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1. 发明授权

US07300946B2 N-(substituted arylmethyl)-4-(disubstituted methyl) piperidines and pyridines 失效
标题翻译： N-（取代的芳基甲基）-4-（二取代的甲基）哌啶和吡啶
公开(公告)号：US07300946B2
公开(公告)日：2007-11-27
申请号：US10538998
申请日：2003-12-08
申请人： Ping Ding , Robert N. Henrie, II , Daniel H. Cohen , John W. Lyga , David S. Rosen , George Theodoridis , Qun Zhang , Walter H. Yeager , Stephen F. Donovan , Steven Shunxiang Zhang , Inna Shulman , Seong Jae Yu , Guozhi Wang , Y. Larry Zhang , Ariamala Gopalsamy , Dennis L. Warkentin , Paul E. Rensner , Ian R. Silverman , Thomas G. Cullen
发明人： Ping Ding , Robert N. Henrie, II , Daniel H. Cohen , John W. Lyga , David S. Rosen , George Theodoridis , Qun Zhang , Walter H. Yeager , Stephen F. Donovan , Steven Shunxiang Zhang , Inna Shulman , Seong Jae Yu , Guozhi Wang , Y. Larry Zhang , Ariamala Gopalsamy , Dennis L. Warkentin , Paul E. Rensner , Ian R. Silverman , Thomas G. Cullen
IPC分类号： A61K31/44 , A61K31/445 , A61K31/4422 , C07D211/06 , C07D211/08 , C07D211/70 , C07D211/82
CPC分类号： C07D405/14 , A01N43/40 , A01N43/54 , A01N43/713 , C07D211/14 , C07D211/18 , C07D211/22 , C07D211/24 , C07D211/26 , C07D211/28 , C07D211/32 , C07D211/94 , C07D401/06 , C07D401/10 , C07D401/12 , C07D401/14 , C07D413/12 , C07D417/12 , C07D451/14 , C07D513/04
摘要： It has now been found that certain novel N-(substituted aryl)-4(disubstituted methyl)piperidine and pyridine derivatives have provided unexpected insecticidal activity. These compounds are represented by formula (I): wherein m, n, q, r, and s are independently selected from 0 or 1; and p is 0, 1, 2, or 3; A is C or CH; and B, D, E, R, R1, R2, R3, R4, R5, R6, R7 and R8 are fully described herein. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula I, and optionally, an effective amount of at least one of a second compound, with at least one insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present
摘要翻译：现在已经发现，某些新的N-（取代的芳基）-4（二取代的甲基）哌啶和吡啶衍生物已经提供了意想不到的杀虫活性。这些化合物由式（I）表示：其中m，n，q，r和s独立地选自0或1; 且p为0,1,2或3; A是C或CH; 和B，D，E，R，R 1，R 2，R 3，R 4，R 本文中充分描述了本发明的第5，第6，第七和第八和第八。此外，还公开了包含杀虫有效量的至少一种式I化合物和任选的有效量的至少一种第二化合物与至少一种与杀虫相容的载体的组合物; 以及控制昆虫的方法，包括将所述组合物施用于存在昆虫或预期存在的场所

2. 发明授权

US07365082B2 N-(substituted arylmethyl)-4-(disubstituted methyl)piperidines and piperazines 失效
标题翻译： N-（取代的芳基甲基）-4-（二取代的甲基）哌啶和哌嗪
公开(公告)号：US07365082B2
公开(公告)日：2008-04-29
申请号：US10538997
申请日：2003-12-08
申请人： Ping Ding , Robert N. Henrie, II , Daniel H. Cohen , John W. Lyga , David S. Rosen , George Theodoridis , Qun Zhang , Walter H. Yeager , Stephen F. Donovan , Steven Shunxiang Zhang , Inna Shulman , Seong Jae Yu , Guozhi Wang , Y. Larry Zhang , Ariamala Gopalsamy , Dennis L. Warkentin , Paul E. Rensner , Ian R. Silverman , Thomas G. Cullen
发明人： Ping Ding , Robert N. Henrie, II , Daniel H. Cohen , John W. Lyga , David S. Rosen , George Theodoridis , Qun Zhang , Walter H. Yeager , Stephen F. Donovan , Steven Shunxiang Zhang , Inna Shulman , Seong Jae Yu , Guozhi Wang , Y. Larry Zhang , Ariamala Gopalsamy , Dennis L. Warkentin , Paul E. Rensner , Ian R. Silverman , Thomas G. Cullen
IPC分类号： A61K31/44 , A61K31/445 , A61K31/4422 , C07D211/06 , C07D211/08 , C07D211/70 , C07D211/82
CPC分类号： C07D405/14 , A01N43/40 , A01N43/54 , A01N43/713 , C07D211/14 , C07D211/18 , C07D211/22 , C07D211/24 , C07D211/26 , C07D211/28 , C07D211/32 , C07D211/94 , C07D401/06 , C07D401/10 , C07D401/12 , C07D401/14 , C07D413/12 , C07D417/12 , C07D451/14 , C07D513/04
摘要： It has now been found that certain novel N-(substituted aryl)-4-(disubstituted methyl)piperidine and pyridine derivatives have provided unexpected insecticidal activity. These compounds are represented by formula (I): wherein m, n, q, r, and s are independently selected from 0 or 1; and p is 0, 1, 2, or 3; A is CH or N; and B, D, E, R, R1, R2, R3, R4, R5, R6, R7 and R8 are fully described herein. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula I, and optionally, an effective amount of at least one of a second compound, with at least one insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present.
摘要翻译：现在已经发现某些新的N-（取代的芳基）-4-（二取代的甲基）哌啶和吡啶衍生物提供了意想不到的杀虫活性。这些化合物由式（I）表示：其中m，n，q，r和s独立地选自0或1; 且p为0,1,2或3; A是CH或N; 和B，D，E，R，R 1，R 2，R 3，R 4，R 本文完全描述了本发明的第5，第6，第七和第八和第八。此外，还公开了包含杀虫有效量的至少一种式I化合物和任选的有效量的至少一种第二化合物与至少一种与杀虫相容的载体的组合物; 以及控制昆虫的方法，包括将所述组合物施用于存在昆虫或预期存在的场所。

3. 发明授权

US07683070B2 N-(substituted arylmethyl)-4-(disubstituted methyl) piperidines and pyridines 有权
标题翻译： N-（取代的芳基甲基）-4-（二取代的甲基）哌啶和吡啶
公开(公告)号：US07683070B2
公开(公告)日：2010-03-23
申请号：US11874015
申请日：2007-10-17
申请人： Ping Ding , Robert N. Henrie, II , Daniel H. Cohen , John W. Lyga , David S. Rosen , George Theodoridis , Qun Zhang , Walter H. Yeager , Stephen F. Donovan , Stephen Shunxiang Zhang , Inna Shulman , Seong Jae Yu , Guozhi Wang , Y. Larry Zhang , Ariamala Gopalsamy , Dennis L. Warkentin , Paul E. Rensner , Ian R. Silverman , Thomas G. Cullen
发明人： Ping Ding , Robert N. Henrie, II , Daniel H. Cohen , John W. Lyga , David S. Rosen , George Theodoridis , Qun Zhang , Walter H. Yeager , Stephen F. Donovan , Stephen Shunxiang Zhang , Inna Shulman , Seong Jae Yu , Guozhi Wang , Y. Larry Zhang , Ariamala Gopalsamy , Dennis L. Warkentin , Paul E. Rensner , Ian R. Silverman , Thomas G. Cullen
IPC分类号： A61K31/4523 , A61K31/4545 , C07D211/06 , C07D239/02
CPC分类号： C07D405/14 , A01N43/40 , A01N43/54 , A01N43/713 , C07D211/14 , C07D211/18 , C07D211/22 , C07D211/24 , C07D211/26 , C07D211/28 , C07D211/32 , C07D211/94 , C07D401/06 , C07D401/10 , C07D401/12 , C07D401/14 , C07D413/12 , C07D417/12 , C07D451/14 , C07D513/04
摘要： It has now been found that certain novel N-(substituted aryl)-4-(disubstituted methyl)piperidine and pyridine derivatives have provided unexpected insecticidal activity. These compounds are represented by formula (I): wherein m, n, q, r, and s are independently selected from 0 or 1; and p is 0, 1, 2, or 3; A is C or CH; and B, D, E, R, R1, R2, R3, R4, R5, R6, R7 and R8 are fully described herein. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula I, and optionally, an effective amount of at least one of a second compound, with at least one insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present.
摘要翻译：现在已经发现某些新的N-（取代的芳基）-4-（二取代的甲基）哌啶和吡啶衍生物提供了意想不到的杀虫活性。这些化合物由式（I）表示：其中m，n，q，r和s独立地选自0或1; 且p为0,1,2或3; A是C或CH; 本文完整地描述了B，D，E，R，R 1，R 2，R 3，R 4，R 5，R 6，R 7和R 8。此外，还公开了包含杀虫有效量的至少一种式I化合物和任选的有效量的至少一种第二化合物与至少一种与杀虫相容的载体的组合物; 以及控制昆虫的方法，包括将所述组合物施用于存在昆虫或预期存在的场所。

4. 发明授权

US06214845B1 Insecticidal N-(substituted arylmethyl)-4[bis(substituted phenyl or pyridyl)methyl] piperidines 失效
标题翻译：杀虫剂N-（取代的芳基甲基）-4 [双（取代的苯基或吡啶基）甲基]哌啶
公开(公告)号：US06214845B1
公开(公告)日：2001-04-10
申请号：US09388592
申请日：1999-09-02
申请人： Ian R. Silverman , Daniel H. Cohen , John W. Lyga , Steven W. Szczepanski , Syed F. Ali , Thomas G. Cullen , Robert N. Henrie, II , Clinton J. Peake
发明人： Ian R. Silverman , Daniel H. Cohen , John W. Lyga , Steven W. Szczepanski , Syed F. Ali , Thomas G. Cullen , Robert N. Henrie, II , Clinton J. Peake
IPC分类号： A01N4340
CPC分类号： C07D401/06 , A01N43/40 , A01N43/50 , A01N43/54 , A01N43/56 , A01N43/60 , A01N43/653 , A01N43/713 , A01N43/76 , A01N43/82 , A01N47/20 , A01N55/00 , C07D211/14 , C07D211/22 , C07D211/24 , C07D211/26 , C07D211/94 , C07D231/12 , C07D233/56 , C07D249/08 , C07D401/10 , C07D401/12 , C07D401/14 , C07D405/06 , C07D405/10 , C07D409/06 , C07D413/06 , C07D413/10 , C07D417/10 , C07D417/12 , C07F7/1804
摘要： Compounds of the following structure, the corresponding N-oxides and agriculturally acceptable salts, are disclosed as effective insecticides: in which U is —(CH2)n—; Q is hydroxy; R is in which V, W, Y, and Z are each hydrogen; X is a five- or six-membered heterocycle; optionally substituted with halogen, cyano, alkyl, haloalkyl, alkoxy, haloalkoxy, alkoxyalkyl, haloalkoxyalkyl, or aminocarbonyl; and the heterocycle is optionally connected to the phenyl ring through a —O—, —S—, —(CH2)p, —C(O)—, or —O—(CR3R4)q linkage; R1 and R2 are independently selected from phenyl or pyridyl substituted with haloalkyl or haloalkoxy; R3 and R4 are independently selected from hydrogen and methyl; n and p are independently 1, 2, or 3; and q is 1 or 2; with the proviso that at least one of R1 and R2 is substituted in the para position; no more than two of R3 and R4 are methyl; each aliphatic moiety contains not more than 4 carbon atoms; halogen means bromine, chlorine, or fluorine; each heterocycle contains from 1 to 4 nitrogen atoms, or 1 or 2 oxygen or sulfur atoms, or 1 or 2 nitrogen atoms and an oxygen or sulfur atom; and the corresponding N-oxides and agriculturally acceptable salts.
摘要翻译：公开了以下结构的化合物，即相应的N-氧化物和农业上可接受的盐作为有效的杀虫剂：其中U是 - （CH 2）n - ; Q是羟基; R 1是其中V，W，Y和Z各自是氢; X是五元或六元杂环; 任选被卤素，氰基，烷基，卤代烷基，烷氧基，卤代烷氧基，烷氧基烷基，卤代烷氧基烷基或氨基羰基取代; 并且杂环任选地通过-O - ， - S - ， - （CH 2）p，-C（O） - 或-O-（CR 3 R 4）q键连接到苯环; R 1和R 2独立地选自苯基或被卤代烷基或卤代烷氧基取代的吡啶基; R3和R4独立地选自氢和甲基; n和p独立地为1,2或3; 且q为1或2;条件是R1和R2中的至少一个在对位取代; R3和R4中不超过两个是甲基; 每个脂族部分含有不超过4个碳原子; 卤素是指溴，氯或氟; 每个杂环含有1至4个氮原子，或1或2个氧或硫原子，或1或2个氮原子和氧或硫原子;以及相应的N-氧化物和农业上可接受的盐。

5. 发明授权

US6030987A Insecticidal N-(substituted arylmethyl)-4-[bis(substituted phenyl or pyridyl)methyl]piperidines 失效
标题翻译：杀虫剂N-（取代的芳基甲基）-4- [双（取代的苯基或吡啶基）甲基]哌啶
公开(公告)号：US6030987A
公开(公告)日：2000-02-29
申请号：US981456
申请日：1998-08-11
申请人： Ian R. Silverman , Daniel H. Cohen , John W. Lyga , Steven W. Szczepanski , Syed F. Ali , Thomas G. Cullen , Robert N. Henrie, II , Clinton J. Peake
发明人： Ian R. Silverman , Daniel H. Cohen , John W. Lyga , Steven W. Szczepanski , Syed F. Ali , Thomas G. Cullen , Robert N. Henrie, II , Clinton J. Peake
IPC分类号： A01N43/40 , A01N43/54 , A01N43/56 , A01N43/653 , A01N43/713 , A01N43/76 , A01N43/82 , C07D401/10 , C07D417/10
CPC分类号： A01N43/713 , A01N43/40 , A01N43/54 , A01N43/56 , A01N43/653 , A01N43/76 , A01N43/82
摘要： Compounds of structure (I) ##STR1## the corresponding N-oxides and agriculturally acceptable salts are disclosed as effective insecticides. In said formula, U is --(CH.sub.2)n--; Q is hydroxy, R is formula (II) ##STR2## in which V, W, Y and Z are hydrogen; X is a five- or six-membered heterocycle optionally substituted; and the heterocycle is optionally connected to the phenyl ring through a --O--, --S-- --CH.sub.2)p--, or --O(CR.sup.3 R.sup.4)q linkage; R.sup.1 and R.sup.2 are independently selected from phenyl or pyridyl substituted with haloalkyl or haloalkoxy; R.sup.3, R.sup.4, n, p, and 1 are as defined in the specification.
摘要翻译： PCT No.PCT / US96 / 07206 Sec。 371日期：1998年8月11日 102（e）1998年8月11日PCT PCT 1996年5月17日PCT公布。公开号WO96 / 36228 PCT 日期：1996年11月21日公开了结构（Ⅰ）化合物对应的N-氧化物和农业上可接受的盐作为有效杀虫剂。在所述式中，U是 - （CH 2）n - ; Q是羟基，R是式（II），其中V，W，Y和Z是氢; X是任选取代的五或六元杂环; 并且杂环任选地通过-O - ， - S--CH 2）对 - 或-O（CR 3 R 4）q键连接到苯环上; R 1和R 2独立地选自苯基或被卤代烷基或卤代烷氧基取代的吡啶基; R3，R4，n，p和1如说明书中所定义。

6. 发明授权

US06184234B2 Insecticidal N-(substituted arylmethyl)-4-[bis(substituted phenyl or pyridyl)methyl]piperidines 失效
标题翻译：杀虫剂N-（取代的芳基甲基）-4- [双（取代的苯基或吡啶基）甲基]哌啶
公开(公告)号：US06184234B2
公开(公告)日：2001-02-06
申请号：US09414375
申请日：1999-10-07
申请人： Ian R. Silverman , Daniel H. Cohen , John W. Lyga , Steven W. Szczepanski , Syed F. Ali , Thomas G. Cullen , Robert N. Henrie, II , Clinton J. Peake
发明人： Ian R. Silverman , Daniel H. Cohen , John W. Lyga , Steven W. Szczepanski , Syed F. Ali , Thomas G. Cullen , Robert N. Henrie, II , Clinton J. Peake
IPC分类号： A01N4340
CPC分类号： C07D231/12 , A01N43/40 , A01N43/50 , A01N43/54 , A01N43/56 , A01N43/60 , A01N43/653 , A01N43/713 , A01N43/76 , A01N43/82 , A01N47/20 , A01N55/00 , C07D211/14 , C07D211/22 , C07D211/24 , C07D211/26 , C07D211/94 , C07D233/56 , C07D249/08 , C07D401/06 , C07D401/10 , C07D401/12 , C07D401/14 , C07D405/06 , C07D405/10 , C07D409/06 , C07D413/06 , C07D413/10 , C07D417/10 , C07D417/12 , C07F7/1804
摘要： Compounds of the following structure, the corresponding N-oxides and agriculturally acceptable salts thereof, are disclosed as effective insecticides: wherein U is —(CH2)n—; Q is hydroxy; and R is: and wherein V, W, Y, and Z are each hydrogen; X is a five- or six-membered heterocycle; optionally substituted with bromine, chlorine, fluorine, cyano, alkyl, haloalkyl, alkoxy, haloalkoxy, alkoxyalkyl, haloalkoxyalkyl, or aminocarbonyl; and the heterocycle is optionally connected to the phenyl ring through a —O—, —S—, —(CH2)p, —C(O)—, or —O—(CR3R4)q linkage; R1 and R2 are independently selected from phenyl or pyridyl substituted with pentahalothio, haloalkylthio, haloalkylsulfinyl, or haloalkylsulfonyl; phenyl substituted with —OC(M)2O—, where M is bromine, chorine or fluorine, to provide a dihalobenzodioxolyl fused ring; or pyridyl substituted with —OC(M)2O— to provide a dihalodioxolenopyridyl fused ring; R3 and R4 are independently selected from hydrogen and methyl; n and p are independently 1, 2, or 3; and q is 1 or 2; with the proviso that at least one of R1 and R2 is substituted in the para position of the phenyl ring or the 5-position of the 2-pyridyl ring; each alkyl portion of said optional substituent on X wherein the optional substituent is alkyl, haloalkyl, alkoxyl, haloalkoxyl, alkoxyalkyl, or haloalkoxyalkyl contains from 1 to 4 carbon atoms; each heterocycle contains from 1 to 4 nitrogen atoms, 1 or 2 oxygen or sulfur atoms, or 1 or 2 nitrogen atoms and an oxygen or sulfur atom; and the corresponding N-oxides and agriculturally acceptable salts.
摘要翻译：以下结构的化合物，其相应的N-氧化物和农业上可接受的盐被公开为有效的杀虫剂：其中U是 - （CH 2）n - ; Q是羟基; 且R为：且其中V，W，Y和Z各自为氢; X为五元或六元杂环; 任选被溴，氯，氟，氰基，烷基，卤代烷基，烷氧基，卤代烷氧基，烷氧基烷基，卤代烷氧基烷基或氨基羰基取代; 并且杂环任选地通过-O - ， - S - ， - （CH 2）p，-C（O） - 或-O-（CR 3 R 4）q键连接到苯环; R 1和R 2独立地选自苯基或被五卤代硫代，卤代烷硫基，卤代烷基亚磺酰基或卤代烷基磺酰基取代的吡啶基; 用-OC（M）2 O-取代的苯基，其中M是溴，氯或氟，得到二卤代二苯甲基稠合环; 或被-OC（M）2 O-取代的吡啶基，以提供二卤代苯并吡啶基稠环; R 3和R 4独立地选自氢和甲基; n和p独立地为1,2或3; 平均值为1或2; 条件是R 1和R 2中的至少一个在苯环的对位或2-吡啶基环的5-位上被取代; X上任选取代基的每个烷基部分，其中任选的取代基是烷基，卤代烷基，烷氧基，卤代烷氧基，烷氧基烷基或卤代烷氧基烷基含有1至4个碳原子; 每个杂环含有1至4个氮原子，1或2个氧或硫原子，或1或2个氮原子和氧或硫原子; 和相应的N-氧化物和农业上可接受的盐。

7. 发明授权

US5534518A Insecticidal substituted-2,4-diaminoquinazolines 失效
公开(公告)号：US5534518A
公开(公告)日：1996-07-09
申请号：US267340
申请日：1994-06-28
申请人： Robert N. Henrie, II , Clinton J. Peake , Thomas G. Cullen , Albert C. Lew , Munirathnam K. Chaguturu , Partha S. Ray , Walter H. Yeager , Ian R. Silverman , John W. Buser , James J. Fiordeliso , John A. Dixson
发明人： Robert N. Henrie, II , Clinton J. Peake , Thomas G. Cullen , Albert C. Lew , Munirathnam K. Chaguturu , Partha S. Ray , Walter H. Yeager , Ian R. Silverman , John W. Buser , James J. Fiordeliso , John A. Dixson
IPC分类号： A01N43/54 , A01N55/00 , C07D239/95 , C07D401/12 , C07D405/04 , C07D409/04 , A61K31/505
CPC分类号： C07D401/12 , A01N43/54 , A01N55/00 , C07D239/95 , C07D405/04 , C07D409/04
摘要： An insecticidal composition comprising, in admixture with an agriculturally acceptable carrier, an insecticidally effective amount of a 2,4-diaminoquinazoline compound of the formula: ##STR1## wherein R.sup.1, R.sup.2, R.sup.6, R.sup.7, W, X, Y, and Z are as defined herein; methods of using the same; novel 2,4-diaminoquinazolines per se; and intermediates in the preparation thereof.

8. 发明授权

US5939438A Insecticidal oximino and hydrazono derivatives of N-benzyl-4-benzhydryl-and N-benzyl-4-benzhydrol-piperidines 失效
标题翻译： N-苄基-4-二苯甲基 - 和N-苄基-4-二苯甲基 - 哌啶的杀虫肟基和亚肼基衍生物
公开(公告)号：US5939438A
公开(公告)日：1999-08-17
申请号：US150424
申请日：1998-09-09
申请人： Walter H. Yeager , Ian R. Silverman , Robert N. Henrie, II , Thomas G. Cullen , Clinton J. Peake
发明人： Walter H. Yeager , Ian R. Silverman , Robert N. Henrie, II , Thomas G. Cullen , Clinton J. Peake
IPC分类号： A01N43/40 , A01N47/02 , A01N47/24 , C07D211/28 , C07D211/94 , C07D211/18 , C07D211/26
CPC分类号： C07D211/28 , A01N43/40 , A01N47/02 , A01N47/24 , C07D211/94
摘要： It has now been found that certain novel oximino and hydrazono derivatives of N-benzyl-4-benzhydryl- and 4-benhydrolpiperidines, and their corresponding N-oxides and agriculturally acceptable salts are useful as insecticides. These compounds are represented by Formula I: where R is hydrogen, halogen, alkyl, alkoxy, dialkylamino; R.sup.1 is hydrogen, alkyl, haloalkyl, alkoxyalkyl, alkylcarbonyl and alkylaminocarbonyl; X is oxygen, or NR.sup.2, Q is fluoro and hydroxy; Z is halogen, haloalkyl, haloalkoxy, pentahalothio, haloalkylthio, haloalkylsulfinyl, haloalkylsulfonyl, and --OCF.sub.2 O-- attached to two adjacent carbon atoms of the phenyl ring; n is 0 or 1; and, when X is NR.sup.2, R.sup.2 is hydrogen, alkyl, alkylcarbonyl, alkoxycarbonyl, or R.sup.1 and R.sup.2 taken together may be --C.sub.m H.sub.2.spsb.m, or --C.sub.2 H.sub.4 OC.sub.2 H.sub.4 --, where m is 3-9. Preferred compounds include those where R is hydrogen; R.sup.1 is alkyl; Q is hydroxy; X is oxygen; and Z is trifluoromethyl or trifluoromethoxy.
摘要翻译：现已发现，N-苄基-4-二苯甲基 - 和4-苯氢哌啶的某些新的肟基和亚氨基衍生物及其相应的N-氧化物和农业上可接受的盐可用作杀虫剂。这些化合物由式I表示：其中R是氢，卤素，烷基，烷氧基，二烷基氨基; R1是氢，烷基，卤代烷基，烷氧基烷基，烷基羰基和烷基氨基羰基; X是氧，或NR 2，Q是氟和羟基; Z是苯环的两个相邻碳原子上的卤素，卤代烷基，卤代烷氧基，五卤代硫代，卤代烷硫基，卤代烷基亚磺酰基，卤代烷基磺酰基和-OCF 2 O-。 n为0或1; 并且当X为NR 2时，R 2为氢，烷基，烷基羰基，烷氧基羰基，或者R 1和R 2一起可以是-C m H 2m或-C 2 H 4 OC 2 H 4 - ，其中m为3-9。优选的化合物包括其中R为氢的化合物; R1是烷基; Q是羟基; X是氧; Z是三氟甲基或三氟甲氧基。

9. 依法登记的发明

USH2007H1 Insecticidal N-heterocyclylalkyl-or N-[(polycyclyl)alkyl]-N′substituted piperazines 失效
公开(公告)号：USH2007H1
公开(公告)日：2001-12-04
申请号：US08780371
申请日：1997-01-09
申请人： Ian R. Silverman , Syed F. Ali , Daniel H. Cohen , John W. Lyga , Kirk A. Simmons , Thomas G. Cullen
发明人： Ian R. Silverman , Syed F. Ali , Daniel H. Cohen , John W. Lyga , Kirk A. Simmons , Thomas G. Cullen
IPC分类号： C07D29500
摘要： Compounds of the following structure are disclosed as effective insecticides: in which: A and B are independently lower alkyl; U is lower alkylidene, lower alkenylidene, or CH—Z, where Z is hydrogen, lower alkyl, lower cycloalkyl, or phenyl; R is phenyl or a dibenzocyclo(C5-8)alkyl, each optionally substituted, or where R3 and R4 are independently selected from phenyl, optionally substituted with, halogen, lower alkyl, lower haloalkyl, lower alkoxy, lower haloalkoxy, lower alkenyl, or phenyl; R1 is selected from a variety of substituents, including 3-R2, where R2 is where D, E, and G are hydrogen, hydroxy, halogen, cyano, hydroxy, lower alkyl, lower haloalkyl, lower alkoxy, nitro, lower haloalkylsuffonyloxy, lower alkylcarboxylato, lower alkylcarbonylamino, lower alkylcarbonyl, lower alkoxycarbonyl, arylcarbonylamino; D and E taken together may form the group —O(CH2)O—; J is hydrogen or lower alkyl; m is 2 or 3, n is 1, 2, or 3; and halogen is chlorine, bromine, or fluorine.

10. 发明授权

US07247756B2 1,4-disubstituted benzenes as insecticides 失效
标题翻译： 1,4-二取代苯作为杀虫剂
公开(公告)号：US07247756B2
公开(公告)日：2007-07-24
申请号：US10353471
申请日：2003-01-29
申请人： George Theodoridis , Edward Barron , Daniel H. Cohen , Ellen M. Crawford , Thomas G. Cullen , Hongyan Qi , Elizabeth Rowley , Syed F. Ali , Walter H. Yeager , Christina B. Duggan
发明人： George Theodoridis , Edward Barron , Daniel H. Cohen , Ellen M. Crawford , Thomas G. Cullen , Hongyan Qi , Elizabeth Rowley , Syed F. Ali , Walter H. Yeager , Christina B. Duggan
IPC分类号： C07C43/20
CPC分类号： C07D215/233 , C07C211/59 , C07C217/20 , C07C217/58 , C07C217/92 , C07C233/43 , C07C235/56 , C07C251/24 , C07C271/28 , C07C275/34 , C07C275/40 , C07C291/04 , C07C2602/08 , C07C2602/10 , C07D209/46 , C07D215/24 , C07D215/38 , C07D215/40 , C07D215/44 , C07D217/22 , C07D295/088 , C07D295/096 , C07D295/205 , C07D491/10
摘要： Compounds of formula I: wherein A, B, D, and R are as defined herein and their agriculturally acceptable salts are disclosed as effective insecticides. In addition, compositions comprising an insecticidally effective amount of a compound of Formula I in admixture with at least one agriculturally acceptable extender or adjuvant and methods of controlling insects comprising applying the compositions to locus on crops where control is desired are disclosed.
摘要翻译：式I化合物：其中A，B，D和R如本文所定义，其农业上可接受的盐被公开为有效的杀虫剂。此外，公开了包含杀虫有效量的式I化合物与至少一种农业上可接受的增量剂或佐剂混合的组合物和控制昆虫的方法，其包括将组合物施用于需要控制的作物上的位点。

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