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1. 发明授权

US07365082B2 N-(substituted arylmethyl)-4-(disubstituted methyl)piperidines and piperazines 失效
标题翻译： N-（取代的芳基甲基）-4-（二取代的甲基）哌啶和哌嗪
公开(公告)号：US07365082B2
公开(公告)日：2008-04-29
申请号：US10538997
申请日：2003-12-08
申请人： Ping Ding , Robert N. Henrie, II , Daniel H. Cohen , John W. Lyga , David S. Rosen , George Theodoridis , Qun Zhang , Walter H. Yeager , Stephen F. Donovan , Steven Shunxiang Zhang , Inna Shulman , Seong Jae Yu , Guozhi Wang , Y. Larry Zhang , Ariamala Gopalsamy , Dennis L. Warkentin , Paul E. Rensner , Ian R. Silverman , Thomas G. Cullen
发明人： Ping Ding , Robert N. Henrie, II , Daniel H. Cohen , John W. Lyga , David S. Rosen , George Theodoridis , Qun Zhang , Walter H. Yeager , Stephen F. Donovan , Steven Shunxiang Zhang , Inna Shulman , Seong Jae Yu , Guozhi Wang , Y. Larry Zhang , Ariamala Gopalsamy , Dennis L. Warkentin , Paul E. Rensner , Ian R. Silverman , Thomas G. Cullen
IPC分类号： A61K31/44 , A61K31/445 , A61K31/4422 , C07D211/06 , C07D211/08 , C07D211/70 , C07D211/82
CPC分类号： C07D405/14 , A01N43/40 , A01N43/54 , A01N43/713 , C07D211/14 , C07D211/18 , C07D211/22 , C07D211/24 , C07D211/26 , C07D211/28 , C07D211/32 , C07D211/94 , C07D401/06 , C07D401/10 , C07D401/12 , C07D401/14 , C07D413/12 , C07D417/12 , C07D451/14 , C07D513/04
摘要： It has now been found that certain novel N-(substituted aryl)-4-(disubstituted methyl)piperidine and pyridine derivatives have provided unexpected insecticidal activity. These compounds are represented by formula (I): wherein m, n, q, r, and s are independently selected from 0 or 1; and p is 0, 1, 2, or 3; A is CH or N; and B, D, E, R, R1, R2, R3, R4, R5, R6, R7 and R8 are fully described herein. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula I, and optionally, an effective amount of at least one of a second compound, with at least one insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present.
摘要翻译：现在已经发现某些新的N-（取代的芳基）-4-（二取代的甲基）哌啶和吡啶衍生物提供了意想不到的杀虫活性。这些化合物由式（I）表示：其中m，n，q，r和s独立地选自0或1; 且p为0,1,2或3; A是CH或N; 和B，D，E，R，R 1，R 2，R 3，R 4，R 本文完全描述了本发明的第5，第6，第七和第八和第八。此外，还公开了包含杀虫有效量的至少一种式I化合物和任选的有效量的至少一种第二化合物与至少一种与杀虫相容的载体的组合物; 以及控制昆虫的方法，包括将所述组合物施用于存在昆虫或预期存在的场所。

2. 发明授权

US5939438A Insecticidal oximino and hydrazono derivatives of N-benzyl-4-benzhydryl-and N-benzyl-4-benzhydrol-piperidines 失效
标题翻译： N-苄基-4-二苯甲基 - 和N-苄基-4-二苯甲基 - 哌啶的杀虫肟基和亚肼基衍生物
公开(公告)号：US5939438A
公开(公告)日：1999-08-17
申请号：US150424
申请日：1998-09-09
申请人： Walter H. Yeager , Ian R. Silverman , Robert N. Henrie, II , Thomas G. Cullen , Clinton J. Peake
发明人： Walter H. Yeager , Ian R. Silverman , Robert N. Henrie, II , Thomas G. Cullen , Clinton J. Peake
IPC分类号： A01N43/40 , A01N47/02 , A01N47/24 , C07D211/28 , C07D211/94 , C07D211/18 , C07D211/26
CPC分类号： C07D211/28 , A01N43/40 , A01N47/02 , A01N47/24 , C07D211/94
摘要： It has now been found that certain novel oximino and hydrazono derivatives of N-benzyl-4-benzhydryl- and 4-benhydrolpiperidines, and their corresponding N-oxides and agriculturally acceptable salts are useful as insecticides. These compounds are represented by Formula I: where R is hydrogen, halogen, alkyl, alkoxy, dialkylamino; R.sup.1 is hydrogen, alkyl, haloalkyl, alkoxyalkyl, alkylcarbonyl and alkylaminocarbonyl; X is oxygen, or NR.sup.2, Q is fluoro and hydroxy; Z is halogen, haloalkyl, haloalkoxy, pentahalothio, haloalkylthio, haloalkylsulfinyl, haloalkylsulfonyl, and --OCF.sub.2 O-- attached to two adjacent carbon atoms of the phenyl ring; n is 0 or 1; and, when X is NR.sup.2, R.sup.2 is hydrogen, alkyl, alkylcarbonyl, alkoxycarbonyl, or R.sup.1 and R.sup.2 taken together may be --C.sub.m H.sub.2.spsb.m, or --C.sub.2 H.sub.4 OC.sub.2 H.sub.4 --, where m is 3-9. Preferred compounds include those where R is hydrogen; R.sup.1 is alkyl; Q is hydroxy; X is oxygen; and Z is trifluoromethyl or trifluoromethoxy.
摘要翻译：现已发现，N-苄基-4-二苯甲基 - 和4-苯氢哌啶的某些新的肟基和亚氨基衍生物及其相应的N-氧化物和农业上可接受的盐可用作杀虫剂。这些化合物由式I表示：其中R是氢，卤素，烷基，烷氧基，二烷基氨基; R1是氢，烷基，卤代烷基，烷氧基烷基，烷基羰基和烷基氨基羰基; X是氧，或NR 2，Q是氟和羟基; Z是苯环的两个相邻碳原子上的卤素，卤代烷基，卤代烷氧基，五卤代硫代，卤代烷硫基，卤代烷基亚磺酰基，卤代烷基磺酰基和-OCF 2 O-。 n为0或1; 并且当X为NR 2时，R 2为氢，烷基，烷基羰基，烷氧基羰基，或者R 1和R 2一起可以是-C m H 2m或-C 2 H 4 OC 2 H 4 - ，其中m为3-9。优选的化合物包括其中R为氢的化合物; R1是烷基; Q是羟基; X是氧; Z是三氟甲基或三氟甲氧基。

3. 发明授权

US5874579A Insecticidal substituted-2.4-diaminoquinazolines related applications 失效
标题翻译：杀虫剂取代-2,4-二氨基喹唑啉
公开(公告)号：US5874579A
公开(公告)日：1999-02-23
申请号：US640610
申请日：1996-05-01
申请人： Robert N. Henrie II , Clinton J. Peake , Thomas G. Cullen , Walter H. Yeager
发明人： Robert N. Henrie II , Clinton J. Peake , Thomas G. Cullen , Walter H. Yeager
IPC分类号： A01N43/54 , A01N55/00 , C07D239/95 , C07D401/12 , C07D405/04 , C07D409/04 , A61K31/505
CPC分类号： C07D401/12 , A01N43/54 , A01N55/00 , C07D239/95 , C07D405/04 , C07D409/04
摘要： An insecticidal composition comprising, in admixture with an agriculturally acceptable carrier, an insecticidally effective amount of a 2,4-diaminoquinazoline compound of the formula: ##STR1## wherein R.sup.1, R.sup.2, R.sup.6, R.sup.7, W, X, Y, and Z are as defined herein; methods of using the same; novel 2,4-diaminoquinazolines per se; and intermediates in the preparation thereof.
摘要翻译：一种杀虫组合物，其包含与农业上可接受的载体的混合物，杀虫有效量的下式的2,4-二氨基喹唑啉化合物：其中R 1，R 2，R 6，R 7，W，X，Y和Z为如本文所定义; 使用方法; 新型2,4-二氨基喹唑啉本身; 和其制备中的中间体。

4. 发明授权

US5593998A 2,4-diamino-5,6-disubstituted-and 5,6,7-trisubstituted-5-deazapteridines as insecticides 失效
标题翻译： 2,4-二氨基-5,6-二取代 - 和5,6,7-三取代-5-脱氮啶啶类作为杀虫剂
公开(公告)号：US5593998A
公开(公告)日：1997-01-14
申请号：US647550
申请日：1996-05-15
申请人： Robert N. Henrie, II , Clinton J. Peake , Thomas G. Cullen , Munirathnam K. Chaguturu , Partha S. Ray , Brian D. Bennett
发明人： Robert N. Henrie, II , Clinton J. Peake , Thomas G. Cullen , Munirathnam K. Chaguturu , Partha S. Ray , Brian D. Bennett
IPC分类号： C07D487/04 , A01N43/54 , A61K31/535
CPC分类号： C07D487/04
摘要： An insecticidal composition comprising, in admixture with an agriculturally acceptable carrier, an insecticidally effective amount of a 5-deazapteridine compound of the formula: ##STR1## wherein R.sup.1, R.sup.2, R.sup.3, R.sup.4, U, V, and W are as defined herein; agriculturally acceptable salts thereof; methods for using the same; and certain novel 5-deazapteridine per se.
摘要翻译：一种杀虫组合物，其包含与农业上可接受的载体的混合物，杀虫有效量的下式的5-去氮萘啶化合物：其中R1，R2，R3，R4，U，V和W为本文定义; 农业上可接受的盐; 使用方法; 和某些新的5-脱氮啶本身。

5. 发明授权

US06214845B1 Insecticidal N-(substituted arylmethyl)-4[bis(substituted phenyl or pyridyl)methyl] piperidines 失效
标题翻译：杀虫剂N-（取代的芳基甲基）-4 [双（取代的苯基或吡啶基）甲基]哌啶
公开(公告)号：US06214845B1
公开(公告)日：2001-04-10
申请号：US09388592
申请日：1999-09-02
申请人： Ian R. Silverman , Daniel H. Cohen , John W. Lyga , Steven W. Szczepanski , Syed F. Ali , Thomas G. Cullen , Robert N. Henrie, II , Clinton J. Peake
发明人： Ian R. Silverman , Daniel H. Cohen , John W. Lyga , Steven W. Szczepanski , Syed F. Ali , Thomas G. Cullen , Robert N. Henrie, II , Clinton J. Peake
IPC分类号： A01N4340
CPC分类号： C07D401/06 , A01N43/40 , A01N43/50 , A01N43/54 , A01N43/56 , A01N43/60 , A01N43/653 , A01N43/713 , A01N43/76 , A01N43/82 , A01N47/20 , A01N55/00 , C07D211/14 , C07D211/22 , C07D211/24 , C07D211/26 , C07D211/94 , C07D231/12 , C07D233/56 , C07D249/08 , C07D401/10 , C07D401/12 , C07D401/14 , C07D405/06 , C07D405/10 , C07D409/06 , C07D413/06 , C07D413/10 , C07D417/10 , C07D417/12 , C07F7/1804
摘要： Compounds of the following structure, the corresponding N-oxides and agriculturally acceptable salts, are disclosed as effective insecticides: in which U is —(CH2)n—; Q is hydroxy; R is in which V, W, Y, and Z are each hydrogen; X is a five- or six-membered heterocycle; optionally substituted with halogen, cyano, alkyl, haloalkyl, alkoxy, haloalkoxy, alkoxyalkyl, haloalkoxyalkyl, or aminocarbonyl; and the heterocycle is optionally connected to the phenyl ring through a —O—, —S—, —(CH2)p, —C(O)—, or —O—(CR3R4)q linkage; R1 and R2 are independently selected from phenyl or pyridyl substituted with haloalkyl or haloalkoxy; R3 and R4 are independently selected from hydrogen and methyl; n and p are independently 1, 2, or 3; and q is 1 or 2; with the proviso that at least one of R1 and R2 is substituted in the para position; no more than two of R3 and R4 are methyl; each aliphatic moiety contains not more than 4 carbon atoms; halogen means bromine, chlorine, or fluorine; each heterocycle contains from 1 to 4 nitrogen atoms, or 1 or 2 oxygen or sulfur atoms, or 1 or 2 nitrogen atoms and an oxygen or sulfur atom; and the corresponding N-oxides and agriculturally acceptable salts.
摘要翻译：公开了以下结构的化合物，即相应的N-氧化物和农业上可接受的盐作为有效的杀虫剂：其中U是 - （CH 2）n - ; Q是羟基; R 1是其中V，W，Y和Z各自是氢; X是五元或六元杂环; 任选被卤素，氰基，烷基，卤代烷基，烷氧基，卤代烷氧基，烷氧基烷基，卤代烷氧基烷基或氨基羰基取代; 并且杂环任选地通过-O - ， - S - ， - （CH 2）p，-C（O） - 或-O-（CR 3 R 4）q键连接到苯环; R 1和R 2独立地选自苯基或被卤代烷基或卤代烷氧基取代的吡啶基; R3和R4独立地选自氢和甲基; n和p独立地为1,2或3; 且q为1或2;条件是R1和R2中的至少一个在对位取代; R3和R4中不超过两个是甲基; 每个脂族部分含有不超过4个碳原子; 卤素是指溴，氯或氟; 每个杂环含有1至4个氮原子，或1或2个氧或硫原子，或1或2个氮原子和氧或硫原子;以及相应的N-氧化物和农业上可接受的盐。

6. 发明授权

US5639753A Insecticidal pteridines and 8-deazapteridines 失效
标题翻译：杀虫蝶啶和8-取代二萜烯
公开(公告)号：US5639753A
公开(公告)日：1997-06-17
申请号：US612657
申请日：1995-11-28
申请人： Robert N. Henrie, II , Clinton J. Peake , Thomas G. Cullen , Albert C. Lew , Ian R. Silverman
发明人： Robert N. Henrie, II , Clinton J. Peake , Thomas G. Cullen , Albert C. Lew , Ian R. Silverman
IPC分类号： A01N43/90 , C07D471/04 , C07D475/08 , A01N43/54 , A01N43/60
CPC分类号： C07D471/04 , A01N43/90 , C07D475/08
摘要： This invention relates to pteridine and 8-deazapteridine compounds and compositions containing the same which are useful for controlling insects in agricultural crops. These pteridines may be represented by the following structure: ##STR1## wherein R and R.sup.1 are independently selected from amino, lower alkylamino, di(lower alkyl)amino (e.g., --N(CH.sub.3).sub.2), or di(lower alkyl)aminomethyleneamino (e.g., --N.dbd.CHN(CH.sub.3).sub.2);R.sup.2 is hydrogen, amino, lower alkyl (e.g., --CH.sub.3, --CH(CH.sub.3).sub.2), di(lower alkyl)aminomethyleneamino, hydroxy, lower alkoxy, phenyl or substituted phenyl, haloalkylphenylalkyl (e.g., 3-trifluoromethylphenylmethyl);Q is N or CH;R.sup.3 is -(n).sub.m -R.sup.4, where m is 0 or 1; wherein, when m is 1,n is a bridging atom or moiety selected from oxygen, sulfur, sulfinyl, sulfonyl, lower alkylene (e.g., --CH.sub.2 --, or --CH.sub.2 CH.sub.2 --), lower alkenylene (e.g., --CH.dbd.CH--), lower alkynylene (e.g., --C.tbd.C--), lower haloalkenylene (e.g., --C(Cl).dbd.CH--), carbonyl, aminomethyl (e.g., --CH.sub.2 NH--), or (substituted amino)methyl (e.g., --CH.sub.2 N(CH.sub.3)--); andR.sup.4 is hydrogen, lower alkyl (e.g., --CH.sub.3, or --CH(CH.sub.3).sub.2), thien-2-yl, pyridin-3-yl, or ##STR2## wherein (i) V, W, X, Y, and Z are as defined herein.
摘要翻译：本发明涉及蝶啶和8-脱氮吡啶化合物及其含有该组合物的组合物，其可用于控制农作物中的昆虫。这些蝶啶可以由以下结构表示：其中R和R 1独立地选自氨基，低级烷基氨基，二（低级烷基）氨基（例如，-N（CH 3）2）或二（低级）烷基）氨基亚甲基氨基（例如，-N = CHN（CH 3）2）; R 2是氢，氨基，低级烷基（例如-CH 3，-CH（CH 3）2），二（低级烷基）氨基亚甲基氨基，羟基，低级烷氧基，苯基或取代的苯基，卤代烷基苯基烷基（例如3-三氟甲基苯基甲基）。 Q是N或CH; R3是 - （n）m-R4，其中m是0或1; 其中，当m为1时，n为选自氧，硫，亚磺酰基，磺酰基，低级亚烷基（例如-CH 2 - 或-CH 2 CH 2 - ）的桥连原子或部分，低级亚烯基（例如-CH = CH-），低级亚炔基（例如-C 3 -C（O） - ），低级卤代亚烯基（例如-C（Cl）= CH-），羰基，氨基甲基（例如-CH 2 NH-）或（取代的氨基）甲基（CH 3） - ）; 和R 4是氢，低级烷基（例如，-CH 3或-CH（CH 3）2），噻吩-2-基，吡啶-3-基或其中（i）V，W，X，Y，和Z如本文所定义。

7. 发明授权

US5534518A Insecticidal substituted-2,4-diaminoquinazolines 失效
公开(公告)号：US5534518A
公开(公告)日：1996-07-09
申请号：US267340
申请日：1994-06-28
申请人： Robert N. Henrie, II , Clinton J. Peake , Thomas G. Cullen , Albert C. Lew , Munirathnam K. Chaguturu , Partha S. Ray , Walter H. Yeager , Ian R. Silverman , John W. Buser , James J. Fiordeliso , John A. Dixson
发明人： Robert N. Henrie, II , Clinton J. Peake , Thomas G. Cullen , Albert C. Lew , Munirathnam K. Chaguturu , Partha S. Ray , Walter H. Yeager , Ian R. Silverman , John W. Buser , James J. Fiordeliso , John A. Dixson
IPC分类号： A01N43/54 , A01N55/00 , C07D239/95 , C07D401/12 , C07D405/04 , C07D409/04 , A61K31/505
CPC分类号： C07D401/12 , A01N43/54 , A01N55/00 , C07D239/95 , C07D405/04 , C07D409/04
摘要： An insecticidal composition comprising, in admixture with an agriculturally acceptable carrier, an insecticidally effective amount of a 2,4-diaminoquinazoline compound of the formula: ##STR1## wherein R.sup.1, R.sup.2, R.sup.6, R.sup.7, W, X, Y, and Z are as defined herein; methods of using the same; novel 2,4-diaminoquinazolines per se; and intermediates in the preparation thereof.

8. 发明授权

US4808722A Pyridinylurea N-oxide compounds and agricultural uses 失效
标题翻译：吡啶基脲N-氧化物和农业用途
公开(公告)号：US4808722A
公开(公告)日：1989-02-28
申请号：US793372
申请日：1985-10-31
申请人： Robert N. Henrie, II
发明人： Robert N. Henrie, II
IPC分类号： A01N47/36 , C07D213/75 , C07D213/89 , A01N47/30
CPC分类号： C07D213/75 , A01N47/36 , C07D213/89
摘要： Pyridinylurea N-oxides of the formula ##STR1## and acid addition salts thereof; wherein R is cycloalkyl (C.sub.3 -C.sub.8), alkenyl (C.sub.3 -C.sub.8), or an alkyl (C.sub.1 -C.sub.6) group optionally substituted with halogen, hydroxy, cycloalkyl (C.sub.3 -C.sub.8) alkoxy (C.sub.1 -C.sub.6), dialkyl (C.sub.1 -C.sub.6)amino or phenyl; R.sup.1 is hydrogen or alkyl (C.sub.1 -C.sub.6); R and R.sup.1 together with the nitrogen atom of the NRR.sup.1 group optionally define a nonaromatic heterocycle containing 4 to 6 ring carbon atoms; each X independently is halogen, alkyl (C.sub.1 -C.sub.6), haloalkyl (C.sub.1 -C.sub.6), alkoxy (C.sub.1 -C.sub.6), hydroxy, 2-pyridinyl, alkyl(C.sub.1 -C.sub.6)thio or alkyl (C.sub.1 -C.sub.6)sulfonyl; A is 1 to 4; and wherein the NHCONRR.sup.1 group is bonded to the pyridinyl ring in the 3- or 4-position. The compounds are useful in agriculture as plant growth regulators.
摘要翻译：吡啶基脲式VII的N-氧化物及其酸加成盐; 其中R是任选被卤素，羟基，环烷基（C 3 -C 8）烷氧基（C 1 -C 6），二烷基（C 1 -C 6）烷基（C 3 -C 8） C6）氨基或苯基; R1是氢或烷基（C1-C6）; R和R 1与NRR1基团的氮原子一起任选地定义含有4-6个环碳原子的非芳族杂环; 每个X独立地是卤素，烷基（C1-C6），卤代烷基（C1-C6），烷氧基（C1-C6），羟基，2-吡啶基，烷基（C1-C6）硫代或烷基（C1-C6） A是1到4; 并且其中NHCONRR1基团键合在3-或4-位的吡啶环上。这些化合物在农业中可用作植物生长调节剂。

9. 发明授权

US08119563B2 N-substituted azacycles 失效
标题翻译： N-取代的azacycles
公开(公告)号：US08119563B2
公开(公告)日：2012-02-21
申请号：US10595298
申请日：2004-10-04
申请人： George Theodoridis , David Rosen , Shunxiang Zhang , Walter H. Yeager , Robert N. Henrie, II , Syed Z. Ahmed , Hongbin Men , Stephen Donovan
发明人： George Theodoridis , David Rosen , Shunxiang Zhang , Walter H. Yeager , Robert N. Henrie, II , Syed Z. Ahmed , Hongbin Men , Stephen Donovan
IPC分类号： A01N43/22 , C07D211/06
CPC分类号： C07D211/48 , A01N43/40 , A01N43/54 , A01N43/58 , A01N43/713 , A01N43/90 , A01N47/06 , A01N47/20 , A01N47/22 , C07D211/94 , C07D401/10 , C07D401/12 , C07D451/02 , C07D471/10
摘要： N-substituted azacycle derivative compounds represented by formula (I): wherein m, q, r, t and u are independently selected from 0 or 1; and p is 0, 1, 2, or 3; and A, B, D, X, Y, R, R1, R2, R3, R4, R5, R6, R7, R8, R9, R10 and R11 are fully described herein. The compounds being particularly useful in compositions comprising an insecticidally effective amount of at least one compound of formula I, and an insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present.
摘要翻译：由式（I）表示的N-取代的azacycle衍生物化合物：其中m，q，r，t和u独立地选自0或1; 且p为0,1,2或3; 并且A，B，D，X，Y，R，R 1，R 2，R 3，R 4，R 5，R 6，R 7，R 8，R 9，R 10和R 11在本文中被完整描述。还公开了特别可用于包含杀虫有效量的至少一种式I化合物和杀虫相容载体的化合物; 以及控制昆虫的方法，包括将所述组合物施用于存在昆虫或预期存在的场所。

10. 发明授权

US07683070B2 N-(substituted arylmethyl)-4-(disubstituted methyl) piperidines and pyridines 有权
标题翻译： N-（取代的芳基甲基）-4-（二取代的甲基）哌啶和吡啶
公开(公告)号：US07683070B2
公开(公告)日：2010-03-23
申请号：US11874015
申请日：2007-10-17
申请人： Ping Ding , Robert N. Henrie, II , Daniel H. Cohen , John W. Lyga , David S. Rosen , George Theodoridis , Qun Zhang , Walter H. Yeager , Stephen F. Donovan , Stephen Shunxiang Zhang , Inna Shulman , Seong Jae Yu , Guozhi Wang , Y. Larry Zhang , Ariamala Gopalsamy , Dennis L. Warkentin , Paul E. Rensner , Ian R. Silverman , Thomas G. Cullen
发明人： Ping Ding , Robert N. Henrie, II , Daniel H. Cohen , John W. Lyga , David S. Rosen , George Theodoridis , Qun Zhang , Walter H. Yeager , Stephen F. Donovan , Stephen Shunxiang Zhang , Inna Shulman , Seong Jae Yu , Guozhi Wang , Y. Larry Zhang , Ariamala Gopalsamy , Dennis L. Warkentin , Paul E. Rensner , Ian R. Silverman , Thomas G. Cullen
IPC分类号： A61K31/4523 , A61K31/4545 , C07D211/06 , C07D239/02
CPC分类号： C07D405/14 , A01N43/40 , A01N43/54 , A01N43/713 , C07D211/14 , C07D211/18 , C07D211/22 , C07D211/24 , C07D211/26 , C07D211/28 , C07D211/32 , C07D211/94 , C07D401/06 , C07D401/10 , C07D401/12 , C07D401/14 , C07D413/12 , C07D417/12 , C07D451/14 , C07D513/04
摘要： It has now been found that certain novel N-(substituted aryl)-4-(disubstituted methyl)piperidine and pyridine derivatives have provided unexpected insecticidal activity. These compounds are represented by formula (I): wherein m, n, q, r, and s are independently selected from 0 or 1; and p is 0, 1, 2, or 3; A is C or CH; and B, D, E, R, R1, R2, R3, R4, R5, R6, R7 and R8 are fully described herein. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula I, and optionally, an effective amount of at least one of a second compound, with at least one insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present.
摘要翻译：现在已经发现某些新的N-（取代的芳基）-4-（二取代的甲基）哌啶和吡啶衍生物提供了意想不到的杀虫活性。这些化合物由式（I）表示：其中m，n，q，r和s独立地选自0或1; 且p为0,1,2或3; A是C或CH; 本文完整地描述了B，D，E，R，R 1，R 2，R 3，R 4，R 5，R 6，R 7和R 8。此外，还公开了包含杀虫有效量的至少一种式I化合物和任选的有效量的至少一种第二化合物与至少一种与杀虫相容的载体的组合物; 以及控制昆虫的方法，包括将所述组合物施用于存在昆虫或预期存在的场所。

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