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1. 发明专利

JP2007297310A Heterocyclic oxyacetic amide compound and bactericide 审中-公开
标题翻译：杂环氧化物酰胺化合物和杀菌剂
公开(公告)号：JP2007297310A
公开(公告)日：2007-11-15
申请号：JP2006125385
申请日：2006-04-28
申请人： Hokko Chem Ind Co Ltd , 北興化学工業株式会社
发明人： ONOE SHINJI , ISHIDA TOMOYUKI , OKITA HIROYUKI , KUTSUMA SEIICHI , MORITA TAKESHI
IPC分类号： C07D213/56 , A01N43/08 , A01N43/10 , A01N43/40 , A01N43/42 , A01N55/00 , A01P3/00 , C07D215/14 , C07D307/52 , C07D333/24 , C07F7/10
摘要： PROBLEM TO BE SOLVED: To provide a novel heterocyclic oxyacetic amide compound that exhibits high effect against plant diseases, particularly against downy mildew and epidemic and shows high safety without drug disaster on the field crops and provide a bactericide including the compound as an active ingredient, particularly a bactericide for agriculture and horticulture. SOLUTION: The heterocyclic oxyacetic amide compound (including optical isomers) is represented by general (I)(wherein Het is a five-membered heterocyclic ring or a six-membered heterocyclic ring; R is H, a halogen, an alkyl, a cycloalkyl, an alkoxy, trialkylsilyl, phenyl which may be substituted or a heterocyclic ring which may be substituted; n is an integer of 1 or 2; z is an alkyl or a cyanoalkyl). COPYRIGHT: (C)2008,JPO&INPIT
摘要翻译：要解决的问题：提供一种对植物病害特别是针对霜霉病和流行病具有高效果的新型杂环氧基乙酰胺化合物，并且在野外作物上表现出高安全性而没有药物灾害，并提供包括该化合物作为活性成分，特别是农业和园艺用杀菌剂。解决方案：杂环氧基乙酰胺化合物（包括光学异构体）由通式（I）表示（其中Het是五元杂环或六元杂环; R是H，卤素，烷基，环烷基，烷氧基，三烷基甲硅烷基，可被取代的苯基或可被取代的杂环; n是1或2的整数; z是烷基或氰基烷基）。版权所有（C）2008，JPO＆INPIT

2. 发明专利

JPS59116272A Imidazole derivative and agricultural and hotricultural fungicide 失效
标题翻译：咪唑衍生物和农业和农村化学品
公开(公告)号：JPS59116272A
公开(公告)日：1984-07-05
申请号：JP22489682
申请日：1982-12-23
申请人： Hokko Chem Ind Co Ltd
发明人： OOYAMA HIROSHI , MORITA TAKESHI , OONO TOSHIJI , WADA TAKUO
IPC分类号： C07D233/61 , A01N43/50
摘要： NEW MATERIAL:The imidazole derivative of formula I (R
1 is lower alkyl; R
2 is R
1 or lower alkenyl) or its salt.
EXAMPLE: 1-[N-(2-Chloro-4-fluorophenyl)-2-ethoxypropaneimidoyl]-imidazole.
USE: An agricultural or horticultural fungicide or seed disinfectant. It has broad fungicidal activity, and exhibits excellent controlling effect against various plant blights, especially rust and powdery mildew of wheat, helminthosporium leaf spot of rice, bean, etc., blast of rice, mildew of cucumber, water melon, etc. at a low rate of application. It is harmless to useful crops, and free from toxicity to man, animal and fish, and can be used safely.
PROCESS: The compound of formula I can be prepared by reacting the compound of formula II (X is halogen) with imidazole of formula III preferably in an or ganic solvent, if necessary in the presence of an acid acceptor such as triethylamine, under ice cooling at 0W100°C for ≤1hr.
COPYRIGHT: (C)1984,JPO&Japio
摘要翻译：新材料：式Ⅰ咪唑衍生物（R1为低级烷基; R2为R1或低级链烯基）或其盐。实施例：1- [N-（2-氯-4-氟苯基）-2- ethoxypropaneimidoyl] - 咪唑。用途：农业或园艺杀菌剂或种子消毒剂。具有广泛的杀菌活性，对各种植物枯萎病，特别是小麦锈病和白粉病，水稻，豆类等等的杀虫剂，水稻，黄瓜，西瓜等霉菌的防治效果优异。使用率低。有用的作物无害，对人，动物和鱼类无毒，可安全使用。方法：式I化合物可以通过使式II化合物（X为卤素）与式III咪唑在惰性溶剂中反应，如果需要，在酸受体如三乙胺存在下，在冰冷却下在0-100℃下<= 1小时。

3. 发明专利

JPS59122473A Imidazole derivative and agricultural and horticultural fungicide 失效
标题翻译：咪唑衍生物和农业和农业化学品
公开(公告)号：JPS59122473A
公开(公告)日：1984-07-14
申请号：JP23056782
申请日：1982-12-29
申请人： Hokko Chem Ind Co Ltd
发明人： OOYAMA HIROSHI , MORITA TAKESHI , OONO TOSHIJI , WADA TAKUO
IPC分类号： C07D233/61 , A01N43/50
摘要： NEW MATERIAL:The compound of formula I (A is lower alkylene; R is lower alkynyl, cycloalkyl, cycloalkylalkyl, lower saturated alkyl or lower unsaturated alkyl which is interrupted by O or S, cyanoalkyl or arylalkyl) and its salt.
EXAMPLE: 1-[N-(2-chloro-4-fluorophenyl)-2-propargyloxyethanimidoyl]imidazole.
USE: An agricultural and horticultural fungicide having little phtotoxicity to useful crops and harmless to man and animal.
PROCESS: The compound of formula I can be prepared by reacting the compound of formula II (X is halogen) with imidazole and an amophoteric substance (e.g. alkali metal salt, inorganic acid salt, organic acid salt, metal complex salt, etc.) in an organic solvent at 0W85°C, optionally in the presence of an acid acceptor.
COPYRIGHT: (C)1984,JPO&Japio
摘要翻译：新材料：式I化合物（A为低级亚烷基; R为低级炔基，环烷基，环烷基烷基，低级饱和烷基或被O或S间隔的低级不饱和烷基，氰基烷基或芳基烷基）及其盐。实施例：1- [N-（2-氯-4-氟苯基）-2-丙酰氧基乙亚氨基]咪唑。用途：农用和园艺杀菌剂对有用作物几乎没有毒性，对人类和动物无害。方法：式I化合物可以通过使式II化合物（X为卤素）与咪唑和amophoteric物质（例如碱金属盐，无机酸盐，有机酸盐，金属络盐等）反应来制备 0-85℃的有机溶剂，任选在酸受体存在下进行。

4. 发明专利

JPS59116271A Imidazole derivative and agricultural and horticultural fungicide 失效
标题翻译：咪唑衍生物和农业和农业化学品
公开(公告)号：JPS59116271A
公开(公告)日：1984-07-05
申请号：JP22489582
申请日：1982-12-23
申请人： Hokko Chem Ind Co Ltd
发明人： OOYAMA HIROSHI , MORITA TAKESHI , OONO TOSHIJI , WADA TAKUO
IPC分类号： C07D233/61 , A01N43/50
摘要： NEW MATERIAL:The imidazole derivative of formula I (R is lower alkyl or lower alkenyl) or its salt.
EXAMPLE: 1-[N-(2-Chloro-4-fluorophenyl)-2-n-propyloxyethaneimidoyl]-imidazole.
USE: An agricultural or horticultural fungicide or seed disinfectant. It has broad fungicidal activity, and exhibits excellent controlling effect against various plant blights, especially rust and powdery mildew of wheat, helminthosporium leaf spot of rice, bean, etc., blast of rice, mildew of cucumber, water melon, etc. at a low rate of application. It is harmless to useful crops, and free from toxicity to man, animal and fish, and can be used safely.
PROCESS: The compound of formula I can be prepared by reacting the compound of formula II (X is halogen) with imidazole of formula III preferably in an organic solvent, if necessary in the presence of an acid acceptor such as triethylamine, under ice cooling at 0W100°C for ≤1hr.
COPYRIGHT: (C)1984,JPO&Japio
摘要翻译：新材料：式I的咪唑衍生物（R是低级烷基或低级烯基）或其盐。实施例：1- [N-（2-氯-4-氟苯基）-2-正丙氧基亚氨基] - 咪唑。用途：农业或园艺杀菌剂或种子消毒剂。具有广泛的杀菌活性，对各种植物枯萎病，特别是小麦锈病和白粉病，水稻，豆类等的防治，防治黄瓜，黄瓜，水瓜等的防治效果显着。使用率低。有用的作物无害，对人，动物和鱼类无毒，可安全使用。方法：式I化合物可以通过使式II的化合物（X为卤素）与式III的咪唑优选在有机溶剂中反应，如果需要，在酸受体如三乙胺的存在下，在冰冷却下， 0-100℃，<= 1小时。

5. 发明专利

JPS5953474A 2-(substituted phenoxy)propionic acid derivative and herbicide containing said derivative as active component 失效
标题翻译： 2-（取代的苯甲酸）含有衍生物和除草剂的含有衍生物作为活性成分
公开(公告)号：JPS5953474A
公开(公告)日：1984-03-28
申请号：JP16319482
申请日：1982-09-21
申请人： Hokko Chem Ind Co Ltd
发明人： OOYAMA HIROSHI , TAKADA SANAE , MORITA TAKESHI , YAMAMURA SABUROU
IPC分类号： A01N43/80 , C07D261/02
摘要： NEW MATERIAL:The 2-(substituted phenoxy)propionic acid derivative of formula I (R
1 is 4-chlorophenyl or 2,4-dichlorophenyl; R
2 is H or lower alkyl).
EXAMPLE: N-{(±)-2-[4-(2,4-Dichlorophenoxy)phenoxy]propionyl}isoxazolidine.
USE: Herbicide effective especially to gramineous weeds, free from phytotoxicity to soybean, beet, radish, cabbage, cotton, etc., having no toxicity to man, animal and fish, and applicable safely.
PROCESS: The objective compound of formula I can be prepared, e.g. by reacting the compound of formula II (X is halogen) with the novel compound of formula IIIin the presence of an acid acceptor. The novel compound of formula III can be obtained easily by the reaction of N-(2-halopropionyl)isoxazolidine with hydroquinone.
COPYRIGHT: (C)1984,JPO&Japio
摘要翻译：新材料：式I的（取代的苯氧基）丙酸衍生物（R1是4-氯苯基或2,4-二氯苯基; R2是H或低级烷基）。实施例：N - {（+或 - ） - 2- [4-（2,4-二氯苯氧基）苯氧基]丙酰基}异恶唑烷。用途：除草剂对禾本科杂草有效，对大豆，甜菜，萝卜，卷心菜，棉花等无植物毒性，对人，动物和鱼类无毒性，安全可用。方法：式I的目标化合物可以制备，例如通过在酸受体的存在下使式II化合物（X是卤素）与新的式III化合物反应。通过N-（2-卤代丙酰基）异恶唑烷与氢醌的反应可以容易地得到式III的新化合物。

6. 发明专利

JPS59116273A Imidazole derivative and agricultural and horticultural fungicide 失效
标题翻译：咪唑衍生物和农业和农业化学品
公开(公告)号：JPS59116273A
公开(公告)日：1984-07-05
申请号：JP22489782
申请日：1982-12-23
申请人： Hokko Chem Ind Co Ltd
发明人： OOYAMA HIROSHI , MORITA TAKESHI , OONO TOSHIJI , WADA TAKUO
IPC分类号： C07D233/61 , A01N43/50
摘要： NEW MATERIAL:The compound of formula 1 (A is straight or branched chain lower alkylene; R is saturated or unsaturated lower alkyl which may be interrupted with O or S, cyanoalkyl, cycloalkyl, benzyl, halobenzyl, or phenyl; n is 0, 1 or 2) and its salt.
EXAMPLE: 1-[N-(2-Chloro-4-fluorophenyl)-2-n-propylthioethaneimidoyl]-imidazole.
USE: An agricultural and horticultural fungicide free from phytotoxicity and harmless to man and animal.
PROCESS: The compound of formula 1 can be prepared by reacting the compound of formula 2 with the compound of formula 3 preferably in an organic solvent such as benzene, chloroform, etc., if necessary in the presence of an acid acceptor, at 0W85°C.
COPYRIGHT: (C)1984,JPO&Japio
摘要翻译：新材料：式1化合物（A为直链或支链低级亚烷基; R为可被O或S间隔的饱和或不饱和低级烷基，氰基烷基，环烷基，苄基，卤代苄基或苯基; n为0,1 或2）及其盐。实施例：1- [N-（2-氯-4-氟苯基）-2-正丙硫基亚氨代] - 咪唑。用途：无植物毒性的农业和园艺杀菌剂，对人类和动物无害。方法：式1的化合物可以通过使式2的化合物与式3的化合物在需要时在酸受体的存在下，在有机溶剂如苯，氯仿等中反应来制备， 85摄氏度

7. 发明专利

JPS61109795A Phenylthiol phosphonic acid derivative, its preparation and insecticide, acaricide and nematocide 失效
标题翻译：苯乙酸磷酸衍生物，其制备和杀虫剂，杀虫剂和杀虫剂
公开(公告)号：JPS61109795A
公开(公告)日：1986-05-28
申请号：JP23034984
申请日：1984-11-02
申请人： Hokko Chem Ind Co Ltd
发明人： OOYAMA HIROSHI , KITAORI KAZUHIKO , MORITA TAKESHI , MORIYAMA SATORU , UCHIYAMA TSUGIO
IPC分类号： A01N57/22 , A01N57/06 , C07F9/38 , C07F9/40
摘要： NEW MATERIAL:A compound of formula I (R
1 is lower alkyl; R
2 is H, lower alkyl, lower alkenyl; R
3 is lower alkyl, lower alkenyl).
EXAMPLE: O-Ethyl-S-(N-methoxyacetimidoyl)phenylathiol phosphate.
USE: Insecticide, acaricide and nematocide in agricultural and horticultural fields.
PREPARATION: The reaction of an O-alkylphenyl phosphonic halide of formula II (X is halogen) such as O-ethylphenyl phosphonic acid chloride with a thiohydroxamic acid derivative of formula III such as O- methylacetothiohydroxamate is carried out, preferably in the presence of a base such as sodium hydroxide in an inert organic solvent such as benzene at 20W80°C.
COPYRIGHT: (C)1986,JPO&Japio
摘要翻译：新物质：式Ⅰ化合物（R1为低级烷基，R2为H，低级烷基，低级烯基，R3为低级烷基，低级烯基）。实施例：O-乙基-S-（N-甲氧基亚氨代乙基）苯基硫醇磷酸酯。用途：农业和园艺领域的杀虫剂，杀螨剂和杀线虫剂。制备：将式II的O-烷基苯基膦酰卤（X为卤素）如O-乙基苯基膦酰氯与式III的硫代异羟肟酸衍生物如O-甲基乙酰基硫代羟基甲酸酯反应进行，优选在碱如氢氧化钠在惰性有机溶剂如苯中，在20-80℃。

8. 发明专利

JPS5962506A Soil fungicide 失效
标题翻译：土壤杀真菌剂
公开(公告)号：JPS5962506A
公开(公告)日：1984-04-10
申请号：JP17099782
申请日：1982-10-01
申请人： Hokko Chem Ind Co Ltd
发明人： OOYAMA HIROSHI , MORITA TAKESHI , ARAKAWA MASAZUMI , SATOU KATSUMI
IPC分类号： C07D249/08 , A01N43/64 , A01N43/653
摘要： PURPOSE: To fungicide extremely effective against infectious blights of soil such as Fusarium wilt of cucumbers, melons, and gourd family, having neither toxicity to men and beasts, nor phytotoxicity to crops, capable of controlling the blights with reduced labor without requiring operation of gas removal, etc., containing one of a 1,2,4-triazole derivative and its salt as an active ingredient.
CONSTITUTION: A fungicide containing one of a 1,2,4-triazole derivative shown by the formula I (X is Cl, or F; Y is H, or Cl) or its salt as an active ingredient. The compound shown by the formula I , for example, is synthesized by reacting a compound shown by the formula II (A is halogen, imidazol-l-yl group, 1,2 4- triazol-1-yl group, alkylsulfone group, or arylsulfone group) with a compound shown by the formula III in an organic solvent such as preferably a hydrocarbon, etc., and, if necessary, in the presence of an acid binder such as triethylamine, etc. 1,2,4-Triazol-l-ylisothioacetic acid-2',4'-dichloroanilido S-p-chlorobenzyl ether, etc. may be cited as a concrete example of the derivative shown by the formula I .
COPYRIGHT: (C)1984,JPO&Japio
摘要翻译：目的：杀菌剂对抗黄瓜，瓜类和葫芦科植物的镰刀菌枯萎病，对人类和野兽没有毒性，对作物没有植物毒性，可以极大地有效地防治病虫害，而不需要操作气体去除等，含有1,2,4-三唑衍生物及其盐之一作为活性成分。构成：含有式I所示的1,2,4-三唑衍生物（X为Cl或F; Y为H或Cl）或其盐作为活性成分的杀真菌剂。式I所示的化合物，例如通过使式II表示的化合物（A是卤素，咪唑-1-基，1,2,4-三唑-1-基，烷基砜基或芳基砜基）与式III化合物反应，在有机溶剂如烃等中，必要时，在酸性粘合剂如三乙胺等的存在下，可以列举出式I所示的衍生物的具体例子，可以举出1-基二硫代乙酸-2'，4'-二氯苯胺基，间氯苄基醚等。

9. 发明专利

JPS5955882A 2-(substituted phenoxy)propionic acid derivative and herbicide containing said derivative as active component 失效
标题翻译： 2-（取代的苯甲酸）含有衍生物和除草剂的含有衍生物作为活性成分
公开(公告)号：JPS5955882A
公开(公告)日：1984-03-31
申请号：JP16496782
申请日：1982-09-24
申请人： Hokko Chem Ind Co Ltd
发明人： OOYAMA HIROSHI , TAKADA SANAE , MORITA TAKESHI , YAMAMURA SABUROU
IPC分类号： A01N43/80 , C07D413/12
摘要： NEW MATERIAL:The compound of formula I (R
1 is 3,5-dichloro-2-pyridyl or 5-trifluoromethyl-2-pyridyl; R
2 is H or lower alkyl).
EXAMPLE: N-{ (±)-2-[ 4-( 3,5-Dichloro-2-pyridyloxy)phenoxy ]propionyl}isoxazolidine.
USE: Herbicide exhibiting excellent activity especially against gramineous weeds, and little phytotxicity to the broad-leaved crops such as soybean, beet, radish, cabbage, etc. or cotton etc., and having high safety.
PROCESS: The compound of formula I can be prepared by reacting the compound of formula R
1 -X (X is halogen) with the novel compound of formula II in an organic solvent in the presence of an acid acceptor (e.g. triethylamine, potassium carbonate, etc.) at room temperature W the boiling point of the solvent. The novel compound of formula II can be obtained easily e.g. by the reaction of N-(2-halopropionyl)-isoxazolidine with hydroquinone.
COPYRIGHT: (C)1984,JPO&Japio
摘要翻译：新物质：式Ⅰ化合物（R1为3,5-二氯-2-吡啶基或5-三氟甲基-2-吡啶基; R2为H或低级烷基）。实施例：N- {（+或 - ） - 2- [4-（3,5-二氯-2-吡啶氧基）苯氧基]丙酰基}异恶唑烷。用途：除草剂表现出优异的活性，特别是对禾本科杂草，对大豆，甜菜，萝卜，卷心菜等棉花等广泛作物的植物毒性小，安全性高。方法：式I化合物可以通过在酸受体（例如三乙胺，碳酸钾等）存在下，在有机溶剂中使式R 1 -X（X为卤素）的化合物与新型式II化合物反应来制备。）在室温下 - 溶剂的沸点。式II的新化合物可以容易地获得，例如，通过N-（2-卤代丙酰基） - 异恶唑烷与氢醌的反应。

10. 发明专利

JPS54147921A Agricultural and horticultural pesticide 失效
标题翻译：农业和农业农药
公开(公告)号：JPS54147921A
公开(公告)日：1979-11-19
申请号：JP5487278
申请日：1978-05-08
申请人： Hokko Chem Ind Co Ltd , Meiji Seika Kaisha Ltd
发明人： NISHIMURA TAMIO , OOYAMA HIROSHI , YAMAMURA HIROSHI , MORITA TAKESHI , MATSUMOTO KUNIOMI , WATANABE TETSUO
IPC分类号： A01N43/56 , C07D403/04
摘要： PURPOSE: An agriculatural and horticultural pesticide effective to rice blast, helminthosporium leaf spot of rice plant, powdery mildew of cucumber, etc., free from phytotoxicity, and harmless to man, beast and fish, containing a specific pyrazolylpyrimidine derivative as an effective component.
CONSTITUTION: A composition containing a pyrazolylpyrimidine derivative of formula [R
1 is lower alkyl, phenyl; R
2 is alkyl, cyclohexyl, phenyl (which may be substituted by lower alkyl or halogen); R
3 is H, alkyl; R
2 and R
3 may together with adjacent N atom form a heterocyclic ring]. For example, a compound wherein all of the R
1-3 are methyl, or a compound where in all of the R
1-3 are methyl, or a compound wherein R
1 is phenyl, R
2 is ethyl, and R
3 is H.
COPYRIGHT: (C)1979,JPO&Japio
摘要翻译：目的：一种对稻瘟病有效的农作物和园艺农药，水稻螟虫斑点，黄瓜白粉病等，无植物毒性，对人体，野兽和鱼类无害，含有特异性吡唑嘧啶衍生物作为有效成分。组成：含有式[R 1的吡唑基嘧啶衍生物的组合物是低级烷基，苯基; R2是烷基，环己基，苯基（其可以被低级烷基或卤素取代）; R3是H，烷基; R2和R3可以与相邻的N原子一起形成杂环]。例如，其中所有R1-3为甲基的化合物，或其中R1-3全部为甲基的化合物或其中R 1为苯基，R 2为乙基且R 3为H的化合物。

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