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1. 发明申请

WO2009007098A1 ISOTHIAZOLE AND PYRAZOLE DERIVATIVES AS FUNGICIDES 审中-公开
标题翻译：异噻唑和吡唑衍生物作为杀真菌剂
公开(公告)号：WO2009007098A1
公开(公告)日：2009-01-15
申请号：PCT/EP2008005589
申请日：2008-07-09
申请人： SYNGENTA PARTICIPATIONS AG , ACKERMANN PETER , BOBBIO CARLA , CORSI CAMILLA , EHRENFREUND JOSEF , MCGINLEY ANN MONICA , VERRAS ANDREAS , TITULAER RUUD
发明人： ACKERMANN PETER , BOBBIO CARLA , CORSI CAMILLA , EHRENFREUND JOSEF , MCGINLEY ANN MONICA , VERRAS ANDREAS , TITULAER RUUD
IPC分类号： C07D401/06 , A01N43/40 , A01N43/54 , C07D417/06 , C07D417/14
CPC分类号： C07D417/06 , A01N43/56 , A01N43/80 , C07D401/06 , C07D417/14
摘要： The present invention relates to compounds of Formula (I) wherein R1, R2, R3 or R4 are as defined in claim 1 or a salt or N-oxide thereof and their use in methods for the control and/or prevention of fungal infection, particularly in plants. The compounds claimed are isothiazole and pyrazole derivatives.
摘要翻译：本发明涉及其中R 1，R 2，R 3或R 4如权利要求1所定义的式（I）化合物或其盐或N-氧化物及其在控制和/或预防真菌感染的方法中的用途，特别是在植物中。所要求的化合物是异噻唑和吡唑衍生物。

2. 发明申请

WO2008155081A3 SUBSTITUTED AROMATIC HETEROCYCLIC COMPOUNDS AS FUNGICIDES 审中-公开
标题翻译：取代的芳香杂环化合物作为防腐剂
公开(公告)号：WO2008155081A3
公开(公告)日：2009-05-07
申请号：PCT/EP2008004831
申请日：2008-06-16
申请人： SYNGENTA PARTICIPATIONS AG , ACKERMANN PETER , BOBBIO CARLA , CORSI CAMILLA , EHRENFREUND JOSEF , MCGINLEY ANN MONICA
发明人： ACKERMANN PETER , BOBBIO CARLA , CORSI CAMILLA , EHRENFREUND JOSEF , MCGINLEY ANN MONICA
IPC分类号： C07D401/06 , A61K31/4025 , A61P43/00 , C07D403/06 , C07D405/14 , C07D409/14
CPC分类号： C07D401/06 , C07D403/06 , C07D405/14 , C07D409/14
摘要： The present invention relates to compounds of formula (I) wherein R1, R2, R3, R4, R5 and R6 are as defined in claim 1 or a salt or N-oxide thereof and their use in methods for the control and/or prevention of fungal infection, particularly in plants.
摘要翻译：本发明涉及其中R 1，R 2，R 3，R 4，R 5和R 6如权利要求1中所定义的式（I）化合物或其盐或N-氧化物及其在控制和/或预防真菌感染，特别是在植物中。

3. 发明申请

WO2007124907A3 HETEROCYCLYL-CARBOXYLIC ACID (BENZONORBORNENE-5-YL)AMIDE DERIVATIVES AS FUNGICIDES FOR AGROCHEMICAL USE 审中-公开
标题翻译：作为农药使用的间苯二酚 - 羧酸（苯并呋喃-5-基）酰胺衍生物
公开(公告)号：WO2007124907A3
公开(公告)日：2008-01-10
申请号：PCT/EP2007003653
申请日：2007-04-25
申请人： SYNGENTA PARTICIPATIONS AG , TOBLER HANS , CORSI CAMILLA , EHRENFREUND JOSEF , WALTER HARALD
发明人： TOBLER HANS , CORSI CAMILLA , EHRENFREUND JOSEF , WALTER HARALD
IPC分类号： C07D231/14 , A01N43/56
CPC分类号： C07D207/34 , C07C205/06 , C07C205/11 , C07C205/12 , C07C211/61 , C07C2602/42 , C07D231/14
摘要： The invention relates to fungicidally active compounds of formula (I): wherein Het, R 1 , R 2 , R 3 , R 4 , R 5 , R 6 , R 7 , R 8 and R 9 are as defined in claim 1, to the preparation of these compounds, to novel intermediates used in the preparation of these compounds, to agrochemical compositions which comprise at least one of the novel compounds as active ingredient, to the preparation of the compositions mentioned and to the use of the active ingredients or compositions in agriculture or horticulture for controlling or preventing infestation of plants by phytopathogenic microorganisms, preferably fungi.
摘要翻译：本发明涉及式（I）的杀真菌活性化合物：其中Het，R 1，R 2，R 3，R 3， R 4，R 5，R 6，R 7，R 8和R 8， 9，如权利要求1中所定义，涉及这些化合物的制备，用于制备这些化合物的新型中间体，其包含至少一种新化合物作为活性成分的农药组合物，所提及的组合物以及在农业或园艺中使用活性成分或组合物来控制或预防植物病原微生物，优选真菌侵染植物。

4. 发明申请

WO2007068417A3 PROCESS FOR THE PREPARATION OF AMINES 审中-公开
标题翻译：制备氨基酸的方法
公开(公告)号：WO2007068417A3
公开(公告)日：2007-10-04
申请号：PCT/EP2006011885
申请日：2006-12-11
申请人： SYNGENTA PARTICIPATIONS AG , TOBLER HANS , WALTER HARALD , CORSI CAMILLA , EHRENFREUND JOSEF , GIORDANO FANNY , ZELLER MARTIN
发明人： TOBLER HANS , WALTER HARALD , CORSI CAMILLA , EHRENFREUND JOSEF , GIORDANO FANNY , ZELLER MARTIN
IPC分类号： C07C209/28 , A01N45/02 , C07C211/31
CPC分类号： C07C209/62 , C07B2200/09 , C07C17/23 , C07C17/30 , C07C17/354 , C07C25/22 , C07C25/24 , C07C209/10 , C07C209/70 , C07C211/61 , C07C2603/66 , C07C23/10
摘要： The present invention relates to a novel a process for the preparation of the compound of the general formula (I), wherein R 1 and R 2 are independently H or C 1-6 alkyl, which comprises treating with a reducing agent either a compound of the general formula (II), wherein R 1 and R 2 have the meanings given for the compound of the formula (I), R 3 is H or C 1-4 alkyl and Ph is phenyl, or a compound of the general formula (III), wherein R 1 , R 2 , R 3 and Ph have the meanings given for the compound of the formula (II), the reducing agent being effective to cleave the benzyl moiety Ph-CH(R 3 )- from the benzylamino moiety PhCH(R 3 )NH- in the compound of the formula (II) or in the compound of the formula (III) to leave an amino group and, in addition, in the case of the compound of the formula (III), to reduce both the 2,3-double bond and the double bond joining the R 1 R 2 C- moiety to the 9-position of the benzonorbornene ring to single bonds. It also relates to processes for the preparation of the compounds (II) and (III) and their precursors and to the compounds (II) and (III) themselves and certain of their precursors, which are novel compounds. The compounds (I) are useful for the preparation of various fungicidal heterocyclyl-carboxylic acid benzonorbornen-5-yl-amides.
摘要翻译：本发明涉及一种制备通式（I）化合物的新方法，其中R 1和R 2独立地为H或C _{1 C-C部分到苯并降冰片烯环的9-位到单键。它还涉及制备化合物（II）和（III）及其前体以及化合物（II）和（III）本身及其某些新型化合物的前体的方法。化合物（I）可用于制备各种杀真菌性杂环基 - 羧酸苯并降冰片烯-5-基 - 酰胺。}

5. 发明申请

WO2007057138A3 PROCESS FOR THE PRODUCTION OF BIPHENYLS 审中-公开
标题翻译：生产联苯的方法
公开(公告)号：WO2007057138A3
公开(公告)日：2007-08-09
申请号：PCT/EP2006010864
申请日：2006-11-13
申请人： SYNGENTA PARTICIPATIONS AG , EHRENFREUND JOSEF , WALTER HARALD , TOBLER HANS , CORSI CAMILLA
发明人： EHRENFREUND JOSEF , WALTER HARALD , TOBLER HANS , CORSI CAMILLA
IPC分类号： C07C201/12 , A01N55/00 , C07C25/18
CPC分类号： C07C201/12 , C07C2601/02 , C07C205/06 , C07C205/11 , C07C205/19 , C07C205/34 , C07C205/42 , C07C205/56
摘要： The present invention relates to a novel process for the preparation of a compound of formula (I): which comprises reacting a compound of formula (II): with a compound of general formula (III): wherein R 1 and R 2 are H or C 1-4 alkyl or R 1 and R 2 join together to form a C 2-3 alkylene group, which is optionally substituted by from 1 to 4 methyl or ethyl groups, or an anhydride of the compound (III), in the presence of a base and of a palladium catalyst which is (a) a palladium (0)- or palladium (I?)-triarylphosphine complex optionally in the presence of additional amounts of a triarylphoshine ligand, or (b) a palladium (II) salt in the presence of a triarylphosphine ligand, or (c) metallic palladium, optionally deposited on a support, in the presence of triarylphosphine; there being used from 0.9 to 2 moles of compound (III) for each mole of compound (II).
摘要翻译：本发明涉及制备式（I）化合物的新方法：其包括使式（II）化合物：与通式（III）化合物反应：其中R 1 = SUP 和R 2是H或C 1-4烷基或R 1和R 2连接在一起形成任选被1至4个甲基或乙基取代的C 2-3亚烷基或化合物（III）的酸酐在碱和钯催化剂存在下反应（a）在三芳基膦配体存在下任选存在额外量的三芳基膦配体或（b）钯（II）盐的情况下，钯（0） - 或钯（I +） - 三芳基膦络合物，或（c）在三芳基膦存在下任选沉积在载体上的金属钯; 每摩尔化合物（II）使用0.9-2摩尔化合物（III）。

6. 发明申请

WO2004018438A3 MICROBIOCIDAL (E.G. FUNGICIDAL) 1,2,3-TRIAZOLE DERIVATIVES 审中-公开
标题翻译： MICROBIOCIDAL（E.G. Fungicidal）1,2,3-三唑衍生物
公开(公告)号：WO2004018438A3
公开(公告)日：2004-08-26
申请号：PCT/EP0309111
申请日：2003-08-18
申请人： SYNGENTA PARTICIPATIONS AG , EHRENFREUND JOSEF , TOBLER HANS , WALTER HARALD
发明人： EHRENFREUND JOSEF , TOBLER HANS , WALTER HARALD
IPC分类号： A01N43/647 , A01N55/00 , C07D249/04 , C07D333/36 , C07D401/12 , C07D405/12 , C07D409/12 , C07D409/14 , C07D411/12 , C07D413/12 , C07D417/12 , C07D487/08 , C07D493/08 , C07D495/08 , C07D209/94 , C07D307/00 , C07D403/12
CPC分类号： C07D401/12 , A01N43/647 , A01N55/00 , C07D249/04 , C07D333/36 , C07D405/12 , C07D409/12 , C07D409/14 , C07D411/12 , C07D413/12 , C07D417/12 , C07D487/08 , C07D493/08 , C07D495/08
摘要： A compound of formula (1):where A is an ortho-substituted ring selected from a number of specified rings; R is halogen, cyano, nitro, C 1-4 alkyl, C 1-4 haloalkyl, C 1-4 alkoxy or C 1-4 haloalkoxy or optionally substituted C 2-4 alkenyl, optionally substituted C 2-4 alkynyl or optionally substituted SO2(C 1-4)alkyl (where the optionally substituted moieties may each have up to 3 substituents, each independently selected from halogen and C 1-4 alkoxy); R is C 1-4 alkyl, C 1-4 haloalkyl, C 1-4 alkoxy(C 1-4)alkyl or C 1-4 alkyltbio(C 1-4)alkyl or [optionally substituted aryl](C 1-4)alkyl- or [optionally substituted aryl]oxy(C l-4)a1kyl(where the optionally substituted aryl moieties may each have up to 3 substituents, each independently selected from halogen and C 1-4 alkoxy); R 3 is hydrogen, CH2C =CR , CH2CR =C(H)R , CH=C=CH2 or COR or optionally substituted C 1-4 alkyl, optionally substituted C 1-4 alkoxy or optionally substituted (C I-4) alkylC(=O)O (where the optionally substituted moieties may each have up to 3 substituents, each independently selected from halogen and C 1-4 alkoxy, C 1-4 alkyl, C 1-2 haloalkoxy, bydroxy, cyano, carboxyl, methoxycarbonyl, ethoxycarbonyl, methylsulfonyl and ethylsulfonyl), The compound of Formula (I) have microbiocidal activity, in particular fungicidal activity.
摘要翻译：式（1）的化合物：其中A是选自多个指定环的邻位取代的环; R 1是卤素，氰基，硝基，C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基或C 1-4卤代烷氧基或任选取代的C 2-4链烯基，任选取代的C 2-4炔基或任选取代的SO 2（C 1-4）烷基（其中任选取代的部分各自可具有至多3个取代基，各自独立地选自卤素和C 1-4烷氧基）; R 2是C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基（C 1-4）烷基或C 1-4烷基二（C 1-4）烷基或[任选取代的芳基]（C 1-4）烷基 - 或[任选取代的芳基]氧基（C 1-4）烷基（其中任选取代的芳基部分可各自具有至多3个取代基，各自独立地选自卤素和C 1-4烷氧基）; R 3是氢，CH 2 C = CR 4，CH 2 CR 4 = C（H）R 4，CH = C = CH 2或COR 5或任选取代的C 1-4烷基，任选取代的C 1- 4烷氧基或任选取代的（C 1-4）烷基C（= O）O（其中任选取代的部分各自可具有至多3个取代基，各自独立地选自卤素和C 1-4烷氧基，C 1-4烷基，C 1-2卤代烷氧基，二羟基，氰基，羧基，甲氧基羰基，乙氧基羰基，甲基磺酰基和乙基磺酰基）。式（I）化合物具有杀微生物活性，特别是杀真菌活性。

7. 发明申请

WO2005028485A8 SILICON COMPOUNDS WITH MICROBIOCIDAL ACTIVITY 审中-公开
标题翻译：具有微生物活性的硅化合物
公开(公告)号：WO2005028485A8
公开(公告)日：2005-06-09
申请号：PCT/EP2004010009
申请日：2004-09-08
申请人： SYNGENTA PARTICIPATIONS AG , EHRENFREUND JOSEF , LAMBERTH CLEMENS , TOBLER HANS , WALTER HARALD
发明人： EHRENFREUND JOSEF , LAMBERTH CLEMENS , TOBLER HANS , WALTER HARALD
IPC分类号： A01N55/00 , A01N55/10 , C07F7/08
CPC分类号： C07F7/0812 , A01N55/00
摘要： Fungicidal compounds of formula (I): where X is O or S; RING is phenyl or thienyl; Het is a 5- or 6-membered heterocyclic ring containing one to three heteroatoms, each independently selected from oxygen, nitrogen and sulphur, the ring being substituted by one to four groups R ; R is hydrogen, optionally substituted (C1-4)alkyl, formyl, optionally substituted (C1-4)alkylC(=O), optionally substituted (C1-4)alkylC(=O)O, optionally substituted (C1-4)alkoxy(C1-4)alkyl, optionally substituted allyl, optionally substituted propargyl or optionally substituted allenyl; each R is, independently, halogen, optionally substituted (C1-4)alkyl, optionally substituted (C1-4)alkoxy or optionally substituted (C1-4)alkoxy(C1-4)alkyl; R is (CR R )m Cy-(CR R )n-Y; each R is, independently, selected from halogen, C1-3 alkyl, C1-3 haloalkyl, C1-3 alkoxy(C1-3)alkyl and cyano; R , R , R and R are each, independently, hydrogen or optionally substituted (C1-4)alkyl; Cy is an optionally substituted carbocyclic or heterocyclic 3-7 membered ring which may be saturated, unsaturated or aromatic and which optionally contains a silicon atom as a ring member; (CR R )m and (CR R )n may be bound either to the same carbon or silicon atom of Cy or to different atoms separated by 1, 2 or 3 ring members; Y is Si(OpZ )(Oq Z )(OsZ) and provided that Cy contains a silicon atom as a ring member then Y may also be hydrogen; Z is C1-4 alkyl or C2-4 alkenyl (each of which is optionally interrupted by one heteroatom selected from O, S and N and is optionally substituted by one to three independently selected halogen atoms); Z and Z are, independently, methyl or ethyl; in and n are each, independently, 0, 1, 2 or 3; p, q and s are each, independently, 0 or 1; and r is 0, 1 or 2; or an N-oxide thereof; novel intermediates used in the preparation of these compounds, agrochemical compositions which comprise at least one of the novel compounds as active ingredient and the use of the active ingredients or compositions in agriculture or horticulture for controlling or preventing infestation of plants by phytopathogenic microorganisms, preferably fungi.
摘要翻译：式（I）的杀真菌化合物：其中X是O或S; RING是苯基或噻吩基; Het是含有1-3个各自独立地选自氧，氮和硫的杂原子的5-或6-元杂环，所述环被1-4个基团R 4取代; R 1是氢，任选取代的（C 1-4）烷基，甲酰基，任选取代的（C 1-4）烷基C（= O），任选取代的（C 1-4）烷基C 4）烷氧基（C 1-4）烷基，任选取代的烯丙基，任选取代的炔丙基或任选取代的丙二烯基; 每个R 2独立地为卤素，任选取代的（C 1-4）烷基，任选取代的（C 1-4）烷氧基或任选取代的（C 1-4）烷氧基（C 1-4）烷基; R 3是（CR a R b）m C y - （CR c R d）n -Y; 每个R 4独立地选自卤素，C 1-3烷基，C 1-3卤代烷基，C 1-3烷氧基（C 1-3）烷基和氰基; R a，R b，R c和R d各自独立地为氢或任选取代的（C 1-4）烷基; Cy是任选取代的碳环或杂环3-7元环，其可以是饱和的，不饱和的或芳族的，并且其任选含有硅原子作为环成员; （CR a R b）m和（CR c R d）n可以与Cy的相同的碳或硅原子结合，或者结合到由1,2或3个环成员分隔的不同原子上; Y是Si（OpZ 1）（Oq Z 2）（OsZ）并且条件是Cy含有硅原子作为环成员，那么Y也可以是氢; Z是C1-4烷基或C2-4链烯基（其每一个任选地被一个选自O，S和N的杂原子间隔，并且任选被1-3个独立选择的卤素原子取代）; Z 1和Z 2独立地为甲基或乙基; in和n各自独立地为0,1,2或3; p，q和s各自独立地为0或1; r是0,1或2; 或其N-氧化物; 用于制备这些化合物的新颖中间体，包含至少一种新化合物作为活性成分的农业化学组合物，以及活性成分或组合物在农业或园艺中用于控制或预防植物病原微生物侵染植物，优选真菌。

8. 发明专利

JP2013035850A Heterocyclic amide derivative useful as microbiocide 有权
标题翻译：杂环酰胺衍生物作为微生物有用
公开(公告)号：JP2013035850A
公开(公告)日：2013-02-21
申请号：JP2012200564
申请日：2012-09-12
申请人： Syngenta Participations Ag , シンジェンタパーティシペーションズアクチェンゲゼルシャフト
发明人： TOBLER HANS , WALTER HARALD , EHRENFREUND JOSEF , CORSI CAMILLA
IPC分类号： C07C205/45
CPC分类号： C07C205/06 , A01N43/32 , A01N43/36 , A01N43/40 , A01N43/56 , A01N43/647 , A01N43/76 , A01N43/78 , C07C205/11 , C07C205/12 , C07C205/37 , C07C205/45 , C07C211/61 , C07C2603/66 , C07D207/34 , C07D207/46 , C07D213/89 , C07D231/14 , C07D249/04 , C07D263/34 , C07D277/56 , C07D327/06
摘要： PROBLEM TO BE SOLVED: To provide a novel intermediate used for tricyclic amine derivative having the microbicidal activity, in particular the fungicidal activity.SOLUTION: A compound is provided which is represented by formula (D) (in the formula, Rand Rare each independently hydrogen, halo, 1-4C alkyl, 1-4C alkoxy, 1-4C haloalkyl or 1-4C haloalkoxy).
摘要翻译：要解决的问题：提供具有杀微生物活性的三环胺衍生物的新型中间体，特别是杀真菌活性。
解决方案：提供由式（D）表示的化合物（在式中，R 2 和R 3

9. 发明申请

WO9518122A3 HETEROARYLPYRROLES 审中-公开
公开(公告)号：WO9518122A3
公开(公告)日：1995-08-10
申请号：PCT/EP9404219
申请日：1994-12-19
申请人： CIBA GEIGY AG , DUERR DIETER , EHRENFREUND JOSEF , HALL ROGER GRAHAM , DANKO PETER
发明人： DUERR DIETER , EHRENFREUND JOSEF , HALL ROGER GRAHAM , DANKO PETER
IPC分类号： C07D207/34 , C07D401/04 , C07D403/04 , C07D409/04 , C07D413/04 , C07D417/04 , A61K31/40 , A61K31/44 , C07D405/04
CPC分类号： C07D401/04 , C07D207/34 , C07D403/04 , C07D409/04 , C07D413/04 , C07D417/04
摘要： Compounds of formula (I) in which R1, R2, R3 and Het are as defined in claim 1, and, where appropriate, tautomers thereof, in each case in free form or in salt form, can be used as agrochemical active ingredients and can be prepared in a manner known per se.

10. 发明专利

CA1281741C PHENYLBENZOYLUREAS 未知
公开(公告)号：CA1281741C
公开(公告)日：1991-03-19
申请号：CA489645
申请日：1985-08-29
申请人： EHRENFREUND JOSEF
发明人： EHRENFREUND JOSEF
IPC分类号： A01N47/34 , C07C67/00 , C07C239/00 , C07C275/54
摘要： Phenylbenzoylureas of the disclosure The invention relates to novel N-¢3-halo-4-(hexafluoropropoxy)-5-trifluoromethyl!phenyl-N'-benzoylureas of the formula wherein R1 is hydrogen or halogen and R2 and R3 are halogen, to a process and intermediate for the preparation of these compounds, and to compositions containing them for use in pest control, in particular for controlling insects and representatives of the order Acarina that attack plants and animals. The novel compounds exhibit in particular larvicidal activity.

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