; ç_{1 -C _{4 烷氧基; 或式（1a）的基团R 6是C 1 -C 6烷基; 并且A是直链或支链C 3 -C 6亚烷基，其任选地被一个或多个* -O- *或* -O-（ CO） - *组; m为0; 或1至5的编号。该化合物可用作化妆品油中具有优异溶解性的化妆品UV过滤器。}}}}

6. 发明申请

WO2008135421A2 CRYSTAL MODIFICATIONS OF TRANSMISSION DYES 审中-公开
标题翻译：传染性染色体的晶体修饰
公开(公告)号：WO2008135421A2
公开(公告)日：2008-11-13
申请号：PCT/EP2008/055139
申请日：2008-04-28
申请人： CIBA HOLDING INC. , VOGT, Martin , MÜLLER, Stefan , GRUMELARD, Julie , DESHAYES, Cyrille , PAUL, Holger , HAASE, Jürg , EHLIS, Thomas
发明人： VOGT, Martin , MÜLLER, Stefan , GRUMELARD, Julie , DESHAYES, Cyrille , PAUL, Holger , HAASE, Jürg , EHLIS, Thomas
IPC分类号： A61K8/49 , A61Q17/04 , A61Q19/08
CPC分类号： C07D295/192 , A61K8/04 , A61K8/494 , A61K31/495 , A61Q17/04 , A61Q19/00 , A61Q19/08 , A61K2300/00
摘要： Disclosed is the use of an aqueous dispersion comprising (a) a micronized sparingly soluble organic benzophenone derivative of formula (1), selected from the crystal modifications (B) and (C), wherein the crystal modification (B) is characterized by a peak in the X-ray diffraction pattern at a d-spacing of about 7.70 Å; and wherein the crystal modification (C) is characterized by a peak in the X-ray diffraction pattern at a d-spacing of about 7.06 Å; and (b) a dispersing agent selected from anionic, non-ionic and amphoteric surfactants; for protecting the human skin from browning and skin aging. The new crystal modification (C) represents a thermodynamically stable compound of formula (1) at 25°C. This modification is therefore suitable in dispersions comprising micro-fine particles.
摘要翻译：公开了含有（a）选自结晶改性物（B）和（C）的式（1）的微粉化的微溶有机二苯甲酮衍生物的水性分散体的用途，其中所述结晶改性（B）的特征在于峰在X射线衍射图中，d-间距约为7.70; 并且其中所述晶体改性（C）的特征在于在约7.06的d间距处的X射线衍射图中的峰; 和（b）选自阴离子，非离子和两性表面活性剂的分散剂; 用于保护人体皮肤免受褐变和皮肤老化。新的结晶改性（C）在25℃下代表热力学稳定的式（1）化合物。因此，该修饰适用于包含微细颗粒的分散体。

7. 发明公开

EP1761237A2 MEROCYANINE DERIVATIVES 审中-公开
标题翻译：部花青衍
公开(公告)号：EP1761237A2
公开(公告)日：2007-03-14
申请号：EP05756874.3
申请日：2005-06-20
申请人： Ciba Specialty Chemicals Holding Inc.
发明人： WAGNER, Barbara , BIENEWALD, Frank , WOLLEB, Heinz , WALLQUIST, Olof , HERZOG, Bernd , EHLIS, Thomas , HAASE, Jürg
IPC分类号： A61K8/35
CPC分类号： A61K8/498 , A61K8/4913 , A61K8/494 , A61Q17/04
摘要： Disclosed is the use of merocyanine derivatives of formula (I) for protecting of human hair and skin against the damaging effect of UV radiation.

8. 发明授权

EP1482904B1 UV ABSORBER COMPOSITIONS COMPRISING A HYDROXYPHENYLTRIAZINE COMPOUND 有权转让
标题翻译： UV吸收组合物含羟苯基
公开(公告)号：EP1482904B1
公开(公告)日：2008-04-02
申请号：EP03709744.1
申请日：2003-03-04
申请人： Ciba Specialty Chemicals Holding Inc.
发明人： HAASE, Jürg , EHLIS, Thomas , BORSOS, Elek , HÜGLIN, Dietmar , HERZOG, Bernd
IPC分类号： A61Q17/04 , A61K8/49
CPC分类号： A61K8/4966 , A61Q17/04
摘要： UV absorber compositions are described, comprising (a) from 1 to 99 % by weight of a hydroxyphenyltriazine compound of formula (I) wherein R1, R2 and R3 are each independently of the others C1-C18alkyl; C2-C10,alkenyl; or phenyl-C,-C4 alkyl; R4 is hydrogen; or C1-C5alkyl; and (b) from 99 to 1 % by weight of a further UV absorber selected from the group of (b) hydroxyphenyltriazines that are different from component (a), (b 2) benzotriazoles, (b3) dibenzoylmethane derivatives and (b4) camphor derivatives. The compositions are suitable as UV filters in cosmetic compositions.

9. 发明公开

EP1482904A1 UV ABSORBER COMPOSITIONS COMPRISING A HYDROXYPHENYLTRIAZINE COMPOUND 有权转让
标题翻译： UV吸收组合物含羟苯基
公开(公告)号：EP1482904A1
公开(公告)日：2004-12-08
申请号：EP03709744.1
申请日：2003-03-04
申请人： Ciba Specialty Chemicals Holding Inc.
发明人： HAASE, Jürg , EHLIS, Thomas , BORSOS, Elek , HÜGLIN, Dietmar , HERZOG, Bernd
IPC分类号： A61K7/42
CPC分类号： A61K8/4966 , A61Q17/04
摘要： UV absorber compositions are described, comprising (a) from 1 to 99 % by weight of a hydroxyphenyltriazine compound of formula (I) wherein R1, R2 and R3 are each independently of the others C1-C18alkyl; C2-C10,alkenyl; or phenyl-C,-C4 alkyl; R4 is hydrogen; or C1-C5alkyl; and (b) from 99 to 1 % by weight of a further UV absorber selected from the group of (b) hydroxyphenyltriazines that are different from component (a), (b 2) benzotriazoles, (b3) dibenzoylmethane derivatives and (b4) camphor derivatives. The compositions are suitable as UV filters in cosmetic compositions.

10. 发明公开

EP1569893A2 AMINO SUBSTITUTED HYDROXYPHENYL BENZOPHENONE DERIVATIVES 有权转让
标题翻译：氨基磺酸羟基苯基苯甲酸酯
公开(公告)号：EP1569893A2
公开(公告)日：2005-09-07
申请号：EP03796081.2
申请日：2003-12-03
申请人： Ciba Specialty Chemicals Holding Inc.
发明人： HAASE, Jürg , EHLIS, Thomas , BORSOS, Elek , MÜLLER, Stefan
IPC分类号： C07C229/52 , C07C237/42 , C07C237/32 , C07C237/34 , C07C237/40 , C07D295/18 , C07D277/66 , C07D277/46 , C07D313/12 , A61K7/44
CPC分类号： C07D295/192 , A61K8/42 , A61K8/44 , A61K8/49 , A61K8/4973 , A61Q17/04 , C07C229/52 , C07C237/32 , C07C237/34 , C07C237/40 , C07C237/42 , C07D277/46 , C07D277/66 , C07D313/12
摘要： Described are amino substituted hydroxyphenyl benzophenone derivatives of formula (I), wherein R1, and R2 independently from each other are; C1,-C20alkyl; C2-C20alkenyl; C3-C10,cycloalkyl; C3-C10cycloalkenyl; or R1, and R2 together with the linking nitogen atom form a 5- or 6-membered heterocyclic ring; n1 is a number from 1 to 4; when n1=1, R3 is a saturated or unsaturated heterocyclic radical; hydroxy-C1-C5alkyl; cyclohexyl optionally substituted with one or more C1,-C5alkyl; phenyl optionally substituted with a heterocyclic radical, aminocarbonyl or C1-C5alkylcarboxy; wenn n1 is 2, R3 is an alkylene-, cycloalkylene- or alkenylene radical which is optionally substituted by a carbonyl- or carboxy group; o R3 together with A forms a bivalent radical of the formula (Ia), wherein n2 is a number from 1 to 3; when n1 is 3, R3 is an alkanetriyl radical; wenn n1 is 4, R3 is an alkanetetrayl radical; A is -O-; or -N(R5)-; and R5 is hydrogen; C1-C5alkyl; or hydroxy-C1-C5alkyl. The compounds are useful as UV filters in sunscreen applications.

你已经成功收藏专利！

检索式保存成功!

IPRDB

热门服务

关于我们

友情链接

联系方式