专利快速检索-快速检索全球专利，免费商用专利数据库-IPRDB

1. 依法登记的发明

USH888H Organophosphorus ester compounds of cyanohydrins as insecticides and nematicides 失效
标题翻译：作为杀虫剂和杀线虫剂的氰醇的有机磷酯化合物
公开(公告)号：USH888H
公开(公告)日：1991-02-05
申请号：US324225
申请日：1989-03-15
申请人： David T. Chou , Gail S. Powell , Philip R. Timmons
发明人： David T. Chou , Gail S. Powell , Philip R. Timmons
IPC分类号： A01N57/12 , C07F9/165
CPC分类号： A01N57/12 , C07F9/1651
摘要： Organophosphorus ester compounds of cyanohydrins of formula (I) ##STR1## wherein R is a hydrogen atom or a methyl group, are useful as insecticides, nematicides or as both. The processes for their preparation, their compositions, and their methods of use are also described.

2. 发明授权

US5223525A Pesticidal 1-arylimidazoles 失效
标题翻译：杀虫剂1-芳基咪唑
公开(公告)号：US5223525A
公开(公告)日：1993-06-29
申请号：US606518
申请日：1990-10-31
申请人： Tai-Teh Wu , David N. Sinodis , Philip R. Timmons , Gail S. Powell , David T. Chou , Peter W. Newsome , Lee S. Hall
发明人： Tai-Teh Wu , David N. Sinodis , Philip R. Timmons , Gail S. Powell , David T. Chou , Peter W. Newsome , Lee S. Hall
IPC分类号： C07D233/68 , A01N43/50 , A01N47/02 , A01P5/00 , A01P7/02 , A01P7/04 , A61K31/415 , C07D233/64 , C07D233/66 , C07D233/70 , C07D233/84 , C07D233/86 , C07D233/88 , C07D233/90 , C07D233/92
CPC分类号： C07D233/84 , A01N43/50 , A01N47/02 , C07D233/86 , C07D233/88
摘要： The invention describes novel 1-arylimidazoles of formula (I) ##STR1## wherein typically preferred substituents are: X is S(O).sub.n R.sub.1, in which R.sub.1 is an alkyl group, preferably a methyl group, which is fully substituted by halogen atoms, and n is 0, 1 and 2;Y is hydrogen, halogen, alkyl, alkoxy, alkoxyalkylideneimino, alkylsulfenyl, alkylsulfinyl or alkylsulfonyl;Z is hydrogen, halogen, alkyl, preferably methyl; andR.sub.2, R.sub.3, R.sub.4, R.sub.5 and R.sub.6 are individually hydrogen, halogen or an unsubstituted or halo-substituted alkyl, alkoxy, alkylsulfenyl, alkylsulfinyl or alkylsulfonyl.The invention further describes intermediates and processes to make the compounds, compositions of the compounds, and methods of use of the compounds for the control of arthropods (especially mites, aphids or insects), nematodes, helminths, or protozoa.
摘要翻译：本发明描述了式（I）的新型1-芳基咪唑，其中通常优选的取代基是：X是S（O）n R 1，其中R 1是烷基，优选甲基，其被完全被卤素原子，n为0,1和2; Y是氢，卤素，烷基，烷氧基，烷氧基亚烷基亚氨基，烷基亚磺酰基，烷基亚磺酰基或烷基磺酰基; Z是氢，卤素，烷基，优选甲基; 并且R 2，R 3，R 4，R 5和R 6分别为氢，卤素或未取代或卤素取代的烷基，烷氧基，烷基亚磺酰基，烷基亚磺酰基或烷基磺酰基。本发明进一步描述了制备化合物，化合物组合物的中间体和方法，以及化合物用于控制节肢动物（特别是螨虫，蚜虫或昆虫），线虫，蠕虫或原生动物的方法。

3. 发明授权

US5306694A Pesticidal 1-(2-pyridyl)-pyrazole 失效
标题翻译：杀虫剂1-（2-吡啶基） - 吡唑
公开(公告)号：US5306694A
公开(公告)日：1994-04-26
申请号：US79221
申请日：1993-06-17
申请人： Jennifer L. Phillips , Philip R. Timmons , Gail S. Powell , Michael T. Pilato , David T. Chou , Jamin Huang
发明人： Jennifer L. Phillips , Philip R. Timmons , Gail S. Powell , Michael T. Pilato , David T. Chou , Jamin Huang
IPC分类号： A01N43/56 , A01N43/40 , A01P5/00 , A01P7/02 , A01P7/04 , C07D213/04 , C07D213/72 , C07D231/14 , C07D401/04 , C07D401/00
CPC分类号： C07D401/04
摘要： The invention describes novel 1-(2-pyridyl)pyrazoles of formula (I) ##STR1## wherein typically preferred substituents are: X is S(O).sub.n R.sub.1, in which R.sub.1 is an alkyl group, preferably a methyl group, which is fully substituted by halogen atoms, and n is 0, 1 and 2;Y is hydrogen, halogen, cyano, alkylsulfenyl, alkylsulfinyl, alkylsulfonyl, alkoxy, amino, alkylamino, dialkylamino, trialkylammonium salt, cyanoalkylamino, alkoxyalkylamino, alkoxycarbonylamino, alkylcarbonylamino, haloalkylcarbonylamino, alkylaminocarbonylamino, dialkylaminocarbonylamino or alkoxyalkylideneimino, wherein the alkyl and alkoxy moieties are a linear or branched chain, containing one to four carbon atoms, and the halo-substitution consists of one or more halogen atoms, which are the same or different, up to full substitution of the alkyl moiety;Z is cyano; andR.sub.2, R.sub.3, R.sub.4, and R.sub.5 are individually hydrogen, halogen or an unsubstituted or halo-substituted alkyl or alkoxy, cyano or nitro; with the proviso that at least one of R.sub.2 to R.sub.5 is other than hydrogen.The invention further describes intermediates and processes to make the compounds, compositions of the compounds, and methods of use of the compounds for the control of arthropods (mites, aphids or insects), nematodes, helminths, or protozoa.
摘要翻译：本发明描述了式（I）的新颖的1-（2-吡啶基）吡唑其中通常优选的取代基是：X是S（O）n R 1，其中R 1是烷基，优选甲基，其完全被卤素原子取代，n为0,1和2; Y是氢，卤素，氰基，烷基亚磺酰基，烷基亚磺酰基，烷基磺酰基，烷氧基，氨基，烷基氨基，二烷基氨基，三烷基铵盐，氰基烷基氨基，烷氧基烷基氨基，烷氧基羰基氨基，烷基羰基氨基，卤代烷基羰基氨基，烷基氨基羰基氨基，二烷基氨基羰基氨基或烷氧基亚烷基亚氨基亚氨基，其中烷基和烷氧基部分是直链或支链，并且卤素取代由一个或多个相同或不同的卤素原子组成，直至烷基部分的完全取代; Z是氰基; 且R 2，R 3，R 4和R 5分别为氢，卤素或未取代或卤素取代的烷基或烷氧基，氰基或硝基; 条件是R 2至R 5中的至少一个不是氢。本发明进一步描述了制备化合物，化合物组合物的中间体和方法以及化合物用于控制节肢动物（螨虫，蚜虫或昆虫），线虫，蠕虫或原生动物的方法。

4. 发明授权

US5079370A 1-arylpyrazoles 失效
标题翻译： 1-芳基吡唑
公开(公告)号：US5079370A
公开(公告)日：1992-01-07
申请号：US681886
申请日：1991-04-08
申请人： Themistocles D. J. D'Silva , Gail S. Powell , Philip R. Timmons , Richard G. Pennicard
发明人： Themistocles D. J. D'Silva , Gail S. Powell , Philip R. Timmons , Richard G. Pennicard
IPC分类号： C07D231/28
CPC分类号： C07D231/28
摘要： The invention describes novel 3-cyano-4-sulfenylated-5-alkoxy-1-arylpyrazoles of general formula(I) ##STR1## wherein typically preferred substituents are: R is C.sub.1 to C.sub.4 alkyl fully substituted by halogen;R.sub.1 is C.sub.1 to C.sub.4 alkyl, C.sub.3 to C.sub.6 alkenyl and alkynyl or aralkyl (each of which may be optionally substituted), dialkylaminocarbonyl or a group --P(.dbd.X)(Oalkyl)(Salkyl) wherein X is oxygen or sulfur;R.sub.2, R.sub.3, R.sub.5 and R.sub.6 are each hydrogen or halogen;R.sub.4 is CF.sub.3, OCF.sub.3, SCF.sub.3, SOCF.sub.3, SO.sub.2 CF.sub.3, OCHF.sub.2, halogen or alkyl; and n is 0, 1 or 2.The invention further relates to intermediates and processes to make the compounds and to compositions thereof and to methods of control of arthopod (especially insect) nematode, helminth, and protozoan pests.
摘要翻译：本发明描述了通式（I）的新的3-氰基-4-亚磺酰基-5-烷氧基-1-芳基吡唑，其中通常优选的取代基是：R是被卤素完全取代的C1-C4烷基; R 1为C 1至C 4烷基，C 3至C 6烯基和炔基或芳烷基（其各自可任选被取代），二烷基氨基羰基或基团-P（= X）（O烷基）（S烷基），其中X为氧或硫; R2，R3，R5和R6各自为氢或卤素; R4是CF3，OCF3，SCF3，SOCF3，SO2CF3，OCHF2，卤素或烷基; 本发明进一步涉及制备化合物及其组合物的中间体和方法以及控制蒿草（尤其是昆虫）线虫，蠕虫和原生动物害虫的方法。

5. 发明授权

US4918085A Pesticidal 3-cyano-5-alkoxy-1-arylpyrazoles, compositions and use 失效
标题翻译：杀虫剂3-氰基-5-烷氧基-1-芳基吡唑，组合物和用途
公开(公告)号：US4918085A
公开(公告)日：1990-04-17
申请号：US317722
申请日：1989-03-02
申请人： Themistocles D. J. D'Silva , Gail S. Powell , Philip R. Timmons , Richard G. Pennicard
发明人： Themistocles D. J. D'Silva , Gail S. Powell , Philip R. Timmons , Richard G. Pennicard
IPC分类号： A01N43/56 , A01N57/18 , A01P5/00 , A01P7/00 , A61K31/415 , A61K31/675 , C07D231/28 , C07F9/6503
CPC分类号： C07F9/65035 , C07D231/28
摘要： The invention describes novel 3-cyano-4-sulfenylated-5-alkoxy-1-arylpyrazoles of general formula (I) ##STR1## wherein typically preferred substituents are: R is C.sub.1 to C.sub.4 alkyl fully substituted by halogen;R.sub.1 is C.sub.1 to C.sub.4 alkyl, C.sub.3 to C.sub.6 alkenyl and alkynyl or aralkyl (each of which may be optionally substituted), dialkylaminocarbonyl or a group --P(=X)(Oalkyl)(Salkyl) wherein X is oxygen or sulfur;R.sub.2, R.sub.3, R.sub.5 and R.sub.6 are each hydrogen or halogen;R.sub.4 is CF.sub.3, OCF.sub.3, SCF.sub.3, SOCF.sub.3, SO.sub.2 CF.sub.3, OCHF.sub.2, halogen or alkyl; and n is 0, 1 or 2.The invention further relates to intermediates and processes to make the compounds and to compositions thereof and to methods of control of arthopod (especially insect) nematode, helminth, and protozoan pests.

6. 发明授权

US06492357B1 Compositions and methods for controlling insects which damage rice and other crops 失效
标题翻译：用于防治大米和其他作物损害昆虫的组成和方法
公开(公告)号：US06492357B1
公开(公告)日：2002-12-10
申请号：US09660777
申请日：2000-09-13
申请人： Norihiko Nakakura , Philip R. Timmons
发明人： Norihiko Nakakura , Philip R. Timmons
IPC分类号： A61K31535
CPC分类号： A01N47/38 , A01N43/56 , A01N2300/00
摘要： Compositions and methods for controlling insect populations, in particular, insects which attack rice crops, are disclosed. The compositions include one or more compounds from the Formula 1A and one or more compounds from the formulas 1B-G described in the specification, and optionally but preferably include a suitable carrier.
摘要翻译：公开了用于防治昆虫种群的组合物和方法，尤其是攻击水稻作物的昆虫。组合物包括一种或多种式1A化合物和一种或多种说明书中所述的式1B-G的化合物，并且任选但优选包括合适的载体。

7. 发明授权

US5187185A Pesticidal 1-arylpyrroles 失效
标题翻译：杀虫1-芳基吡咯
公开(公告)号：US5187185A
公开(公告)日：1993-02-16
申请号：US533470
申请日：1990-06-05
申请人： Russell J. Outcalt , Philip R. Timmons , Susan M. Cramp , Patricia L. Kwiatkowski , Anibal Lopes , Paul A. Cain , David N. Sinodis , Lee S. Hall , Jean-Pierre A. Vors
发明人： Russell J. Outcalt , Philip R. Timmons , Susan M. Cramp , Patricia L. Kwiatkowski , Anibal Lopes , Paul A. Cain , David N. Sinodis , Lee S. Hall , Jean-Pierre A. Vors
IPC分类号： A01N43/36 , A01N47/02 , A01P7/02 , C07C255/30 , C07C255/33 , C07D207/09 , C07D207/34 , C07D207/36 , C07D211/34 , C07D295/145
CPC分类号： C07D295/145 , A01N43/36 , A01N47/02 , C07C255/30 , C07D207/34 , C07D207/36
摘要： Substituted-1-arylpyrrole compounds of general formula (I) below, are useful as pesticides, in particular for the control of insects, arachnids, and nematodes. Processes to make the compounds and intermediates used for their preparation are described. Additionally, compositions containing the compounds and methods of use therefore are provided. Preferred compounds are the compounds of general formula (I) ##STR1## wherein typically preferred substituents are: X is halogen or a group R.sup.5 S(O).sub.n, in which n is 0, 1, or 2 and R.sup.5 is CH.sub.3, CF.sub.3, CCl.sub.3, CF.sub.2 Cl, CFCl.sub.2, CF.sub.2 Br, CHF.sub.2, CHCl.sub.2 or CHClF;R.sup.1 is H, F, Cl, Br, OCH.sub.3, SCH.sub.3, or CH.sub.3 optionally substituted;R.sup.2 is CN;R.sup.3 is H, F, Cl, Br, OCH.sub.3, or CH.sub.3 optionally substituted;Y is CF.sub.3, CF.sub.3 O, H, F, Cl or Br;X.sup.1 and X.sup.4 are individually H, F, Cl, Br, CH.sub.3, OCH.sub.3 or SCH.sub.3 ; andX.sup.2 and X.sup.3 are each H.
摘要翻译：以下通式（I）的取代的1-芳基吡咯化合物可用作农药，特别是用于防治昆虫，蜘蛛和线虫。描述了制备用于制备化合物和中间体的方法。另外，提供含有这些化合物的组合物和使用方法。优选的化合物是通式（I）的化合物其中通常优选的取代基是：X是卤素或基团R 5 S（O）n，其中n是0,1或2，R 5是CH 3， CF 3，CCl 3，CF 2 Cl，CFCl 2，CF 2 Br，CHF 2，CHCl 2或CHClF; R1是任选取代的H，F，Cl，Br，OCH 3，SCH 3或CH 3; R2为CN; R3是任选取代的H，F，Cl，Br，OCH 3或CH 3; Y是CF 3，CF 3 O，H，F，Cl或Br; X1和X4分别为H，F，Cl，Br，CH3，OCH3或SCH3; X2和X3各自为H.

8. 发明授权

US5506260A Pesticidal 1-arylpyrrole compositions and method of use thereas 失效
标题翻译：杀虫剂1-芳基吡咯组合物及其使用方法
公开(公告)号：US5506260A
公开(公告)日：1996-04-09
申请号：US16102
申请日：1993-02-10
申请人： Russell J. Outcalt , Philip R. Timmons , Susan M. Cramp , Patricia L. Kwiatkowski , Anibal Lopes , Paul A. Cain , David N. Sinodis , Lee S. Hall , Jean-Pierre A. Vors
发明人： Russell J. Outcalt , Philip R. Timmons , Susan M. Cramp , Patricia L. Kwiatkowski , Anibal Lopes , Paul A. Cain , David N. Sinodis , Lee S. Hall , Jean-Pierre A. Vors
IPC分类号： A01N43/36 , A01N47/02 , A01P7/02 , C07C255/30 , C07C255/33 , C07D207/09 , C07D207/34 , C07D207/36 , C07D211/34 , C07D295/145
CPC分类号： C07D295/145 , A01N43/36 , A01N47/02 , C07C255/30 , C07D207/34 , C07D207/36
摘要： Substituted-1-arylpyrrole compounds of general formula (I) below, are useful as pesticides, in particular for the control of insects, arachnids, and nematodes. Processes to make the compounds and intermediates used for their preparation are described. Additionally, compositions containing the compounds and methods of use therefore are provided. Preferred compounds are the compounds of general formula (I) ##STR1## wherein typically preferred substituents are: X is halogen or a group R.sup.5 S(O).sub.n, in which n is 0, 1, or 2 and R.sup.5 is CH.sub.3, CF.sub.3, CCl.sub.3, CF.sub.2 Cl, CFCl.sub.2, CF.sub.2 Br, CHF.sub.2, CHCl.sub.2 or CHClF;R.sup.1 is H, F, Cl, Br, OCH.sub.3, SCH.sub.3, or CH.sub.3 optionally substituted;R.sup.2 is CN;R.sup.3 is H, F, Cl, Br, OCH.sub.3, or CH.sub.3 optionally substituted;Y is CF.sub.3, CF.sub.3 O, H, F, Cl or Br;X.sup.1 and X.sup.4 are individually H, F, Cl, Br, CH.sub.3, OCH.sub.3 or SCH.sub.3 ; andX.sup.2 and X.sup.3 are each H.
摘要翻译：以下通式（I）的取代的1-芳基吡咯化合物可用作农药，特别是用于防治昆虫，蜘蛛和线虫。描述了制备用于制备化合物和中间体的方法。另外，提供含有这些化合物的组合物和使用方法。优选的化合物是通式（I）的化合物其中通常优选的取代基是：X是卤素或基团R 5 S（O）n，其中n是0,1或2，R 5是CH 3， CF 3，CCl 3，CF 2 Cl，CFCl 2，CF 2 Br，CHF 2，CHCl 2或CHClF; R1是任选取代的H，F，Cl，Br，OCH 3，SCH 3或CH 3; R2为CN; R3是任选取代的H，F，Cl，Br，OCH 3或CH 3; Y是CF 3，CF 3 O，H，F，Cl或Br; X1和X4分别为H，F，Cl，Br，CH3，OCH3或SCH3; X2和X3各自为H.

9. 发明授权

US5236938A Pesticidal 1-aryl-5-(substituted alkylideneimino)pyrazoles 失效
标题翻译：杀虫剂1-芳基-5-（取代的亚烷基亚氨基）吡唑
公开(公告)号：US5236938A
公开(公告)日：1993-08-17
申请号：US693580
申请日：1991-04-30
申请人： Jamin Huang , Hafez M. Ayad , Philip R. Timmons
发明人： Jamin Huang , Hafez M. Ayad , Philip R. Timmons
IPC分类号： A01N43/56 , A01P7/02 , A01P7/04 , C07D231/44 , C07D401/04 , C07D401/12 , C07D401/14
CPC分类号： C07D401/04 , C07D231/44 , C07D401/12 , C07D401/14
摘要： The invention describes novel 1-aryl-5-(substituted alkylideneimino)pyrazoles of formula (I) ##STR1## wherein typically preferred substituents are: R.sup.1 is cyano, nitro, or halogen;R.sup.2 is R.sup.9 S(O).sub.n in which n is 0, 1 or 2 and R.sup.9 is alkyl, preferably methyl which is substituted by halogen atoms which are the same or different up to full substitution of the alkyl moiety;R.sup.3 is hydrogen or alkyl;R.sup.4 is phenyl or heteroaryl, optionally substituted by one or more hydroxy, halogen, alkoxy, alkylthio, cyano or alkyl or combinations thereof;R.sup.5 is hydrogen, alkyl or halogen;R.sup.6 and R.sup.8 are hydrogen;R.sup.7 is halogen, alkyl, haloalkyl or haloalkoxy; andX is a nitrogen atom or CR.sup.14 in which R.sup.14 is hydrogen, halogen, cyano, alkyl, alkylthio or alkoxy.The invention further describes processes to make the compounds, compositions of the compounds, and methods of use of the compounds for the control of arthropods (mites, aphids or insects), nematodes, helminths, or protozoa.
摘要翻译：本发明描述了式（I）的新型1-芳基-5-（取代的亚烷基亚氨基）吡唑其中通常优选的取代基是：R 1是氰基，硝基或卤素; R2是R9S（O）n，其中n是0,1或2，R9是烷基，优选被烷基部分完全取代的相同或不同的卤素原子取代的甲基; R3是氢或烷基; R4是任选被一个或多个羟基，卤素，烷氧基，烷硫基，氰基或烷基或其组合取代的苯基或杂芳基; R5是氢，烷基或卤素; R6和R8是氢; R7是卤素，烷基，卤代烷基或卤代烷氧基; X为氮原子或CR 14，其中R 14为氢，卤素，氰基，烷基，烷硫基或烷氧基。本发明还描述了使化合物，化合物的组合物和化合物用于控制节肢动物（螨虫，蚜虫或昆虫），线虫，蠕虫或原生动物的方法。

10. 发明授权

US5360910A Pesticidal 1-aryl-5-(substituted alkylideneimino)pyrazoles 失效
标题翻译：杀虫剂1-芳基-5-（取代的亚烷基亚氨基）吡唑
公开(公告)号：US5360910A
公开(公告)日：1994-11-01
申请号：US842431
申请日：1992-03-04
申请人： Jamin Huang , Hafez M. Ayad , Philip R. Timmons
发明人： Jamin Huang , Hafez M. Ayad , Philip R. Timmons
IPC分类号： C07D231/44 , C07D401/04 , C07D401/14
CPC分类号： C07D401/04 , C07D231/44 , C07D401/14
摘要： The invention describes novel 1-aryl-5-(substituted alkylideneimino)pyrazoles of formula (I) ##STR1## wherein typically preferred substituents are: R.sup.1 is cyano, nitro, or halogen;R.sup.2 is R.sup.9 S(O).sub.n in which n is 0, 1 or 2 and R.sup.9 is alkyl, preferably methyl which is substituted by halogen atoms which are the same or different up to full substitution of the alkyl moiety;R.sup.3 is hydrogen or alkyl;R.sup.4 is phenyl or heteroaryl, optionally substituted by one or more hydroxy, halogen, alkoxy, alkylthio, cyano or alkyl or combinations thereof; preferably R.sup.4 is phenyl, which is at least substituted by 3-hydroxy or 4-hydroxy;R.sup.5 is hydrogen, alkyl or halogen;R.sup.6 and R.sup.8 are hydrogen;R.sup.7 is halogen, alkyl, haloalkyl or haloalkoxy; andX is a nitrogen atom or CR.sup.14 in which R.sup.14 is hydrogen, halogen, cyano, alkyl, alkylthio or alkoxy.The invention further describes processes to make the compounds, compositions of the compounds, and methods of use of the compounds for the control of arthropods (mites, aphids or insects), nematodes, helminths, or protozoa.
摘要翻译：本发明描述了式（I）的新型1-芳基-5-（取代的亚烷基亚氨基）吡唑其中通常优选的取代基是：R 1是氰基，硝基或卤素; R2是R9S（O）n，其中n是0,1或2，R9是烷基，优选被烷基部分完全取代的相同或不同的卤素原子取代的甲基; R3是氢或烷基; R4是任选被一个或多个羟基，卤素，烷氧基，烷硫基，氰基或烷基或其组合取代的苯基或杂芳基; 优选R4是至少被3-羟基或4-羟基取代的苯基; R5是氢，烷基或卤素; R6和R8是氢; R7是卤素，烷基，卤代烷基或卤代烷氧基; X为氮原子或CR 14，其中R 14为氢，卤素，氰基，烷基，烷硫基或烷氧基。本发明还描述了使化合物，化合物的组合物和化合物用于控制节肢动物（螨虫，蚜虫或昆虫），线虫，蠕虫或原生动物的方法。

你已经成功收藏专利！

检索式保存成功!

IPRDB

热门服务

关于我们

友情链接

联系方式