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11. 发明授权

US5532367A Insecticidal pteridines and 8-deazapteridines 失效
标题翻译：杀虫蝶啶和8-取代二萜烯
公开(公告)号：US5532367A
公开(公告)日：1996-07-02
申请号：US416017
申请日：1995-03-31
申请人： Robert N. Henrie, II , Clinton J. Peake , Thomas G. Cullen , Albert C. Lew , Ian R. Silverman
发明人： Robert N. Henrie, II , Clinton J. Peake , Thomas G. Cullen , Albert C. Lew , Ian R. Silverman
IPC分类号： A01N43/90 , C07D471/04 , C07D475/08 , C07D487/04
CPC分类号： C07D471/04 , A01N43/90 , C07D475/08
摘要： This invention relates to pteridine and 8-deazapteridine compounds which are useful for controlling insects in agricultural crops. These pteridines may be represented by the following structure: ##STR1## wherein R and R.sup.1 are amino;R.sup.2 is hydrogen or lower alkyl;Q is N or CH;R.sup.3 is --(n).sub.m --R.sup.4, andR.sup.4 is ##STR2## wherein n, m, V, W, X, Y, and Z are as defined in the specification.
摘要翻译：本发明涉及可用于防治农作物昆虫的蝶啶和8-脱氮啶啶化合物。这些蝶啶可以由以下结构表示：其中R和R 1是氨基; R2是氢或低级烷基; Q是N或CH; R3是 - （n）m-R4，R4是＆lt; IMAGE＆gt;其中n，m，V，W，X，Y和Z如说明书中所定义。

12. 发明授权

US5521190A Insecticidal pterdines and 8-deazapteridines 失效
标题翻译：杀虫蝶啶和8-去甲基吡啶
公开(公告)号：US5521190A
公开(公告)日：1996-05-28
申请号：US067897
申请日：1993-05-27
申请人： Robert N. Henrie, II , Clinton J. Peake , Thomas G. Cullen , Albert C. Lew , Ian R. Silverman
发明人： Robert N. Henrie, II , Clinton J. Peake , Thomas G. Cullen , Albert C. Lew , Ian R. Silverman
IPC分类号： A01N43/90 , C07D471/04 , C07D475/08 , A61K31/505
CPC分类号： C07D471/04 , A01N43/90 , C07D475/08
摘要： This invention relates to pteridine and 8-deazapteridine compounds and compositions containing the same which are useful for controlling insects in agricultural crops. These pteridines may be represented by the following structure: ##STR1## wherein R and R.sup.1 are independently selected from amino, lower alkylamino, di(lower alkyl)amino (e.g., --N(CH.sub.3).sub.2), or di(lower alkyl)aminomethyleneamino (e.g., --N.dbd.CHN(CH.sub.3).sub.2);R.sup.2 is hydrogen, amino, lower alkyl (e.g., --CH.sub.3, --CH(CH.sub.3).sub.2), di(lower alkyl)aminomethyleneamino, hydroxy, lower alkoxy, phenyl or substituted phenyl, haloalkylphenylalkyl (e.g., 3-trifluoromethylphenylmethyl);Q is N or CH;R.sup.3 is --(n).sub.m --R.sup.4, where m is 0 or 1; wherein, when m is 1,n is a bridging atom or moiety selected from oxygen, sulfur, sulfinyl, sulfonyl, lower alkylene (e.g., --CH.sub.2 --, or --CH.sub.2 CH.sub.2 --), lower alkenylene (e.g., --CH.dbd.CH--), lower alkynylene (e.g., --C.dbd.C--), lower haloalkenylene (e.g., --C(Cl).dbd.CH--), carbonyl, aminomethyl (e.g.,--CH.sub.2 NH--), or (substituted amino)methyl (e.g.,--CH.sub.2 N(CH.sub.3)--); andR.sup.4 is hydrogen, lower alkyl (e.g., --CH.sub.3, or --CH(CH.sub.3).sub.2), thien-2-yl, pyridin-3-yl, or ##STR2## wherein (i) V, W, X, Y, and Z are as defined herein.
摘要翻译：本发明涉及蝶啶和8-脱氮吡啶化合物及其含有该组合物的组合物，其可用于控制农作物中的昆虫。这些蝶啶可以由以下结构表示：其中R和R 1独立地选自氨基，低级烷基氨基，二（低级烷基）氨基（例如，-N（CH 3）2）或二（低级）烷基）氨基亚甲基氨基（例如，-N = CHN（CH 3）2）; R 2是氢，氨基，低级烷基（例如-CH 3，-CH（CH 3）2），二（低级烷基）氨基亚甲基氨基，羟基，低级烷氧基，苯基或取代的苯基，卤代烷基苯基烷基（例如3-三氟甲基苯基甲基）。 Q是N或CH; R3是 - （n）m-R4，其中m是0或1; 其中，当m为1时，n为选自氧，硫，亚磺酰基，磺酰基，低级亚烷基（例如-CH 2 - 或-CH 2 CH 2 - ）的桥连原子或部分，低级亚烯基（例如-CH = CH-），低级亚炔基（例如-C = C-），低级卤代亚烯基（例如-C（Cl）= CH-），羰基，氨基甲基（例如-CH 2 NH-）或（取代的氨基）甲基（例如-CH 2 N （CH 3） - ）; 和R 4是氢，低级烷基（例如，-CH 3或-CH（CH 3）2），噻吩-2-基，吡啶-3-基或其中（i）V，W，X，Y，和Z如本文所定义。

13. 发明授权

US5696259A 2,4-diamino-5-iodopyrimidines useful as pesticide intermediates 失效
标题翻译：可用作农药中间体的2,4-二氨基-5-碘嘧啶
公开(公告)号：US5696259A
公开(公告)日：1997-12-09
申请号：US681032
申请日：1996-07-22
申请人： Robert N. Henrie, II , Clinton J. Peake , Thomas G. Cullen , Walter H. Yeager , Mary E. Brown , John W. Buser
发明人： Robert N. Henrie, II , Clinton J. Peake , Thomas G. Cullen , Walter H. Yeager , Mary E. Brown , John W. Buser
IPC分类号： C07D239/48 , C07D401/04 , C07D413/04
CPC分类号： C07D239/49
摘要： This invention describes 2,4-diamino-5-iodopyrimidines II where R, R1, R2, and R3 are independently selected from hydrogen, alkyl, cycloalkyl, alkoxyalkyl, alkoxyalkoxyalkyl, and arylalkyl; or, R1 and R2, and R3 and R, each independently, when taken together with pentylene or 3-oxapentylene, form piperidine and morpholine ring systems respectively; and R4 is hydrogen or lower alkyl. These compounds are useful intermediates in the preparation of insecticides I where U is an optionally substituted alkenylene. ##STR1##
摘要翻译：本发明描述了2,4-二氨基-5-碘嘧啶II，其中R，R 1，R 2和R 3独立地选自氢，烷基，环烷基，烷氧基烷基，烷氧基烷氧基烷基和芳基烷基; 或者R 1和R 2以及R 3和R 3各自独立地与亚戊基或3-氧杂萘基一起形成哌啶和吗啉环体系; R4是氢或低级烷基。这些化合物是制备杀虫剂I的有用的中间体，其中U是任选取代的亚烯基。 II。图像II

14. 发明授权

US5622954A 5[W(substituted aryl)alkenylene and alkynylene]-2,4-diaminopyrimidines as pesticides 失效
标题翻译： 5 [W（取代的芳基）亚烯基和亚炔基] -2,4-二氨基嘧啶作为农药
公开(公告)号：US5622954A
公开(公告)日：1997-04-22
申请号：US398205
申请日：1995-03-02
申请人： Robert N. Henrie, II , Clinton J. Peake , Thomas G. Cullen , Walter H. Yeager , Mary E. Brown , John W. Buser
发明人： Robert N. Henrie, II , Clinton J. Peake , Thomas G. Cullen , Walter H. Yeager , Mary E. Brown , John W. Buser
IPC分类号： A01N43/54 , C07D239/48 , C07D239/49 , C07D401/06 , C07D401/14 , C07F7/08
CPC分类号： C07D239/49 , A01N43/54 , C07D401/06 , C07D401/14 , C07F7/0812
摘要： 5-Substituted-2,4-diaminopyrimidines, and agriculturally acceptable salts thereof, when present in insecticidally or acaricidally effective amounts, and with a suitable agricultural carrier, are useful as active ingredients in novel insecticidal and acaricidal compositions. These pyrimidines may be represented by the following formula: ##STR1## wherein Ar is ##STR2## and wherein U is an alkenylene or alkynylene moiety, and R, R.sup.1, R.sup.2, R.sup.3, R.sup.4, V, W, X, Y, Z and n are as defined herein; also disclosed and claimed are novel intermediates thereof.
摘要翻译： 5-取代的2,4-二氨基嘧啶及其农业上可接受的盐当以杀虫或杀螨有效量存在时，并且与合适的农业载体一起可用作新的杀虫和杀螨组合物中的活性成分。这些嘧啶可以由下式表示：其中Ar为“IMA”，其中U为亚烯基或亚炔基部分，R 1，R 2，R 3，R 4，V，W，X，Y Z和n如本文所定义; 还公开并要求保护的是其新颖的中间体。

15. 发明授权

US5874579A Insecticidal substituted-2.4-diaminoquinazolines related applications 失效
标题翻译：杀虫剂取代-2,4-二氨基喹唑啉
公开(公告)号：US5874579A
公开(公告)日：1999-02-23
申请号：US640610
申请日：1996-05-01
申请人： Robert N. Henrie II , Clinton J. Peake , Thomas G. Cullen , Walter H. Yeager
发明人： Robert N. Henrie II , Clinton J. Peake , Thomas G. Cullen , Walter H. Yeager
IPC分类号： A01N43/54 , A01N55/00 , C07D239/95 , C07D401/12 , C07D405/04 , C07D409/04 , A61K31/505
CPC分类号： C07D401/12 , A01N43/54 , A01N55/00 , C07D239/95 , C07D405/04 , C07D409/04
摘要： An insecticidal composition comprising, in admixture with an agriculturally acceptable carrier, an insecticidally effective amount of a 2,4-diaminoquinazoline compound of the formula: ##STR1## wherein R.sup.1, R.sup.2, R.sup.6, R.sup.7, W, X, Y, and Z are as defined herein; methods of using the same; novel 2,4-diaminoquinazolines per se; and intermediates in the preparation thereof.
摘要翻译：一种杀虫组合物，其包含与农业上可接受的载体的混合物，杀虫有效量的下式的2,4-二氨基喹唑啉化合物：其中R 1，R 2，R 6，R 7，W，X，Y和Z为如本文所定义; 使用方法; 新型2,4-二氨基喹唑啉本身; 和其制备中的中间体。

16. 发明授权

US06214845B1 Insecticidal N-(substituted arylmethyl)-4[bis(substituted phenyl or pyridyl)methyl] piperidines 失效
标题翻译：杀虫剂N-（取代的芳基甲基）-4 [双（取代的苯基或吡啶基）甲基]哌啶
公开(公告)号：US06214845B1
公开(公告)日：2001-04-10
申请号：US09388592
申请日：1999-09-02
申请人： Ian R. Silverman , Daniel H. Cohen , John W. Lyga , Steven W. Szczepanski , Syed F. Ali , Thomas G. Cullen , Robert N. Henrie, II , Clinton J. Peake
发明人： Ian R. Silverman , Daniel H. Cohen , John W. Lyga , Steven W. Szczepanski , Syed F. Ali , Thomas G. Cullen , Robert N. Henrie, II , Clinton J. Peake
IPC分类号： A01N4340
CPC分类号： C07D401/06 , A01N43/40 , A01N43/50 , A01N43/54 , A01N43/56 , A01N43/60 , A01N43/653 , A01N43/713 , A01N43/76 , A01N43/82 , A01N47/20 , A01N55/00 , C07D211/14 , C07D211/22 , C07D211/24 , C07D211/26 , C07D211/94 , C07D231/12 , C07D233/56 , C07D249/08 , C07D401/10 , C07D401/12 , C07D401/14 , C07D405/06 , C07D405/10 , C07D409/06 , C07D413/06 , C07D413/10 , C07D417/10 , C07D417/12 , C07F7/1804
摘要： Compounds of the following structure, the corresponding N-oxides and agriculturally acceptable salts, are disclosed as effective insecticides: in which U is —(CH2)n—; Q is hydroxy; R is in which V, W, Y, and Z are each hydrogen; X is a five- or six-membered heterocycle; optionally substituted with halogen, cyano, alkyl, haloalkyl, alkoxy, haloalkoxy, alkoxyalkyl, haloalkoxyalkyl, or aminocarbonyl; and the heterocycle is optionally connected to the phenyl ring through a —O—, —S—, —(CH2)p, —C(O)—, or —O—(CR3R4)q linkage; R1 and R2 are independently selected from phenyl or pyridyl substituted with haloalkyl or haloalkoxy; R3 and R4 are independently selected from hydrogen and methyl; n and p are independently 1, 2, or 3; and q is 1 or 2; with the proviso that at least one of R1 and R2 is substituted in the para position; no more than two of R3 and R4 are methyl; each aliphatic moiety contains not more than 4 carbon atoms; halogen means bromine, chlorine, or fluorine; each heterocycle contains from 1 to 4 nitrogen atoms, or 1 or 2 oxygen or sulfur atoms, or 1 or 2 nitrogen atoms and an oxygen or sulfur atom; and the corresponding N-oxides and agriculturally acceptable salts.
摘要翻译：公开了以下结构的化合物，即相应的N-氧化物和农业上可接受的盐作为有效的杀虫剂：其中U是 - （CH 2）n - ; Q是羟基; R 1是其中V，W，Y和Z各自是氢; X是五元或六元杂环; 任选被卤素，氰基，烷基，卤代烷基，烷氧基，卤代烷氧基，烷氧基烷基，卤代烷氧基烷基或氨基羰基取代; 并且杂环任选地通过-O - ， - S - ， - （CH 2）p，-C（O） - 或-O-（CR 3 R 4）q键连接到苯环; R 1和R 2独立地选自苯基或被卤代烷基或卤代烷氧基取代的吡啶基; R3和R4独立地选自氢和甲基; n和p独立地为1,2或3; 且q为1或2;条件是R1和R2中的至少一个在对位取代; R3和R4中不超过两个是甲基; 每个脂族部分含有不超过4个碳原子; 卤素是指溴，氯或氟; 每个杂环含有1至4个氮原子，或1或2个氧或硫原子，或1或2个氮原子和氧或硫原子;以及相应的N-氧化物和农业上可接受的盐。

17. 发明授权

US06184234B2 Insecticidal N-(substituted arylmethyl)-4-[bis(substituted phenyl or pyridyl)methyl]piperidines 失效
标题翻译：杀虫剂N-（取代的芳基甲基）-4- [双（取代的苯基或吡啶基）甲基]哌啶
公开(公告)号：US06184234B2
公开(公告)日：2001-02-06
申请号：US09414375
申请日：1999-10-07
申请人： Ian R. Silverman , Daniel H. Cohen , John W. Lyga , Steven W. Szczepanski , Syed F. Ali , Thomas G. Cullen , Robert N. Henrie, II , Clinton J. Peake
发明人： Ian R. Silverman , Daniel H. Cohen , John W. Lyga , Steven W. Szczepanski , Syed F. Ali , Thomas G. Cullen , Robert N. Henrie, II , Clinton J. Peake
IPC分类号： A01N4340
CPC分类号： C07D231/12 , A01N43/40 , A01N43/50 , A01N43/54 , A01N43/56 , A01N43/60 , A01N43/653 , A01N43/713 , A01N43/76 , A01N43/82 , A01N47/20 , A01N55/00 , C07D211/14 , C07D211/22 , C07D211/24 , C07D211/26 , C07D211/94 , C07D233/56 , C07D249/08 , C07D401/06 , C07D401/10 , C07D401/12 , C07D401/14 , C07D405/06 , C07D405/10 , C07D409/06 , C07D413/06 , C07D413/10 , C07D417/10 , C07D417/12 , C07F7/1804
摘要： Compounds of the following structure, the corresponding N-oxides and agriculturally acceptable salts thereof, are disclosed as effective insecticides: wherein U is —(CH2)n—; Q is hydroxy; and R is: and wherein V, W, Y, and Z are each hydrogen; X is a five- or six-membered heterocycle; optionally substituted with bromine, chlorine, fluorine, cyano, alkyl, haloalkyl, alkoxy, haloalkoxy, alkoxyalkyl, haloalkoxyalkyl, or aminocarbonyl; and the heterocycle is optionally connected to the phenyl ring through a —O—, —S—, —(CH2)p, —C(O)—, or —O—(CR3R4)q linkage; R1 and R2 are independently selected from phenyl or pyridyl substituted with pentahalothio, haloalkylthio, haloalkylsulfinyl, or haloalkylsulfonyl; phenyl substituted with —OC(M)2O—, where M is bromine, chorine or fluorine, to provide a dihalobenzodioxolyl fused ring; or pyridyl substituted with —OC(M)2O— to provide a dihalodioxolenopyridyl fused ring; R3 and R4 are independently selected from hydrogen and methyl; n and p are independently 1, 2, or 3; and q is 1 or 2; with the proviso that at least one of R1 and R2 is substituted in the para position of the phenyl ring or the 5-position of the 2-pyridyl ring; each alkyl portion of said optional substituent on X wherein the optional substituent is alkyl, haloalkyl, alkoxyl, haloalkoxyl, alkoxyalkyl, or haloalkoxyalkyl contains from 1 to 4 carbon atoms; each heterocycle contains from 1 to 4 nitrogen atoms, 1 or 2 oxygen or sulfur atoms, or 1 or 2 nitrogen atoms and an oxygen or sulfur atom; and the corresponding N-oxides and agriculturally acceptable salts.
摘要翻译：以下结构的化合物，其相应的N-氧化物和农业上可接受的盐被公开为有效的杀虫剂：其中U是 - （CH 2）n - ; Q是羟基; 且R为：且其中V，W，Y和Z各自为氢; X为五元或六元杂环; 任选被溴，氯，氟，氰基，烷基，卤代烷基，烷氧基，卤代烷氧基，烷氧基烷基，卤代烷氧基烷基或氨基羰基取代; 并且杂环任选地通过-O - ， - S - ， - （CH 2）p，-C（O） - 或-O-（CR 3 R 4）q键连接到苯环; R 1和R 2独立地选自苯基或被五卤代硫代，卤代烷硫基，卤代烷基亚磺酰基或卤代烷基磺酰基取代的吡啶基; 用-OC（M）2 O-取代的苯基，其中M是溴，氯或氟，得到二卤代二苯甲基稠合环; 或被-OC（M）2 O-取代的吡啶基，以提供二卤代苯并吡啶基稠环; R 3和R 4独立地选自氢和甲基; n和p独立地为1,2或3; 平均值为1或2; 条件是R 1和R 2中的至少一个在苯环的对位或2-吡啶基环的5-位上被取代; X上任选取代基的每个烷基部分，其中任选的取代基是烷基，卤代烷基，烷氧基，卤代烷氧基，烷氧基烷基或卤代烷氧基烷基含有1至4个碳原子; 每个杂环含有1至4个氮原子，1或2个氧或硫原子，或1或2个氮原子和氧或硫原子; 和相应的N-氧化物和农业上可接受的盐。

18. 发明授权

US6030987A Insecticidal N-(substituted arylmethyl)-4-[bis(substituted phenyl or pyridyl)methyl]piperidines 失效
标题翻译：杀虫剂N-（取代的芳基甲基）-4- [双（取代的苯基或吡啶基）甲基]哌啶
公开(公告)号：US6030987A
公开(公告)日：2000-02-29
申请号：US981456
申请日：1998-08-11
申请人： Ian R. Silverman , Daniel H. Cohen , John W. Lyga , Steven W. Szczepanski , Syed F. Ali , Thomas G. Cullen , Robert N. Henrie, II , Clinton J. Peake
发明人： Ian R. Silverman , Daniel H. Cohen , John W. Lyga , Steven W. Szczepanski , Syed F. Ali , Thomas G. Cullen , Robert N. Henrie, II , Clinton J. Peake
IPC分类号： A01N43/40 , A01N43/54 , A01N43/56 , A01N43/653 , A01N43/713 , A01N43/76 , A01N43/82 , C07D401/10 , C07D417/10
CPC分类号： A01N43/713 , A01N43/40 , A01N43/54 , A01N43/56 , A01N43/653 , A01N43/76 , A01N43/82
摘要： Compounds of structure (I) ##STR1## the corresponding N-oxides and agriculturally acceptable salts are disclosed as effective insecticides. In said formula, U is --(CH.sub.2)n--; Q is hydroxy, R is formula (II) ##STR2## in which V, W, Y and Z are hydrogen; X is a five- or six-membered heterocycle optionally substituted; and the heterocycle is optionally connected to the phenyl ring through a --O--, --S-- --CH.sub.2)p--, or --O(CR.sup.3 R.sup.4)q linkage; R.sup.1 and R.sup.2 are independently selected from phenyl or pyridyl substituted with haloalkyl or haloalkoxy; R.sup.3, R.sup.4, n, p, and 1 are as defined in the specification.
摘要翻译： PCT No.PCT / US96 / 07206 Sec。 371日期：1998年8月11日 102（e）1998年8月11日PCT PCT 1996年5月17日PCT公布。公开号WO96 / 36228 PCT 日期：1996年11月21日公开了结构（Ⅰ）化合物对应的N-氧化物和农业上可接受的盐作为有效杀虫剂。在所述式中，U是 - （CH 2）n - ; Q是羟基，R是式（II），其中V，W，Y和Z是氢; X是任选取代的五或六元杂环; 并且杂环任选地通过-O - ， - S--CH 2）对 - 或-O（CR 3 R 4）q键连接到苯环上; R 1和R 2独立地选自苯基或被卤代烷基或卤代烷氧基取代的吡啶基; R3，R4，n，p和1如说明书中所定义。

19. 发明授权

US07365082B2 N-(substituted arylmethyl)-4-(disubstituted methyl)piperidines and piperazines 失效
标题翻译： N-（取代的芳基甲基）-4-（二取代的甲基）哌啶和哌嗪
公开(公告)号：US07365082B2
公开(公告)日：2008-04-29
申请号：US10538997
申请日：2003-12-08
申请人： Ping Ding , Robert N. Henrie, II , Daniel H. Cohen , John W. Lyga , David S. Rosen , George Theodoridis , Qun Zhang , Walter H. Yeager , Stephen F. Donovan , Steven Shunxiang Zhang , Inna Shulman , Seong Jae Yu , Guozhi Wang , Y. Larry Zhang , Ariamala Gopalsamy , Dennis L. Warkentin , Paul E. Rensner , Ian R. Silverman , Thomas G. Cullen
发明人： Ping Ding , Robert N. Henrie, II , Daniel H. Cohen , John W. Lyga , David S. Rosen , George Theodoridis , Qun Zhang , Walter H. Yeager , Stephen F. Donovan , Steven Shunxiang Zhang , Inna Shulman , Seong Jae Yu , Guozhi Wang , Y. Larry Zhang , Ariamala Gopalsamy , Dennis L. Warkentin , Paul E. Rensner , Ian R. Silverman , Thomas G. Cullen
IPC分类号： A61K31/44 , A61K31/445 , A61K31/4422 , C07D211/06 , C07D211/08 , C07D211/70 , C07D211/82
CPC分类号： C07D405/14 , A01N43/40 , A01N43/54 , A01N43/713 , C07D211/14 , C07D211/18 , C07D211/22 , C07D211/24 , C07D211/26 , C07D211/28 , C07D211/32 , C07D211/94 , C07D401/06 , C07D401/10 , C07D401/12 , C07D401/14 , C07D413/12 , C07D417/12 , C07D451/14 , C07D513/04
摘要： It has now been found that certain novel N-(substituted aryl)-4-(disubstituted methyl)piperidine and pyridine derivatives have provided unexpected insecticidal activity. These compounds are represented by formula (I): wherein m, n, q, r, and s are independently selected from 0 or 1; and p is 0, 1, 2, or 3; A is CH or N; and B, D, E, R, R1, R2, R3, R4, R5, R6, R7 and R8 are fully described herein. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula I, and optionally, an effective amount of at least one of a second compound, with at least one insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present.
摘要翻译：现在已经发现某些新的N-（取代的芳基）-4-（二取代的甲基）哌啶和吡啶衍生物提供了意想不到的杀虫活性。这些化合物由式（I）表示：其中m，n，q，r和s独立地选自0或1; 且p为0,1,2或3; A是CH或N; 和B，D，E，R，R 1，R 2，R 3，R 4，R 本文完全描述了本发明的第5，第6，第七和第八和第八。此外，还公开了包含杀虫有效量的至少一种式I化合物和任选的有效量的至少一种第二化合物与至少一种与杀虫相容的载体的组合物; 以及控制昆虫的方法，包括将所述组合物施用于存在昆虫或预期存在的场所。

20. 发明授权

US07683070B2 N-(substituted arylmethyl)-4-(disubstituted methyl) piperidines and pyridines 有权
标题翻译： N-（取代的芳基甲基）-4-（二取代的甲基）哌啶和吡啶
公开(公告)号：US07683070B2
公开(公告)日：2010-03-23
申请号：US11874015
申请日：2007-10-17
申请人： Ping Ding , Robert N. Henrie, II , Daniel H. Cohen , John W. Lyga , David S. Rosen , George Theodoridis , Qun Zhang , Walter H. Yeager , Stephen F. Donovan , Stephen Shunxiang Zhang , Inna Shulman , Seong Jae Yu , Guozhi Wang , Y. Larry Zhang , Ariamala Gopalsamy , Dennis L. Warkentin , Paul E. Rensner , Ian R. Silverman , Thomas G. Cullen
发明人： Ping Ding , Robert N. Henrie, II , Daniel H. Cohen , John W. Lyga , David S. Rosen , George Theodoridis , Qun Zhang , Walter H. Yeager , Stephen F. Donovan , Stephen Shunxiang Zhang , Inna Shulman , Seong Jae Yu , Guozhi Wang , Y. Larry Zhang , Ariamala Gopalsamy , Dennis L. Warkentin , Paul E. Rensner , Ian R. Silverman , Thomas G. Cullen
IPC分类号： A61K31/4523 , A61K31/4545 , C07D211/06 , C07D239/02
CPC分类号： C07D405/14 , A01N43/40 , A01N43/54 , A01N43/713 , C07D211/14 , C07D211/18 , C07D211/22 , C07D211/24 , C07D211/26 , C07D211/28 , C07D211/32 , C07D211/94 , C07D401/06 , C07D401/10 , C07D401/12 , C07D401/14 , C07D413/12 , C07D417/12 , C07D451/14 , C07D513/04
摘要： It has now been found that certain novel N-(substituted aryl)-4-(disubstituted methyl)piperidine and pyridine derivatives have provided unexpected insecticidal activity. These compounds are represented by formula (I): wherein m, n, q, r, and s are independently selected from 0 or 1; and p is 0, 1, 2, or 3; A is C or CH; and B, D, E, R, R1, R2, R3, R4, R5, R6, R7 and R8 are fully described herein. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula I, and optionally, an effective amount of at least one of a second compound, with at least one insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present.
摘要翻译：现在已经发现某些新的N-（取代的芳基）-4-（二取代的甲基）哌啶和吡啶衍生物提供了意想不到的杀虫活性。这些化合物由式（I）表示：其中m，n，q，r和s独立地选自0或1; 且p为0,1,2或3; A是C或CH; 本文完整地描述了B，D，E，R，R 1，R 2，R 3，R 4，R 5，R 6，R 7和R 8。此外，还公开了包含杀虫有效量的至少一种式I化合物和任选的有效量的至少一种第二化合物与至少一种与杀虫相容的载体的组合物; 以及控制昆虫的方法，包括将所述组合物施用于存在昆虫或预期存在的场所。

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