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1. 发明授权

US4659363A N-(2-nitrophenyl)-2-aminopyrimidine derivatives, the preparation and use thereof 失效
标题翻译： N-（2-硝基苯基）-2-氨基嘧啶衍生物，的制备及应用
公开(公告)号：US4659363A
公开(公告)日：1987-04-21
申请号：US632161
申请日：1984-07-18
申请人： Adolf Hubele , Helmut Zondler , Peter Riebli , Wolfgang Eckhardt
发明人： Adolf Hubele , Helmut Zondler , Peter Riebli , Wolfgang Eckhardt
IPC分类号： A01N43/54 , C07D239/42 , C07D239/46 , C07D239/47 , C07D239/52 , C07D239/56 , C07D401/12
CPC分类号： C07D239/42 , A01N43/54 , C07D239/47 , C07D239/52 , C07D239/56 , C07D401/12
摘要： The invention discloses novel N-(2-nitrophenyl)-2-aminopyrimidine derivatives of the general formula I ##STR1## wherein R.sub.1 and R.sub.2 are each independently NO.sub.2 or CF.sub.3, with the proviso that only R.sub.1 or R.sub.2 can be NO.sub.2R.sub.3 is halogen,R.sub.4 is hydrogen or the --C(O)R' group, in which R' is C.sub.1 -C.sub.4 alkyl which is unsubstituted or substituted by halogen, C.sub.1 -C.sub.3 alkoxy or C.sub.1 -C.sub.3 alkylthio,R.sub.5, R.sub.6 and R.sub.7 are each independently hydrogen, halogen, nitro, cyano, thiocyano, C.sub.1 -C.sub.12 alkyl, C.sub.3 -C.sub.8 cycloalkyl, C.sub.1 -C.sub.8 alkylthio, C.sub.1 -C.sub.6 alkylsulfonyl, C.sub.1 -C.sub.6 alkylsulfoxyl, C.sub.3 -C.sub.6 alkenyl, C.sub.3 -C.sub.6 haloalkenyl, C.sub.3 -C.sub.6 alkynyl, C.sub.3 -C.sub.6 haloalkynyl, C.sub.3 -C.sub.6 alkenyloxy, C.sub.3 -C.sub.6 -haloalkenyloxy, C.sub.3 -C.sub.6 alkenylthio, C.sub.3 -C.sub.6 alkynyloxy, C.sub.3 -C.sub.6 haloalkynyloxy, C.sub.1 -C.sub.8 alkyl which is substituted by halogen, cyano and/or C.sub.1 -C.sub.4 alkoxy, unsubstituted C.sub.1 -C.sub.8 alkoxy or halogen-substituted C.sub.1 -C.sub.8 alkoxy, the alkyl moiety of which may be interrupted by one or more single oxygen atoms; or are the Q--(E).sub.n --(X).sub.m -group, in which n is 0 or 1, m is 0 or 1, Q is phenyl which is unsubstituted or substituted by halogen, nitro, C.sub.1 -C.sub.3 alkyl, CF.sub.3 and/or C.sub.1 -C.sub.3 alkoxy, or is a saturated or unsaturated heterocyclic radical containing one or more hetero atoms, E is a C.sub.1 -C.sub.3 alkylene bridge, and X is oxygen or sulfur.Also disclosed are methods of preparing these compounds, and also agrochemical compositions which contain one such compound as active ingredient. The invention further relates to the use of the novel compounds, or, compositions containing them, in agriculture and related fields.
摘要翻译：本发明公开了通式I（I）的新型N-（2-硝基苯基）-2-氨基嘧啶衍生物，其中R 1和R 2各自独立地为NO 2或CF 3，条件是仅R 1或R 2可为NO 2 R 3 C 1 -C 3烷氧基或C 1 -C 3烷硫基，R 5，R 6和R 7各自独立地为氢，R 4为氢或-C（O）R'基团，其中R'为未被取代或被卤素取代的C 1 -C 4烷基，卤素，硝基，氰基，硫氰基，C 1 -C 12烷基，C 3 -C 8环烷基，C 1 -C 8烷硫基，C 1 -C 6烷基磺酰基，C 1 -C 6烷基亚磺酰基，C 3 -C 6烯基，C 3 -C 6卤代烯基，C 3 -C 6炔基，C 3 -C 6卤代炔基，C 3 -C 6烯氧基， C 6-卤代链烯氧基，C 3 -C 6烯基硫基，C 3 -C 6炔氧基，C 3 -C 6卤代炔氧基，被卤素，氰基和/或C 1 -C 4烷氧基取代的C 1 -C 8烷基，未取代的C 1 -C 8烷氧基或卤素取代的C 1 -C 8烷氧基，其可被一个或多个单个氧原子中断; 或者是Q-（E）n-（X）m-基，其中n为0或1，m为0或1，Q为未被取代或被卤素，硝基，C 1 -C 3烷基，CF 3和或C1-C3烷氧基，或是含有一个或多个杂原子的饱和或不饱和杂环基，E是C1-C3亚烷基桥，X是氧或硫。还公开了制备这些化合物的方法，以及含有一种这样的化合物作为活性成分的农药组合物。本发明还涉及在农业和相关领域中新颖化合物或含有它们的组合物的用途。

2. 发明授权

US4694009A Pesticidal compositions 失效
标题翻译：杀虫剂组合物
公开(公告)号：US4694009A
公开(公告)日：1987-09-15
申请号：US746432
申请日：1985-06-19
申请人： Adolf Hubele , Helmut Zondler , Peter Riebli , Wolfgang Eckhardt
发明人： Adolf Hubele , Helmut Zondler , Peter Riebli , Wolfgang Eckhardt
IPC分类号： A01N43/54 , C07D239/42 , C07D239/46 , C07D239/47 , C07D239/52 , A61K31/505
CPC分类号： C07D239/42 , A01N43/54 , C07D239/47
摘要： The invention discloses novel N-(2-nitrophenyl)-2-aminopyrimidine derivatives of the general formula I ##STR1## wherein R.sub.1 and R.sub.2 are hydrogen, NO.sub.2 or CF.sub.3, with the proviso that only R.sub.1 or R.sub.2 can be NO.sub.2 ;R.sub.4 is hydrogen or the --C(O)R' group, in which R' is C.sub.1 -C.sub.4 alkyl which is unsubstituted or substituted by halogen, C.sub.1 -C.sub.3 alkoxy or C.sub.1 -C.sub.3 alkylthio;R.sub.5, R.sub.6 and R.sub.7 are each independently halogen, nitro, cyano, thiocyano, C.sub.1 -C.sub.12 alkyl, C.sub.3 -C.sub.8 cycloalkyl, C.sub.1 -C.sub.8 alkylthio, C.sub.1 -C.sub.6 alkylsulfonyl, C.sub.1 -C.sub.6 alkylsulfoxyl, C.sub.3 -C.sub.6 alkenyl, C.sub.3 -C.sub.6 haloalkenyl, C.sub.3 -C.sub.6 alkynyl, C.sub.3 -C.sub.6 haloalkynyl, C.sub.3 -C.sub.6 alkenyloxy, C.sub.3 -C.sub.6 haloalkenyloxy, C.sub.3 -C.sub.6 alkenylthio, C.sub.3 -C.sub.6 alkynyloxy, C.sub.3 -C.sub.6 haloalkynyloxy, C.sub.1 -C.sub.8 alkyl which is substituted by halogen, cyano and/or C.sub.1 -C.sub.4 alkoxy, or are unsubstituted C.sub.1 -C.sub.8 alkoxy or halogen-substituted C.sub.1 -C.sub.8 alkoxy, the alkyl moiety of which may be interrupted by one or more single oxygen atoms, or are the Q--(E).sub.n --(X).sub.m group, in which n is 0 or 1, m is 0 or 1, Q is phenyl which is unsubstituted or substituted by halogen, nitro, C.sub.1 -C.sub.3 alkyl, CF.sub.3 and/or C.sub.1 -C.sub.3 alkoxy, or is a saturated or unsaturated heterocyclic radical containing one or more hetero atoms, E is a C.sub.1 -C.sub.3 alkylene bridge, and X is oxygen or sulfur, and R.sub.6 and/or one of the radicals R.sub.5 or R.sub.7 can also be hydrogen.Also disclosed are methods of preparing these compounds, and agrochemical compositions which contain one such compound as active ingredient. The invention further relates to the use of the novel compounds, or compositions containing them, in agriculture and related fields.
摘要翻译：本发明公开了通式I（I）的新型N-（2-硝基苯基）-2-氨基嘧啶衍生物，其中R 1和R 2是氢，NO 2或CF 3，条件是只有R 1或R 2可以是NO 2; R 4是氢或-C（O）R'基团，其中R'是未被取代或被卤素，C 1 -C 3烷氧基或C 1 -C 3烷硫基取代的C 1 -C 4烷基; R5，R6和R7各自独立地为卤素，硝基，氰基，氰基，C1-C12烷基，C3-C8环烷基，C1-C8烷硫基，C1-C6烷基磺酰基，C1-C6烷基亚磺酰基，C3-C6链烯基，C3-C6卤代烯基，C3-C6炔基， C 6卤代炔基，C 3 -C 6烯氧基，C 3 -C 6卤代烯氧基，C 3 -C 6烯基硫基，C 3 -C 6炔氧基，C 3 -C 6卤代炔氧基，被卤素，氰基和/或C 1 -C 4烷氧基取代的C 1 -C 8烷基，或未取代的C 1 -C 8烷氧基或卤素取代的C 1 C 1-8烷氧基，其烷基部分可被一个或多个单个氧原子间隔，或是Q-（E）n-（X）m基团，其中n为0或1，m为0或1，Q 是未取代的或被卤素，硝基，C 1 -C 3烷基，CF 3和/或C 1 -C 3烷氧基取代的苯基，或是含有一个或多个杂原子的饱和或不饱和杂环基，E是C 1 -C 3亚烷基桥，X是氧或硫，R6和/或基团R5或R7之一也可以是氢。还公开了制备这些化合物的方法和含有一种这样的化合物作为活性成分的农药组合物。本发明还涉及在农业和相关领域中使用含有它们的新化合物或组合物。

3. 发明授权

US4428964A Sulfinyl- and sulfonylacetanilides and their use as microbicides 失效
标题翻译：亚磺酰基和磺酰乙酰苯胺及其作为杀微生物剂的用途
公开(公告)号：US4428964A
公开(公告)日：1984-01-31
申请号：US182197
申请日：1980-08-28
申请人： Adolf Hubele , Peter Riebli , Wolfgang Eckhardt , Walter Kunz
发明人： Adolf Hubele , Peter Riebli , Wolfgang Eckhardt , Walter Kunz
IPC分类号： A01N37/46 , A01N41/10 , C07C67/00 , C07C313/00 , C07C317/44 , C07C147/13 , C07C147/14
CPC分类号： A01N41/10
摘要： There are described novel compounds of the formula I defined herein: ##STR1## which have valuable microbicidal properties. The novel compounds can be used for combating microorganisms harmful to plants, particularly for combating phytopathogenic fungi. The compounds of the formula I thus have a very favorable curative and preventive action for practical requirements for the protection of cultivated plants, without the plants being impaired as a result of undesirable secondary effects. The compounds can be used in practice on their own or in the form of pesticidal compositions.
摘要翻译：描述了本文定义的式I的新颖化合物：其具有有价值的杀微生物性质。新型化合物可用于对抗对植物有害的微生物，特别是用于防治植物病原真菌。因此，式I化合物对于保护栽培植物的实际需要具有非常有利的治疗和预防作用，而不会由于不期望的二次效应而损害植物。这些化合物可以在实践中以其本身或以杀虫组合物的形式使用。

4. 发明授权

US4442117A Homoserine derivatives and their use as microbicides 失效
标题翻译：高丝氨酸衍生物及其作为杀微生物剂的用途
公开(公告)号：US4442117A
公开(公告)日：1984-04-10
申请号：US199903
申请日：1980-10-23
申请人： Walter Kunz , Wolfgang Eckhardt , Adolf Hubele , Peter Riebli
发明人： Walter Kunz , Wolfgang Eckhardt , Adolf Hubele , Peter Riebli
IPC分类号： C07C231/12 , A01N37/46 , A01N41/04 , A01N43/08 , A01N43/50 , A01N43/56 , A01N43/653 , A01N47/12 , A01N47/16 , A01N47/20 , A01N53/00 , C07C233/54 , C07D307/24 , C07D521/00 , A01N37/22 , C07C103/66 , C07C103/737
CPC分类号： C07D231/12 , A01N37/46 , A01N41/04 , A01N43/08 , A01N43/50 , A01N43/56 , A01N43/653 , A01N47/12 , A01N47/16 , A01N47/20 , A01N53/00 , C07D233/56 , C07D249/08 , C07D307/24
摘要： There are described novel homoserine derivatives of the formula (I) ##STR1## which possess valuable microbicidal properties. In the formula: Ar is substituted phenyl or naphthyl; R.sub.1 is C.sub.2 -C.sub.6 alkyl optionally interrupted by oxygen or sulfur, 2-furyl, 2-tetrahydrofuryl, 1H-1,2,4-triazolylmethyl, 1-imidazolylmethyl, 1-pyrazolylmethyl, C.sub.2 -C.sub.4 alkenyl or cyclopropyl, each of which is optionally substituted by halogen; R.sub.2 is hydrogen or methyl; R.sub.3 is hydrogen or C.sub.1 -C.sub.4 alkyl; and B is halogen or an ester, thioester, sulfonic acid ester or sulfonic acid amide group. Additionally, where B is halogen, R.sub.1 may be halomethyl. The novel derivatives can be used for combating microorganisms harmful to plants, particularly for combating phytopathogenic fungi, and they have for practical requirements a very favorable curative and protective action for protecting cultivating plants, without the plants being impaired as a result of undesirable secondary effects. A notable feature is their stability to heat and to solar irradiation. They can be used in practice on their own or in the form of pesticidal compositions.
摘要翻译：描述了具有有价值的杀微生物性质的式（I）的新颖高丝氨酸衍生物。式中Ar是取代的苯基或萘基; R1是任选被氧或硫中断的C 2 -C 6烷基，2-呋喃基，2-四氢呋喃基，1H-1,2,4-三唑基甲基，1-咪唑基甲基，1-吡唑基甲基，C 2 -C 4烯基或环丙基，任选被卤素取代; R2是氢或甲基; R3是氢或C1-C4烷基; 和B是卤素或酯，硫酯，磺酸酯或磺酸酰胺基。另外，当B是卤素时，R 1可以是卤代甲基。新型衍生物可用于对抗对植物有害的微生物，特别是用于防治植物病原性真菌，并且它们具有非常有利的治疗和保护作用，用于保护栽培植物，而不会由于不期望的二次作用而损害植物。它的一个显着特点是它们对热和太阳辐射的稳定性。它们可以自己使用或以农药组合物的形式使用。

5. 发明授权

US4438125A Arylamine derivatives and use as microbicides 失效
标题翻译：芳胺衍生物，用作杀菌剂
公开(公告)号：US4438125A
公开(公告)日：1984-03-20
申请号：US417232
申请日：1982-09-13
申请人： Adolf Hubele , Wolfgang Eckhardt , Peter Riebli
发明人： Adolf Hubele , Wolfgang Eckhardt , Peter Riebli
IPC分类号： C07C231/02 , A01N37/22 , A01N37/24 , A01N37/36 , A01N37/44 , A01N37/46 , A01N41/04 , A01N41/08 , A01N41/10 , A01N43/08 , A01N43/653 , A01N53/00 , A01N53/12 , C07C231/12 , C07D249/10 , C07D307/16 , C07D307/24 , C07D307/68 , C07D521/00 , C07K5/00 , C07K5/06 , A01N37/34 , C07C121/78
CPC分类号： A01N37/22 , A01N37/24 , A01N37/36 , A01N37/44 , A01N37/46 , A01N41/04 , A01N41/08 , A01N41/10 , A01N43/08 , A01N43/653 , A01N53/00 , C07D231/12 , C07D233/56 , C07D249/08 , C07D307/24 , C07D307/68
摘要： The invention relates to novel microbicides of the general formula I ##STR1## wherein R is hydrogen or methyl, Ar is a phenyl or .alpha.-naphthyl group which is substituted by NH.sub.2 or NO.sub.2 and further radicals, W is a cyano, ester, alkenyl or alkynyl group, and B is alkyl, alkenyl, cyclopropyl, 2-furyl, 2-tetrahydrofuryl, .beta.-(alkoxy)ethyl, triazolylmethyl, methylsulfonylmethyl, alkoxymethyl, alkenyloxymethyl, alkynylmethyl, alkylthiomethyl, alkenylthiomethyl, alkynylthiomethyl, --OSO.sub.2 -alkyl, --OSO.sub.2 NH(alkyl) or --N(alkyl).sub.2. The invention also describes plant protection compositions which contain these compounds, a process for the production of the novel compounds and compositions, and a method of controlling phytopathogenic microorganisms which comprises the use thereof.
摘要翻译：本发明涉及通式I的新型杀微生物剂，其中R是氢或甲基，Ar是被NH 2或NO 2取代的苯基或α-萘基，以及其它基团，W是氰基，酯，烯基或乙炔基，三唑基甲基，甲基磺酰基甲基，烷氧基甲基，烯氧基甲基，炔基甲基，烷基硫代甲基，链烯基硫代甲基，炔基硫代甲基，-OSO 2 - 烷基，-OSO 2 NH （烷基）或-N（烷基）2。本发明还描述了含有这些化合物的植物保护组合物，用于生产新化合物和组合物的方法，以及控制植物病原微生物的方法，其包括其用途。

6. 发明授权

US4377587A Arylamine derivatives and use thereof as microbicides 失效
标题翻译：芳胺衍生物及其作为杀微生物剂的用途
公开(公告)号：US4377587A
公开(公告)日：1983-03-22
申请号：US285652
申请日：1981-07-21
申请人： Adolf Hubele , Wolfgang Eckhardt , Peter Riebli
发明人： Adolf Hubele , Wolfgang Eckhardt , Peter Riebli
IPC分类号： C07C231/02 , A01N37/22 , A01N37/24 , A01N37/36 , A01N37/44 , A01N37/46 , A01N41/04 , A01N41/08 , A01N41/10 , A01N43/08 , A01N43/653 , A01N53/00 , A01N53/12 , C07C231/12 , C07D249/10 , C07D307/16 , C07D307/24 , C07D307/68 , C07D521/00 , C07K5/00 , C07K5/06 , C07C103/32
CPC分类号： A01N37/22 , A01N37/24 , A01N37/36 , A01N37/44 , A01N37/46 , A01N41/04 , A01N41/08 , A01N41/10 , A01N43/08 , A01N43/653 , A01N53/00 , C07D231/12 , C07D233/56 , C07D249/08 , C07D307/24 , C07D307/68
摘要： The invention relates to novel microbicides of the general formula I ##STR1## wherein R is hydrogen or methyl, Ar is a phenyl or .alpha.-naphthyl group which is substituted by NH.sub.2 or NO.sub.2 and further radicals, W is a cyano, ester, alkenyl or alkynyl group, and B is alkyl, alkenyl, cyclopropyl, 2-furyl, 2-tetrahydrofuryl, .beta.-(alkoxy)ethyl, triazolylmethyl, methylsulfonylmethyl, alkoxymethyl, alkenyloxymethyl, alkynyloxymethyl, alkylthiomethyl, alkenylthiomethyl, alkynylthiomethyl, --OSO.sub.2 -alkyl, --OSO.sub.2 NH(alkyl) or --N(alkyl).sub.2. The invention also describes plant protection compositions which contain these compounds, a process for the production of the novel compounds and compositions, and a method of controlling phytopathogenic microorganisms which comprises the use thereof.
摘要翻译：本发明涉及通式I的新型杀微生物剂，其中R是氢或甲基，Ar是被NH 2或NO 2取代的苯基或α-萘基，以及其它基团，W是氰基，酯，烯基或炔基，链烯基，环丙基，2-呋喃基，2-四氢呋喃基，β-（烷氧基）乙基，三唑基甲基，甲基磺酰基甲基，烷氧基甲基，烯氧基甲基，炔氧基甲基，烷硫基甲基，链烯基硫代甲基，炔硫基甲基，-OSO 2烷基，-OSO 2 NH （烷基）或-N（烷基）2。本发明还描述了含有这些化合物的植物保护组合物，用于生产新化合物和组合物的方法，以及控制植物病原微生物的方法，其包括其用途。

7. 发明授权

US4479004A 1-[2-(4-Diphenyl)-1,3-dioxolan-2-yl-methyl]-1-H-triazoles 失效
标题翻译： 1- [2-（4-二苯基）-1,3-二氧戊环-2-基 - 甲基] -1H-三唑
公开(公告)号：US4479004A
公开(公告)日：1984-10-23
申请号：US423391
申请日：1982-09-24
申请人： Adolf Hubele , Peter Riebli
发明人： Adolf Hubele , Peter Riebli
IPC分类号： A01N43/50 , A01N43/653 , C07D405/06 , C07D521/00 , A01N43/64
CPC分类号： C07D231/12 , A01N43/50 , A01N43/653 , C07D233/56 , C07D249/08 , C07D405/06 , Y10S514/937
摘要： A description is given of new compounds of the formula defined herein: ##STR1## which display valuable microbicidal properties. The compounds can be used for combatting microorganisms harmful to plants, especially phytopathogenic fungi. The compounds of formula I thus possess a curative, systemic, and preventive action very useful for practical requirements for the protection of cultivated plants, without causing these to suffer any undesirable side effects. In practice, the compounds can be used by themselves or in the form of pesticides.
摘要翻译：给出了本文定义的新化合物的描述：显示有价值的杀菌性质的图像（I）。该化合物可用于对有害于植物，特别是植物病原真菌的微生物进行防治。因此，式I化合物具有对保护栽培植物的实际需要非常有用的治疗性，系统性和预防性作用，而不会使它们遭受任何不期望的副作用。实际上，这些化合物可以自己或以农药的形式使用。

8. 发明授权

US4840662A N-(2-nitrophenyl)-5-aminopyrimidine derivatives and useful for controlling harmful micro-organisms 失效
标题翻译： N-（2-硝基苯基）-5-氨基嘧啶衍生物，可用于控制有害微生物
公开(公告)号：US4840662A
公开(公告)日：1989-06-20
申请号：US631272
申请日：1984-07-16
申请人： Helmut Zondler , Adolf Hubele , Robert Nyfeler
发明人： Helmut Zondler , Adolf Hubele , Robert Nyfeler
IPC分类号： A01N43/54 , C07D239/42 , C07D239/46 , C07D239/47 , C07D239/48 , C07D239/50 , C07D239/52 , C07D239/56 , C07D239/58 , C07D239/60
CPC分类号： C07D239/42 , A01N43/54 , C07D239/47 , C07D239/48 , C07D239/50 , C07D239/52 , C07D239/56 , C07D239/58 , C07D239/60
摘要： The invention discloses novel N-(2-nitrophenyl)-5-aminopyrimidine derivatives of the general formula ##STR1## wherein R.sub.1 and R.sub.2 are each independently NO.sub.2 or CF.sub.3, or one of R.sub.1 and R.sub.2 is hydrogen,R.sub.3 is hydrogen or halogen,R.sub.4 is hydrogen or the --C(O)R' group, in which R' is C.sub.1 -C.sub.4 alkyl which is unsubstituted or substituted by halogen, C.sub.1 -C.sub.3 alkoxy or C.sub.1 -C.sub.3 alkylthio,R.sub.5, R.sub.6 and R.sub.7 are each independently hydrogen, halogen, nitro, cyano, thiocyano, mercapto, C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.6 haloalkyl, C.sub.1 -C.sub.6 alkoxy, C.sub.1 -C.sub.6 alkoxy which is substituted by halogen, nitro, cyano, C.sub.1 -C.sub.3 alkoxy, C.sub.1 -C.sub.3 alkylthio and/or N(C.sub.1 -C.sub.4 alkyl).sub.2 ; or are C.sub.3 -C.sub.6 cycloalkoxy, C.sub.3 -C.sub.6 alkenyloxy, C.sub.3 -C.sub.6 alkynyloxy, C.sub.1 -C.sub.6 alkylthio, C.sub.3 -C.sub.6 alkenylthio, C.sub.1 -C.sub.6 alkylsulfonyl, C.sub.1 -C.sub.6 alkylsulfoxyl, C.sub.3 -C.sub.6 alkenyl, C.sub.3 -C.sub.6 haloalkenyl, C.sub.3 -C.sub.6 alkynyl, C.sub.3 -C.sub.6 haloalkynyl or the N(C.sub.1 -C.sub.4 alkyl).sub.2 group, and R.sub.5 may additionally be a phenyl or benzyl group which is unsubstituted or substituted by one to three identical or different members selected from halogen, nitro, cyano, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.3 haloalkyl, N--(C.sub.1 -C.sub.3 alkyl).sub. 2, and/or C.sub.1 -C.sub.3 alkoxy.The preparation of these compounds and their use in agriculture are also disclosed.
摘要翻译：本发明公开了通式（I）的新型N-（2-硝基苯基）-5-氨基嘧啶衍生物，其中R 1和R 2各自独立地为NO 2或CF 3，或者R 1和R 2中的一个为氢，R 3为氢或卤素，R 4是氢或-C（O）R'基团，其中R'是未被取代或被卤素取代的C 1 -C 4烷基，C 1 -C 3烷氧基或C 1 -C 3烷硫基，R 5，R 6和R 7各自独立地为氢，卤素，硝基，氰基，硫氰基，巯基，C1-C6烷基，C1-C6卤代烷基，C1-C6烷氧基，被卤素，硝基，氰基，C1-C3烷氧基，C1-C3烷硫基和/或N（C1-C4烷基））2; 或者是C 3 -C 6环烷氧基，C 3 -C 6烯氧基，C 3 -C 6炔氧基，C 1 -C 6烷硫基，C 3 -C 6烯基硫基，C 1 -C 6烷基磺酰基，C 1 -C 6烷基亚磺酰基，C 3 -C 6烯基，C 3 -C 6卤代烯基，C 3 -C 6炔基，C 3 -C 6卤代炔基或N -C 1-4烷基）2基团，并且R 5可另外为未取代的或被一至三个相同或不同的选自卤素，硝基，氰基，C 1 -C 4烷基，C 1 -C 3卤代烷基，N-（C 1 -C 4烷基） C3烷基）2和/或C1-C3烷氧基。还公开了这些化合物的制备及其在农业中的应用。

9. 发明授权

US5175293A Pesticides 失效
标题翻译：农药
公开(公告)号：US5175293A
公开(公告)日：1992-12-29
申请号：US677352
申请日：1991-03-22
申请人： Helmut Zondler , Adolf Hubele
发明人： Helmut Zondler , Adolf Hubele
IPC分类号： A01N43/54 , C07D239/30 , C07D239/34 , C07D239/42 , C07D401/12 , C07D403/12 , C07D405/12 , C07D409/12
CPC分类号： C07D401/12 , A01N43/54 , C07D239/34 , C07D239/42 , C07D403/12 , C07D405/12 , C07D409/12
摘要： Compounds of the formula ##STR1## wherein: R.sub.1 is phenyl or phenyl mono- to tri-substituted by R.sub.4 ; R.sub.2 is hydrogen, C.sub.1 -C.sub.5 alkyl, C.sub.1 -C.sub.5 alkyl substituted by the radical OR.sub.5 or by the radical SR.sub.5, C.sub.3 -C.sub.6 cycloalkyl, C.sub.3 -C.sub.6 cycloalkyl mono- to tri-substituted by C.sub.1 -C.sub.4 alkyl or by halogen, C.sub.2 -C.sub.5 alkenyl, C.sub.2 -C.sub.5 alkynyl or the formyl radical; R.sub.3 is hydrogen, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkyl substituted by halogen, cyano or by the radical OR.sub.5 or by the radical SR.sub.5, C.sub.3 -C.sub.6 cycloalkyl or C.sub.3 -C.sub.6 cycloalkyl mono- to tri-substituted by C.sub.1 -C.sub.4 alkyl or by halogen; R.sub.4 is halogen; C.sub.1 -C.sub.3 alkyl, C.sub.1 -C.sub.2 haloalkyl, C.sub.1 -C.sub.3 alkoxy or C.sub.1 -C.sub.3 haloalkoxy; R.sub.5 is hydrogen, C.sub.1 -C.sub.5 alkyl, C.sub.3 -C.sub.5 alkenyl, C.sub.3 -C.sub.5 alkynyl or the radical (CH.sub.2).sub.n -X-C.sub.1 -C.sub.3 -alkyl;R.sub.7 is the group -NH.sub.2, ##STR2## and where R.sub.8 -R.sub.11 are as defined hereafter.
摘要翻译：式（I）的化合物其中：R 1是苯基或被R4单 - 三取代的苯基; R 2是氢，C 1 -C 5烷基，被基团OR 5取代的C 1 -C 5烷基或被基团SR 5，C 3 -C 6环烷基，被C 1 -C 4烷基单取代至三取代的C 3 -C 6环烷基或被卤素，C 2 -C 5烯基，C 2 -C 5炔基或甲酰基; R3是氢，C1-C4烷基，被卤素，氰基或基团OR5取代的C 1 -C 4烷基或被C 1 -C 4烷基或被卤素单 - 三取代的基团SR 5，C 3 -C 6环烷基或C 3 -C 6环烷基取代; R4是卤素; C 1 -C 3烷基，C 1 -C 2卤代烷基，C 1 -C 3烷氧基或C 1 -C 3卤代烷氧基; R5是氢，C1-C5烷基，C3-C5链烯基，C3-C5炔基或基团（CH2）n-X-C1-C3-烷基; R 7是基团-NH 2，，其中R 8 -R 11如下文所定义。

10. 发明授权

US4992458A 1-phenoxyphenyl-1-triazolylmethyl-carbinol compound as microbicides 失效
标题翻译： 1-苯氧基苯基-1-三唑基甲基 - 甲醇化合物作为杀微生物剂
公开(公告)号：US4992458A
公开(公告)日：1991-02-12
申请号：US376185
申请日：1989-07-06
申请人： Peter Riebli , Adolf Hubele
发明人： Peter Riebli , Adolf Hubele
IPC分类号： A01N43/653 , C07D249/08 , C07D521/00
CPC分类号： C07D231/12 , A01N43/653 , C07D233/56 , C07D249/08
摘要： Novel 1-phenoxyphenyl-1-triazolylmethyl-carbinols of formula I ##STR1## in which R.sub.1 is fluorine, chlorine or bromine and R.sub.2 is fluorine, chlorine, bromine or methyl,and the phytophysiologically tolerable acid addition salts thereof have excellent microbicidal, in particular phytofungicidal, properties. They can be used for controlling and/or preventing infections caused by microorganisms in useful plants. The preparation of these compounds and compositions containing them is described.
摘要翻译：式I的1-苯氧基苯基-1-三唑基甲基 - 甲醇其中R1是氟，氯或溴，R2是氟，氯，溴或甲基，其植物生理学上可耐受的酸加成盐具有优异的杀微生物剂，特别是植物杀灭剂的性质。它们可用于控制和/或预防有用植物中的微生物引起的感染。描述了这些化合物和含有它们的组合物的制备。

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