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1. 发明授权

US5530021A Hydrazine derivative and pesticidal composition comprising said derivative as an effective ingredient 失效
标题翻译：肼衍生物和包含所述衍生物作为有效成分的农药组合物
公开(公告)号：US5530021A
公开(公告)日：1996-06-25
申请号：US308643
申请日：1994-09-19
申请人： Mikio Yanagi , Hiroyasu Sugizaki , Tetsuya Toya , Yasuhito Kato , Hidetoshi Shirakura , Tetsuo Watanabe , Yoshimi Yajima , Seiichirou Kodama , Akio Masui , Toshiaki Yanai , Yoshihisa Tsukamoto , Yoshihiro Sawada , Shinji Yokoi
发明人： Mikio Yanagi , Hiroyasu Sugizaki , Tetsuya Toya , Yasuhito Kato , Hidetoshi Shirakura , Tetsuo Watanabe , Yoshimi Yajima , Seiichirou Kodama , Akio Masui , Toshiaki Yanai , Yoshihisa Tsukamoto , Yoshihiro Sawada , Shinji Yokoi
IPC分类号： A01N43/16 , A01N43/18 , A01N43/24 , A01N43/32 , A01N43/42 , A01N43/46 , A01N43/60 , A01N43/62 , A01N43/72 , A01N43/84 , A01P7/04 , C07D223/16 , C07D241/42 , C07D241/44 , C07D243/12 , C07D265/36 , C07D267/14 , C07D279/16 , C07D281/10 , C07D311/12 , C07D311/22 , C07D311/58 , C07D311/68 , C07D313/08 , C07D319/16 , C07D319/18 , C07D319/20 , C07D321/10 , C07D327/06 , C07D335/06 , C07D337/08 , C07D339/00 , C07D339/08 , C07D493/10 , C07F7/18
CPC分类号： C07D493/10 , A01N43/16 , A01N43/24 , A01N43/32 , A01N43/84 , C07D265/36 , C07D311/22 , C07D311/58 , C07D311/68 , C07D319/18 , C07D319/20 , C07D321/10 , C07D327/06 , C07F7/1844
摘要： A novel hydrazine derivative and a pesticidal composition containing the hydrazine derivative as the effecting ingredient. The hydrazine derivative show high pesticidal activity against harmful pests which are resistant to known pesticides such as organophosphorus pesticides, pyrethroids, etc., especially against Lepidoptera harmful pests such as Plutella xylostella, Spodoptera litura, Cnaphalocrocis medinalis, Adoxophyes orana, etc., and is effective for controlling harmful pests in paddy field, upland field, orchard, forest or places to be kept environmentally hygienic.
摘要翻译：一种新颖的肼衍生物和含有肼衍生物作为有效成分的农药组合物。肼衍生物对杀虫剂具有很强的杀虫活性，对有机磷杀虫剂，拟除虫菊酯等已知的农药具有抗性，特别是针对鳞翅目有害害虫如小菜蛾（Plutella xylostella），斜纹夜蛾（Spodoptera litura），Cnaphalocrocis medinalis，Adoxophyes orana等，有效控制水田，旱田，果园，森林或环境卫生的有害害虫。

2. 发明授权

US5378726A New hydrazine derivative and pesticidal composition comprising said derivative as an effective ingredient 失效
标题翻译：包含所述衍生物作为有效成分的新肼衍生物和杀虫组合物
公开(公告)号：US5378726A
公开(公告)日：1995-01-03
申请号：US152877
申请日：1993-11-15
申请人： Mikio Yanagi , Hiroyasu Sugizaki , Tetsuya Toya , Yasuhito Kato , Hidetoshi Shirakura , Tetsuo Watanabe , Yoshimi Yajima , Seiichirou Kodama , Akio Masui , Toshiaki Yanai , Yoshihisa Tsukamoto , Yoshihiro Sawada , Shinji Yokoi
发明人： Mikio Yanagi , Hiroyasu Sugizaki , Tetsuya Toya , Yasuhito Kato , Hidetoshi Shirakura , Tetsuo Watanabe , Yoshimi Yajima , Seiichirou Kodama , Akio Masui , Toshiaki Yanai , Yoshihisa Tsukamoto , Yoshihiro Sawada , Shinji Yokoi
IPC分类号： A01N43/16 , A01N43/18 , A01N43/24 , A01N43/32 , A01N43/42 , A01N43/46 , A01N43/60 , A01N43/62 , A01N43/72 , A01N43/84 , A01P7/04 , C07D223/16 , C07D241/42 , C07D241/44 , C07D243/12 , C07D265/36 , C07D267/14 , C07D279/16 , C07D281/10 , C07D311/12 , C07D311/22 , C07D311/58 , C07D311/68 , C07D313/08 , C07D319/16 , C07D319/18 , C07D319/20 , C07D321/10 , C07D327/06 , C07D335/06 , C07D337/08 , C07D339/00 , C07D339/08 , C07D493/10 , C07F7/18
CPC分类号： C07D493/10 , A01N43/16 , A01N43/24 , A01N43/32 , A01N43/84 , C07D265/36 , C07D311/22 , C07D311/58 , C07D311/68 , C07D319/18 , C07D319/20 , C07D321/10 , C07D327/06 , C07F7/1844
摘要： A novel hydrazine derivative and a pesticidal composition containing the hydrazine derivative as the effecting ingredient. The hydrazine derivative show high pesticidal activity against harmful pests which are resistant to known pesticides such as organophosphorus pesticides, pyrethroids, etc., especially against Lepidopters harmful pests such as Plutella xylostella, Spodoptera litura, Cnaphalocrocis medinalis, Adoxophyes orana, etc., and is effective for controlling harmful pests in paddy field, upland field, orchard, forest or places to be kept environmentally hygienic.
摘要翻译：一种新颖的肼衍生物和含有肼衍生物作为有效成分的农药组合物。肼衍生物对杀虫剂具有较高的杀虫活性，对有机磷杀虫剂，拟除虫菊酯等已知的农药具有抗性，特别是针对小菜蛾，斜纹夜蛾，白僵菌，Adoxophyes orana等对鳞翅目害虫有害害虫的杀虫活性，有效控制水田，旱田，果园，森林或环境卫生的有害害虫。

3. 发明授权

US5276033A 13-(substituted thio)acetoxymilbemycin derivatives, their preparation and their agrochemical uses 失效
标题翻译： 13-（取代硫代）乙酰氧基米尔伯霉素衍生物，其制备方法及其农用化学品用途
公开(公告)号：US5276033A
公开(公告)日：1994-01-04
申请号：US992865
申请日：1992-12-17
申请人： Toshiaki Yanai , Soji Sugai , Hideo Takeshiba , Junzo Tobitsuka , Kazuo Sato , Shinji Yokoi , Shinya Niimi , Akio Saito
发明人： Toshiaki Yanai , Soji Sugai , Hideo Takeshiba , Junzo Tobitsuka , Kazuo Sato , Shinji Yokoi , Shinya Niimi , Akio Saito
IPC分类号： A01N43/90 , A01P7/04 , C07D493/22 , C07H19/01 , A61K31/53 , A61K31/505 , C07D239/38
CPC分类号： C07H19/01 , A01N43/90
摘要： Compounds having the formula (I) ##STR1## wherein: R.sup.1 is methyl, ethyl or isopropyl; R.sup.2 is alkyl, aralkyl, cycloalkyl, cycloalkylmethyl, aryl, heterocyclic, or heterocyclic-substituted thio; R.sup.3 is hydrogen, methyl or ethyl; or R.sup.2 together with R.sup.3 is --(CH.sub.2).sub.n --, wherein n is 3,4 or 5; and A is aromatic heterocyclic; and salts thereof, are valuable agricultural and horticultural anthelmintic, acaricidal and insecticidal agents.
摘要翻译：具有式（I）的化合物（I）其中：R1是甲基，乙基或异丙基; R2是烷基，芳烷基，环烷基，环烷基甲基，芳基，杂环或杂环取代的硫代; R3是氢，甲基或乙基; 或R 2与R 3一起为 - （CH 2）n - ，其中n为3,4或5; A是芳族杂环; 和其盐是有价值的农业和园艺驱虫剂，杀螨剂和杀虫剂。

4. 发明授权

US5614470A 13-substituted milbemycin derivatives, their preparation and their use 失效
标题翻译： 13-取代的米尔倍霉素衍生物，其制备及其应用
公开(公告)号：US5614470A
公开(公告)日：1997-03-25
申请号：US412687
申请日：1995-03-29
申请人： Hideo Takeshiba , Kazuo Sato , Toshiaki Yanai , Shinji Yokoi , Reiji Ichinose , Kinji Tanizawa
发明人： Hideo Takeshiba , Kazuo Sato , Toshiaki Yanai , Shinji Yokoi , Reiji Ichinose , Kinji Tanizawa
IPC分类号： C07D493/22 , A01N20060101 , A01N43/90 , A01P7/02 , A01P7/04 , C07D20060101 , C07H20060101 , C07H19/01 , A01N43/04 , A61K31/335
CPC分类号： C07H19/01 , A01N43/90
摘要： 13-Substituted milbemycin derivatives having the formula (I): ##STR1## wherein: R.sup.1 is methyl, ethyl, isopropyl or sec-butyl;R.sup.2 is hydrogen or alkyl;X is (.alpha.-hydroxyimino- or .alpha.-alkoxyimino-substituted)-arylmethyl or (.alpha.-hydroxyimino- or .alpha.-alkoxyimino-substituted)-heterocyclylmethyl, N-substituted-aminophenyl or N-substituted-aminophenoxy;m is 0 or 1; and n is 0 or 1;are valuable as agricultural and horticultural anthelmintic, acaricidal and insecticidal agents.
摘要翻译： 13-取代的具有式（I）的密尔伯霉素衍生物：其中：R1是甲基，乙基，异丙基或仲丁基; R2是氢或烷基; X是（α-羟基亚氨基 - 或α-烷氧基亚氨基取代的） - 芳基甲基或（α-羟基亚氨基或α-烷氧基亚氨基取代的） - 杂环基甲基，N-取代的 - 氨基苯基或N-取代的 - 氨基苯氧基; m为0或1; 并且n为0或1; 作为农业和园艺驱虫剂，杀螨剂和杀虫剂是有价值的。

5. 发明授权

US5208349A Process for preparing milbemycin derivatives and certain novel compounds employed therein 失效
标题翻译：米尔霉素衍生物及其中所用的某些新化合物的制备方法
公开(公告)号：US5208349A
公开(公告)日：1993-05-04
申请号：US644880
申请日：1991-01-24
申请人： Kazuo Sato , Takao Kinoto , Shigeru Mio , Toshiaki Yanai
发明人： Kazuo Sato , Takao Kinoto , Shigeru Mio , Toshiaki Yanai
IPC分类号： C07H19/01
CPC分类号： C07H19/01
摘要： 13-Hydroxy-5-ketomilbemycin derivatives are prepared by oxidizing a 5-ketomilbemycin with selenium dioxide in the presence of a lower aliphatic carboxylic acid. A range of new 13-acyloxy-5-ketomilbemycins and a method of preparing them are also disclosed.
摘要翻译：通过在低级脂肪族羧酸的存在下用二氧化硒氧化5-酮米尔贝霉素来制备13-羟基-5-酮米尔贝霉素衍生物。还公开了一系列新的13-酰氧基-5-酮基尔贝莫霉素及其制备方法。

6. 发明授权

US4835290A Process for preparing 13-hydroxy-5-ketomibemycin derivatives having acaricidal, insecticidal and anthelmintic activity 失效
标题翻译：制备具有杀螨，杀虫和驱虫活性的13-羟基-5-酮基霉素衍生物的方法
公开(公告)号：US4835290A
公开(公告)日：1989-05-30
申请号：US115642
申请日：1987-10-26
申请人： Kazuo Sato , Takao Kinoto , Shigeru Mio , Toshiaki Yanai
发明人： Kazuo Sato , Takao Kinoto , Shigeru Mio , Toshiaki Yanai
IPC分类号： C07H19/01
CPC分类号： C07H19/01
摘要： 13-Hydroxy-5-ketomilbemycin derivatives are prepared by oxidizing a 5-ketomilbemycin with selenium dioxide in the presence of a lower aliphatic carboxylic acic. A range of new 13-acyloxy-5-ketomilbemycins and a method or preparing them are also disclosed.
摘要翻译：通过在低级脂肪族羧酸存在下，用二氧化硒氧化5-酮米尔贝霉素来制备13-羟基-5-酮米尔贝霉素衍生物。还公开了一系列新的13-酰氧基-5-酮基尔贝莫霉素及其制备方法或制备方法。

7. 发明授权

US5212322A Macrolide compounds, their preparation and their use 失效
标题翻译：大环内酯类化合物，其制备及其用途
公开(公告)号：US5212322A
公开(公告)日：1993-05-18
申请号：US644100
申请日：1991-01-22
申请人： Takao Okazaki , Shuji Takahashi , Seigo Iwado , Keiji Tanaka , Toshiaki Yanai , Hisaki Kajino
发明人： Takao Okazaki , Shuji Takahashi , Seigo Iwado , Keiji Tanaka , Toshiaki Yanai , Hisaki Kajino
IPC分类号： A01N49/00 , C07H19/01 , C12P17/18
CPC分类号： C07H19/01 , A01N49/00 , C12P17/181 , Y02P20/55 , Y10S424/08
摘要： Compounds with acaricidal, insecticidal and anthelmintic activities have the formula: ##STR1## wherein: --X--Y-- is selected from the group consisting of --CH.sub.2 --CH.sub.2 --, --CH.sub.2 --CHOH--, --CH.dbd.CH--, and --CH.sub.2 --C(.dbd.O)--;R.sup.1 is selected from the group consisting of a methyl group, an ethyl group, an isopropyl group, a sec-butyl group and groups of formula --C(CH.sub.3).dbd.CHR.sup.5 in which R.sup.5 is selected from the group consisting of a methyl group, an ethyl group and an isopropyl group;R.sup.2 represents a group of formula --(CH.sub.2).sub.n --C(R.sup.6).dbd.C(R.sup.7)(R.sup.8) in which n is 0, 1 or 2, R.sup.6 and R.sup.7 each is selected from the group consisting of a hydrogen atom and a methyl group and R.sup.8 is selected from the group consisting of a hydrogen atom, a C.sub.1-4 alkyl group, a phenyl group and a phenyl group substituted with at least one substituent selected from the group consisting of halogen, methyl and nitro substituents;R.sup.3 is selected from the group consisting of a hydrogen atom, a methyl group, a hydroxy-protecting group, an ester-forming carboxylic acid residue, and an ester-forming carbonic acid residue; andR.sup.4 is selected from the group consisting of a hydrogen atom and an .alpha.-L-oleandrosyl-.alpha.-L-oleandrosyloxy group, with the proviso that R.sup.4 represents a hydrogen atom when the group R.sup.1 is selected from the group consisting of a methyl group, an ethyl group, and groups of formula --C(CH.sub.3).dbd.CHR.sup.5 in which R.sup.5 is selected from the group consisting of a methyl group, an ethyl group and an isopropyl group.
摘要翻译：具有杀螨，杀虫和驱虫活性的化合物具有下式：其中：-XY-选自-CH 2 -CH 2 - ， - CH 2 -CHOH - ， - CH = CH-和 - CH2-C（= O） - ; R 1选自甲基，乙基，异丙基，仲丁基和式-C（CH 3）= CHR 5的基团，其中R 5选自甲基，乙基和异丙基; R 2表示式 - （CH 2）n C（R 6）= C（R 7）（R 8）的基团，其中n为0,1或2，R 6和R 7各自为氢原子和甲基并且R 8选自氢原子，C 1-4烷基，苯基和被至少一个选自卤素，甲基和硝基取代基的取代基取代的苯基; R3选自氢原子，甲基，羟基保护基，成酯羧酸残基和形成酯的碳酸残基; 并且R 4选自氢原子和α-L-甘氨酰基-α-L-胆碱基氧基，条件是当R 1选自甲基时，R 4表示氢原子，乙基和式-C（CH 3）= CHR 5基团，其中R 5选自甲基，乙基和异丙基。

8. 发明授权

US4945105A 13-Halomilbemycin derivatives, their preparation and compositions containing them 失效
标题翻译： 13-哈美列霉素衍生物，其制备方法和含有它们的组合物
公开(公告)号：US4945105A
公开(公告)日：1990-07-31
申请号：US290835
申请日：1988-12-28
申请人： Kazuo Sato , Toshiaki Yanai , Noritoshi Kitano , Akira Nishida , Bruno Frei , Anthony O'Sullivan
发明人： Kazuo Sato , Toshiaki Yanai , Noritoshi Kitano , Akira Nishida , Bruno Frei , Anthony O'Sullivan
IPC分类号： C07D493/22 , A01N43/90 , A01P5/00 , A01P7/02 , A01P7/04 , A61K31/365 , A61P33/10 , C07D307/00 , C07D309/00 , C07H19/01
CPC分类号： C07H19/01 , A01N43/90
摘要： Derivatives of milbemycins D, A.sub.3 and A.sub.4 and of the corresponding sec-butyl compound have a halogen atom at the 13-position; at the 5-position, they have an oxygen (keto) atom, an oxime group or a substituted oxime group. They may be prepared from known compounds by any appropriate combination of halogenation, ketonization and oximation.
摘要翻译：米尔倍霉素D，A3和A4及相应的仲丁基化合物的衍生物在13位具有卤素原子; 在5位，它们具有氧（酮）原子，肟基或取代的肟基。它们可以通过卤化，酮化和肟化的任何适当组合由已知化合物制备。

9. 发明授权

US4963582A Macrolide compounds, their preparation and their use 失效
标题翻译：大环内酯类化合物，其制备及其用途
公开(公告)号：US4963582A
公开(公告)日：1990-10-16
申请号：US30217
申请日：1987-03-24
申请人： Kazuo Sato , Toshiaki Yanai , Takao Kinoto , Keiji Tanaka , Akira Nishida , Toshimitsu Toyama , Bruno Frei , Anthony O'Sullivan
发明人： Kazuo Sato , Toshiaki Yanai , Takao Kinoto , Keiji Tanaka , Akira Nishida , Toshimitsu Toyama , Bruno Frei , Anthony O'Sullivan
IPC分类号： A01N43/90 , A01N47/06 , A01P5/00 , A01P7/02 , A01P7/04 , A61K31/365 , C07D493/22 , C07H19/01
CPC分类号： C07D493/22 , A01N43/90 , A01N47/06 , C07H19/01
摘要： Compounds having a 16-membered macrolide ring, and related to the milbemycins and avermectins, with substituents at positions 5, 13, 25 and optionally also 23, have acaricidal, insecticidal and anthelmintic properties. They are useful for treating various pests in plants and animals.

10. 发明授权

US4460597A Herbicidal 5-aminoalkoxy-4-benzoyl-1,3-dimethyl-pyrazole derivatives 失效
标题翻译：除草剂5-氨基烷氧基-4-苯甲酰基-1,3-二甲基 - 吡唑衍生物
公开(公告)号：US4460597A
公开(公告)日：1984-07-17
申请号：US496815
申请日：1983-05-23
申请人： Toshiaki Yanai , Teruomi Jojima , Katsuhiko Kawakubo , Toyokuni Honma , Masahiro Shindo
发明人： Toshiaki Yanai , Teruomi Jojima , Katsuhiko Kawakubo , Toyokuni Honma , Masahiro Shindo
IPC分类号： A01N43/56 , C07D231/20
CPC分类号： C07D231/20 , A01N43/56
摘要： Pyrazole derivatives of formula (I): ##STR1## (R.sup.1 is methyl, halogen or nitro; n is 2 or 3; R.sup.2 is hydrogen, C.sub.1-4 alkyl, C.sub.3-4 alkenyl or aralkyl; R.sup.3 is C.sub.1-4 alkyl, C.sub.3-4 alkenyl or phenyl; A is C.sub.1-5 alkylene) are of use as herbicides.
摘要翻译：式（I）的吡唑衍生物：（I）（R1是甲基，卤素或硝基; n是2或3; R2是氢，C1-4烷基，C3-4链烯基或芳烷基; R3是C1-4 烷基，C3-4烯基或苯基; A为C1-5亚烷基）可用作除草剂。

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