专利快速检索-快速检索全球专利，免费商用专利数据库-IPRDB

2. 发明授权

US4645678A Sweetening agents 失效
标题翻译：甜味剂
公开(公告)号：US4645678A
公开(公告)日：1987-02-24
申请号：US532499
申请日：1983-09-15
申请人： Claude Nofre , Jean-Marie Tinti
发明人： Claude Nofre , Jean-Marie Tinti
IPC分类号： A23L27/30 , C07C67/00 , C07C239/00 , C07C275/42 , C07C279/18 , C07C313/00 , C07C317/28 , C07C317/30 , C07C317/42 , C07C325/00 , C07C335/16 , C07K5/072 , C07K5/075 , A23L1/236 , C07C127/00 , C07C147/13 , C07C149/43
CPC分类号： C07K5/06113 , A23L27/32 , C07K5/0613
摘要： Compounds of the formula: ##STR1## in which: X represents at least one lone-electron pair donor group;A represents an oxygen or a sulfur atom, or an optionally substituted imino or methylene group;R represents a hydrogen atom or an alkyl group of 1 to 4 carbon atoms;n represents a number equal to zero or to one;B represents a COOH or COOM group (M designating a cation);Y represents either a lone-electron pair donor group, or an alkyl group R' of 1 to 4 carbon atoms;Z representseither an optionally substituted hydrophobic group R", R" designating an alkyl, cycloalkyl or aryl group of 1 to 12 carbon atoms;or a lone-electron pair donor group on which a hydrophobic group R" is fixed;are useful as sweetening agents.
摘要翻译：下式的化合物：其中：X表示至少一个单电子对供体基团; A表示氧或硫原子，或任选取代的亚氨基或亚甲基; R表示氢原子或1〜4个碳原子的烷基; n表示等于零或1的数; B表示COOH或COOM基团（M表示阳离子）; Y表示单电子对给体基团或1〜4个碳原子的烷基R'; Z表示任选取代的疏水基团R“，R”表示1至12个碳原子的烷基，环烷基或芳基; 或其上固定有疏水基团R“的单电子对供体基团; 可用作甜味剂。

3. 发明授权

US4230874A N-(Benzenesulfonyl) carbamates-herbicidal antidotes 失效
标题翻译： N-（苯磺酰基）氨基甲酸酯 - 除草剂
公开(公告)号：US4230874A
公开(公告)日：1980-10-28
申请号：US721721
申请日：1976-09-13
申请人： Ferenc M. Pallos , Edmund J. Gaughan
发明人： Ferenc M. Pallos , Edmund J. Gaughan
IPC分类号： A01N47/12 , A01N25/32 , A01N47/16 , A01N47/18 , A01P13/02 , C07D319/06 , C07F9/38 , C07C147/13
CPC分类号： C07D319/06 , C07F9/3808
摘要： N-(substituted benzenesulfonyl) carbamates as new compositions of matter useful as active herbicidal antidotes to protect against and decrease crop injury when used with a thiocarbamate herbicide when applied in various methods; improved herbicidal compositions and utility of said compositions to protect against and decrease phytotoxic crop injury when employing thiocarbamate herbicides and a two-part herbicide system comprising a first-part of one or more thiocarbamate herbicide and a second part of an effective antidote therefor compound said antidote compounds of the class N-benzene sulfonyl carbamates having the formula ##STR1## wherein X is hydrogen, bromo, chloro, methoxy, trifluoromethyl, and methyl; n is an integer from 1 to 3 inclusive, provided that when X is bromo, trifluoromethyl, or methoxy, n is 1; and R is selected from alkyl, haloalkyl wherein halo is chloro or fluoro, alkenyl, haloalkenyl and wherein halo is chloro, alkynyl, trifluoroacetamidomethyl, dialkylamino cyanoalkylthioalkyl, phosphonomethyl, lower alkyl substituted phenyl, 4-chlorophenylthiomethyl, alkoxyalkyl, alkylthioalkyl, cyanoalkyl, alkoxycarbonylalkyl, formamidoalkyl, alkoxycarbonylalkenyl, alkylcarbonylalkyl, 1,3-dioxacyclohexane-5,5-methylene, phenyl, chlorophenyl, benzyl, 4-chlorobenzyl, 4-methoxybenzyl, 3-pyridylmethyl, phenoxyethyl, 3-phenylpropyn-2-yl, methylthioacetimino, acetone imino and benzaldimino.
摘要翻译： N-（取代的苯磺酰基）氨基甲酸酯作为活性除草剂的新组合物，用于当以各种方法施用时用于与硫代氨基甲酸酯除草剂一起使用时防止和减少作物损伤; 改进的除草组合物和所述组合物在使用硫代氨基甲酸酯除草剂时防止和减少植物毒性作物损伤的效用以及包含一种或多种硫代氨基甲酸酯除草剂的第一部分的两部分除草剂系统和其中一种有效解毒剂的第二部分化合物所述解毒剂具有式“IMAGE”的N-苯磺酰基氨基甲酸酯类化合物，其中X是氢，溴，氯，甲氧基，三氟甲基和甲基; n为1〜3的整数，条件是当X为溴，三氟甲基或甲氧基时，n为1; 其中卤素为氯或氟，烯基，卤代烯基，其中卤素为氯，炔基，三氟乙酰胺基甲基，二烷基氨基氰基烷基硫代烷基，膦酰基甲基，低级烷基取代的苯基，4-氯苯硫基甲基，烷氧基烷基，烷硫基烷基，氰基烷基，烷氧羰基烷基，甲酰氨基烷基，烷氧基羰基烯基，烷基羰基烷基，1,3-二氧杂环己烷-5,5-亚甲基，苯基，氯苯基，苄基，4-氯苄基，4-甲氧基苄基，3-吡啶基甲基，苯氧基乙基，3-苯基丙炔-2-基，甲硫基乙酰亚氨基，和苯达拉霉素。

4. 发明授权

EP0002182B1 Bis-Azidophthalsäurederivate und Verfahren zu ihrer Herstellung 失效
标题翻译： BIS-AZIDO-PHTHALIC酸衍生物及其制备方法
公开(公告)号：EP0002182B1
公开(公告)日：1981-04-08
申请号：EP78101084.8
申请日：1978-10-06
申请人： CIBA-GEIGY AG
发明人： Kvita, Vratislav, Dr. , Zweifel, Hans, Dr. , Greber, Gerd, Prof. Dr.
IPC分类号： C07D209/48 , C07C149/43 , C07C147/13 , C07C117/08
CPC分类号： C07D209/48 , G03F7/008

5. 发明授权

US4663484A Diaminoalkyldiphenyl ethers, a process for their preparation and their use 失效
标题翻译：二氨基烷基二苯醚，其制备方法及其用途
公开(公告)号：US4663484A
公开(公告)日：1987-05-05
申请号：US801527
申请日：1985-11-25
申请人： Walter Horstmann
发明人： Walter Horstmann
IPC分类号： C08G18/00 , C07C67/00 , C07C213/00 , C07C217/90 , C08G18/76 , C08G18/77 , C07C147/13
CPC分类号： C08G18/771
摘要： New diaminoalkyldiphenyl ethers of the formula ##STR1## wherein R.sup.1 and R.sup.2 are identical or different and denote hydrogen or methyl, but R.sup.1 and R.sup.2 do not simultaneously represent methyl,are prepared by a process wherein alkyldiphenyl ethers of the formula ##STR2## wherein R.sup.1 and R.sup.2 have the above-mentioned meaning are acetylated, the diacetyl compounds obtained, in aqueous-alcoholic solution or suspension, are converted to the corresponding dioximes with hydroxylamine, the dried dioximes are subjected to a Beckmann rearrangement and thereafter the diacetylaminoalkyldiphenyl ethers formed are hydrolyzed by means of aqueous mineral acids or alkali metal hydroxide solutions to give the diamines.The new diaminoalkyldiphenyl ethers are used in the preparation of dyestuffs and polyurethanes and serve as monomers for the preparation of polymers.
摘要翻译：新的式（II）的二氨基烷基二苯基醚，其中R 1和R 2相同或不同并且表示氢或甲基，但R 1和R 2不同时表示甲基，其通式为其中R1和 R2具有上述含义是乙酰化的，在水溶液或悬浮液中获得的二乙酰基化合物用羟胺转化成相应的二肟，将干燥的二肟进行贝克曼重排，然后形成的二乙酰基氨基烷基二苯基醚被水解含水无机酸或碱金属氢氧化物溶液的方法，得到二胺。新的二氨基烷基二苯醚用于制备染料和聚氨酯，并用作制备聚合物的单体。

6. 发明授权

US4537896A Thrombin inhibiting arylsulfonyl guanidinophenylalanine amides 失效
标题翻译：凝血酶抑制芳基磺酰胍胍苯丙氨酸酰胺
公开(公告)号：US4537896A
公开(公告)日：1985-08-27
申请号：US504338
申请日：1983-06-14
申请人： Carl G. Claeson , Stig I. Gustavsson
发明人： Carl G. Claeson , Stig I. Gustavsson
IPC分类号： A61K31/18 , A61K31/445 , A61P7/02 , C07C67/00 , C07C301/00 , C07C303/38 , C07C311/18 , C07C311/42 , C07D211/14 , C07D295/185 , G01N33/86 , A61K31/16 , C07C147/13 , C07D211/16
CPC分类号： C07D295/185 , C07C311/42
摘要： New thrombin inhibiting N.sup..alpha. -arylsulfonyl-p-guanidinophenylalanine amides of the formula ##STR1## wherein Ar is a substituted aryl and R.sub.1 and R.sub.2 are an alkyl group having 1-5 carbon atoms or together with the amine nitrogen form an heterocyclic ring, in racemate form as well as in form of optical active antipodes, theirs pharmaceutically acceptable salts, methods for their preparation, pharmaceutical composition and diagnostical preparation containing these compounds, use of the compounds in treatments of thrombosis and methods of treatment of thrombosis as well as methods for determination of thrombin concentration in blood.
摘要翻译：新型凝血酶抑制式为“IMAGE”的Nα - 芳基磺酰基 - 对胍胍苯丙氨酸酰胺，其中Ar为取代的芳基，R 1和R 2为具有1-5个碳原子的烷基或与胺氮一起形成杂环，外消旋形式以及光学活性对映体的形式，它们的药学上可接受的盐，其制备方法，含有这些化合物的药物组合物和诊断制剂，治疗血栓形成的用途以及血栓形成治疗方法测定血液中凝血酶浓度。

7. 发明授权

US4144225A Novel aromatic diamine compounds and flame-resistant polyamide compositions containing said compounds 失效
标题翻译：新型芳族二胺化合物和含有所述化合物的阻燃聚酰胺组合物
公开(公告)号：US4144225A
公开(公告)日：1979-03-13
申请号：US713651
申请日：1976-08-12
申请人： Keio Yamanaka , Kazuo Okamoto , Yoshikatsu Mizukami
发明人： Keio Yamanaka , Kazuo Okamoto , Yoshikatsu Mizukami
IPC分类号： C08K5/20 , C08K5/41 , C07C103/127 , C07C147/13
CPC分类号： C08K5/20 , C08K5/41
摘要： Novel N,N,N',N'-tetraacetyl aromatic diamine compounds shown by the general formula (1) ##STR1## wherein R is ##STR2## X is Br or Cl, Y is alkylene group or akylidene group having 1-3 carbon atoms, carbonyl group, sulfonyl group or oxygen atom and m and n is 0 or an integer of 1-4, are produced by reacting 1 mole of aromatic diamine having the general formulaH.sub.2 N--R--NH.sub.2 (2)with at least 4 moles of acetic anhydride. These compounds are used as a flame retardant for polyamides.
摘要翻译：由通式（1）表示的新型N，N，N'，N'-四乙酰芳族二胺化合物，其中R为Br或Cl，Y为亚烷基具有1-3个碳原子的基团或亚烷基，羰基，磺酰基或氧原子，m和n为0或1-4的整数，通过使1摩尔具有通式H2N-R- NH 2（2）与至少4摩尔乙酸酐反应。这些化合物用作聚酰胺的阻燃剂。

8. 发明授权

US4467101A Compounds with terminal aminocarboxylic acid grouping 失效
标题翻译：具有末端氨基羧酸分子的化合物
公开(公告)号：US4467101A
公开(公告)日：1984-08-21
申请号：US420534
申请日：1982-09-20
申请人： Karoly Kocsis , Peter Schneider , Bruno Fechtig , Riccardo Scartazzini
发明人： Karoly Kocsis , Peter Schneider , Bruno Fechtig , Riccardo Scartazzini
IPC分类号： C07D499/06 , A61K31/545 , A61K31/546 , A61P31/04 , C07D307/34 , C07D307/52 , C07D307/54 , C07D333/04 , C07D333/24 , C07D501/00 , C07D501/20 , C07D501/32 , C07D501/34 , C07D501/57 , C07D501/59 , C07C143/52 , C07C147/13 , C07C153/00
CPC分类号： C07D333/24 , C07D307/52 , C07D307/54
摘要： Acylamido-3-cephem-4-carboxylic acid compounds of the formula ##STR1## in which the index n represents an integer of from 1 to 4,the index m represents 0 or 1,X represents oxygen, sulphur or an --NH-- group,W represents a --CO--, --CO--NHSO.sub.2 -- or --SO.sub.2 NH--CO-- group, orX-W together represent a --CO-- or --CO--NHSO.sub.2 -- group,A represents optionally substituted phenylene, thienylene or furylene,Y represents hydrogen, hydroxyl, formyloxy, amino or sulpho optionally present in salt form, andZ represents hydrogen, orY and Z together represent an oxo group or an .dbd.N--O--R.degree. group in which R.degree. represents hydrogen or optionally substituted lower alkyl,R.sub.1 represents hydrogen, lower alkyl, lower alkoxy, halogen or a group of the formula --CH.sub.2 --R.sub.2 in which R.sub.2 is a free, esterified or etherified hydroxy or mercapto group or a quaternary ammonium group, andR.sub.3 represents hydrogen or methoxy,wherein the carboxyl groups are optionally esterified in a form that can be split under physiological conditions, and the salts thereof, are obtained by liberating the functional group(s) in a starting compound of the formula I in which at least one of the functional groups present is protected.The compounds are effective in vitro and in vivo against gram-positive and gram-negative bacteria and cocci.
摘要翻译：酰亚胺基-3-头孢烯-4-羧酸化合物，其中指数n表示1至4的整数，指数m表示0或1，X表示氧，硫或-NH-基团，W表示-CO-，-CO-NHSO2-或-SO2NH-CO-基团，或XW一起表示-CO-或-CO-NHSO2-基团，A表示任选取代的亚苯基，亚噻吩基或呋喃基，Y表示氢，羟基，甲酰氧基，任选以盐形式存在的氨基或磺基，Z表示氢，或Y和Z一起表示氧代基或= NOROR基，其中R DEG表示氢或任选取代的低级烷基，R 1表示氢，低级烷基，低级烷氧基，卤素或式-CH 2 -R 2的基团，其中R 2是游离的，酯化的或醚化的羟基或巯基或季铵基团，R 3表示氢或甲氧基，其中羧基任选地以可在生理学上分裂的形式进行酯化定义及其盐通过释放其中存在至少一个官能团被保护的式I起始化合物中的官能团而获得。这些化合物在体外和体内对革兰氏阳性和革兰氏阴性细菌和球菌有效。

9. 发明授权

US4428964A Sulfinyl- and sulfonylacetanilides and their use as microbicides 失效
标题翻译：亚磺酰基和磺酰乙酰苯胺及其作为杀微生物剂的用途
公开(公告)号：US4428964A
公开(公告)日：1984-01-31
申请号：US182197
申请日：1980-08-28
申请人： Adolf Hubele , Peter Riebli , Wolfgang Eckhardt , Walter Kunz
发明人： Adolf Hubele , Peter Riebli , Wolfgang Eckhardt , Walter Kunz
IPC分类号： A01N37/46 , A01N41/10 , C07C67/00 , C07C313/00 , C07C317/44 , C07C147/13 , C07C147/14
CPC分类号： A01N41/10
摘要： There are described novel compounds of the formula I defined herein: ##STR1## which have valuable microbicidal properties. The novel compounds can be used for combating microorganisms harmful to plants, particularly for combating phytopathogenic fungi. The compounds of the formula I thus have a very favorable curative and preventive action for practical requirements for the protection of cultivated plants, without the plants being impaired as a result of undesirable secondary effects. The compounds can be used in practice on their own or in the form of pesticidal compositions.
摘要翻译：描述了本文定义的式I的新颖化合物：其具有有价值的杀微生物性质。新型化合物可用于对抗对植物有害的微生物，特别是用于防治植物病原真菌。因此，式I化合物对于保护栽培植物的实际需要具有非常有利的治疗和预防作用，而不会由于不期望的二次效应而损害植物。这些化合物可以在实践中以其本身或以杀虫组合物的形式使用。

10. 发明授权

US3981910A Sulfur containing trialkoxybenzoylamino carboxylic acids 失效
标题翻译：含有三烷氧基苯甲酰氨基羧酸的硫
公开(公告)号：US3981910A
公开(公告)日：1976-09-21
申请号：US468087
申请日：1974-05-08
申请人： Heribert Offermanns , Klaus Posselt
发明人： Heribert Offermanns , Klaus Posselt
IPC分类号： C07C323/58 , A61K31/215 , A61K31/38 , A61K31/381 , A61P9/06 , A61P9/08 , A61P9/10 , C07C231/02 , C07C235/52 , C07D333/36 , C07C147/13 , C07C149/31
CPC分类号： C07D333/36 , Y10S514/821
摘要： Compounds are prepared of the formula: ##SPC1##Wherein A is a straight or branched chain alkylene or alkylidene radical having 2 to 5 carbon atoms and which is substituted by an alkylthio group having 1 to 4 carbon atoms, a carboxymethyl thio group, a carboxyethyl thio group, an alkylsulfonyl group having 1 to 4 carbon atoms, a mercapto group, or the substituent on A together with --COR.sub.4 forms a 4 to 7 membered thiolactone ring, or A is substituted by an acylmercapto group wherein the acyl is benzoyl, a benzoyl radical substituted with one, two or three alkoxy groups with 1 to 6 carbon atoms, an alkanoyl radical of 1 to 6 carbon atoms, an alkenoyl radical of 3 to 6 carbon atoms, R.sub.1, R.sub.2 and R.sub.3 are the same or different and are alkyl groups of 1 to 5 carbon atoms and one of R.sub.1, R.sub.2 and R.sub.3 also can be hydrogen or the acyl radical of an alkanoic acid of 2 to 4 carbon atoms and R.sub.4 is a hydroxy group or an alkoxy group with 1 to 5 carbon atoms and their pharmacologically acceptable salts. The compounds are pharmacodynamically active and are suited for prophylaxis and treatment of heart illnesses such as cardiac ischemia, cardiac infarct, heart rhythm and circulatory disturbances.
摘要翻译：化合物由下式制备：

你已经成功收藏专利！

检索式保存成功!

IPRDB

热门服务

关于我们

友情链接

联系方式