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1. 发明授权

US6060485A Arylacetic amide derivative or salt thereof, and pharmaceutical comprising it 失效
标题翻译：芳酰乙酰胺衍生物或其盐，以及包含它的药物
公开(公告)号：US6060485A
公开(公告)日：2000-05-09
申请号：US181091
申请日：1998-10-28
申请人： Terumitsu Kaihoh , Tomomi Okada , Yoshinori Takahashi , Hiroyuki Mizuno , Haruyoshi Honda , Susumu Sato
发明人： Terumitsu Kaihoh , Tomomi Okada , Yoshinori Takahashi , Hiroyuki Mizuno , Haruyoshi Honda , Susumu Sato
IPC分类号： C07D211/58 , C07D211/94 , C07D401/12 , A61K31/445
CPC分类号： C07D401/12 , C07D211/58 , C07D211/94
摘要： Described is an arylacetic amide derivative represented by the following formula (1): ##STR1## wherein R.sup.1 represents an aryl group or the like, R.sup.2 and R.sup.3 each independently represents an alkyl group, a cycloalkyl group or the like, and R.sup.4 represents an aralkyl group, an alkyl group or the like; or salt thereof. The compound according to the present invention has both excellent anticholinergic action and calcium antagonism and at the same time has high selectivity to bladder, so that it is useful as a preventive or remedy for urinary disorders.
摘要翻译：描述了由下式（1）表示的芳基乙酰胺衍生物：其中R 1表示芳基等，R 2和R 3各自独立地表示烷基，环烷基等，R 4表示芳烷基，烷基等; 或其盐。根据本发明的化合物具有优异的抗胆碱能作用和钙拮抗作用，同时对膀胱具有高选择性，因此可用作尿障碍的预防或治疗方法。

2. 发明授权

US06174900B1 Substituted piperidine derivative for treating urinary disturbance 失效
标题翻译：用于治疗尿失禁的替代哌啶衍生物
公开(公告)号：US06174900B1
公开(公告)日：2001-01-16
申请号：US09332444
申请日：1999-06-14
申请人： Tomomi Okada , Fujiko Konno , Terumitsu Kaihoh , Masago Ishikawa , Yoshinori Takahashi , Hiroyuki Mizuno , Haruyoshi Honda , Susumu Sato , Hideaki Matsuda
发明人： Tomomi Okada , Fujiko Konno , Terumitsu Kaihoh , Masago Ishikawa , Yoshinori Takahashi , Hiroyuki Mizuno , Haruyoshi Honda , Susumu Sato , Hideaki Matsuda
IPC分类号： A61K31445
CPC分类号： C07D401/12 , C07D211/58 , C07D409/12
摘要： Disclosed herein is a substituted piperidine derivative represented by the following general formula (1): wherein R1 means an aryl or heteroaryl group which may have at least one substituent, R2 denotes an alkyl, alkenyl or aralkyl group, R3 stands for a hydrogen atom or an alkyl group, and R4 is a hydrogen atom, an alkyl group, or an aryl, heteroaryl, aralkyl, aralkenyl or heteroaralkyl group which may have at least one substituent, or a salt thereof. A medicine including this compound is also disclosed. The compound has excellent anticholinergic effect and calcium antagonism and inhibits reflex bladder contraction and is hence useful for prophylaxis of and treatment for a urinary disturbance such as pollakiuria.
摘要翻译：本文公开了由以下通式（1）表示的取代的哌啶衍生物：其中R 1表示可具有至少一个取代基的芳基或杂芳基，R 2表示烷基，烯基或芳烷基，R 3表示氢原子或烷基，可以具有至少一个取代基的芳基，杂芳基，芳烷基，芳烯基或杂芳烷基，或其盐。还公开了包含该化合物的药物。该化合物具有优异的抗胆碱能作用和钙拮抗作用并抑制反射膀胱收缩，因此可用于预防和治疗尿频紊乱如尿频。

3. 发明授权

US5968956A Substituted piperidine derivative and medicine comprising the same 失效
标题翻译：取代的哌啶衍生物及含有它们的药物
公开(公告)号：US5968956A
公开(公告)日：1999-10-19
申请号：US672058
申请日：1996-06-26
申请人： Tomomi Okada , Fujiko Konno , Terumitsu Kaihoh , Masago Ishikawa , Yoshinori Takahashi , Hiroyuki Mizuno , Haruyoshi Honda , Susumu Sato , Hideaki Matsuda
发明人： Tomomi Okada , Fujiko Konno , Terumitsu Kaihoh , Masago Ishikawa , Yoshinori Takahashi , Hiroyuki Mizuno , Haruyoshi Honda , Susumu Sato , Hideaki Matsuda
IPC分类号： C07D211/58 , C07D401/12 , C07D409/12 , A61K31/445 , C07D211/56
CPC分类号： C07D401/12 , C07D211/58 , C07D409/12
摘要： Disclosed herein is a substituted piperidine derivative represented by the following general formula (1): ##STR1## wherein R.sup.1 means an aryl or heteroaryl group which may have at least one substituent, R.sup.2 denotes an alkyl, alkenyl or aralkyl group, R.sup.3 stands for a hydrogen atom or an alkyl group, and R.sup.4 is a hydrogen atom, an alkyl group, or an aryl, heteroaryl, aralkyl, aralkenyl or heteroaralkyl group which may have at least one substituent, or a salt thereof. A medicine including this compound is also disclosed. The compound has excellent anticholinergic effect and calcium antagonism and inhibits reflex bladder contraction and is hence useful for prophylaxis of and treatment for a urinary disturbance such as pollakiuria.
摘要翻译：本文公开了由以下通式（1）表示的取代的哌啶衍生物：其中R 1表示可具有至少一个取代基的芳基或杂芳基，R 2表示烷基，烯基或芳烷基，R 3表示氢原子或烷基，可以具有至少一个取代基的芳基，杂芳基，芳烷基，芳烯基或杂芳烷基，或其盐。还公开了包含该化合物的药物。该化合物具有优异的抗胆碱能作用和钙拮抗作用并抑制反射膀胱收缩，因此可用于预防和治疗尿频紊乱如尿频。

4. 发明授权

US07214672B2 Preventives/remedies for inflammatory airway diseases 有权
标题翻译：炎症性气道疾病的预防/补救措施
公开(公告)号：US07214672B2
公开(公告)日：2007-05-08
申请号：US10451061
申请日：2001-12-21
申请人： Teruo Komoto , Hiroyuki Mizuno , Yoshinori Takahashi , Koichi Takahashi , Susumo Sato
发明人： Teruo Komoto , Hiroyuki Mizuno , Yoshinori Takahashi , Koichi Takahashi , Susumo Sato
IPC分类号： A61K31/56 , A61K31/58
CPC分类号： C07J5/00 , A61K31/57 , A61K31/573 , C07J7/00
摘要： A preventive and/or therapeutic agent for inflammatory respiratory tract diseases containing, as an active ingredient, a steroid derivative represented by the following formula (1): (wherein R represents a hydrogen atom, a halogen atom, a hydroxy group, or —OCOR1 (wherein R1 represents a linear or branched alkyl group which may be substituted by a halogen atom or a cycloalkyl group; a cycloalkyl group; or an aryl group)). These compounds can continuously suppress respiratory tract inflammation and respiratory tract hyperreaction and show a high site selectivity and little systemic effect when administered directly to the respiratory tract. By virtue of these characteristics, these compounds are remarkably useful in clinical medicine as highly safe preventive and/or therapeutic agents for inflammatory respiratory tract diseases which can be administered for a long period of time.
摘要翻译：一种炎性呼吸道疾病的预防和/或治疗剂，含有下式（1）表示的类固醇衍生物作为活性成分：（式中，R表示氢原子，卤素原子，羟基或-OCOR （其中R 1表示可被卤素原子或环烷基取代的直链或支链烷基;环烷基;或芳基））。这些化合物可以连续抑制呼吸道炎症和呼吸道高反应，并且当直接施用于呼吸道时显示出高的选择性和很小的全身效应。由于这些特征，这些化合物在临床医学中非常有用，作为可长期施用的炎症性呼吸道疾病的高度安全的预防和/或治疗剂。

5. 发明申请

US20140376434A1 START SIGNAL GENERATING APPARATUS 有权
标题翻译：开始信号发生装置
公开(公告)号：US20140376434A1
公开(公告)日：2014-12-25
申请号：US14369028
申请日：2013-02-25
申请人： Akihito Hirai , Yoshinori Takahashi , Eiji Taniguchi
发明人： Akihito Hirai , Yoshinori Takahashi , Eiji Taniguchi
IPC分类号： H04W52/02
CPC分类号： H04W52/0225 , H04B1/16 , H04B17/318 , H04W52/0229 , H04W52/0245 , Y02D70/142 , Y02D70/40
摘要： Besides a time constant circuit 5 that imposes a frequency limit on a wireless signal detected by a power detecting circuit 4 at a preset time constant Ta, there is provided a time constant circuit 8 that imposes a frequency limit on the wireless signal at a time constant Tb greater than the time constant Ta. When the signal level of an intermittent operation signal supplied from a signal input terminal 1 is H level or when a threshold processing circuit 6 decides that the level of the wireless signal is higher than a threshold Th, a logic unit 3 supplies a control signal that instructs starting to the power detecting circuit 4, time constant circuits 5 and 8 and threshold processing circuits 6 and 9.
摘要翻译：除了在预设时间常数Ta对由功率检测电路4检测到的无线信号施加频率限制的时间常数电路5之外，还提供了时间常数电路8，其以时间常数对无线信号施加频率限制 Tb大于时间常数Ta。当从信号输入端子1提供的间歇操作信号的信号电平为H电平时，或者当阈值处理电路6判定无线信号的电平高于阈值Th时，逻辑单元3提供控制信号指示开始到功率检测电路4，时间常数电路5和8以及阈值处理电路6和9。

6. 发明授权

US08914068B2 Array antenna apparatus 有权
标题翻译：阵列天线装置
公开(公告)号：US08914068B2
公开(公告)日：2014-12-16
申请号：US13581507
申请日：2011-02-22
申请人： Ryoji Hayashi , Yoshihito Hirano , Kiyohide Sakai , Mitsuhiro Shimozawa , Akira Inoue , Morishige Hieda , Hiroyuki Joba , Kenichi Tajima , Yoshinori Takahashi , Kazutomi Mori , Tomohiro Akiyama
发明人： Ryoji Hayashi , Yoshihito Hirano , Kiyohide Sakai , Mitsuhiro Shimozawa , Akira Inoue , Morishige Hieda , Hiroyuki Joba , Kenichi Tajima , Yoshinori Takahashi , Kazutomi Mori , Tomohiro Akiyama
IPC分类号： H04M1/00 , H01Q3/42 , H04B17/00 , H01Q3/30 , H01Q21/00
CPC分类号： H01Q3/42 , H01Q3/30 , H01Q21/0025 , H04B17/0085
摘要： An array antenna apparatus in which an SN ratio is improved. Antenna elements having transmission modules, respectively, are arranged in plurality, wherein the plurality of transmission modules respectively have transmission signal generators that each output a transmission intermediate frequency signal, local oscillation signal generators that each output a local oscillation signal, and transmission mixers that each mix the transmission intermediate frequency signal and the local oscillation signal with each other, thereby to carry out frequency conversion to a transmission high frequency signal. A reference signal source inputs a reference signal to the transmission signal generators and the local oscillation signal generators. The transmission intermediate frequency signal and the local oscillation signal are synchronized with each other by the reference signal.
摘要翻译：提高SN比的阵列天线装置。分别具有发送模块的天线元件分别配置有多个发送模块，其中，所述多个发送模块分别具有各自输出发送中频信号的发送信号发生器，各自输出本地振荡信号的本地振荡信号发生器以及各自输出本地振荡信号的发送混频器将发送中频信号和本地振荡信号彼此混合，从而对发送高频信号进行频率转换。参考信号源将参考信号输入到发送信号发生器和本地振荡信号发生器。发送中频信号和本地振荡信号通过参考信号彼此同步。

7. 发明授权

US08774737B2 Transmission module and phased array antenna apparatus 失效
标题翻译：传输模块和相控阵天线装置
公开(公告)号：US08774737B2
公开(公告)日：2014-07-08
申请号：US13582237
申请日：2010-03-04
申请人： Kazutomi Mori , Hiroyuki Joba , Yoshinori Takahashi , Tomohiro Akiyama , Ryoji Hayashi , Mitsuhiro Shimozawa , Akira Inoue , Morishige Hieda , Kiyohide Sakai , Yoshihito Hirano
发明人： Kazutomi Mori , Hiroyuki Joba , Yoshinori Takahashi , Tomohiro Akiyama , Ryoji Hayashi , Mitsuhiro Shimozawa , Akira Inoue , Morishige Hieda , Kiyohide Sakai , Yoshihito Hirano
IPC分类号： H04B1/04 , H01Q11/12 , H03F1/32 , H03F1/02 , H03G3/00 , H03G3/30
CPC分类号： H03F1/3247 , H01Q3/26 , H01Q3/267 , H03F1/02 , H03F1/0211 , H03F1/0227 , H03F1/0238 , H03F3/24 , H03F2200/211 , H03F2200/411 , H03F2200/451 , H03G3/004 , H03G3/3042 , H04B1/0483 , H04B17/13 , H04B2001/045
摘要： A transmission module including a power supply voltage control unit that sets a power supply voltage to the high frequency amplifier in a variable manner, and a control circuit that controls an amplitude control unit, a phase control unit and the power supply voltage control unit. The control circuit and the power supply voltage control unit control the power supply voltage in accordance with an output power of the high frequency amplifier. The transmission module can carry out not only phase control but also amplitude control in a continuous manner, while suppressing amplitude and phase variation, and a high frequency amplifier in the transmission module is made highly efficient. In addition, a large directional gain, a low side lobe level and a low power consumption are achieved, as a phased array antenna apparatus using a transmission module.
摘要翻译：一种传输模块，包括以可变方式设置高频放大器的电源电压的电源电压控制单元和控制振幅控制单元，相位控制单元和电源电压控制单元的控制电路。控制电路和电源电压控制单元根据高频放大器的输出功率来控制电源电压。传输模块不仅可以在抑制幅度和相位变化的同时进行相位控制，而且可以连续进行幅度控制，并且使传输模块中的高频放大器高效。此外，作为使用传输模块的相控阵天线装置，实现了大的方向增益，低旁瓣电平和低功耗。

8. 发明授权

US08530504B2 Pyrazolothiazole compound 失效
标题翻译：吡唑并噻唑化合物
公开(公告)号：US08530504B2
公开(公告)日：2013-09-10
申请号：US12900026
申请日：2010-10-07
申请人： Kogyoku Shin , Taro Terauchi , Yoshinori Takahashi , Minako Hashizume , Kunitoshi Takeda , Kodo Shikata , Akira Inomata
发明人： Kogyoku Shin , Taro Terauchi , Yoshinori Takahashi , Minako Hashizume , Kunitoshi Takeda , Kodo Shikata , Akira Inomata
IPC分类号： A61K31/429 , A61P25/24
CPC分类号： C07D513/04
摘要： A compound represented by the formula (I) or pharmacologically acceptable salt thereof exhibits an excellent CRF receptor antagonism wherein X is a nitrogen atom or CH; R1 is -A11-A12; A11 is a single bond or a C1-6 alkylene group; A12 is a hydrogen atom, a C1-6 alkyl group or a C3-6 cycloalkyl group, etc.; R2 is -A21-A22; A21 is a single bond or a C1-6 alkylene group; A22 is a hydrogen atom, a C1-6 alkyl group, a C3-6 cycloalkyl group, a non-aromatic heterocyclic group, or a heteroaryl group, etc.; R3 is a C1-6 alkyl group, a C3-6 cycloalkyl group, a C1-6 alkoxy group, a C3-6 cycloalkoxy C1-6 alkyl group, di-C1-6 alkyl amino group, a halogen atom, a cyano group, a formyl group, or a carboxyl group, etc; R4 is a hydrogen atom or a C1-6 alkoxy group; R5 is a halogen atom, a C1-6 alkyl group, or a C1-6 alkoxy group; R6 is a hydrogen atom, a C1-6 alkyl group, a C1-6 alkoxy group, a C1-6 alkylthio group, or a C1-6 alkyl sulfinyl group etc.; and R7 is a C1-6 alkyl group, a C1-6 alkoxy group, or a C1-6 alkylthio group.
摘要翻译：由式（I）表示的化合物或其药理学上可接受的盐表现出优异的CRF受体拮抗作用，其中X为氮原子或CH; R1为-A11-A12; A11是单键或C1-6亚烷基; A12是氢原子，C1-6烷基或C3-6环烷基等; R2为-A21-A22; A21是单键或C1-6亚烷基; A22为氢原子，C1-6烷基，C3-6环烷基，非芳族杂环基或杂芳基等; R3是C1-6烷基，C3-6环烷基，C1-6烷氧基，C3-6环烷氧基C1-6烷基，二C1-6烷基氨基，卤素原子，氰基，甲酰基或羧基等; R4是氢原子或C1-6烷氧基; R5是卤素原子，C1-6烷基或C1-6烷氧基; R6是氢原子，C1-6烷基，C1-6烷氧基，C1-6烷硫基或C1-6烷基亚磺酰基等; 且R 7为C 1-6烷基，C 1-6烷氧基或C 1-6烷硫基。

9. 发明申请

US20120326781A1 TRANSMISSION MODULE AND PHASED ARRAY ANTENNA APPARATUS 失效
标题翻译：传输模块和相位阵列天线装置
公开(公告)号：US20120326781A1
公开(公告)日：2012-12-27
申请号：US13582237
申请日：2010-03-04
申请人： Kazutomi Mori , Hiroyuki Joba , Yoshinori Takahashi , Tomohiro Akiyama , Ryoji Hayashi , Mitsuhiro Shimozawa , Akira Inoue , Morishige Hieda , Kiyohide Sakai , Yoshihito Hirano
发明人： Kazutomi Mori , Hiroyuki Joba , Yoshinori Takahashi , Tomohiro Akiyama , Ryoji Hayashi , Mitsuhiro Shimozawa , Akira Inoue , Morishige Hieda , Kiyohide Sakai , Yoshihito Hirano
IPC分类号： H03G3/20
CPC分类号： H03F1/3247 , H01Q3/26 , H01Q3/267 , H03F1/02 , H03F1/0211 , H03F1/0227 , H03F1/0238 , H03F3/24 , H03F2200/211 , H03F2200/411 , H03F2200/451 , H03G3/004 , H03G3/3042 , H04B1/0483 , H04B17/13 , H04B2001/045
摘要： A transmission module including a power supply voltage control unit that sets a power supply voltage to the high frequency amplifier in a variable manner, and a control circuit that controls an amplitude control unit, a phase control unit and the power supply voltage control unit. The control circuit and the power supply voltage control unit control the power supply voltage in accordance with an output power of the high frequency amplifier. The transmission module can carry out not only phase control but also amplitude control in a continuous manner, while suppressing amplitude and phase variation, and a high frequency amplifier in the transmission module is made highly efficient. In addition, a large directional gain, a low side lobe level and a low power consumption are achieved, as a phased array antenna apparatus using a transmission module.
摘要翻译：一种传输模块，包括以可变方式设置高频放大器的电源电压的电源电压控制单元和控制振幅控制单元，相位控制单元和电源电压控制单元的控制电路。控制电路和电源电压控制单元根据高频放大器的输出功率来控制电源电压。传输模块不仅可以在抑制幅度和相位变化的同时进行相位控制，而且可以连续进行幅度控制，并且使传输模块中的高频放大器高效。此外，作为使用传输模块的相控阵天线装置，实现了大的方向增益，低旁瓣电平和低功耗。

10. 发明申请

US20100283177A1 PROCESS FOR PRODUCING PRECURSOR FILM FOR RETARDATION FILM MADE OF POLYPROPYLENE RESIN 审中-公开
标题翻译：生产用于聚丙烯树脂延伸膜的前置膜的方法
公开(公告)号：US20100283177A1
公开(公告)日：2010-11-11
申请号：US12679079
申请日：2008-09-18
申请人： Hiroaki Takahata , Yoshinori Takahashi , Kyoko Hino , Yoshiaki Ishigami , Shuji Ozaki , Shuji Fujioka
发明人： Hiroaki Takahata , Yoshinori Takahashi , Kyoko Hino , Yoshiaki Ishigami , Shuji Ozaki , Shuji Fujioka
IPC分类号： B29C47/52
CPC分类号： B29C48/9155 , B29C48/08 , B29C48/914
摘要： There is provided a process for producing a precursor film for a polypropylene-based resin retardation film that can yield films with almost no orientation and with high transparency.The process for producing a precursor film for a polypropylene-based resin retardation film comprises a step of pressing a molten sheet formed by extruding a molten polypropylene-based resin from a T-shaped die 12 at 180° C. or higher and 300° C. or lower between a cooling roll 16 having a surface temperature regulated to −5° C. or higher and 30° C. or lower and a touch roll 14 having a surface temperature regulated to 80° C. or higher and 150° C. or lower, whereby the molten sheet is cooled and solidified.
摘要翻译：提供了一种用于制造聚丙烯基树脂延迟膜的前体膜的方法，其可以产生几乎没有取向和高透明度的膜。制造聚丙烯类树脂延迟膜用前体膜的方法包括：将来自T型模具12的熔融聚丙烯类树脂挤出成形为180℃以上且300℃以下的熔融片材的工序在表面温度调节为-5℃以上且30℃以下的冷却辊16和表面温度调节为80℃以上且150℃以下的接触辊14之间或之下。或更低，由此熔融的片材被冷却和固化。

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