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1. 发明公开

EP3896058A3 ENANTIONSELECTIVE PROCESSES TO INSECTICIDAL 3-ARYL-3-TRIFLUOROMETHYL-SUBSTITUTED PYRROLIDINES 审中-公开
公开(公告)号：EP3896058A3
公开(公告)日：2022-01-12
申请号：EP21175826.3
申请日：2012-09-28
申请人： SYNGENTA PARTICIPATIONS AG
发明人： SMEJKAL, Tomas , SMITS, Helmars , WENDEBORN, Sebastian, Volker , BERTHON, Guillaume , CASSAYRE, Jérôme, Yves , EL QACEMI, Myriem
IPC分类号： C07D207/08 , C07D207/267 , C07D207/333 , C07D207/40 , C07D307/46 , C07D409/12
摘要： The present invention relates to processes for the enantio-selective preparation of spyrrolidine derivatives useful in the manufacture of pesticidally active compounds, as well as to intermedates in the processes. The processes include those comprising
(a-i) reacting a compound of formula Ia

wherein
P is alkyl, aryl or heteroaryl, each optionally substituted, wherein the heteroaryl is connected at P via a ring carbon atom;
R 1 is chlorodifluoromethyl or trifluoromethyl;
R 2 is aryl or heteroaryl, each optionally substituted;
with a source of cyanide in the presence a chiral catalyst to give a compound of formula IIa

wherein P, R 1 and R 2 are as defined for the compound of formula Ia; and
(a-ii) oxidising the compound of formula IIa with a peroxy acid, or peroxide in the presence of an acid to give a compound of formula VI

wherein R 1 and R 2 are as defined for the compound of formula Ia.

2. 发明公开

EP3692031A1 PESTICIDALLY ACTIVE PYRROLE DERIVATIVES 失效
公开(公告)号：EP3692031A1
公开(公告)日：2020-08-12
申请号：EP18782438.8
申请日：2018-10-04
申请人： Syngenta Participations AG
发明人： BIGOT, Aurelien , EL QACEMI, Myriem , GRIBKOV, Denis , STOLLER, André
IPC分类号： C07D401/14 , C07D403/04 , C07D409/14 , C07D413/04 , A01N43/56 , A01N43/80

3. 发明公开

EP3601275A1 INSECTICIDAL COMPOUNDS 无效
公开(公告)号：EP3601275A1
公开(公告)日：2020-02-05
申请号：EP18712896.2
申请日：2018-03-22
申请人： Syngenta Participations AG
发明人： CASSAYRE, Jérôme, Yves , EL QACEMI, Myriem , STOLLER, André
IPC分类号： C07D413/14 , A01N43/80 , C07D413/12 , C07D417/12

4. 发明授权

EP2709983B1 INSECTICIDAL COMPOUNDS BASED ON ARYLTHIOACETAMIDE DERIVATIVES 失效
标题翻译：基于芳基乙酰胺衍生物的杀虫活性化合物
公开(公告)号：EP2709983B1
公开(公告)日：2018-04-18
申请号：EP12720526.8
申请日：2012-05-15
申请人： Syngenta Participations AG
发明人： CASSAYRE, Jérôme Yves , EL QACEMI, Myriem , LUKSCH, Torsten , RENOLD, Peter
IPC分类号： C07D207/20 , C07D261/04 , A01N33/24 , A01N43/36
CPC分类号： C07D307/28 , A01N43/08 , A01N43/10 , A01N43/36 , A01N43/40 , A01N43/78 , A01N43/80 , C07D207/20 , C07D261/04 , C07D405/12 , C07D407/12 , C07D409/12 , C07D413/04 , C07D413/12 , C07D417/12
摘要： The present invention provides compounds of formula (I) wherein R1, R2, R3, R4, G1, n, A1, A2, A3, A4, Y1, Y2, and Y3 are as defined in the claims. The invention also relates to processes and intermediates for preparing these compounds, to insecticidal, acaricidal, nematicidal and molluscicidal compositions comprising these compounds and to methods of using these compounds to control insect, acarine, nematode and mollusc pests.

5. 发明授权

EP2445906B1 INSECTICIDAL COMPOUNDS 有权
公开(公告)号：EP2445906B1
公开(公告)日：2014-07-23
申请号：EP10726052.3
申请日：2010-06-11
申请人： Syngenta Participations AG , Syngenta Limited
发明人： RENOLD, Peter , CASSAYRE, Jérôme Yves , EL QACEMI, Myriem , PABBA, Jagadish , PITTERNA, Thomas
IPC分类号： C07D413/12 , C07D413/14 , C07D417/14 , A01N43/80 , C07D207/20 , C07D401/04 , C07D403/04 , C07D409/12 , C07D409/14 , A01N43/36 , A01N43/40
CPC分类号： C07D409/12 , A01N43/36 , C07D207/20 , C07D401/04 , C07D403/04 , C07D409/14 , C07F7/0812
摘要： The invention relates to compounds of formula (I) where A1, A2, A3, A4, G, R1, R2, R3 and R4 are as defined in claim 1; or a salt or JV-oxide thereof. Furthermore, the present invention relates to processes and intermediates for preparing compounds of formula (I), to insecticidal, acaricidal, nematicidal and molluscicidal compositions comprising the compounds of formula (I) and to methods of using the compounds of formula (I) to control insect, acarine, nematode and mollusc pests.

6. 发明公开

EP2748155A1 ISOXAZOLINE DERIVATIVES AS INSECTICIDAL COMPOUNDS 有权
标题翻译：异恶唑啉衍生物作为杀虫化合物
公开(公告)号：EP2748155A1
公开(公告)日：2014-07-02
申请号：EP12748717.1
申请日：2012-08-24
申请人： Syngenta Participations AG
发明人： CASSAYRE, Jérôme, Yves , RENOLD, Peter , PITTERNA, Thomas , EL QACEMI, Myriem
IPC分类号： C07D331/04 , C07D409/12 , C07D413/12 , A01N43/36 , A01N43/80
CPC分类号： A01N43/20 , A01N43/40 , A01N43/54 , A01N43/80 , C07D331/04 , C07D413/12
摘要： The present invention provides compounds of formula (I), wherein G
1 is oxygen; R
1 is hydrogen; R
2 is group P (P) L is a bond, methylene or ethylene; one of A
1 and A
2 is S, SO or SO
2 and the other is -C(R
4 )R
4 -R
3 is hydrogen or methyl; each R
4 is independently hydrogen or methyl; Y
1 is C-R
6 , CH or nitrogen; Y
2 and Y
3 are independently CH or nitrogen; wherein no more than two of Y
1 , Y
2 and Y
3 are nitrogen and wherein Y
2 and Y
3 are not both nitrogen; R
5 is hydrogen, halogen, cyano, nitro, NH
2 , C
1 -C
2 alkyl, C
1 -C
2 haloalkyl, C
3 -C
5 cycloalkyl, C
3 -C
5 halocycloalkyl, C
1 -C
2 alkoxy, C
1 -C
2 haloalkoxy; R
6 together with R
5 forms a -CH=CH-CH=CH- bridge; X
2 is C-X
6 or nitrogen; X
1 , X
3 and X
6 are independently hydrogen, halogen or trihalomethyl, wherein at least two of X
1 , X
3 and X
6 are not hydrogen; X
4 is trifluoromethyl, difluoromethyl or chlorodifluoromethyl. The invention also provides intermediates useful for the preparation of compounds of formula (I), as well as methods of controlling insects, acarines, nematodes or molluscs using the compounds of formula (I).
摘要翻译：本发明提供了式（I）的化合物，其中G 1是氧; R 1是氢; R 2是基团P（P）L是键，亚甲基或亚乙基; A 1和A 2中的一个是S，SO或SO 2，另一个是-C（R 4）R 4 -R 3是氢或甲基; 每个R 4独立地为氢或甲基; Y 1是C-R 6，CH或氮; Y 2和Y 3独立地为CH或氮; 其中Y 1，Y 2和Y 3中不多于两个是氮，并且其中Y 2和Y 3不都是氮; 卤素，氰基，硝基，NH 2，C 1 -C 2烷基，C 1 -C 2卤代烷基，C 3 -C 5环烷基，C 3 -C 5卤代环烷基，C 1 -C 2烷氧基，C 1 -C 2卤代烷氧基; R 6与R 5一起形成-CH = CH-CH = CH-桥; X 2是C-X 6或氮; X 1，X 3和X 6独立地为氢，卤素或三卤代甲基，其中X 1，X 3和X 6中的至少两个不是氢; X 4是三氟甲基，二氟甲基或氯二氟甲基。本发明还提供可用于制备式（I）化合物的中间体，以及使用式（I）化合物防治昆虫，螨，线虫或软体动物的方法。

7. 发明公开

EP2670248A2 METHODS OF PEST CONTROL IN SOYBEAN 审中-公开
标题翻译：方法大豆农药
公开(公告)号：EP2670248A2
公开(公告)日：2013-12-11
申请号：EP12703052.6
申请日：2012-02-01
申请人： Syngenta Participations AG , Syngenta Limited
发明人： VOCK, Christoph , CASSAYRE, Jérôme Yves , EL QACEMI, Myriem
IPC分类号： A01P7/04
CPC分类号： A01N43/80 , C07D231/06 , C07D261/04 , C07D413/12 , A01N2300/00
摘要： The present invention provides methods comprising applying to a crop of soybean plants, the locus thereof, or propagation material thereof, a compound a compound of formula III wherein A3, A4, A4' and A5' are independently C-H, or nitrogen and wherein #1 indicates the bond to X and #2 indicates the bond to cycle B; cycle B is selected from B1 to B6 wherein #1 indicates the bond to cycle A, #2 indicates the bond to R7 and #3 indicates the bond to cycle C; cycle C is phenyl; R5 is chloro, bromo, CF3 or methyl; R7 is chlorodifluoromethyl or trifluoromethyl; each R8 is independently bromo, chloro, fluoro or trifluoromethyl; p is 2 or 3; and wherein X is defined in the claims. The methods are preferably for the control of stinkbugs, in particular Euschistus.

8. 发明公开

EP2651220A1 PESTICIDAL MIXTURES 审中-公开
标题翻译：混配农药
公开(公告)号：EP2651220A1
公开(公告)日：2013-10-23
申请号：EP11801705.2
申请日：2011-12-15
申请人： Syngenta Participations AG
发明人： RENOLD, Peter , CASSAYRE, Jérôme Yves , EL QACEMI, Myriem , PABBA, Jagadish , PITTERNA, Thomas
IPC分类号： A01N43/36 , A01N43/40 , A01N43/90 , A01N57/16 , A01N43/56 , A01N53/00 , A01N43/707 , A01N47/06 , A01N51/00 , A01P9/00 , A01P7/04 , A01P7/02 , A01P7/00 , A01P5/00
CPC分类号： A01N43/36 , A01N43/40 , A01N2300/00 , A01N43/56 , A01N43/707 , A01N43/90 , A01N47/06 , A01N51/00 , A01N53/00 , A01N57/16
摘要： The present invention relates to pesticidal mixtures comprising a component A and a component B, wherein component A is a compound of formula I wherein one of Y
1 and Y
2 is S, SO or SO
2 and the other is CH
2 ; L is a direct bond or methylene; A
1 and A
2 are C-H, or one of A
1 and A
2 is C-H and the other is N; R
1 is hydrogen or methyl; R
2 is chlorodifluoromethyl or trifluoromethyl; R
3 is 3,5-dibromo-phenyl, 3,5-dichloro-phenyl, 3,4-dichloro-phenyl, or 3,4,5-trichloro- phenyl, 3,5-dichloro-4-fluoro-phenyl, or 3,5-bis-trifluoromethylphenyl; R
4 is methyl or chlorine; R
5 is hydrogen; or R
4 and R
5 together form a bridging 1,3-butadiene group; and wherein component B is an insecticide. The invention also relates to methods of controlling insects, acarines, nematodes or molluscs which comprises applying to a pest, to a locus of a pest, or to a plant susceptible to attack by a pest a combination of components A and B.

9. 发明授权

EP2331515B1 INSCETICIDAL COMPOUNDS 无效
标题翻译： INSCETICIDAL化合物
公开(公告)号：EP2331515B1
公开(公告)日：2013-07-10
申请号：EP09781036.0
申请日：2009-07-24
申请人： Syngenta Participations AG , Syngenta Limited
发明人： PITTERNA, Thomas , EL QACEMI, Myriem , BOBOSIK, Vladimir , RENOLD, Peter , CASSAYRE, Jérôme, Yves , JUNG, Pierre, Joseph, Marcel.
IPC分类号： C07D261/02 , C07D413/12 , A01N43/80 , A61P29/00
CPC分类号： C07D261/02 , A01N43/80 , C07D413/12

10. 发明公开

EP3606918A1 PESTICIDALLY ACTIVE PYRAZOLE DERIVATIVES 审中-实审转让
公开(公告)号：EP3606918A1
公开(公告)日：2020-02-12
申请号：EP18717876.9
申请日：2018-04-04
申请人： Syngenta Participations AG
发明人： EL QACEMI, Myriem , BIGOT, Aurelien , EDMUNDS, Andrew , GAGNEPAIN, Julien, Daniel, Henri , JEANGUENAT, André , PITTERNA, Thomas , STOLLER, André , SABBADIN, Davide , MONDIERE, Régis, Jean, Georges , GRIBKOV, Denis
IPC分类号： C07D409/14 , A01N43/10 , A01N43/36

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