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1. 发明授权

US07211572B2 Nitrogen-containing fused ring compound and use thereof as HIV integrase inhibitor 有权
标题翻译：含氮稠环化合物及其作为HIV整合酶抑制剂的用途
公开(公告)号：US07211572B2
公开(公告)日：2007-05-01
申请号：US11255605
申请日：2005-10-13
申请人： Susumu Miyazaki , Susumu Katoh , Kaoru Adachi , Hirotaka Isoshima , Satoru Kobayashi , Yuji Matsuzaki , Wataru Watanabe , Kazunobu Yamataka , Shinichi Kiyonari , Shuichi Wamaki
发明人： Susumu Miyazaki , Susumu Katoh , Kaoru Adachi , Hirotaka Isoshima , Satoru Kobayashi , Yuji Matsuzaki , Wataru Watanabe , Kazunobu Yamataka , Shinichi Kiyonari , Shuichi Wamaki
IPC分类号： A01N43/00 , A01N43/58 , A61K31/55 , A61K31/553 , A61K31/554
CPC分类号： C07D471/04 , C07D487/04
摘要： The present invention relates to a nitrogen-containing fused ring compound represented by the following formula [I] wherein each symbol is as defined in the specification, or a pharmaceutically acceptable salt thereof, and an anti-HIV agent containing such compound. The compound of the present invention has an HIV integrase inhibitory activity, and is useful as an agent for the prophylaxis or treatment of AIDS, or as an anti-HIV agent. In addition, by the combined use with other anti-HIV agents such as a protease inhibitor, a reverse transcriptase inhibitor and the like, it can be a more effective anti-HIV agent. Because it shows integrase-specific high inhibitory activity, the compound can be a pharmaceutical agent safe on human body, which causes only a fewer side effects.
摘要翻译：本发明涉及由下式[I]表示的含氮稠环化合物，其中每个符号如说明书中所定义，或其药学上可接受的盐和含有该化合物的抗HIV剂。本发明的化合物具有HIV整合酶抑制活性，可用作预防或治疗AIDS或作为抗HIV剂的药剂。此外，通过与其它抗HIV剂如蛋白酶抑制剂，逆转录酶抑制剂等的组合使用，它可以是更有效的抗HIV剂。因为它显示出整合酶特异性的高抑制活性，所以化合物可以是对人体安全的药剂，其副作用较小。

2. 发明申请

US20060052361A1 Nitrogen-containing fused ring compound and use thereof as HIV integrase inhibitor 有权
标题翻译：含氮稠环化合物及其作为HIV整合酶抑制剂的用途
公开(公告)号：US20060052361A1
公开(公告)日：2006-03-09
申请号：US11255605
申请日：2005-10-13
申请人： Susumu Miyazaki , Susumu Katoh , Kaoru Adachi , Hirotaka Isoshima , Satoru Kobayashi , Yuji Matsuzaki , Wataru Watanabe , Kazunobu Yamataka , Shinichi Kiyonari , Shuichi Wamaki
发明人： Susumu Miyazaki , Susumu Katoh , Kaoru Adachi , Hirotaka Isoshima , Satoru Kobayashi , Yuji Matsuzaki , Wataru Watanabe , Kazunobu Yamataka , Shinichi Kiyonari , Shuichi Wamaki
IPC分类号： A61K31/55 , A61K31/503 , A61K31/553 , A61K31/519
CPC分类号： C07D471/04 , C07D487/04
摘要： The present invention relates to a nitrogen-containing fused ring compound represented by the following formula [I] wherein each symbol is as defined in the specification, or a pharmaceutically acceptable salt thereof, and an anti-HIV agent containing such compound. The compound of the present invention has an HIV integrase inhibitory activity, and is useful as an agent for the prophylaxis or treatment of AIDS, or as an anti-HIV agent. In addition, by the combined use with other anti-HIV agents such as a protease inhibitor, a reverse transcriptase inhibitor and the like, it can be a more effective anti-HIV agent. Becuae it shows integrase-specific high inhibitory activity, the compound can be a pharmaceutical agent safe on human body, which causes only a fewer side effects.
摘要翻译：本发明涉及由下式[I]表示的含氮稠环化合物，

3. 发明申请

US20050054645A1 Nitrogen-containing fused ring compound and use thereof as HIV integrase inhibitor 审中-公开
标题翻译：含氮稠环化合物及其作为HIV整合酶抑制剂的用途
公开(公告)号：US20050054645A1
公开(公告)日：2005-03-10
申请号：US10958225
申请日：2004-10-05
申请人： Susumu Miyazaki , Susumu Katoh , Kaoru Adachi , Hirotaka Isoshima , Satoru Kobayashi , Yuji Matsuzaki , Wataru Watanabe , Kazunobu Yamataka , Shinichi Kiyonari , Shuichi Wamaki
发明人： Susumu Miyazaki , Susumu Katoh , Kaoru Adachi , Hirotaka Isoshima , Satoru Kobayashi , Yuji Matsuzaki , Wataru Watanabe , Kazunobu Yamataka , Shinichi Kiyonari , Shuichi Wamaki
IPC分类号： A61K31/4985 , A61K31/519 , A61K31/53 , A61K31/551 , A61P31/12 , A61P31/18 , A61P43/00 , C07D471/04 , C07D487/04
CPC分类号： C07D471/04 , C07D487/04
摘要： The present invention relates to a nitrogen-containing fused ring compound represented by the following formula [I] wherein each symbol is as defined in the specification, or a pharmaceutically acceptable salt thereof, and an anti-HIV agent containing such compound. The compound of the present invention has an HIV integrase inhibitory activity, and is useful as an agent for the prophylaxis or treatment of AIDS, or as an anti-HIV agent. In addition, by the combined use with other anti-HIV agents such as a protease inhibitor, a reverse transcriptase inhibitor and the like, it can be a more effective anti-HIV agent. Becuae it shows integrase-specific high inhibitory activity, the compound can be a pharmaceutical agent safe on human body, which causes only a fewer side effects.
摘要翻译：本发明涉及由下式[I]表示的含氮稠环化合物，其中每个符号如说明书中所定义，或其药学上可接受的盐和含有该化合物的抗HIV剂。本发明的化合物具有HIV整合酶抑制活性，可用作预防或治疗AIDS或作为抗HIV剂的药剂。此外，通过与其它抗HIV剂如蛋白酶抑制剂，逆转录酶抑制剂等的组合使用，它可以是更有效的抗HIV剂。它表现出整合酶特异性的高抑制活性，该化合物可以作为人体安全的药物，这只会减少副作用。

4. 发明申请

US20080161311A1 Nitrogen-containing fused ring compound and use thereof as HIV integrase inhibitor 审中-公开
标题翻译：含氮稠环化合物及其作为HIV整合酶抑制剂的用途
公开(公告)号：US20080161311A1
公开(公告)日：2008-07-03
申请号：US11783270
申请日：2007-04-06
申请人： Susumu Miyazaki , Susumu Katoh , Kaoru Adachi , Hirotaka Isoshima , Satoru Kobayashi , Yuji Matsuzaki , Wataru Watanabe , Kazunobu Yamataka , Shinichi Kiyonari , Shuichi Wamaki
发明人： Susumu Miyazaki , Susumu Katoh , Kaoru Adachi , Hirotaka Isoshima , Satoru Kobayashi , Yuji Matsuzaki , Wataru Watanabe , Kazunobu Yamataka , Shinichi Kiyonari , Shuichi Wamaki
IPC分类号： A61K31/519 , A61K31/503
CPC分类号： C07D471/04 , C07D487/04
摘要： The present invention relates to a nitrogen-containing fused ring compound represented by the following formula [I] wherein each symbol is as defined in the specification, or a pharmaceutically acceptable salt thereof, and an anti-HIV agent containing such compound. The compound of the present invention has an HIV integrase inhibitory activity, and is useful as an agent for the prophylaxis or treatment of AIDS, or as an anti-HIV agent. In addition, by the combined use with other anti-HIV agents such as a protease inhibitor, a reverse transcriptase inhibitor and the like, it can be a more effective anti-HIV agent. Because it shows integrase-specific high inhibitory activity, the compound can be a pharmaceutical agent safe on human body, which causes only a fewer side effects.
摘要翻译：本发明涉及由下式[I]表示的含氮稠环化合物，其中每个符号如说明书中所定义，或其药学上可接受的盐和含有该化合物的抗HIV剂。本发明的化合物具有HIV整合酶抑制活性，可用作预防或治疗AIDS或作为抗HIV剂的药剂。此外，通过与其它抗HIV剂如蛋白酶抑制剂，逆转录酶抑制剂等的组合使用，它可以是更有效的抗HIV剂。因为它显示出整合酶特异性的高抑制活性，所以化合物可以是对人体安全的药剂，其副作用较小。

5. 发明授权

US10065950B2 Substituted thiazoles as HIV integrase inhibitors 有权
公开(公告)号：US10065950B2
公开(公告)日：2018-09-04
申请号：US13034866
申请日：2011-02-25
申请人： Susumu Miyazaki , Yuki Bessho , Kaoru Adachi , Seiji Kawashita , Hirotaka Isoshima , Kengo Oshita , Shunichi Fukuda
发明人： Susumu Miyazaki , Yuki Bessho , Kaoru Adachi , Seiji Kawashita , Hirotaka Isoshima , Kengo Oshita , Shunichi Fukuda
IPC分类号： A61K31/427 , C07D277/20 , C07D471/04 , A61K31/4985 , A61K31/5377
摘要： [Problem] Provided is a novel 1,3,4,8-tetrahydro-2H-pyrido[1,2-a]pyrazine derivative or a pharmaceutically acceptable salt thereof, or a solvate thereof, which is useful as an anti-HIV agent.[Solving Means] The present invention provides a compound represented by the following formula [I] wherein each symbol is as defined in the specification, or a pharmaceutically acceptable salt thereof, or a solvate thereof.

6. 发明授权

US5428389A Image data storage/processing apparatus 失效
标题翻译：图像数据存储/处理装置
公开(公告)号：US5428389A
公开(公告)日：1995-06-27
申请号：US104928
申请日：1993-08-12
申请人： Kenji Ito , Kaoru Adachi , Osamu Saito
发明人： Kenji Ito , Kaoru Adachi , Osamu Saito
IPC分类号： G11C7/10 , H04N1/21 , H04N7/30 , H04N5/76 , H04N9/64
CPC分类号： H04N1/2137 , G11C7/1027 , H04N1/2112 , H04N1/2158 , H04N19/60
摘要： An image data storage/processing apparatus is provided, which is particularly applicable to an electronic still camera, for example. The image data storage apparatus uses a dynamic RAM as a frame memory for temporarily storing image data representative of a field of an image to be recorded. The frame memory includes at least first and second memories. In the apparatus, there is provided a control so that the image data corresponding to the adjacent two pixel lines on the field are continuously read out in such a manner that they are simultaneously read out from the first and second memories, and the image data corresponding to one of the two pixel lines are read out with delay by the time required for reading out of the image data corresponding to the other pixel line. The image signal processing apparatus is capable of performing processing for writing in and reading out of various types of image data with a single memory.
摘要翻译：提供了一种特别适用于电子静态照相机的图像数据存储/处理装置。图像数据存储装置使用动态RAM作为帧存储器，用于临时存储表示要记录的图像的场的图像数据。帧存储器至少包括第一和第二存储器。在该装置中，提供了一种控制，使得对应于场上的相邻两个像素线的图像数据以从第一和第二存储器同时读出的方式连续地读出，并且图像数据对应到两个像素线中的一个被延迟地读出对应于另一个像素线的图像数据所需的时间。图像信号处理装置能够执行用单个存储器写入和读出各种图像数据的处理。

7. 发明授权

US5352538A Surface hardened aluminum part and method of producing same 失效
标题翻译：表面硬化铝部件及其制造方法
公开(公告)号：US5352538A
公开(公告)日：1994-10-04
申请号：US937266
申请日：1992-08-31
申请人： Toshihide Takeda , Kaoru Adachi
发明人： Toshihide Takeda , Kaoru Adachi
IPC分类号： C23C24/08 , B22F7/08 , C23C24/10 , C23C26/00 , C23C26/02 , F02F3/12 , B22F7/04
CPC分类号： B22F7/08 , C23C24/103 , C23C26/02 , F02F3/12 , F05C2201/021 , F05C2201/0448 , Y10T428/12014 , Y10T428/12049 , Y10T428/12056 , Y10T428/12063 , Y10T428/12139
摘要： A surface hardened aluminum part having excellent heat resistance and abrasion resistance obtained by forming, on the surface of an aluminum base material, an alloy layer that has a uniform composition and uniform hardness, being free from cracks. An aluminum alloy powder made of aluminum and metals each of which forms an intermetallic compound of high hardness with aluminum is prepared. This aluminum alloy powder is supplied onto the aluminum base material and the aluminum or aluminum alloy contained in the aluminum base material is alloyed with the aluminum alloy powder using a high-density energy heat source to form an alloy layer. The alloy layer thus formed has an intermetallic compound of high hardness uniformly distributed throughout the layer so that the hardness of the alloy layer is uniform and cracking is unlikely to occur.
摘要翻译：通过在铝基材的表面上形成具有均匀组成和均匀硬度的合金层，没有裂纹而获得的具有优异的耐热性和耐磨性的表面硬化铝部分。制备由铝和金属制成的铝合金粉末，每种铝粉均与铝形成高硬度的金属间化合物。将该铝合金粉末供给到铝基材上，使用高密度能量热源将包含在铝基材中的铝或铝合金与铝合金粉末合金化，形成合金层。如此形成的合金层具有均匀分布在整个层中的高硬度的金属间化合物，使得合金层的硬度是均匀的，并且不可能发生开裂。

8. 发明授权

US5303198A Method of recording data in memory card having EEPROM and memory card system using the same 失效
标题翻译：在具有EEPROM的存储卡和使用其的存储卡系统中记录数据的方法
公开(公告)号：US5303198A
公开(公告)日：1994-04-12
申请号：US726173
申请日：1991-07-05
申请人： Kaoru Adachi , Kouichi Gouhara
发明人： Kaoru Adachi , Kouichi Gouhara
IPC分类号： G06K19/07 , G11C16/10 , G11C7/00
CPC分类号： G11C16/105 , G06K19/07 , G11C16/102 , G06F2212/2022
摘要： A method of recording data in a memory card having an EEPROM, and a memory card system using the same are provided. A memory card has at least two collective erasure type EEPROM chips where at least one of which is conditioned for a spare memory. When an access of the kind needing overwriting is made to the memory card, data stored in memory locations of the addresses of a corresponding EEPROM chip, except for the address where overwriting is to occur, are copied in the spare memory, and then the EEPROM chip of interest and the spare memory are replaced with each other. The EEPROM chips may be replaced with a plurality of memory blocks or clusters defined in a block erasure type EEPROM.
摘要翻译：提供了一种在具有EEPROM的存储卡中记录数据的方法和使用其的存储卡系统。存储卡具有至少两个集体擦除型EEPROM芯片，其中至少一个被调节为备用存储器。当对存储卡进行需要覆盖的存取时，存储在相应的EEPROM芯片的地址的存储位置中的数据除了要进行重写的地址之外，被复制到备用存储器中，然后EEPROM 感兴趣的芯片和备用存储器被彼此替换。 EEPROM芯片可以用在块擦除型EEPROM中定义的多个存储器块或簇代替。

9. 发明授权

US06727944B1 Digital electronic still-video camera and method of controlling operation of same 有权
标题翻译：数字电子静态摄像机及其操作方法
公开(公告)号：US06727944B1
公开(公告)日：2004-04-27
申请号：US09258423
申请日：1999-02-26
申请人： Kaoru Adachi
发明人： Kaoru Adachi
IPC分类号： H04N576
CPC分类号： H04N5/772 , H04N5/907
摘要： Consumption of power in a digital electronic still-video camera is reduced. Specifically, a digital electronic still-video camera includes a first memory module circuit and a second memory module circuit controlled by a memory module circuit so as to be placed in active and standby states. When one memory module circuit is in the active state, the other memory module circuit is placed in the standby state, thereby making it possible to reduce power consumption.
摘要翻译：在数字电子静态摄像机中的功率消耗降低。具体地，数字电子静态摄像机包括由存储器模块电路控制以便处于主动和待机状态的第一存储器模块电路和第二存储器模块电路。当一个存储器模块电路处于活动状态时，另一个存储器模块电路处于待机状态，从而可以降低功耗。

10. 发明授权

US06433821B1 Digital electronic still-video camera, and method of controlling same 失效
标题翻译：数字电子静态摄像机及其控制方法
公开(公告)号：US06433821B1
公开(公告)日：2002-08-13
申请号：US09500485
申请日：2000-02-09
申请人： Kouichi Gouhara , Kaoru Adachi , Kenji Moronaga
发明人： Kouichi Gouhara , Kaoru Adachi , Kenji Moronaga
IPC分类号： H04N576
CPC分类号： H04N1/2141 , H04N1/2112 , H04N1/215 , H04N1/2158 , H04N5/907 , H04N5/9261
摘要： A digital electronic still-video camera is capable of performing rapid-sequence photography at high speeds. When a rapid-sequence photographic mode has been set, each of a plurality of frames of image data obtained by such photography is compressed. Image data which forms a single multiple-frame picture is constructed by a set of image data composed of the compressed plurality of frames. Thinning out is performed in order to compress the image data. The image data is successively stored, while being thinned out, at corresponding addresses of an image memory in such a manner that a multiple-frame picture is constructed in the image memory. After photography in the rapid-sequence mode ends, the image data in the image memory is subjected to data compression and then recorded on a memory card.
摘要翻译：数字电子静态摄像机能够以高速执行快速拍摄。当已经设置了快速拍摄模式时，通过这种摄影获得的多个图像数据帧中的每一个被压缩。由一组由压缩的多个帧组成的图像数据构成形成单个多帧图像的图像数据。为了压缩图像数据，执行稀疏化。在图像存储器的相应地址以图像存储器中构成多帧图像的方式，连续地存储图像数据。在快速顺序模式拍摄结束后，图像存储器中的图像数据经受数据压缩，然后记录在存储卡上。

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