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1. 发明授权

US6028032A 1,3-oxazin-4-one derivatives as herbicides 失效
标题翻译： 1,3-恶嗪-4-酮衍生物作为除草剂
公开(公告)号：US6028032A
公开(公告)日：2000-02-22
申请号：US981569
申请日：1998-04-13
申请人： Michael Colin Cramp , Yoshihiro Usui , Keiichi Hayashizaki
发明人： Michael Colin Cramp , Yoshihiro Usui , Keiichi Hayashizaki
IPC分类号： A01N43/86 , C07D265/06 , C07F7/18
CPC分类号： C07D265/06 , A01N43/86
摘要： 1,3-oxazin-4-ones of formula (I), ##STR1## wherein R.sup.1 represents phenyl optionally substituted; R.sup.2 represents: a straight- or branched-chain alkyl having from one to ten carbon atoms which is substituted by one or more groups R.sup.8 which may be the same or different; a straight- or branched-chain optionally halogenated alkenyl or alkynyl group having up to ten carbon atoms; or a group selected from cyano, --CHO, --COR.sup.7, --CO.sub.2 H, --CO.sub.2 R.sup.7, --COSR.sup.7, --CONR.sup.9 R.sup.10, --CH.dbd.NOH, --CH.dbd.NOR.sup.7, --CH.dbd.NOCOR.sup.7, --CH.dbd.NNR.sup.9 R.sup.10, --CH.sub.2 CN, --CH.sub.2 NO.sub.2 and oxiranyl; R.sup.3 represents phenyl optionally substituted or R.sup.3 represents a first five to seven membered heteroaromatic ring; said first ring being optionally fused and said first ring being linked to the nitrogen atom of the group NR.sup.6 via one of the ring carbon atoms; R.sup.4 and R.sup.5 independently represent lower alkyl; W represents --NR.sup.6 --; R.sup.6 represents hydrogen, lower alkyl, haloalkyl, alkenyl, alkynyl, --COR.sup.7 or --CO.sub.2 R.sup.7 ; and their use as herbicides.
摘要翻译： PCT No.PCT / EP96 / 02616 371日期：1998年4月13日 102（e）1998年4月13日PCT PCT 1996年6月18日PCT公布。出版物WO97 / 00865 日本1991年1月9日公开了式（I）的1,3-二嗪-4-酮，其中R 1表示任选取代的苯基; R2表示：具有1至10个碳原子的直链或支链烷基，其被一个或多个可以相同或不同的基团R 8取代; 具有至多10个碳原子的直链或支链任选卤代的烯基或炔基; 或选自氰基，-CHO，-COR 7，-CO 2 H，-CO 2 R 7，-COSR 7，-CONR 9 R 10，-CH = NOH，-CH = NOR 7，-CH = NOCOR 7，-CH = NNR 9 R 10，-CH 2 CN，-CH 2 NO 2 和环氧乙烷基; R3代表任意取代的苯基或R3代表第一个五至七元杂芳环; 所述第一环任选地稠合，并且所述第一环通过环碳原子之一与NR6的氮原子连接; R4和R5独立地表示低级烷基; W代表-NR6-; R6代表氢，低级烷基，卤代烷基，烯基，炔基，-COR7或-COO2R7; 及其作为除草剂的用途。

2. 发明授权

US6046135A 1,3-oxazin-4-one derivatives as herbicides 失效
标题翻译： 1,3-恶嗪-4-酮衍生物作为除草剂
公开(公告)号：US6046135A
公开(公告)日：2000-04-04
申请号：US77745
申请日：1998-09-02
申请人： Michael Colin Cramp , Yoshihiro Usui , Sachio Kudo
发明人： Michael Colin Cramp , Yoshihiro Usui , Sachio Kudo
IPC分类号： A01N43/86 , C07D265/06 , C07D413/04 , C07D413/06 , C07D417/06
CPC分类号： C07D413/04 , A01N43/86 , C07D265/06 , C07D413/06
摘要： 1,3-Oxazin-4-one derivatives of formula (I): ##STR1## wherein Q represents --C(.dbd.O)--, --CH(OH)-- or --C(OR.sup.11)(OR.sup.11)--, in which R.sup.11 represents lower alkyl; or the two groups --OR.sup.11, together with the carbon atom to which they are attached, form a five or six membered cyclic ketal group; and their use as herbicides.
摘要翻译： PCT No.PCT / EP96 / 05404 Sec。 371日期：1998年9月2日 102（e）1998年9月2日PCT 1996年12月4日PCT PCT。公开号WO97 / 21688 日期：19,1971年3-式（I）的恶嗪-4-酮衍生物：其中Q表示-C（= O） - ， - CH（OH） - 或-C（OR 11）（OR 11）其中R11表示低级烷基; 或两个基团-OR 11与它们所连接的碳原子一起形成五或六元环缩酮基团; 及其作为除草剂的用途。

3. 发明授权

US5977025A 1,3-oxazin-4-one derivative, herbicide containing same, and intermediate for preparing same 失效
标题翻译： 1,3-恶嗪-4-酮衍生物，含有它们的除草剂及其制备中间体
公开(公告)号：US5977025A
公开(公告)日：1999-11-02
申请号：US663118
申请日：1996-06-20
申请人： Keiichi Hayashizaki , Yoshihiro Usui , Koichi Araki , Norishige Toshima , Tetsuya Murata , Takako Aoki , Atsushi Go , Hideshi Mukaida , Rika Higurashi
发明人： Keiichi Hayashizaki , Yoshihiro Usui , Koichi Araki , Norishige Toshima , Tetsuya Murata , Takako Aoki , Atsushi Go , Hideshi Mukaida , Rika Higurashi
IPC分类号： A01N43/86 , A01P13/00 , C07C229/12 , C07C251/08 , C07D265/06 , A01N43/32
CPC分类号： C07C251/08 , C07D265/06
摘要： This invention provides 1,3-oxazin-4-one derivatives represented by following general formula (I): ##STR1## in which R.sup.1 represents a phenyl group which may be substituted; R.sup.2 represents a hydrogen atom or a lower alkyl group; R.sup.3 represents a hydrogen atom, a lower alkyl group, an aralkyl group or a phenyl group which may be substituted; R.sup.4 and R.sup.5 each independently represent a lower alkyl group; and W represents an oxygen atom or a group represented by the formula --N(R.sup.6)-- in which R.sup.6 represents a hydrogen atom, a lower alkyl group, a lower alkenyl group or a lower alkynyl group. There are also provided herbicidal compositions containing the derivatives and intermediates for preparing them. The compounds according to the present invention exhibit strong herbicidal activities and thus they are useful as active ingredients of agricultural chemicals.
摘要翻译： PCT No.PCT / JP94 / 02152 Sec。 371日期：1996年6月20日 102（e）1996年6月20日PCT 1994年12月20日PCT PCT。 WO95 / 18113 PCT出版物日期：1995年7月6日本发明提供由以下通式（I）表示的1,3-恶嗪-4-酮衍生物：其中R1表示可被取代的苯基; R2表示氢原子或低级烷基; R3表示氢原子，低级烷基，芳烷基或可被取代的苯基; R4和R5各自独立地表示低级烷基; W表示氧原子或式-N（R6） - 表示的基团，其中R6表示氢原子，低级烷基，低级烯基或低级炔基。还提供含有用于制备它们的衍生物和中间体的除草组合物。根据本发明的化合物表现出强烈的除草活性，因此它们可用作农药的活性成分。

4. 发明授权

US5436224A 1,3-oxazin-4-one derivatives, herbicides containing the same, and novel intermediates for preparing the same 失效
标题翻译： 1,3-恶嗪-4-酮衍生物，含有它们的除草剂及其制备新颖的中间体
公开(公告)号：US5436224A
公开(公告)日：1995-07-25
申请号：US122563
申请日：1993-09-30
申请人： Takeshi Hamatani , Hirokazu Hasebe , Keiichi Hayashizaki , Yoshihiro Usui , Chiharu Yasumoto , Atsushi Go , Mitsuru Hikido , Kumiko Tamura , Kazuo Jikihara
发明人： Takeshi Hamatani , Hirokazu Hasebe , Keiichi Hayashizaki , Yoshihiro Usui , Chiharu Yasumoto , Atsushi Go , Mitsuru Hikido , Kumiko Tamura , Kazuo Jikihara
IPC分类号： C07D265/06 , A01N43/86 , C07C251/04 , C07D265/10 , C07D319/06
CPC分类号： A01N43/86 , C07C251/04 , C07D265/06 , C07D265/10 , C07D319/06
摘要： 1,3-Oxazin-4-one derivatives represented by general formula (I) ##STR1## wherein R.sup.1 is a lower alkyl group, a lower alkenyl group, an aryl group which may be substituted, or an aralkyl group which may be substituted;R.sup.2 is a hydrogen atom or a lower alkyl group;R.sup.3 is a lower alkyl group, an aryl group which may be substituted, or an aralkyl group which may be substituted; andR.sup.4 and R.sup.5, independently, each is a lower alkyl group, or R.sup.4 and R.sup.5, taken together with the carbon atom to which they are bonded, combine to form a 3- to 8-membered carbocyclic group which may have a branch of a lower alkyl group. These compounds have broad herbicidal spectra and potent herbicidal activities and in addition high safety to useful crops, so that they are useful as herbicides.
摘要翻译： PCT No.PCT / JP93 / 00105 Sec。 371日期：1993年9月30日 102（e）1993年9月30日PCT PCT 1993年1月28日PCT公布。出版物WO93 / 15064 日本8月5日，1993.1通式（I）表示的1,3-恶嗪-4-酮衍生物其中R 1为低级烷基，低级烯基，可被取代的芳基，或可被取代的芳烷基; R2是氢原子或低级烷基; R3是低级烷基，可被取代的芳基或可被取代的芳烷基; 并且R 4和R 5独立地是低级烷基，或者R 4和R 5与它们所键合的碳原子一起结合形成3-8元碳环基，其可以具有低级烷基。这些化合物具有广泛的除草光谱和有效的除草活性，另外对有用作物的安全性高，因此它们可用作除草剂。

5. 发明授权

US08569294B2 2-(cyclic amino)-pyrimidone derivatives 失效
标题翻译： 2-（环状氨基） - 嘧啶酮衍生物
公开(公告)号：US08569294B2
公开(公告)日：2013-10-29
申请号：US12282396
申请日：2007-03-14
申请人： Kenji Fukunaga , Toshiyuki Kohara , Kazutoshi Watanabe , Yoshihiro Usui , Fumiaki Uehara , Satoshi Yokoshima , Daiki Sakai , Shin-ichi Kusaka , Kazuki Nakayama
发明人： Kenji Fukunaga , Toshiyuki Kohara , Kazutoshi Watanabe , Yoshihiro Usui , Fumiaki Uehara , Satoshi Yokoshima , Daiki Sakai , Shin-ichi Kusaka , Kazuki Nakayama
IPC分类号： A61K31/535
CPC分类号： C07D413/14 , C07D401/04 , C07D401/14 , C07D403/14 , C07D409/14 , C07D453/06 , C07D493/04
摘要： A compound represented by the formula (I), an optically active isomer thereof, or a pharmaceutical acceptable salt thereof: wherein R2 represents a hydrogen or the like; R3 represents methyl group or the like; R20 represents a halogen atom or the like; q represents an integer of 0 to 3; Z represent nitrogen atom, CH, or the like; R4 represents hydrogen or the like; R5 represents hydrogen or the like; R6 represents a substituted alkyloxy and the like; p represents an integer of 0 to 3; X represents bond, CH2, oxygen atom, NH, or the like; any one or more of R5 and R6, R5 and R4, R6 and R4, X and R5, X and R4, X and R6, and R6 and R6 may combine to each other to form a ring, which is used for preventive and/or therapeutic treatment of a disease caused by tau protein kinase 1 hyperactivity such as a neurodegenerative diseases (e.g. Alzheimer disease).
摘要翻译：由式（I）表示的化合物或其光学活性异构体或其药学上可接受的盐：其中R2表示氢等; R3表示甲基等; R 20表示卤素原子等; q表示0〜3的整数， Z表示氮原子，CH等; R4表示氢等; R5表示氢等; R6表示取代的烷氧基等; p表示0〜3的整数， X表示键，CH2，氧原子，NH等; R 5和R 6，R 5和R 4，R 6和R 4，X和R 5，X和R 4，X和R 6以及R 6和R 6中的任何一个或多个可以彼此结合形成环，其用于预防和/ 或治疗由tau蛋白激酶1多动症如神经变性疾病（例如阿尔茨海默病）引起的疾病。

6. 发明授权

US5696054A Herbicidal 1,3-oxazin-4-one derivatives and intermediates thereto 失效
标题翻译：除草剂1,3-恶嗪-4-酮衍生物及其中间体
公开(公告)号：US5696054A
公开(公告)日：1997-12-09
申请号：US403433
申请日：1995-03-14
申请人： Atsushi Go , Rika Higurashi , Miki Komine , Yoshimi Tsutsumi , Yoshihiro Usui
发明人： Atsushi Go , Rika Higurashi , Miki Komine , Yoshimi Tsutsumi , Yoshihiro Usui
IPC分类号： A01N43/86 , C07D265/06 , C07D319/06 , A01N43/72 , C07D413/02
CPC分类号： C07D319/06 , A01N43/86 , C07D265/06
摘要： Novel 1,3-oxazin-4-one derivatives of the formula ##STR1## wherein R.sup.1 to R.sup.5 are hydrocarbyl radicals which are optionally substituted, and herbicidal compositions comprising the same as active ingredients and their use in controlling the growth of weeds. The compounds can be produced by reacting substituted 1,3-dioxin-4-one derivatives and N-methylene-alkylamine.
摘要翻译：式（I）的新的1,3-恶嗪-4-酮衍生物，其中R 1至R 5为任选取代的烃基，以及包含与活性成分相同的除草组合物及其在控制杂草生长中的用途。化合物可以通过使取代的1,3-二恶英-4-酮衍生物和N-亚甲基 - 烷基胺反应来制备。

7. 发明授权

US4419553A Vacuum type circuit breaker 失效
标题翻译：真空式断路器
公开(公告)号：US4419553A
公开(公告)日：1983-12-06
申请号：US336433
申请日：1981-12-31
申请人： Masayuki Ohshita , Toshiaki Horiuchi , Takashi Yamanaka , Yoshihiro Usui
发明人： Masayuki Ohshita , Toshiaki Horiuchi , Takashi Yamanaka , Yoshihiro Usui
IPC分类号： H01H33/66 , H01H33/666 , H01H33/00
CPC分类号： H01H33/666 , H01H2001/5827 , H01H2033/6667 , H01H33/668
摘要： A vacuum type circuit breaker which has an operating lever (31) connected at one end thereof to the movable electrode (102) of a vacuum switch tube (1) and at the other end to a closing spring (55) through an energy storage link mechanism (54). The operating lever (31) functions to drive the movable electrode (102). The energy storage link mechanism (54) is provided with an energy storage crank (52) pivotally supported on a shaft (2051). The force which the energy storage link mechanism (54) applies to the operating lever (31) is set such that it is less than a force on the operating lever (31) which is produced by the difference between the internal pressure of the vacuum switch tube (1) and atmospheric pressure. This arrangement makes it possible, upon occurrence of vacuum loss, to detect the vacuum shortage, whereupon the closing of the switch is prevented to thereby avoid an accident due to vacuum degradation.
摘要翻译：一种真空式断路器，其具有在其一端连接到真空开关管（1）的可动电极（102）的操作杆（31），另一端通过能量存储连杆机构（54）。操作杆（31）用于驱动可动电极（102）。能量存储连杆机构（54）设置有枢转地支撑在轴（2051）上的储能曲柄（52）。能量存储连杆机构54施加到操作杆31的力被设定为小于由真空开关的内部压力之间的差异产生的操作杆（31）上的力管（1）和大气压力。这种布置使得在发生真空损失时可以检测真空不足，从而防止开关的闭合，从而避免由于真空劣化而引起的事故。

8. 发明授权

US07067668B2 4-quinolinol derivatives and fungicides containing the same as an active ingredient used for agriculture and horticulture 失效
标题翻译：含有与用于农业和园艺的活性成分相同的4-羟基喹啉衍生物和杀真菌剂
公开(公告)号：US07067668B2
公开(公告)日：2006-06-27
申请号：US10715846
申请日：2003-11-19
申请人： Kazumi Yamamoto , Takeshi Teraoka , Michiaki Iwata , Keiichi Imamura , Hiroshi Kurihara , Norio Sasaki , Yoshihiro Usui , Nobumitsu Sawai
发明人： Kazumi Yamamoto , Takeshi Teraoka , Michiaki Iwata , Keiichi Imamura , Hiroshi Kurihara , Norio Sasaki , Yoshihiro Usui , Nobumitsu Sawai
IPC分类号： C07D215/16 , C07D221/22
CPC分类号： C07D215/233 , A01N43/42
摘要： A new agricultural and horticultural fungicide having an excellent control effect is provided.4-Quinolinol derivatives represented by the following formula: or agriculturally and horticulturally acceptable acid addition salts thereof.
摘要翻译：提供了一种具有良好控制效果的新型农业和园艺杀真菌剂。由下式表示的4-喹啉醇衍生物：或其农业上和园艺上可接受的酸加成盐。

9. 发明授权

US06784215B2 Production process of non-flying plastic mircoballoons 有权
标题翻译：非飞行塑料微气球的生产工艺
公开(公告)号：US06784215B2
公开(公告)日：2004-08-31
申请号：US09988145
申请日：2001-11-19
申请人： Yoshihiro Shigemori , Osamu Saito , Yoshihiro Usui
发明人： Yoshihiro Shigemori , Osamu Saito , Yoshihiro Usui
IPC分类号： C08J916
CPC分类号： B01F17/0057 , B01F17/0021 , B01F17/0028 , B01F17/0064 , C08J9/22
摘要： Non-flying plastic microballoons are produced by bringing unexpanded, expandable plastic microballoons, which have been heated to a temperature lower than an expansion starting temperature thereof, and a mixture of a wetting agent and gas, the mixture having been heated to a temperature at least equal to the expansion starting temperature of the expandable plastic microballoons, into contact with each other to cause expansion of the expandable plastic balloons, and then cooling the resulting expanded plastic balloons.
摘要翻译：通过将未膨胀的可膨胀塑料微球加热到低于其膨胀起始温度的温度和润湿剂和气体的混合物来制造非飞行塑料微球，该混合物已被加热到至少的温度等于可膨胀塑料微球的膨胀起始温度彼此接触以引起可膨胀塑料球的膨胀，然后冷却所形成的膨胀塑料球。

10. 发明授权

US5753156A Process for producing non-scattering hollow plastic balloons 失效
标题翻译：生产非散射中空塑料气球的方法
公开(公告)号：US5753156A
公开(公告)日：1998-05-19
申请号：US675799
申请日：1996-07-05
申请人： Yoshihiro Shigemori , Osamu Saito , Yoshihiro Usui
发明人： Yoshihiro Shigemori , Osamu Saito , Yoshihiro Usui
IPC分类号： B01J13/02 , C08J9/22
CPC分类号： B01J13/02
摘要： A process for producing non-scattering hollow plastic balloons which comprises: (a) heating a mixture (A) of non-foamed plastic balloons and a first wetting agent, which is a plasticizer, to a temperature from 40.degree. C. to a temperature which is 40.degree. C. below an exit temperature of a heat exchanger, (b) contacting the mixture (A) with a second wetting agent being heated to a temperature equal to or above the foaming starting temperature of the non-foamed plastic balloons, wherein a ratio of the mixture (A) to the second wetting agent (B) is 1:0.5 to 1:1.5, the contacting being within 1 minute after heating the mixture (A) by the heat exchanger to a temperature ranging from 20.degree. to 50.degree. C. below the foaming starting temperature of the non-foamed plastic balloons, (c) foaming the non-foamed plastic balloons, and (d) cooling the resultant mixture from step (c) containing the foamed plastic balloons. Non-scattering foamed plastic balloons can thus be obtained simultaneously with the foaming. The present process needs a smaller amount of a plasticizer than the conventional process of wetting foamed plastic balloons with a plasticizer.
摘要翻译：一种制造非散射中空塑料球的方法，包括：（a）将非发泡塑料球的混合物（A）和作为增塑剂的第一润湿剂加热至40℃至其在热交换器的出口温度以下为40℃，（b）使混合物（A）与加热至等于或高于非泡沫塑料气囊的起泡温度的温度的第二润湿剂接触，其中混合物（A）与第二润湿剂（B）的比例为1:0.5至1:1.5，接触在通过热交换器将混合物（A）加热至20℃之后的1分钟内至低于非发泡塑料球泡的发泡起始温度至50℃，（c）使非发泡塑料球泡沫发泡，和（d）从含有发泡塑料球的步骤（c）中冷却得到的混合物。因此，可以与发泡同时获得非散射的泡沫塑料气囊。与使用增塑剂润湿发泡塑料球的常规方法相比，本方法需要更少量的增塑剂。

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