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1. 发明专利

IL217078D0 4-(3-BUTYNYL) AMINOPYRIMIDINE DERIVATIVES AS PEST CONTROL AGENTS FOR AGRICULTURAL AND HORTICULTURAL USE 未知
公开(公告)号：IL217078D0
公开(公告)日：2012-02-29
申请号：IL21707811
申请日：2011-12-19
申请人： SDS BIOTECH CORP , SAKAI MASAAKI , MATSUMURA TOMOAKI , MIDORIKAWA SATOHIRO , NOMOTO TAKASHI , KATSUKI RYUTARO
IPC分类号： C07D20060101
摘要： Novel 4-(3-butynyl)aminopyrimidine derivatives represented by general formula [I] are useful as pest control agents. In general formula [I], R 1 is a mono- or bi-cyclic ring which may contain 0 to 3 heteroatoms, for example, phenyl or oxazolyl; R 2 is a hydrogen atom, -R, -OR, -C(O)OR, -C(O)NHR, -CONR 2 (wherein R is straight-chain or branched C 1-8 alkyl, or the like), hydroxyalkyl, or the like; R 3 is a hydrogen atom, a halogen atom, acyloxy represented by (straight-chain or branched C 1-8 aliphatic hydrocarbon group) -CO-O-, or the like; and R 4 is a hydrogen atom, a halogen atom, C 1-6 alkyl, or the like, or alternatively, R 4 and R 3 together with the carbon atoms on the pyrimidine ring may form a thiophene ring, a pyrrole ring, an imidazole ring, a benzene ring, a pyrimidine ring, a furan ring, a pyrazine ring, or a pyrrolidine ring.

2. 发明专利

IL227460D0 Agri- horicultural pest control compositiions comprising 4 - (3 - butynyl) aminopyrimidine derivatives 未知
公开(公告)号：IL227460D0
公开(公告)日：2013-09-30
申请号：IL22746013
申请日：2013-07-11
申请人： SDS BIOTECH CORP , SAKAI MASAAKI , MATSUMURA TOMOAKI , MIDORIKAWA SATOHIRO , KATSUKI RYUTARO , MURAKI TOMOKO , NOMOTO TAKASHI
IPC分类号： A01N20060101

3. 发明专利

IL217078A 4-(3-butynyl) aminopyrimidine derivatives as pest control agents for agricultural and horticultural use 未知
公开(公告)号：IL217078A
公开(公告)日：2015-05-31
申请号：IL21707811
申请日：2011-12-19
申请人： SDS BIOTECH CORP , SAKAI MASAAKI , MATSUMURA TOMOAKI , MIDORIKAWA SATOHIRO , NOMOTO TAKASHI , KATSUKI RYUTARO , MURAKI TOMOKO
发明人： SAKAI MASAAKI , MATSUMURA TOMOAKI , MIDORIKAWA SATOHIRO , NOMOTO TAKASHI , KATSUKI RYUTARO , MURAKI TOMOKO
IPC分类号： A01N20060101 , C07D20060101 , C07F20060101
摘要： Novel 4-(3-butynyl)aminopyrimidine derivatives represented by general formula [I] are useful as pest control agents. In general formula [I], R 1 is a mono- or bi-cyclic ring which may contain 0 to 3 heteroatoms, for example, phenyl or oxazolyl; R 2 is a hydrogen atom, -R, -OR, -C(O)OR, -C(O)NHR, -CONR 2 (wherein R is straight-chain or branched C 1-8 alkyl, or the like), hydroxyalkyl, or the like; R 3 is a hydrogen atom, a halogen atom, acyloxy represented by (straight-chain or branched C 1-8 aliphatic hydrocarbon group) -CO-O-, or the like; and R 4 is a hydrogen atom, a halogen atom, C 1-6 alkyl, or the like, or alternatively, R 4 and R 3 together with the carbon atoms on the pyrimidine ring may form a thiophene ring, a pyrrole ring, an imidazole ring, a benzene ring, a pyrimidine ring, a furan ring, a pyrazine ring, or a pyrrolidine ring.

4. 发明申请

WO2011122714A1 Absorbent Product 审中-公开
标题翻译：吸收产品
公开(公告)号：WO2011122714A1
公开(公告)日：2011-10-06
申请号：PCT/JP2011/058754
申请日：2011-03-31
申请人： UNICHARM CORPORATION , NOMOTO, Takashi , ONOZUKA, Takashi
发明人： NOMOTO, Takashi , ONOZUKA, Takashi
IPC分类号： A61F13/15 , A61F13/472
CPC分类号： A61F13/5514 , A61F13/475 , A61F13/476
摘要： The skin contact side sheet is protected and fastening of the absorbent body is secured while reliably suppressing liquid leakage. The sanitary napkin 1 is provided with an absorbent body 2 including a liquid permeable skin contact side sheet 3, a liquid impermeable non-skin contact side sheet, and an absorbent core 5 arranged between these skin contact side sheet 3 and non-skin contact side sheet. A cover sheet which covers the surface of the skin contact side sheet 3 is provided. At the cover sheet, partition lines are used to define a front wing 10F and back wing 10B for fastening the absorbent body 2 to the clothing. At the time of use, the front wing and back wing are folded and extended at the front folded region 14F and the back folded region 14B and fastened to the clothing. The partition lines are formed so that the front folded region 14F is positioned at the outside in the longitudinal direction from the front end edge 5F of the absorbent core 5 and so that the back folded region 14B is positioned at the inside in the longitudinal direction from the back end edge 5B of the absorbent core 5.
摘要翻译：皮肤接触侧片被保护，并且确保吸收体的紧固而可靠地抑制液体泄漏。卫生巾1设置有吸收体2，其包括透液性皮肤接触侧片3，不透液性非皮肤接触侧片和设置在这些皮肤接触侧片3和非皮肤接触侧之间的吸收芯5 片。设置覆盖皮肤接触侧片材3的表面的覆盖片。在盖板上，分隔线用于限定用于将吸收体2紧固到衣服上的前翼10F和后翼10B。在使用时，前翼和后翼在前折叠区域14F和后折叠区域14B处被折叠并延伸并紧固到衣服上。分隔线形成为使得前折叠区域14F从吸收芯5的前端边缘5F沿长度方向定位在外侧，并且使得后折叠区域14B位于从纵向方向的内侧吸收芯5的后端缘5B。

5. 发明申请

WO2011122713A1 Individually Wrapped Absorbent Product 审中-公开
标题翻译：单独包裹的吸收产品
公开(公告)号：WO2011122713A1
公开(公告)日：2011-10-06
申请号：PCT/JP2011/058753
申请日：2011-03-31
申请人： UNICHARM CORPORATION , NOMOTO, Takashi , ONOZUKA, Takashi , OBA, Kenji
发明人： NOMOTO, Takashi , ONOZUKA, Takashi , OBA, Kenji
IPC分类号： A61F13/15 , A61F13/472 , A61F13/56
CPC分类号： A61F13/5514
摘要： A sanitary napkin is provided with an absorbent body (2) which includes a liquid permeable skin contact side sheet (3), a liquid impermeable non-skin contact side sheet (4), and an absorbent core (5) which is arranged between these skin contact side sheet (3) and non-skin contact side sheet (4) and with a cover sheet (8) which covers the surface of the skin contact side sheet (3). An individually wrapped product (1W) is formed by wrapping the napkin (1R) in the ready-to-wrap state by the wrapping material (20). The wrapping material (20) includes a belt-shaped material (21) which surrounds the ready-to-wrap napkin (1R) across the entire circumference of the ready-to-wrap napkin (1R). A width (LW) of the belt-shaped material (21) is shorter than a length (LN) of the ready-to-wrap napkin (1R) in the width direction of the belt-shaped material (21).
摘要翻译：卫生巾设置有吸收体（2），其包括透液性皮肤接触侧片（3），不透液性非皮肤接触侧片（4）和吸收芯（5）皮肤接触侧片（3）和非皮肤接触侧片（4）以及覆盖皮肤接触侧片（3）的表面的覆盖片（8）。单独包装的产品（1W）通过用包装材料（20）将卫生巾（1R）包裹在即将包装状态中而形成。包装材料（20）包括穿过即将包装的卫生巾（1R）的整个圆周包围即将包裹的卫生巾（1R）的带状材料（21）。带状材料（21）的宽度（LW）比带状材料（21）的宽度方向上的即将包装的卫生巾（1R）的长度（LN）短。

6. 发明申请

WO1998005641A1 FLUORINATED 1,4-DISUBSTITUTED PIPERIDINE DERIVATIVES 审中-公开
标题翻译：氟化1,4-取代的哌啶衍生物
公开(公告)号：WO1998005641A1
公开(公告)日：1998-02-12
申请号：PCT/JP1997002600
申请日：1997-07-28
申请人： BANYU PHARMACEUTICAL CO., LTD. , TSUCHIYA, Yoshimi , NOMOTO, Takashi , OHSAWA, Hirokazu , KAWAKAMI, Kumiko , OHWAKI, Kenji , NISHIKIBE, Masaru
发明人： BANYU PHARMACEUTICAL CO., LTD.
IPC分类号： C07D211/46
CPC分类号： C07D401/06 , C07D211/58 , C07D405/06 , C07D409/06
摘要： Novel fluorinated 1,4-disubstituted piperidine derivatives represented by general formula (I) or pharmaceutically acceptable salts thereof, wherein Ar represents aryl or heteroaryl having 1 or 2 heteroatoms selected from the group consisting of nitrogen, oxygen and sulphur in which one to three hydrogen atoms on the aryl or heteroaryl ring may be substituted by lower alkyl, etc.; R represents C1-3 cycloalkyl in which one to four arbitrary hydrogen atoms may be substituted by fluorine; R represents saturated or unsaturated, aliphatic C5-15 hydrocarbon in which one to six arbitrary hydrogen atoms may be substituted by fluorine, aralkyl, arylalkenyl, or heteroarylalkyl or heteroarylalkenyl having one or two heteroatoms selected from the group consisting of nitrogen, oxygen and sulfur, in which one to three hydrogen atoms on the aralkyl, arylalkenyl, heteroarylalkyl or heteroarylalkenyl ring may be substituted by lower alkyl, trifluoromethyl, cyano, hydroxy, nitro, lower alkoxycarbonyl, halogeno, lower alkoxy, amino, etc.; and X represents O or NH, provided that at least one of R and R has one or more fluorine atoms. Because of having selective muscarinic receptor antagonism and being excellent in oral activity, persistence of the action and dynamic in vivo, these compounds are useful as efficacious and safe remedies or preventives with little side effects for respiratory, urologic and digestive diseases.
摘要翻译：由通式（I）表示的新型氟化1,4-二取代哌啶衍生物或其药学上可接受的盐，其中Ar表示具有1或2个选自氮，氧和硫的杂原子的芳基或杂芳基，其中一至三个氢芳基或杂芳基环上的原子可以被低级烷基等取代; R 1表示其中一至四个任意氢原子可被氟取代的C 1-3环烷基; R 2表示饱和或不饱和的脂族C 5-15烃，其中一至六个任意氢原子可被氟，芳烷基，芳基烯基或具有一个或两个选自氮，氧的杂芳基烷基或杂芳基烯基取代和其中芳烷基，芳基烯基，杂芳基烷基或杂芳基烯基环上的一至三个氢原子可被低级烷基，三氟甲基，氰基，羟基，硝基，低级烷氧基羰基，卤代，低级烷氧基，氨基等取代的硫。并且X表示O或NH，条件是R 1和R 2中的至少一个具有一个或多个氟原子。由于具有选择性的毒蕈碱受体拮抗作用，口服活性优异，作用持久，体内动态，因此这些化合物作为呼吸系统，泌尿系统和消化系统疾病副作用少的有效和安全的补救措施或预防措施是有用的。

7. 发明申请

WO1997045414A1 1,4-DISUBSTITUTED PIPERIDINE DERIVATIVES 审中-公开
标题翻译： 1,4-取代的哌啶衍生物
公开(公告)号：WO1997045414A1
公开(公告)日：1997-12-04
申请号：PCT/JP1997001770
申请日：1997-05-27
申请人： BANYU PHARMACEUTICAL CO., LTD. , TSUCHIYA, Yoshimi , NOMOTO, Takashi , OHSAWA, Hirokazu , KAWAKAMI, Kumiko , OHWAKI, Kenji , NISHIKIBE, Masaru
发明人： BANYU PHARMACEUTICAL CO., LTD.
IPC分类号： C07D211/58
CPC分类号： C07D211/58
摘要： 1,4-Disubstituted piperidine derivatives represented by general formula (I) and pharmaceutically acceptable salts thereof, wherein Ar represents heteroaryl having one or two heteroatoms selected from the group consisting of nitrogen, oxygen and sulfur and optionally fused to aryl or benzene (wherein each hydrogen on the aryl and heteroaryl rings may be substituted by lower alkyl, halogeno, lower alkoxy, amino or hydroxymethyl); R represents C3-6 cycloalkyl having one or two hydroxyl groups on the ring; R represents heteroarylalkyl having one or two heteroatoms selected from the group consisting of nitrogen, oxygen and sulfur and optionally fused to saturated or unsaturated aliphatic C5-15 hydrocarbon, aralkyl, arylalkenyl or benzene (wherein each hydrogen on the aralkyl, arylalkenyl and heteroarylalkyl rings may be substituted by lower alkyl, halogeno, lower alkoxy, amino or hydroxymethyl); and X represents O or NH. Because of having a selective muscarine M3 receptor antagonism, these compounds are useful as safe remedies or preventives with little side effects for respiratory diseases such as asthma, chronic respiratory obstruction and pulmonary fibrosis; urologic diseases in association with urination disorders such as frequent urination, urgency of micturition and urinary incontinence; and digestive diseases such as irritable bowel syndrome and convulsion or motor hyperenergia of digestive tracts.
摘要翻译：由通式（I）表示的1,4-二取代哌啶衍生物及其药学上可接受的盐，其中Ar表示具有一个或两个选自氮，氧和硫并且任选地与芳基或苯稠合的杂原子的杂芳基（其中每个芳基和杂芳基环上的氢可以被低级烷基，卤代，低级烷氧基，氨基或羟甲基取代）; R 1表示在环上具有一个或两个羟基的C 3-6环烷基; R 2表示具有一个或两个选自氮，氧和硫的杂原子的杂芳基烷基，并且任选地与饱和或不饱和的脂族C 5-15烃，芳烷基，芳基烯基或苯稠合（其中芳烷基上的每个氢，芳烯基烯基和杂芳基烷基环可以被低级烷基，卤代，低级烷氧基，氨基或羟甲基取代）; X表示O或NH。由于具有选择性的毒蕈碱M3受体拮抗作用，这些化合物可用作对哮喘，慢性呼吸阻塞和肺纤维化等呼吸系统疾病具有副作用的安全补救措施或预防药物; 泌尿系统疾病与排尿障碍如排尿紧急，排尿紧急和尿失禁有关; 消化道疾病如肠易激综合征，消化道惊厥或运动过敏等。

8. 发明申请

WO1996033973A1 1,4-DISUBSTITUTED PIPERIDINE DERIVATIVES 审中-公开
标题翻译： 1,4-取代的哌啶衍生物
公开(公告)号：WO1996033973A1
公开(公告)日：1996-10-31
申请号：PCT/JP1996001128
申请日：1996-04-25
申请人： BANYU PHARMACEUTICAL CO., LTD. , TSUCHIYA, Yoshimi , NOMOTO, Takashi , OHSAWA, Hirokazu , KAWAKAMI, Kumiko , OHWAKI, Kenji , NISHIKIBE, Masaru
发明人： BANYU PHARMACEUTICAL CO., LTD.
IPC分类号： C07D211/46
CPC分类号： C07D401/12 , C07D211/46 , C07D211/58 , C07D405/12 , C07D409/12 , C07D417/12
摘要： Novel 1,4-disubstituted piperidine derivatives represented by general formula (I) and pharmaceutically acceptable salts thereof, wherein Ar represents phenyl wherein one or two arbitrary hydrogen atoms on its ring may be substituted by substituent(s) selected from the group consisting of halogeno and lower alkyl or an aromatic 5- or 6-membered heterocycle having one or two heteroatoms selected from the group consisting of oxygen, nitrogen and sulfur; R represents C3-6 cycloalkyl or C3-6 cycloalkenyl; R represents saturated or unsaturated aliphatic C5-15 hydrocarbon group; and X represents O or NH. The compounds have a selective antagonism against the muscarine M3 receptor and a high safety with little side effect. Thus they are useful in the treatment or prevention of respiratory diseases such as asthma, chronic respiratory obstruction and pulmonary fibrosis, urological diseases accompanied with urination disorders such as frequent urination, urgency of micturition and urinary incontinence and digestive diseases such as convulsion or motion hyperenergia of the digestive tracts and irritable large intestine.
摘要翻译：由通式（I）表示的新的1,4-二取代哌啶衍生物及其药学上可接受的盐，其中Ar表示苯基，其中其一个或两个任意的氢原子可以被选自以下的取代基取代：卤代和具有一个或两个选自氧，氮和硫的杂原子的低级烷基或芳族5-或6-元杂环; R 1表示C 3-6环烷基或C 3-6环烯基; R 2表示饱和或不饱和的脂族C 5-15烃基; X表示O或NH。这些化合物对毒蕈碱M3受体具有选择性拮抗作用，安全性高，副作用小。因此，它们可用于治疗或预防呼吸系统疾病如哮喘，慢性呼吸阻塞和肺纤维化，泌尿系统疾病伴随排尿障碍，例如尿频，排尿紧急和尿失禁以及消化系统疾病如惊厥或运动过敏消化道和易怒大肠。

9. 发明申请

WO1993024478A1 SUBSTITUTED HETEROCYCLIC DERIVATIVE HAVING SQUALENE EPOXIDASE INHIBITORY EFFECT AND USE THEREOF 审中-公开
标题翻译：具有平均环氧化酶抑制作用的取代的杂环衍生物及其用途
公开(公告)号：WO1993024478A1
公开(公告)日：1993-12-09
申请号：PCT/JP1993000723
申请日：1993-05-28
申请人： BANYU PHARMACEUTICAL CO., LTD. , TSUCHIYA, Yoshimi , NOMOTO, Takashi , MITSUYA, Morihiro , NONOSHITA, Katsumasa , HAYASHI, Masahiro , SATO, Toshihiko , SAWASAKI, Yoshio , KAMEI, Toshio
发明人： BANYU PHARMACEUTICAL CO., LTD.
IPC分类号： C07D333/16
CPC分类号： C07D333/08 , C07D333/16 , C07D333/18 , C07D333/24
摘要： A substituted heterocyclic derivative represented by general formula (I), wherein R represents a 5- or 6-membered heterocyclic group containing one or two heteroatoms selected from among nitrogen and other atoms; Q represents (II), (III), -CH=CH-CH2-, etc., -CH2-O-CH2-, or thrimethylene; X and Y may be the same or different from each other and each represents methylene, oxygen, etc., or alternatively X and Y may be combined together to represent vinylene, etc.; Q represents either (a) a 5- or 6-membered aromatic group represented by (IV) wherein A &cir& _, B &cir& _, D &cir& _ and E &cir& _ represent each nitrogen, etc., or =CH-; and p represents an integer of 0 or 1, or (b) a group represented by -F &cir& _-G &cir& _-I &cir& _- wherein F &cir& _, G &cir& _ and I &cir& _ may be the same or different from each other and each represents oxygen, etc., or =CH-; R represents lowr alkyl, etc.; Q represents ethylene, etc.; Q represents vinylene, etc.; R and R may be the same or different from each other and each represents lower alkyl, or alternatively R and R are combined together with the adjacent carbon atom to represent cycloalkyl; and R represents hydrogen, lower alkyl, etc.
摘要翻译：由通式（I）表示的取代的杂环衍生物，其中R表示含有一个或两个选自氮原子和其它原子的杂原子的5-或6-元杂环基; Q 1表示（II），（III），-CH = CH-CH 2 - 等，-CH 2 -O-CH 2 - 或三亚甲基; X和Y可以相同或不同，各自表示亚甲基，氧等，或者X和Y可以组合在一起代表亚乙烯基等; Q 2表示（a）由（IV）表示的5或6元芳族基团，其中A 1和R 3各自表示每个氮等，或= CH- ; 并且p表示0或1的整数，或（b）由-F 1和R 3表示的基团，其中F 1和R 3可以相同或不同彼此各自表示氧等，或= CH-; R 1表示低级烷基等; Q 3表示乙烯等。 Q 4表示亚乙烯基等; R 2和R 3可以彼此相同或不同，并且各自表示低级烷基，或者R 2和R 3与相邻的碳原子一起代表环烷基; R 4表示氢，低级烷基等。

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