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71. 发明授权

US4312859A Sisomicin derivatives, processes for their production and their medicinal use 失效
标题翻译：西索米星衍生物，其生产方法及其药用
公开(公告)号：US4312859A
公开(公告)日：1982-01-26
申请号：US147908
申请日：1980-05-08
申请人： Uwe Petersen , Karl G. Metzger , Hans-Joachim Zeiler , Peter Stadler , Eckart Voss
发明人： Uwe Petersen , Karl G. Metzger , Hans-Joachim Zeiler , Peter Stadler , Eckart Voss
IPC分类号： A61K31/70 , A61K31/7028 , A61K31/7034 , A61K31/7036 , A61P31/04 , C07H15/236 , A61K31/71 , C07H15/22
CPC分类号： C07H15/236
摘要： The invention relates to sesomycin derivatives of Formula I, infra as well as processes for preparing said sisomycin derivatives. Also included in the invention are compositions containing said sisomycin derivatives and methods for the use of said compounds and compositions. The sisomycon derivatives are useful as antibacterial agents of broad activity and reduced side effects.
摘要翻译：本发明涉及式I的芝霉素衍生物，以及制备所述西沙星霉素衍生物的方法。本发明还包括含有所述顺式霉素衍生物的组合物和使用所述化合物和组合物的方法。 sisomycon衍生物可用作具有广泛活性和减少副作用的抗菌剂。

72. 发明授权

US4235888A Pseudotrissaccharides, a process for their production and their use as medicaments 失效
标题翻译：伪三糖，其生产过程及其作为药物的用途
公开(公告)号：US4235888A
公开(公告)日：1980-11-25
申请号：US52871
申请日：1979-06-28
申请人： Peter Stadler , Karl-Georg Metzger , Eckart Voss , Uwe Petersen , Hans-Joachim Zeiler , Hans-Joachim Kabbe
发明人： Peter Stadler , Karl-Georg Metzger , Eckart Voss , Uwe Petersen , Hans-Joachim Zeiler , Hans-Joachim Kabbe
IPC分类号： A61K31/70 , A61K31/7028 , A61K31/7034 , A61K31/7036 , A61P31/04 , C07D317/72 , C07H15/236 , C07H17/08
CPC分类号： C07D317/72 , C07H15/236
摘要： Pseudotrisaccharides of the sisomycin type are provided which are effective an antibacterial agents, particularly against gram-negative microorganisms. The invention also includes methods for the manufacture of the pseudotrisaccharides, compositions containing said pseudotrisaccharides and methods for the treatment of warm-blooded animals using said compounds and compositions.
摘要翻译：提供了具有抗菌剂，特别是抗革兰氏阴性微生物的抗生素，具有抗生素的类型。本发明还包括制备假三糖的方法，含有所述假三糖的组合物和使用所述化合物和组合物治疗温血动物的方法。

73. 发明授权

US4190722A 4,6-Di-O-(aminoglycosyl)-1,3-diaminocyclitols, process for their production and their use 失效
标题翻译： 4,6-二-O-（氨基糖基）-1,3-二氨基二醇，其制备及其用途
公开(公告)号：US4190722A
公开(公告)日：1980-02-26
申请号：US913135
申请日：1978-06-06
申请人： Eckart Voss , Peter Stadler , Uwe Petersen , Hans-Joachim Kabbe , Karl G. Metzger
发明人： Eckart Voss , Peter Stadler , Uwe Petersen , Hans-Joachim Kabbe , Karl G. Metzger
IPC分类号： C07H15/234 , A61K31/70 , A61K31/7028 , A61K31/7034 , A61K31/7036 , A61P31/04 , C07H15/236 , A61K31/71 , C07H15/22
CPC分类号： C07H15/236
摘要： The invention includes selectively acylated or sulphenylated 4,6-O-(aminoglycosyl)-1,3-diaminocyclitols (and methods for their preparation). Also included in the invention are 1-N-acylated-derivatives, such as 1-N-formyl-sisomicin, useful because of the anti-bacterial effects (and methods for their procurement). The invention includes, furthermore, methods for the procurement of said 1-N-acylated or sulphenylated derivatives, compositions containing them and methods for their use.
摘要翻译：本发明包括选择性酰化或磺基化的4,6-O-（氨基糖基）-1,3-二氨基二醇（及其制备方法）。本发明还包括1-N-酰化衍生物，例如1-N-甲酰基西索米星，因为其具有抗菌作用（及其采购方法）。此外，本发明还包括采购所述1-N-酰化或磺化衍生物的方法，含有它们的组合物及其使用方法。

74. 发明授权

US3997533A Process for the preparation of 7-acylamino-desacetoxycephalosporanic derivatives 失效
标题翻译：制备7-酰氨基 - 去乙酸基头孢烷衍生物的方法
公开(公告)号：US3997533A
公开(公告)日：1976-12-14
申请号：US442810
申请日：1974-02-14
申请人： Hans-Joachim Kabbe , Uwe Petersen
发明人： Hans-Joachim Kabbe , Uwe Petersen
IPC分类号： A61K31/545 , B01J27/00 , C07B61/00 , C07D20060101 , C07D205/00 , C07D279/00 , C07D401/04 , C07D499/04 , C07D501/10 , C07D501/22 , C07D501/28 , C07D501/30 , C07D501/34
CPC分类号： C07D499/00
摘要： 7-Acylaminodesacetoxycephalosporanic acid derivatives are produced by heating a penicillin ester S-oxide to a temperature between 60.degree. C and 150.degree. C in the presence of a heavy metal salt.
摘要翻译：通过在重金属盐的存在下将青霉素酯S-氧化物加热至60℃至150℃的温度来制备7-酰基乙酰氧基头孢烷酸衍生物。

75. 发明申请

US20120010215A1 Treatment of bacterial diseases of the respiratory organs 审中-公开
标题翻译：治疗呼吸器官细菌性疾病
公开(公告)号：US20120010215A1
公开(公告)日：2012-01-12
申请号：US13192893
申请日：2011-07-28
申请人： Rainer Endermann , Harald Labischinski , Christoph Ladel , Uwe Petersen , Ben Newton
发明人： Rainer Endermann , Harald Labischinski , Christoph Ladel , Uwe Petersen , Ben Newton
IPC分类号： A61K31/496 , A61P11/08 , A61P11/00 , A61P31/04
CPC分类号： A61K9/0075 , A61K31/496
摘要： The invention relates to inhalable quinolonecarboxylic acid derivative compositions for local control of diseases of the respiratory organs, in particular of lung diseases.
摘要翻译：本发明涉及用于局部控制呼吸器官疾病，特别是肺部疾病的吸入性喹诺酮羧酸衍生物组合物。

76. 发明申请

US20060220908A1 Method and device for supporting the driver of a vehicle during an emergency braking 审中-公开
标题翻译：在紧急制动期间支撑车辆驾驶员的方法和装置
公开(公告)号：US20060220908A1
公开(公告)日：2006-10-05
申请号：US10566834
申请日：2004-07-28
申请人： Uwe Petersen , Volker Schmid , Thomas Unselt
发明人： Uwe Petersen , Volker Schmid , Thomas Unselt
IPC分类号： G08G1/16
CPC分类号： B60T8/3275 , B60T7/22 , B60T2201/02 , B60T2201/03
摘要： The invention relates to a method and device for supporting the driver of a vehicle during an emergency braking process in order to prevent the vehicle from colliding with an object which is located in a detection zone in front of the vehicle in the direction of travel, in particular a preceding vehicle. In the method according to the invention braking means for braking the vehicle (50) are actuated independently of the driver if a predefined emergency braking condition is met and if it is determined that the driver wishes to carry out the emergency braking process, emergency braking information to the driver of the vehicle (50) being issued when the emergency braking condition is met. According to the invention information to the driver is issued even when the emergency braking condition is not met, said information informing the driver of the vehicle (50) about the current situation in the surroundings or the traffic situation in the detection zone (54), the information to the driver being adjusted as a function of predefined information conditions being met.
摘要翻译：本发明涉及一种用于在紧急制动过程中支撑车辆驾驶员的方法和装置，以便防止车辆与位于车辆前方的检测区域中的物体沿行驶方向相撞，特别是前一车辆。在根据本发明的方法中，如果满足预定义的紧急制动条件，则独立于驾驶员致动用于制动车辆（50）的制动装置，并且如果确定驾驶员希望执行紧急制动过程，紧急制动信息在满足紧急制动条件时向车辆（50）的驾驶员发出。根据本发明，即使当不满足紧急制动条件时，也向驾驶员发出信息，所述信息通知车辆（50）的驾驶员关于周围环境中的当前情况或检测区（54）中的交通情况，作为根据预定信息条件的函数调整驱动程序的信息。

77. 发明授权

US06308959B1 Elastic sealing element in the form of bellows 有权
标题翻译：波纹管形式的弹性密封元件
公开(公告)号：US06308959B1
公开(公告)日：2001-10-30
申请号：US09254263
申请日：1999-03-01
申请人： Dirk Sokolihs , Uwe Petersen
发明人： Dirk Sokolihs , Uwe Petersen
IPC分类号： F16J1538
CPC分类号： F16J3/046 , Y10T403/315
摘要： An elastic sealing element in the form of bellows, which is used to seal the contact surface between at least two components movable in relation to one another is described, which has low-elasticity contact zones as well as a deformation zone whose elasticity is higher than that of the contact zones, wherein the said deformation zone defines a chamber for accommodating lubricants on its inner side facing the movable components. An overpressure relief means (14) is arranged at least in the area of one of the two low-elasticity contact zones (6 or 7). The overpressure relief means (14) has at least one relief opening (15) connecting the lubricant chamber (11) with the outside of the sealing element (1) and a closing element (16) covering the said relief opening. The closing element (16) is in turn made in one piece with the sealing element (1) and closes the relief opening (15) up to an overpressure limit in the lubricant chamber (11) due to the intrinsic elasticity of the material of the sealing element.
摘要翻译：描述了波纹管形式的弹性密封元件，其用于密封可相对于彼此移动的至少两个部件之间的接触表面，其具有低弹性接触区域以及弹性高于所述接触区域的所述变形区域限定用于在其面向所述可移动部件的内侧容纳润滑剂的腔室。至少在两个低弹性接触区域（6或7）之一的区域中布置有超压释放装置（14）。超压释放装置（14）具有将润滑剂室（11）与密封元件（1）的外部连接的至少一个释放开口（15）和覆盖所述浮雕开口的封闭元件（16）。关闭元件（16）又与密封元件（1）一体制成，并且由于所述材料的固有弹性而将所述释放开口（15）封闭到所述润滑剂室（11）中的超压极限密封元件。

78. 发明授权

US06271342B1 Sugar-modified cytostatics 失效
标题翻译：糖改性细胞抑制剂
公开(公告)号：US06271342B1
公开(公告)日：2001-08-07
申请号：US08930546
申请日：1997-09-25
申请人： Hans-Georg Lerchen , Karsten von dem Bruch , Uwe Petersen , Jörg Baumgarten , Norbert Piel , Horst-Peter Antonicek , Walter Weichel , Michael Sperzel , Klaus Dieter Bremm
发明人： Hans-Georg Lerchen , Karsten von dem Bruch , Uwe Petersen , Jörg Baumgarten , Norbert Piel , Horst-Peter Antonicek , Walter Weichel , Michael Sperzel , Klaus Dieter Bremm
IPC分类号： A61K3814
CPC分类号： C07D401/04 , A61K31/02 , C07D487/04 , C07H15/203 , C07K9/001 , Y02P20/55
摘要： The invention relates to cytostatics which, by modification with sugar, are tumor-specific. Suitable spacers ensure serum stability and at the same time an intracellular action.
摘要翻译：本发明涉及通过用糖改性的肿瘤特异性的细胞抑制剂。合适的间隔物确保血清稳定性，并同时进行细胞内作用。

79. 发明授权

US6004956A Enantiomerically pure 2-oxa-5,8-dizaabicyclo[4.3.0] nonanes and process for their preparation 失效
标题翻译：对映异构体纯的2-氧杂-5,8-二氮杂双环[4.3.0]壬烷和其制备方法
公开(公告)号：US6004956A
公开(公告)日：1999-12-21
申请号：US628437
申请日：1996-04-05
申请人： Thomas Schenke , Andreas Krebs , Uwe Petersen
发明人： Thomas Schenke , Andreas Krebs , Uwe Petersen
IPC分类号： C07D498/04 , A61K31/535 , C07D265/36
CPC分类号： C07D498/04
摘要： The invention relates to enantiomerically pure 2-oxa-5,8-diazabicyclo[4.3.0]nonanes and processes for their preparation.
摘要翻译：本发明涉及对映体纯的2-氧杂-5,8-二氮杂双环[4.3.0]壬烷及其制备方法。

80. 发明授权

US5703094A Quinolone- and naphthyridonecarboxylic acid derivatives 失效
标题翻译：喹诺酮和萘啶酮羧酸衍生物
公开(公告)号：US5703094A
公开(公告)日：1997-12-30
申请号：US583685
申请日：1996-01-05
申请人： Uwe Petersen , Michael Ruther , Thomas Schenke , Klaus Dieter Bremm , Rainer Endermann
发明人： Uwe Petersen , Michael Ruther , Thomas Schenke , Klaus Dieter Bremm , Rainer Endermann
IPC分类号： A61K31/47 , A61P31/04 , C07D209/44 , C07D401/04 , C07D471/04 , C07D513/04 , C07D513/14 , C07D215/233
CPC分类号： C07D401/04 , C07D209/44 , C07D471/04 , C07D513/04
摘要： The invention relates to new quinolone- and naphthyridonecarboxylic acid derivatives which are substituted in the 7-position by an unsaturated bicyclic amine radical, their salts, processes for their preparation and antibacterial compositions comprising these compounds
摘要翻译：本发明涉及在7-位被不饱和双环胺基取代的新喹诺酮和萘啶酮羧酸衍生物，其盐，其制备方法和包含这些化合物的抗菌组合物

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