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1. 发明申请

WO2005005376A8 FUNGICIDAL PHENOXYPHENYLHYDRAZINE DERIVATIVES 审中-公开
标题翻译：杀真菌剂苯氧基衍生物
公开(公告)号：WO2005005376A8
公开(公告)日：2007-01-18
申请号：PCT/US2004016324
申请日：2004-05-25
申请人： UNIROYAL CHEM CO INC , CROMPTON CO CIE , CHEE GAIK-LEE , DEKEYSER MARK A , SEEBOLD KENNETH W JR , OSIKA EWA MARIA , BROUWER WALTER G , PARK SHELDON B , LAI HOI KIONG
发明人： CHEE GAIK-LEE , DEKEYSER MARK A , SEEBOLD KENNETH W JR , OSIKA EWA MARIA , BROUWER WALTER G , PARK SHELDON B , LAI HOI KIONG
IPC分类号： C07C323/48 , C07D213/77 , C07D249/08
CPC分类号： C07D213/77 , C07C243/22 , C07C243/28 , C07C281/02 , C07C281/20 , C07C323/48 , C07D249/08
摘要： A fungicidally active compound of the formula: wherein Q is -NY-NH-,-N=N-,or X is oxygen, sulfur, sulfoxide, or sulfone; n is 0 or 1; Y is hydrogen, C 1 -C 4 alkanoyl, C 1 -C 6 haloalkanoyl, C 1 -C 6 straight chain or branched alkoxycarbonyl, C 1 -C 4 alkoxy(C 1 -C 4 ) alkoxycarbonyl, C 1 -C 4 alkyl, or C 1 -C 4 haloalkyl; R 1 is C 1 -C 6 alkoxy, C 3 -C 6 branched alkoxy, C 3 -C 6 cycloalkoxy, phenoxy, benzyloxy, C 2 -C 6 alkenyloxy, C 2 -C 6 alkynyloxy, C 1 -C 6 haloalkoxy, silyloxy, (C 1 -C 6 alkoxy)-carbonylmethoxy, C 1 -C 6 thioalkoxy, C 1 -C 6 alkylamino, C 1 -C 6 alkyl, C 3 -C 6 branched alkyl, (C 1 -C 6 alkoxy) C 1 -C 6 alkoxy, or (C 1 -C 6 alkoxy)carbonyl; R 2 and R 3 are each, independently, hydrogen, halogen, C 1 -C 6 alkyl, C 3 -C 6 branched alkyl, C 1 -C 6 haloalkyl, C 1 -C 6 alkoxy, C 1 -C 6 haloalkoxy, cyano, or (C 1 -C 6 alkoxy) carbonyl; R 4 is C 1 -C 6 alkyl; and Z 1 and Z 2 are each independently, carbon or nitrogen with the proviso that when Z 1 is carbon, X is oxygen, and R 2 is hydrogen, then R 3 cannot be hydrogen; wherein R 5 is C 1 -C 6 alkoxy; an R 6 and R 7 are, independently halo or C 1 -C 6 haloalkyl, or wherein R 8 is C 1 -C 6 alkyl; and R 9 and R 10 , independently, are halo or C 1 -C 6 haloalkyl, and a method for controlling fungi using the compound.
摘要翻译：一种杀真菌活性的下式化合物：其中Q为-NY-NH - ， - N = N-，或X为氧，硫，亚砜或砜; n为0或1; Y是氢，C 1 -C 4烷酰基，C 1 -C 6卤代烷酰基，C 1 -C 4烷基， C 1 -C 6直链或支链烷氧基羰基，C 1 -C 4烷氧基（C 1 -C 12 - C 1 -C 4烷氧基羰基，C 1 -C 4烷基或C 1 -C 4烷基， 4卤代烷基; R 1是C 1 -C 6烷氧基，C 3 -C 6烷基，C 1 -C 6烷基，C 1 -C 6烷基，支链烷氧基，C 3 -C 6环烷氧基，苯氧基，苄氧基，C 2 -C 6链烯氧基，C C 1 -C 6烷氧基，C 1 -C 6卤代烷氧基，甲硅烷氧基，（C 1 -C 6）烷氧基， C 1 -C 6烷氧基） - 羰基甲氧基，C 1 -C 6硫代烷氧基，C 1 -C C 1 -C 6烷基氨基，C 1 -C 6烷基，C 3 -C 6烷基，C 1 -C 6 - 支链烷基，（C 1 -C 6烷氧基）C 1 -C 6烷氧基，或（C 1 -C 6 - C 1 -C 6烷氧基）羰基; R 2和R 3各自独立地为氢，卤素，C 1 -C 6烷基，C C 3 -C 6支链烷基，C 1 -C 6卤代烷基，C 1 -C 12 C 1 -C 6烷氧基，C 1 -C 6卤代烷氧基，氰基或（C 1 -C 3 - C 6 -C 6烷氧基）羰基; R 4是C 1 -C 6烷基; R 4是C 1 -C 6烷基; Z 1和Z 2各自独立地为碳或氮，条件是当Z 1是碳时，X是氧，R H 2是氢，则R 3不能是氢; 其中R 5是C 1 -C 6烷氧基; R 6和R 7独立地是卤素或C 1 -C 6卤代烷基，或其中R 1， SUP> 8是C 1 -C 6烷基; 和R 9和R 10独立地是卤素或C 1 -C 6卤代烷基，以及一种方法用于控制使用该化合物的真菌。

2. 发明申请

WO2005005376A2 FUNGICIDAL PHENOXYPHENYLHYDRAZINE DERIVATIVES 审中-公开
标题翻译：杀真菌苯氧基苯基肼衍生物
公开(公告)号：WO2005005376A2
公开(公告)日：2005-01-20
申请号：PCT/US2004016324
申请日：2004-05-25
申请人： UNIROYAL CHEM CO INC , CROMPTON CO CIE , CHEE GAIK-LEE , DEKEYSER MARK A , SEEBOLD KENNETH W JR , OSIKA EWA MARIA , BROUWER WALTER G , PARK SHELDON B , LAI HOI KIONG
发明人： CROMPTON CO CIE , CHEE GAIK-LEE , DEKEYSER MARK A , SEEBOLD KENNETH W JR , OSIKA EWA MARIA , BROUWER WALTER G , PARK SHELDON B , LAI HOI KIONG
IPC分类号： C07C323/48 , C07D213/77 , C07D249/08 , C07C281/02 , A01N37/28
CPC分类号： C07D213/77 , C07C243/22 , C07C243/28 , C07C281/02 , C07C281/20 , C07C323/48 , C07D249/08
摘要： A fungicidally active compound of the formula: wherein Q is -NY-NH-,-N=N-,or X is oxygen, sulfur, sulfoxide, or sulfone; n is 0 or 1; Y is hydrogen, C1-C4 alkanoyl, C1-C6 haloalkanoyl, C1-C6 straight chain or branched alkoxycarbonyl, C1-C4 alkoxy(C1-C4) alkoxycarbonyl, C1-C4 alkyl, or C1-C4 haloalkyl; R is C1-C6 alkoxy, C3-C6 branched alkoxy, C3-C6 cycloalkoxy, phenoxy, benzyloxy, C2-C6 alkenyloxy, C2-C6 alkynyloxy, C1-C6 haloalkoxy, silyloxy, (C1-C6 alkoxy)-carbonylmethoxy, C1-C6 thioalkoxy, C1-C6 alkylamino, C1-C6 alkyl, C3-C6 branched alkyl, (C1-C6 alkoxy) C1-C6 alkoxy, or (C1-C6 alkoxy)carbonyl; R and R are each, independently, hydrogen, halogen, C1-C6 alkyl, C3-C6 branched alkyl, C1-C6 haloalkyl, C1-C6 alkoxy, C1-C6 haloalkoxy, cyano, or (C1-C6 alkoxy) carbonyl; R is C1-C6 alkyl; and Z and Z are each independently, carbon or nitrogen with the proviso that when Z is carbon, X is oxygen, and R is hydrogen, then R cannot be hydrogen; wherein R is C1-C6 alkoxy; an R and R7 are, independently halo or C1-C6 haloalkyl, or wherein R is C1-C6 alkyl; and R and R , independently, are halo or C1-C6 haloalkyl, and a method for controlling fungi using the compound.
摘要翻译：具有下式的杀真菌活性化合物：其中Q是-NY-NH - ， - N = N-或X是氧，硫，亚砜或砜; n是0或1; Y是氢，C 1 -C 4烷酰基，C 1 -C 6卤代烷酰基，C 1 -C 6直链或支链烷氧基羰基，C 1 -C 4烷氧基（C 1 -C 4）烷氧基羰基，C 1 -C 4烷基或C 1 -C 4卤代烷基; R 1是C 1 -C 6烷氧基，C 3 -C 6支链烷氧基，C 3 -C 6环烷氧基，苯氧基，苄氧基，C 2 -C 6烯氧基，C 2 -C 6炔氧基，C 1 -C 6卤代烷氧基，甲硅烷氧基，（C 1 -C 6烷氧基） C 1 -C 6烷基氨基，C 1 -C 6烷基，C 3 -C 6支链烷基，（C 1 -C 6烷氧基）C 1 -C 6烷氧基或（C 1 -C 6烷氧基）羰基; R 2和R 3各自独立地为氢，卤素，C 1 -C 6烷基，C 3 -C 6支链烷基，C 1 -C 6卤代烷基，C 1 -C 6烷氧基，C 1 -C 6卤代烷氧基，氰基或（C 1 -C 6） C6烷氧基）羰基; R 4是C 1 -C 6烷基; Z 1和Z 2各自独立地为碳或氮，条件是当Z 1为碳时，X为氧且R 2为氢，则R 3不能为氢; 其中R 5是C 1 -C 6烷氧基; R 6和R 7独立地为卤代或C 1 -C 6卤代烷基，或者其中R 8为C 1 -C 6烷基; 并且R 9和R 10独立地为卤代或C 1 -C 6卤代烷基，和使用该化合物防治真菌的方法。

3. 发明申请

WO2012024083A9 OXATHIAZINE AND DITHIINE OXIDES AS INHIBITORS OF SULFHYDRYL-DEPENDENT BIOMOLECULES 审中-公开
标题翻译：作为巯基依赖性生物分子抑制剂的硫嘌呤和酪氨酸氧化物
公开(公告)号：WO2012024083A9
公开(公告)日：2012-10-04
申请号：PCT/US2011046355
申请日：2011-08-03
申请人： CHEMTURA CORP , UNIV MANITOBA , CHEE GAIK-LEAN , BROUWER WALTER G , OSIKA EWA , HASINOFF BRIAN B , BREWER A DAVID
发明人： CHEE GAIK-LEAN , BROUWER WALTER G , OSIKA EWA , HASINOFF BRIAN B , BREWER A DAVID
IPC分类号： C07D291/06 , A61K31/385 , A61K31/54 , A61P35/00 , C07D339/08
CPC分类号： C07D291/06 , A61K31/385 , A61K31/54 , C07D339/08
摘要： Novel derivatives of dihydro-l,4,2-oxathiazine and dihydro-l,4-dithiine oxides, more particularly, novel derivatives of dihydro-l,4,2-oxathiazine and dmydro-l,4-dithiine oxides that target cysteine residues of biomolecules of pharmacological importance are provided as pharmaceutically useful compounds, for example, as anticancer, antiinfectious, antigastric acid secretion, antiosteoporosic, and antiinflammatory agents.
摘要翻译：二氢-1,4,2-氧杂噻嗪和二氢-1,4-二硫杂环己烯氧化物的新衍生物，更具体地说是靶向半胱氨酸残基的二氢-1,4,2-氧杂噻嗪和二氢-1,4-二硫基氧化物的新衍生物提供药理学重要性的生物分子作为药学上有用的化合物，例如，作为抗癌剂，抗感染剂，抗胃酸分泌剂，抗骨质疏松剂和抗炎剂。

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