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61. 发明公开

EP0212550A2 Substituted dipeptide amides 失效
标题翻译：取代二哌啶酰胺。
公开(公告)号：EP0212550A2
公开(公告)日：1987-03-04
申请号：EP86111143.3
申请日：1986-08-12
申请人： G.D. Searle & Co.
发明人： Hansen, Donald Willis, Jr. , Pilipauskas, Daniel Richard , Clare, Michael
IPC分类号： C07K5/06 , A61K37/02
CPC分类号： C07D333/48 , A61K38/00 , C07D333/20 , C07D333/38 , C07D335/02 , C07K5/06078
摘要： The invention relates to novel substituted tyrosyl alanine dipeptide amides of the formula:
and the pharmaceutically acceptable acid addition salts thereof wherein R¹ is hydrogen, lower alkyl, hydroxy, lower alkoxy, -O(CH₂) n phenyl with the phenyl optionally substituted by halogen, -NO₂, -CN, -NH₂ or lower alkyl wherein n is 1 to 4; R² and R³ represent lower alkyl, halogen, or lower alkoxy, or either one of R² or R³ is hydrogen and the other is lower alkyl, lower alkoxy or halogen; R⁴, R⁵, R⁶, and R⁹ may be the same or different and represent hydrogen, lower alkyl, cycloalkyl having 3 to 8 carbons, unsaturated lower alkyl, or -(CH₂) m cycloalkyl with the cycloalkyl having 3 to 8 carbons and m is 1 to 4; R 10 is hydrogen or -(CH₂) p phenyl or with the phenyl optionally substituted with -NH₂, -OH, halogen, -NO₂, or lower alkyl or -(CH₂) p thienyl wherein p is 1 to 4; one of R⁷ or R⁸ is -(CH₂) f -S(O) z -(CH₂) q -CH₃ where f is 1 to 3 and q is 0 to 3, z is 0, 1 or 2 and the other is hydrogen or lower alkyl, or R⁷ and R⁸ together with carbon w is
where x and y are independently 1 to 3 and z is 0, or 2. V represents an asymmetric carbon that may be recemic or have the D or L configuration; W represents an asymmetric carbon when R⁷ and R⁸ are not the same that may be recemic or have the D or L configuration.
The compounds of this invention are useful as analgesic and/or antihypertensive agents.
摘要翻译：本发明涉及下式的新型取代的酪氨酰丙氨酸二肽酰胺：其中R 1是氢，低级烷基，羟基，低级烷氧基，-O（CH 2）n苯基与苯基任选地被卤素，-NO 2，-CN，-NH 2或其中n为1至4的低级烷基取代; R 2和R 3代表低级烷基，卤素或低级烷氧基，R 2或R 3中的任一个是氢，另一个是低级烷基，低级烷氧基或卤素; R 4，R 5，R 6和R 9可以相同或不同，表示氢，低级烷基，具有3-8个碳的环烷基，不饱和低级烷基或 - （CH 2）m环烷基环烷基具有3至8个碳原子，m为1至4; R 10为氢或 - （CH 2）p苯基或与-NH 2，-OH，卤素，-NO 2或低级烷基或 - （CH 2）p噻吩基取代的苯基，其中p为1至4; R 7或R 8中的一个为 - （CH 2）f S（O）z - （CH 2）q -CH 3，其中f为1至3，q为0至3，z为0,1或2，且另一个是氢或低级烷基，或R 7和R 8与碳w一起是，其中x和y独立地为1〜3，z为0或2.V表示可以是接收或具有D或L配置; 当R 7和R 8不同时，W表示不对称碳，可以是可接受的或具有D或L构型。本发明的化合物可用作镇痛和/或抗高血压药。

62. 发明公开

EP0158496A2 Substituted oxime carbamates 失效
标题翻译：取代的肟氨基甲酸酯。
公开(公告)号：EP0158496A2
公开(公告)日：1985-10-16
申请号：EP85302256.4
申请日：1985-04-01
申请人： UNIROYAL, INC.
发明人： Strunk, Richard J. , Moore, Richard C.
IPC分类号： C07D333/48 , C07D333/22 , C07D409/06 , A01N43/10
CPC分类号： C07D333/48 , A01N43/10 , C07C323/00 , C07D333/22 , C07D409/06
摘要： A compound having the formula
wherein R is C 1 -C 4 alkyl, cyclopropyl, C 2 -C 4 alkoxyalkyl, C 4 -C 8 dialkylaminoalkyl, C 2 -C 4 alkylthioalkyl, C 2 -C 4 alkylsulfinylalkyl, C 2 -C 4 alkylsulfonylalkyl, phenyl, C 7 -C 9 aralkyl, C 7 -C 9 alkaryl, furyl, thienyl or pyridyl; R 1 is hydrogen or C 1 -C 4 alkyl; R 2 is hydrogen or C 1 -C 4 alkyl; R 3 , R 4 and R 5 are the same or different and the hydrogen or C 1 -C 4 alkyl; R 6 and R 7 are the same or different and are hydrogen, C 1 -C 4 alkyl, allyl, benzyl or tolyl with the proviso that both R 6 and R 7 are not hydrogen; and n is 0, 1 or 2 and methods of making same are disclosed. This compound is useful as a pesticide.
Intermediates useful in synthesizing this pesticidally effective compound are also taught. These intermediate compounds have the structural formulas

where R, R', R 2 , R 3 , R 4 , R 5 and n have the same meanings as the pesticidally effective compound recited above; and Q is a leaving group. Methods of making these intermediate compounds are described.

63. 发明公开

EP0109575A3 Benzoic-acid derivatives, process and means for its production 失效
标题翻译：苯甲酸衍生物，其生产方法和手段
公开(公告)号：EP0109575A3
公开(公告)日：1984-09-05
申请号：EP83110605
申请日：1983-10-24
申请人： F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft
发明人： Frater, Georg, Dr. , Suchy, Milos, Dr. , Wenger, Jean, Dr. , Winternitz, Paul, Dr.
IPC分类号： C07C161/00 , C07D213/64 , C07D333/46 , A01N41/02 , A01N43/40 , A01N43/10
CPC分类号： C07D213/643 , A01N41/02 , A01N43/10 , A01N43/40 , C07D333/48
摘要： Benzoesäurederivate der allgemeinen Formel worin AN oder CR³,
R¹ Halogen oder Trifluormethyl,
R² und R³, unabhängig voneinander, Wasserstoff oder Halogen,
R⁴ Halogen, Nitro oder Cyano,
R⁵ Wasserstoff oder Methyl,
R⁶-Alkyl und R⁷-Alkyl oder gegebenenfalls mit Halogen, -Alkyl, -Alkoxy und/oder Nitro substituiertes Aryl, oder R⁶ und R⁷ zusammen Tetra-, Penta- oder Hexa methylen,
n 0 oder 1,
X Sauerstoff oder -NR⁸-
und R⁸ Wasserstoff oder -Alkyl bedeuten.
Verfahren zu deren Herstellung, Unkrautbekämpfungs mittel, die diese Verbindungen als Wirkstoffe enthalten, sowie die Verwendung solcher Verbindungen bzw. Mittel zur Bekämpfung von Unkräutern. Zudem betrifft sie zur Herstel lung dieser Verbindungen dienende Ausgangsmaterialien.

64. 发明授权

EP0027940B1 Verfahren zur Herstellung von Urethanen 失效
标题翻译：制备URETHANES的方法
公开(公告)号：EP0027940B1
公开(公告)日：1983-09-14
申请号：EP80106196.1
申请日：1980-10-11
申请人： BAYER AG
发明人： König, Klaus, Dr. , Findeisen, Kurt, Dr. , Sundermann, Rudolf, Dr. , Penninger, Stefan, Dr. , Fauss, Rudolf, Dr.
IPC分类号： C07C125/065 , C07C125/073 , C07D213/75 , C07D295/22 , C07D307/82 , C07D333/48
CPC分类号： C07D213/75 , C07D295/205 , C07D307/91 , C07D333/48

65. 发明公开

EP3395171A1 N-ARYLAMIDINE-SUBSTITUIERTE TRIFLUOROETHYLSULFID-DERIVATE ALS AKARIZIDE UND INSEKTIZIDE 审中-公开
公开(公告)号：EP3395171A1
公开(公告)日：2018-10-31
申请号：EP18168893.8
申请日：2012-12-12
申请人： Bayer CropScience Aktiengesellschaft
发明人： KÖHLER, Adeline , ALIG, Bernd , BECKER, Angela , VOERSTE, Arnd , GÖRGENS, Ulrich , FISCHER, Reiner , MORADI, Wahed Ahmed , CEREZO-GALVEZ, Silvia , HAHN, Julia Johanna , ILG, Kerstin , SCHWARZ, Hans-Georg , GOMIBUCHI, Takuya , ITO, Masahito , YAMAZAKI, Daiei , SHIBUYA, Katsuhiko , SHIMOJO, Eiichi
IPC分类号： A01N37/52 , C07C317/42 , C07C323/36 , C07C323/44 , C07C323/63
CPC分类号： A01N41/10 , A01N41/12 , A01N43/08 , A01N43/10 , A01N43/36 , A01N43/40 , A01N43/60 , A01N43/84 , A01N43/86 , C07C315/02 , C07C317/34 , C07C317/40 , C07C319/14 , C07C319/20 , C07C323/36 , C07C323/41 , C07C323/44 , C07C323/45 , C07C335/16 , C07C2601/02 , C07C2601/04 , C07C2601/08 , C07C2601/14 , C07D207/22 , C07D207/34 , C07D211/38 , C07D211/72 , C07D211/98 , C07D213/61 , C07D213/78 , C07D239/28 , C07D241/24 , C07D263/28 , C07D277/16 , C07D277/18 , C07D277/38 , C07D277/54 , C07D279/06 , C07D285/08 , C07D295/125 , C07D295/13 , C07D305/08 , C07D307/24 , C07D307/68 , C07D331/04 , C07D333/38 , C07D333/48 , C07D401/06
摘要： Die vorliegende Erfindung betrifft neue N-Arylamidine-substituierte Trifluoroethylsulfid-Derivate der Formel (I),

- in welcher X 1 , X 2 , X 3 , X 4 , R 1 , R 2 , R 3 , n die in der Beschreibung angegebenen Bedeutungen haben- deren Anwendung als Akarizide und Insektizide zur Bekämpfung tierischer Schädlinge und Verfahren sowie Zwischenprodukte zu ihrer Herstellung

67. 发明公开

EP3283460A1 MOLECULES HAVING PESTICIDAL UTILITY, AND INTERMEDIATES, COMPOSITION, AND PROCESSES, RELATED THERETO 有权转让
标题翻译：具有杀虫剂功效的分子，以及中间体，组合物和过程，与其相关的那些
公开(公告)号：EP3283460A1
公开(公告)日：2018-02-21
申请号：EP16718785.5
申请日：2016-04-07
申请人： Dow Agrosciences LLC
发明人： ECKELBARGER, Joseph D. , KNUEPPEL, Daniel I. , HEEMSTRA, Ronald J. , ROSS, Ronald , DEKORVER, Kyle A. , GARY, Kaitlyn , VEDNOR, Peter , MARTIN, Timothy P. , HUNTER, Ricky , DEMETER, David A. , TRULLINGER, Tony K. , BAUM, Erich W. , BENKO, Zoltan L. , CHOY, Nakyen , CROUSE, Gary D. , DAEUBLE, John F. , LI, Fangzheng , NISSEN, Jeffrey , RIENER, Michelle , SPARKS, Thomas C. , WESSELS, Frank J. , YAP, Maurice C.
IPC分类号： C07C237/42 , C07C255/46 , C07D205/04 , C07D295/32 , C07D305/08 , C07D309/14 , C07D333/36 , C07D331/04 , A01N37/18
CPC分类号： A01N53/00 , A01N37/22 , A01N37/34 , A01N41/10 , A01N43/40 , A01N43/60 , A01N43/653 , A01N43/707 , A01N43/82 , A01N43/90 , C07C233/63 , C07C233/65 , C07C237/22 , C07C237/42 , C07C255/29 , C07C255/46 , C07C255/57 , C07C255/60 , C07C259/10 , C07C271/28 , C07C271/66 , C07C311/08 , C07C311/46 , C07C317/14 , C07C317/28 , C07C317/40 , C07C317/50 , C07C323/41 , C07C323/42 , C07C323/59 , C07C331/12 , C07C381/10 , C07C2601/02 , C07C2601/04 , C07C2601/08 , C07C2601/14 , C07D205/04 , C07D207/10 , C07D207/273 , C07D207/452 , C07D209/49 , C07D213/56 , C07D213/75 , C07D213/81 , C07D213/84 , C07D213/89 , C07D215/227 , C07D215/38 , C07D231/12 , C07D231/56 , C07D233/36 , C07D233/80 , C07D235/30 , C07D241/20 , C07D249/08 , C07D253/07 , C07D261/12 , C07D263/26 , C07D277/30 , C07D277/36 , C07D285/06 , C07D295/32 , C07D305/08 , C07D307/33 , C07D307/52 , C07D309/14 , C07D331/04 , C07D333/36 , C07D333/48 , C07D333/60 , C07D487/04
摘要： This disclosure relates to the field of molecules having pesticidal utility against pests in Phyla Arthropoda, Mollusca, and Nematoda, processes to produce such molecules, intermediates used in such processes, pesticidal compositions containing such molecules, and processes of using such pesticidal compositions against such pests. These pesticidal compositions may be used, for example, as acaricides, insecticides, miticides, molluscicides, and nematicides. This document discloses molecules having the following formula ("Formula One").

68. 发明公开

EP3283458A1 MOLECULES HAVING PESTICIDAL UTILITY, AND INTERMEDIATES, COMPOSITIONS, AND PROCESSES, RELATED THERETO 有权转让
标题翻译：具有杀虫活性的分子，以及与其相关的中间体，组合物和过程
公开(公告)号：EP3283458A1
公开(公告)日：2018-02-21
申请号：EP16718097.5
申请日：2016-04-07
申请人： Dow Agrosciences LLC
发明人： MARTIN, Timothy P. , ECKELBARGER, Joseph D. , ROSS, Ronald , DEKORVER, Kyle A. , HEEMSTRA, Ronald J. , KNUEPPEL, Daniel I. , VEDNOR, Peter , HUNTER, Ricky , DEMETER, David A. , TRULLINGER, Tony K. , BAUM, Erich W. , BENKO, Zoltan L. , CHOY, Nakyen , CROUSE, Gary D. , DAEUBLE, John F. , LI, Fangzheng , NISSEN, Jeffrey , RIENER, Michelle , SPARKS, Thomas C. , WESSELS, Frank J. , YAP, Maurice C.
IPC分类号： C07C237/42 , A01N37/18 , C07C255/29 , C07C255/46 , C07C255/57 , C07C255/60
CPC分类号： A01N53/00 , A01N37/22 , A01N37/34 , A01N41/10 , A01N43/40 , A01N43/60 , A01N43/653 , A01N43/707 , A01N43/82 , A01N43/90 , C07C233/63 , C07C233/65 , C07C237/22 , C07C237/42 , C07C255/29 , C07C255/46 , C07C255/57 , C07C255/60 , C07C259/10 , C07C271/28 , C07C271/66 , C07C311/08 , C07C311/46 , C07C317/14 , C07C317/28 , C07C317/40 , C07C317/50 , C07C323/41 , C07C323/42 , C07C323/59 , C07C331/12 , C07C381/10 , C07C2601/02 , C07C2601/04 , C07C2601/08 , C07C2601/14 , C07D205/04 , C07D207/10 , C07D207/273 , C07D207/452 , C07D209/49 , C07D213/56 , C07D213/75 , C07D213/81 , C07D213/84 , C07D213/89 , C07D215/227 , C07D215/38 , C07D231/12 , C07D231/56 , C07D233/36 , C07D233/80 , C07D235/30 , C07D241/20 , C07D249/08 , C07D253/07 , C07D261/12 , C07D263/26 , C07D277/30 , C07D277/36 , C07D285/06 , C07D295/32 , C07D305/08 , C07D307/33 , C07D307/52 , C07D309/14 , C07D331/04 , C07D333/36 , C07D333/48 , C07D333/60 , C07D487/04
摘要： This disclosure relates to the field of molecules having pesticidal utility against pests in Phyla Arthropoda, Mollusca, and Nematoda, processes to produce such molecules, intermediates used in such processes, pesticidal compositions containing such molecules, and processes of using such pesticidal compositions against such pests. These pesticidal compositions may be used, for example, as acaricides, insecticides, miticides, molluscicides, and nematicides. This document discloses molecules having the following formula ("Formula One").

69. 发明授权

EP1686125B1 3-Alkoxy-tetraalkylene Sulfone and Derivatives as Seal Swelling Agents and a Process for their Preparation 有权
标题翻译： 3-烷氧基tetraalkylensulfon和衍生物作为密封溶胀剂，以及它们的制备方法
公开(公告)号：EP1686125B1
公开(公告)日：2017-05-17
申请号：EP06250501.1
申请日：2006-01-30
申请人： Afton Chemical Corporation
发明人： Kadkhodayan, Abbas , Ozbalik, Nubar
IPC分类号： C07D333/48 , C10M135/34
CPC分类号： C07D333/48 , C10M135/34 , C10M2219/102 , C10N2230/36 , C10N2240/042

70. 发明公开

EP2800470A4 SKIN LIGHTENING COMPOSITIONS 审中-公开
标题翻译：组合物美白肌肤
公开(公告)号：EP2800470A4
公开(公告)日：2015-11-04
申请号：EP13733800
申请日：2013-01-04
申请人： MERZ NORTH AMERICA INC
发明人： KVALNES KALLA LYNN , EWELL KEVIN R , DELONG MITCHELL A , WITWIT MOE , CHAMBOURNIER GILLES
IPC分类号： A01N43/04 , A61K8/34 , A61K8/41 , A61K8/49 , A61K31/70 , A61Q5/08 , A61Q19/02
CPC分类号： A61K8/602 , A61K8/347 , A61K8/41 , A61K8/4926 , A61K8/4973 , A61K8/498 , A61K8/4986 , A61Q5/08 , A61Q19/02 , C07C43/23 , C07D215/227 , C07D307/20 , C07D309/10 , C07D311/02 , C07D311/20 , C07D313/04 , C07D313/18 , C07D319/12 , C07D333/32 , C07D333/48 , C07D333/64 , C07D335/02 , C07D493/04 , C07H15/203

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