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1. 发明授权

US06506939B1 Production of acrylic monomers 失效
标题翻译：生产丙烯酸单体
公开(公告)号：US06506939B1
公开(公告)日：2003-01-14
申请号：US09889281
申请日：2001-07-13
申请人： Peter Stuart Littlewood , Michael Singh
发明人： Peter Stuart Littlewood , Michael Singh
IPC分类号： C07C23309
CPC分类号： C07C231/12 , C07C209/62
摘要： A process for the preparation of a mixture comprising a compound of formula (1) and a compound of formula (2) wherein R1 is an optionally substituted C1-20 alkyl, optionally substituted C3-4 alkenyl, optionally substituted C5-7 cycloalkyl or optionally substituted benzyl, R2 is an optionally substituted C1-20 alkyl, optionally substituted C3-4 alkenyl or optionally substituted C5-7 cycloalkyl, A is either S or NR3, R3 is an optionally substituted C1-20 alkyl, optionally substituted C3-4 alkenyl or optionally substituted C5-7 cycloalkyl, or R2 and R3 together form a 5-7 membered ring which can contain an oxygen atom, R4 is hydrogen or methyl, R5 is an optionally substituted C1-20 alkyl, optionally substituted C3-4 alkenyl, optionally substituted C5-7 cycloalkyl or optionally substituted benzyl and, R6 is hydrogen or an optionally substituted C1-20 alkyl, optionally substituted C3-4 alkenyl or optionally substituted C5-7 cycloalkyl, or R5 and R6 together form a 5-7 membered ring which can contain an oxygen atom, which comprises reacting in an alkaline or base medium a compound of formula (3) wherein X− is an anion, R1, R2, R3, R4, R5 and R6 have the same meaning as above, A+ is S+ or N+R3.
摘要翻译：一种制备包含式（1）化合物和式（2）化合物的混合物的方法，其中R 1是任选取代的C 1-20烷基，任选取代的C 3-4烯基，任选取代的C 5-7环烷基或任选地取代的苄基，R2是任选取代的C 1-20烷基，任选取代的C 3-4烯基或任选取代的C 5-7环烷基，A是S或NR 3，R 3是任选取代的C 1-20烷基，任选取代的C 3-4烯基或任选取代的C 5-7环烷基，或R 2和R 3一起形成可含有氧原子的5-7元环，R 4为氢或甲基，R 5为任选取代的C 1-20烷基，任选取代的C 3-4烯基，任选取代的C 5-7环烷基或任选取代的苄基，R 6是氢或任选取代的C 1-20烷基，任选取代的C 3-4烯基或任选取代的C 5-7环烷基，或者R 5和R 6一起形成5-7元环哪个行包含氧原子，其包括在碱性或碱性介质中使式（3）化合物（其中X是阴离子）R1，R2，R3，R4，R5和R6具有与上述相同的含义，A +是S +或 N + R3。

2. 发明授权

US06504057B2 Fluorophenyl-substituted alkenylcarboxylic acid guanidides, process for their preparation, their use as a medicament or diagnostic, and medicament containing them 失效
标题翻译：氟苯基取代的烯基羧酸胍苷，其制备方法，它们作为药物或诊断剂的用途，以及含有它们的药物
公开(公告)号：US06504057B2
公开(公告)日：2003-01-07
申请号：US10024388
申请日：2001-12-20
申请人： Jan-Robert Schwark , Hans-Jochen Lang , Heinz-Werner Kleemann , Andreas Weichert , Wolfgang Scholz , Udo Albus
发明人： Jan-Robert Schwark , Hans-Jochen Lang , Heinz-Werner Kleemann , Andreas Weichert , Wolfgang Scholz , Udo Albus
IPC分类号： C07C23309
CPC分类号： C07C279/22
摘要： This invention relates to fluorophenyl-substituted alkenylcarboxylic acid guanidides, process for their preparation, their use as a medicament or diagnostic, and medicament containing them. An embodiment of the invention embraces compounds of the formula I: and the pharmaceutically tolerated salts thereof. The disclosed compounds are valuable inhibitors of the cellular sodium/proton exchanger (Na+ /H+ exchanger) . They are therefore outstandingly suitable for the treatment of all diseases attributable to increased Na+ /H+ exchange.
摘要翻译：本发明涉及氟苯基取代的烯基羧酸胍，其制备方法，它们作为药物或诊断剂的用途，以及含有它们的药物。本发明的一个实施方案包括式I化合物及其药学上可耐受的盐。所公开的化合物是细胞钠/质子交换剂（Na + / H +交换剂）的有价值的抑制剂。因此，它们非常适合用于治疗由于增加的Na + / H +交换而引起的所有疾病。

3. 发明授权

US06787670B1 Glyoxyl acid amides, method for producing them and their use for controlling harmful organisms 失效
标题翻译：乙氧基酰胺，它们的制备方法及其用于控制有害生物的用途
公开(公告)号：US06787670B1
公开(公告)日：2004-09-07
申请号：US10130899
申请日：2002-05-23
申请人： Christiane Boie , Thomas Seitz , Ulrich Heinemann , Reiner Fischer , Martin Vaupel , Ulrike Wachendorff-Neumann , Karl-Heinz Kuck
发明人： Christiane Boie , Thomas Seitz , Ulrich Heinemann , Reiner Fischer , Martin Vaupel , Ulrike Wachendorff-Neumann , Karl-Heinz Kuck
IPC分类号： C07C23309
CPC分类号： C07C251/48 , C07C2602/08 , C07C2602/10
摘要： The invention relates to novel gloyoxylic acid amides, to a process for their preparation and to their use for controlling harmful organisms.
摘要翻译：本发明涉及新型的羟丙酸酰胺，其制备方法及其用于控制有害生物体的用途。

4. 发明授权

US06696607B2 Use of phenethyl acrylamides, novel phenethyl acrylamides, method for the production thereof and agents containing the same 失效
标题翻译：使用苯乙基丙烯酰胺，新型苯乙基丙烯酰胺，其制备方法和含有它们的试剂
公开(公告)号：US06696607B2
公开(公告)日：2004-02-24
申请号：US10297287
申请日：2002-12-04
申请人： Wassilios Grammenos , Hubert Sauter , Oliver Cullmann , Markus Gewehr , Bernd Müller , Jordi Tormo i Blasco , Norbert Götz , Thorsten Volk , Gisela Lorenz , Eberhard Ammermann , Reinhard Stierl , Siegfried Strathmann
发明人： Wassilios Grammenos , Hubert Sauter , Oliver Cullmann , Markus Gewehr , Bernd Müller , Jordi Tormo i Blasco , Norbert Götz , Thorsten Volk , Gisela Lorenz , Eberhard Ammermann , Reinhard Stierl , Siegfried Strathmann
IPC分类号： C07C23309
CPC分类号： A01N37/36 , A01N37/18 , A01N37/38 , C07C231/02 , C07C233/22
摘要： Use of phenethylacrylamides of the formula I: in which the substituents have the following meanings: X is halogen, alkyl, haloalkyl, alkoxy, haloalkoxy and —O—C(Ra,Rb)—C≡C—R6; Ra,Rb and Rc have the meanings given in the description; m,n independently of one another are 1 to 4, it being possible for the radicals X or Y to be different if m or n is greater than 1; Y is halogen, nitro, cyano, alkyl, CF3, alkoxy and phenyl; R1,R2 independently of one another are hydrogen, halogen, alkyl, alkoxy, haloalkoxy and CF3; R3,R4,R5,R6 independently of one another are hydrogen, halogen, alkyl, alkoxy, or R3 and R4 together form a cyclopropyl ring, it being possible for the C—R5— and C—R6 bonds can be in the E- or Z-position relative to each other; for controlling phytopathogenic fungal pests, novel phenethylacrylamides, their preparation, and compositions comprising them.
摘要翻译：使用式I的苯乙基丙烯酰胺：其中取代基具有以下含义：X是卤素，烷基，卤代烷基，烷氧基，卤代烷氧基和-OC（R a，R b）-C = CR 6; R a，R b和R c具有说明书中给出的含义; m，n彼此独立地为1至4，如果m或n可以使基团X或Y不同大于1; Y是卤素，硝基，氰基，烷基，CF 3，烷氧基和苯基; R 1，R 2彼此独立地是氢，卤素，烷基，烷氧基，卤代烷氧基和CF 3; R 3 R 4，R 5，R 6彼此独立地是氢，卤素，烷基，烷氧基或R 3和R 4一起形成环丙基环，其中CR <5> - 和CR 6键可以相对于彼此位于E-或Z-位;用于控制植物病原性真菌害虫，新型苯乙基丙烯酰胺，它们的制备和包含它们的组合物。

5. 发明授权

US06469209B1 Acrylate-type fungicide 失效
标题翻译：丙烯酸酯类杀菌剂
公开(公告)号：US06469209B1
公开(公告)日：2002-10-22
申请号：US10009701
申请日：2001-12-14
申请人： Hong Lim , Bong Jin Chung , Jong Sang Chung , In Young Choi , Dae Jong Park , Chang Il Hwang
发明人： Hong Lim , Bong Jin Chung , Jong Sang Chung , In Young Choi , Dae Jong Park , Chang Il Hwang
IPC分类号： C07C23309
CPC分类号： A01N37/50
摘要： The present invention relates to novel acrylate-type N-methyl E-2-(2-methylphenyl)oxymethyl)-6-methylphenyl-glyoxylamide O-methyl oxime represented by formula (1), its preparation method and its use as fungicides. The compound of the present invention has not only stronger fungicidal effect on plant pathogens at low concentrations but also broader fungicidal spectrum than the conventional fungicides. Especially, because the compound has excellent systemic and curative effect as well as no toxicity, it can be used as an efficacious agricultural fungicide. In addition, the compound of the present invention can be useful as environmental-friendly fungicide capable of causing less environmental pollution fungicide due to its strong fungicidal effect at low concentrations.
摘要翻译：本发明涉及由式（1）表示的新型丙烯酸酯型N-甲基E-2-（2-甲基苯基）氧甲基）-6-甲基苯基 - 乙醛酰胺O-甲基肟，其制备方法及其作为杀真菌剂的用途。本发明的化合物不仅具有比常规杀真菌剂在低浓度下对植物病原体更强的杀真菌作用，而且具有更广泛的杀真菌作用。特别是因为该化合物具有优异的全身和治疗效果以及无毒性，因此可用作有效的农药杀菌剂。此外，本发明的化合物由于其在低浓度下具有强烈的杀真菌作用，因此可用作能够减少环境污染杀真菌剂的环保杀真菌剂。

6. 发明授权

US06426435B1 Substantive water-soluble bis-quaternary salts of cinnamidoalkylamines 失效
标题翻译：肉桂酰胺基烷基胺的实质性水溶性双季盐
公开(公告)号：US06426435B1
公开(公告)日：2002-07-30
申请号：US09917953
申请日：2001-07-31
申请人： Nirmal Madhukar Koshti , Arun Harchandra Jawale , Bharat Bhikaji Parab , Shubhangi Dattaram Naik , Manasi Dattatraya Moghe , Tanaji Shamrao Jadhav , Subhash Shivling Nashte
发明人： Nirmal Madhukar Koshti , Arun Harchandra Jawale , Bharat Bhikaji Parab , Shubhangi Dattaram Naik , Manasi Dattatraya Moghe , Tanaji Shamrao Jadhav , Subhash Shivling Nashte
IPC分类号： C07C23309
CPC分类号： C07C233/40 , A61K8/416 , A61Q5/02 , A61Q5/12 , A61Q17/04 , C11D3/28
摘要： Substantive UV-absorbing water-soluble quaternary salts of cinnamidoalkylamine of formula I. Hair, skin and fabric care compositions containing the compounds of formula I; wherein R1 represents up to four substituents, same or different, selected from H, halo, —OH, —NH2, —NO2, —OCH3, —N(CH3)2, alkyl groups containing up to 6 carbon atoms, alkoxy groups containing up to 6 carbon atoms, alkylamino or N,N-dialkylamino groups containing up to 6 carbon atoms; R2 is selected from hydrogen, alkyl group containing up to 6 carbon atoms; R3 and R4 are independently selected from benzyl, alkyl group containing up to 6 carbon atoms; n is an integer from 1 to 6; m is an integer from 1 to 10; X− is a counter anion of quaternary centres selected from halides including chloride, bromide, iodide and methane sulphonate and its derivatives such as trifluoro methane sulphonate, benzene sulphonates including its p-bromo, nitro and methyl derivative.
摘要翻译：含有式I的肉桂酰胺基烷基胺的实质性紫外线吸收水溶性季盐。含有式I化合物的头发，皮肤和织物护理组合物;其中R1代表至多四个相同或不同的选自H，卤素，-OH， -NH 2，-NO 2，-OCH 3，-N（CH 3）2，含有至多6个碳原子的烷基，含有至多6个碳原子的烷氧基，含有至多6个碳原子的烷基氨基或N，N-二烷基氨基; R2选自氢，最多含6个碳原子的烷基; R3和R4独立地选自苄基，含有至多6个碳原子的烷基; n是1至6的整数; m为1〜10的整数; X-是选自卤化物（包括氯化物，溴化物，碘化物和甲磺酸盐）及其衍生物如三氟甲烷磺酸盐，苯磺酸盐，包括其对溴，硝基和甲基衍生物的季铵盐的抗衡阴离子。

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