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1. 发明申请

WO2007068417A3 PROCESS FOR THE PREPARATION OF AMINES 审中-公开
标题翻译：制备氨基酸的方法
公开(公告)号：WO2007068417A3
公开(公告)日：2007-10-04
申请号：PCT/EP2006011885
申请日：2006-12-11
申请人： SYNGENTA PARTICIPATIONS AG , TOBLER HANS , WALTER HARALD , CORSI CAMILLA , EHRENFREUND JOSEF , GIORDANO FANNY , ZELLER MARTIN
发明人： TOBLER HANS , WALTER HARALD , CORSI CAMILLA , EHRENFREUND JOSEF , GIORDANO FANNY , ZELLER MARTIN
IPC分类号： C07C209/28 , A01N45/02 , C07C211/31
CPC分类号： C07C209/62 , C07B2200/09 , C07C17/23 , C07C17/30 , C07C17/354 , C07C25/22 , C07C25/24 , C07C209/10 , C07C209/70 , C07C211/61 , C07C2603/66 , C07C23/10
摘要： The present invention relates to a novel a process for the preparation of the compound of the general formula (I), wherein R 1 and R 2 are independently H or C 1-6 alkyl, which comprises treating with a reducing agent either a compound of the general formula (II), wherein R 1 and R 2 have the meanings given for the compound of the formula (I), R 3 is H or C 1-4 alkyl and Ph is phenyl, or a compound of the general formula (III), wherein R 1 , R 2 , R 3 and Ph have the meanings given for the compound of the formula (II), the reducing agent being effective to cleave the benzyl moiety Ph-CH(R 3 )- from the benzylamino moiety PhCH(R 3 )NH- in the compound of the formula (II) or in the compound of the formula (III) to leave an amino group and, in addition, in the case of the compound of the formula (III), to reduce both the 2,3-double bond and the double bond joining the R 1 R 2 C- moiety to the 9-position of the benzonorbornene ring to single bonds. It also relates to processes for the preparation of the compounds (II) and (III) and their precursors and to the compounds (II) and (III) themselves and certain of their precursors, which are novel compounds. The compounds (I) are useful for the preparation of various fungicidal heterocyclyl-carboxylic acid benzonorbornen-5-yl-amides.
摘要翻译：本发明涉及一种制备通式（I）化合物的新方法，其中R 1和R 2独立地为H或C _{1 C-C部分到苯并降冰片烯环的9-位到单键。它还涉及制备化合物（II）和（III）及其前体以及化合物（II）和（III）本身及其某些新型化合物的前体的方法。化合物（I）可用于制备各种杀真菌性杂环基 - 羧酸苯并降冰片烯-5-基 - 酰胺。}

2. 发明专利

CA2687176C PROCESS FOR THE PRODUCTION OF PYRAZOLES 未知
公开(公告)号：CA2687176C
公开(公告)日：2015-06-30
申请号：CA2687176
申请日：2008-05-13
申请人： SYNGENTA LTD , SYNGENTA PARTICIPATIONS AG
发明人： GIORDANO FANNY , VETTIGER THOMAS , WISS JUERG GUSTAV , WANG LINHUA
IPC分类号： C07D231/14
摘要： A process for the production of a compound of formula (I), which comprises a) reacting a compound of formula (II), wherein R1 and R2 are both independently C1-C6 alkyl, with methylhydrazine in the presence of water and a water-immiscible organic solvent being inert in saponification reactions, to form a compound of formula (III) wherein R1 is as defined for formula (II) and b) saponifying that compound in sit.upsilon. leading to the formation of the compound of formula (I) by b1) adding a base to form the anion of the compound of formula (I) and then adding an; acid to form the compound of formula (I); or b2) adding an acid to form the compound of formula (I).

3. 发明专利

CA2631973C PROCESS FOR THE PREPARATION OF AMINES 未知
公开(公告)号：CA2631973C
公开(公告)日：2015-02-03
申请号：CA2631973
申请日：2006-12-11
申请人： SYNGENTA PARTICIPATIONS AG
发明人： TOBLER HANS , WALTER HARALD , CORSI CAMILLA , EHRENFREUND JOSEF , GIORDANO FANNY , ZELLER MARTIN
IPC分类号： C07C209/28 , A01N45/02 , C07C211/31
摘要： The present invention relates to a novel a process for the preparation of the compound of the general formula (I), wherein R1 and R2 are independently H or C1-6 alkyl, which comprises treating with a reducing agent either a compound of the general formula (II), wherein R1 and R2 have the meanings given for the compound of the formula (I), R3 is H or C1-4alkyl and Ph is phenyl, or a compound of the general formula (III), wherein R1, R2, R3 and Ph have the meanings given for the compound of the formula (II), the reducing agent being effective to cleave the benzyl moiety Ph-CH(R3)- from the benzylamino moiety PhCH(R3)NH- in the compound of the formula (II) or in the compound of the formula (III) to leave an amino group and, in addition, in the case of the compound of the formula (III), to reduce both the 2,3-double bond and the double bond joining the R1R2C- moiety to the 9-position of the benzonorbornene ring to single bonds. It also relates to processes for the preparation of the compounds (II) and (III) and their precursors and to the compounds (II) and (III) themselves and certain of their precursors, which are novel compounds. The compounds (I) are useful for the preparation of various fungicidal heterocyclyl-carboxylic acid benzonorbornen-5-yl-amides.

4. 发明专利

EA019039B1 СПОСОБ ПОЛУЧЕНИЯ БЕНЗОНОРБОРНЕНОВ 未知
公开(公告)号：EA019039B1
公开(公告)日：2013-12-30
申请号：EA201100665
申请日：2009-09-28
申请人： SYNGENTA PARTICIPATIONS AG
发明人： GRIBKOV DENIS , ANTELMANN BJOERN , GIORDANO FANNY , WALTER HARALD , DE MESMAEKER ALAIN
IPC分类号： C07C205/12 , C07C17/25 , C07C22/02 , C07C23/08 , C07C211/61
摘要： Визобретенииописанновыйспособполучения 9-дихлорметилен-1,2,3,4-тетрагидро-1,4-метанонафталин-5-иламина, которыйвключаета) реакциюциклопентадиенав присутствиирадикальногоинициатораи CXCl, где X обозначаетхлорилибром, сполучениемсоединенияформулы (II), илиаа) реакциюциклопентадиенас CXCl, где X обозначаетхлор, вприсутствииметаллсодержащегокатализаторас получениемсоединенияформулы (II), вкоторой X обозначаетхлор, b) реакциюсоединенияформулы (II) соснованиемв присутствииподходящегорастворителяс получениемсоединенияформулы (III); с) превращениесоединенияформулы (III) вприсутствии 1,2-дигидро-6-нитробензолав соединениеформулы (IV) и d) гидрированиесоединенияформулы (IV) вприсутствииметаллсодержащегокатализатора.

5. 发明专利

ES2391904T3 Procedimiento para la preparación de aminas 未知
公开(公告)号：ES2391904T3
公开(公告)日：2012-11-30
申请号：ES06829477
申请日：2006-12-11
申请人： SYNGENTA PARTICIPATIONS AG
发明人： TOBLER HANS , WALTER HARALD , CORSI CAMILLA , EHRENFREUND JOSEF , GIORDANO FANNY , ZELLER MARTIN
IPC分类号： C07C17/23 , C07C17/30 , C07C17/354 , C07C23/10 , C07C25/22 , C07C25/24 , C07C209/10 , C07C209/62 , C07C209/70 , C07C211/61
摘要： Un procedimiento para la preparación del compuesto de la fórmula general (I):en la que R1 y R2 son independientemente H o alquilo de C1-6, que comprende tratar con un agente reductor uncompuesto de la fórmula general (II):en la que R1 y R2 tienen los significados dados anteriormente, R3 es H o alquilo de C1-4 y Ph es fenilo, oun compuesto de la fórmula general (III):en la que R1, R2, R3 y Ph tienen los significados dados anteriormente, siendo el agente reductor eficaz para escindirel resto bencilo Ph-CH(R3)- del resto bencilamino PhCH(R3)NH- en el compuesto de la fórmula (II) o en el compuestode la fórmula (III) para dejar un grupo amino, y, además, en el caso del compuesto de la fórmula (III), para reducirtanto el doble enlace de 2,3 como el doble enlace que une el resto R1R2C- a la posición 9 del anillobenzonorbornénico a enlaces sencillos, y en el que dicho agente reductor es hidrógeno en presencia de uncatalizador de la hidrogenación metálico.

6. 发明专利

DK1963251T3 Fremgangsmåde til fremstilling af aminer 未知
公开(公告)号：DK1963251T3
公开(公告)日：2012-11-26
申请号：DK06829477
申请日：2006-12-11
申请人： SYNGENTA PARTICIPATIONS AG
发明人： TOBLER HANS , WALTER HARALD , CORSI CAMILLA , EHRENFREUND JOSEF , GIORDANO FANNY , ZELLER MARTIN
IPC分类号： C07C17/23 , C07C17/30 , C07C17/354 , C07C23/10 , C07C25/22 , C07C25/24 , C07C209/10 , C07C209/62 , C07C209/70 , C07C211/61

7. 发明专利

ZA201200413B PROCESS FOR THE PREPARATION OF PYRAZOLE CARBOXYLIC ACID AMIDES 未知
公开(公告)号：ZA201200413B
公开(公告)日：2012-10-31
申请号：ZA201200413
申请日：2012-01-18
申请人： SYNGENTA PARTICIPATIONS AG
发明人： GRIBKOV DENIS , LAGGER MARTIN , MULLER ADRIAN , GIORDANO FANNY
IPC分类号： C07C20060101 , C07D20060101
摘要： The invention relates to a process for the preparation of 3-difluoromethyl-1-methyl-1H-pyrazole-4-carboxylic acid (9-dichloromethylene-1,2,3,4-tetrahydro-1,4-methano-naphthalen-5-yl)-amide.

8. 发明专利

AU2006291419B2 Process for the production of amides 未知
公开(公告)号：AU2006291419B2
公开(公告)日：2012-06-14
申请号：AU2006291419
申请日：2006-09-14
申请人： SYNGENTA LTD , SYNGENTA PARTICIPATIONS AG
发明人： ZELLER MARTIN , GEORGE NEIL , CORSI CAMILLA , JONES IAN , WALTER HARALD , EHRENFREUND JOSEF , TOBLER HANS , SEIFERT GOTTFRIED , GIORDANO FANNY , SHAH SHAILESH C , BONNETT PAUL
IPC分类号： C07D231/14 , A01N43/26 , C07C205/06 , C07C211/45
摘要： The present invention relates to a process for the preparation of compounds of formula (I) wherein R and R are each independently of the other hydrogen or C-Calkyl and R is CFor CFH, by a) reaction of a compound of formula (Il) wherein R and R are as defined for formula (I), with at least one reducing agent to form a compound of formula (III) wherein R and Rare as defined for formula (I), and b) reaction of that compound with at least one reducing agent to form a compound of formula (IV) wherein R and R are as defined for formula (I), and (c) reaction of that compound with a compound of formula (V) wherein Q is chlorine, fluorine, bromine, iodine, hydroxy or C-Calkoxy and R is as defined for formula (I), to form the compound of formula (I); and to novel intermediates for use in that process.

9. 发明专利

UA98062C2 КРИСТАЛЛИЧЕСКАЯ МОДИФИКАЦИЯ В (9-ИЗОПРОПИЛ-1,2,3,4-ТЕТРАГИДРО-1,4-МЕТАНОНАФТАЛЕН-5-ИЛ)АМИДА, КОМПОЗИЦИЯ НА ЕЕ ОСНОВЕ И СПОСОБ БОРЬБЫ С БОЛЕЗНЯМИ, ВЫЗВАННЫМИ ФИТОПАТОГЕНАМИ 未知
公开(公告)号：UA98062C2
公开(公告)日：2012-04-10
申请号：UAA201102589
申请日：2006-09-14
申请人： SYNGENTA PARTICIPATIONS AG , SYNGENTA LTD
发明人： TOBLER HANS , WALTER HARALD , EHRENFREUND JOSEF , CORSI CAMILLA , GIORDANO FANNY , ZELLER MARTIN , SEIFERT GOTTFRIED , SHAH SHAILESH C , GEORGE NEIL , JONES IAN , BONNETT PAUL
IPC分类号： C07D231/14 , A01N43/26 , C07C205/00 , C07C211/45
摘要： Настоящееизобретениеотноситсяк кристаллическоймодификацииВ (9-изопропил-1,2,3,4-тетрагидро-1,4-метанонафтален-5-ил)амидасин-3-дифторметил-1-метил-1Н-пиразол-4-карбоновойкислоты, приэтомуказаннаякристаллическаямодификацияхарактеризуетсяпорошковойрентгенограммой, выраженнойв значенияхмежплоскостныхрасстояний d иотносительныхинтенсивностей, иуказаннаяпорошковаярентгенограммасодержитследующиехарактеристическиелинии: 13,42 Ǻ (сильная), 9,76 Ǻ (средняя), 6,93 Ǻ (средняя), 6,74 Ǻ (средняя), 4,79 Ǻ (средняя), 4,73 Ǻ (средняя) i 3,66 Ǻ (средняя) сиспользованием CuKα1 вкачествеисточникарентгеновскихлучей, изображенанафиг. 1. КомпозициянаосновекристаллическоймодификацииВ (9-изолропил-1,2,3,4-тетрагидро-1,4-метанонафтален-5-ил)амидасин-3-дифторметил-1-метил-1Н-п

10. 发明专利

BRPI0619629A2 未知
公开(公告)号：BRPI0619629A2
公开(公告)日：2011-10-04
申请号：BRPI0619629
申请日：2006-12-11
申请人： SYNGENTA PARTICIPATIONS AG
发明人： TOBLER HANS , WALTER HARALD , CORSI CAMILLA , EHRENFREUND JOSEF , ZELLER MARTIN , GIORDANO FANNY
IPC分类号： C07C209/28 , A01N45/02 , C07C211/31
摘要： The present invention relates to processes for the preparation of compounds of formula (VII) wherein X is chloro or bromo. Compounds of formula (VII) are useful intermediates for the preparation of various fungicidal heterocyclyl-carboxylic acid benzonorbornen-5-yl-amides.

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