专利快速检索-快速检索全球专利，免费商用专利数据库-IPRDB

1. 发明申请

WO2012069633A1 MICROBICIDAL HETEROCYCLES 审中-公开
标题翻译：微生物杂交
公开(公告)号：WO2012069633A1
公开(公告)日：2012-05-31
申请号：PCT/EP2011/071037
申请日：2011-11-25
申请人： SYNGENTA PARTICIPATIONS AG , SULZER-MOSS, Sarah , LAMBERTH, Clemens , RESPONDEK, Mathias, Stephan , QUARANTA, Laura , CEDERBAUM, Fredrik , BERTHON, Guillaume
发明人： SULZER-MOSS, Sarah , LAMBERTH, Clemens , RESPONDEK, Mathias, Stephan , QUARANTA, Laura , CEDERBAUM, Fredrik , BERTHON, Guillaume
IPC分类号： C07D401/14 , C07D413/14 , C07D417/14 , C07D513/04 , A01N43/80
CPC分类号： A01N43/82 , A01N43/60 , A01N43/80 , C07D401/14 , C07D413/14 , C07D417/14 , C07D513/04
摘要： Compounds of the formula I Formula (I) wherein the substituents are as defined in claim 1, are useful as active ingredients, which have microbiocidal activity, in particular fungicidal activity.
摘要翻译：其中取代基如权利要求1中所定义的式I化学式（I）的化合物可用作具有杀微生物活性，特别是杀真菌活性的活性成分。

2. 发明申请

WO2011018415A3 MICROBIOCIDAL HETEROCYCLES 审中-公开
标题翻译：微生物杂环
公开(公告)号：WO2011018415A3
公开(公告)日：2011-08-18
申请号：PCT/EP2010061464
申请日：2010-08-06
申请人： SYNGENTA PARTICIPATIONS AG , SULZER SARAH , LAMBERTH CLEMENS , QUARANTA LAURA , RESPONDEK MATHIAS STEPHAN
发明人： SULZER SARAH , LAMBERTH CLEMENS , QUARANTA LAURA , RESPONDEK MATHIAS STEPHAN
IPC分类号： C07D231/12 , C07D401/04 , C07D401/06 , C07D401/12 , C07D401/14
CPC分类号： C07D401/14 , C07D231/12 , C07D401/04 , C07D401/06 , C07D401/12
摘要： The present invention relates to heterocyclic compounds of formula I which have microbiocidal activity, in particular fungicidal activity as well as methods of using the compounds of formula (I) to control microbes: wherein A is x-C(R10R11)-C(=O)-, x-C(R12R13)-C(=S)-, x-O-C(=O)-, x-O-C(=S)-, x-N(R14)-C(=O)-, x-N(R15)-C(=S)-,x-C(R16R17)-SO2- or X-N=C(R30)-,, in each case x indicates the bond that is connected to R1; T is CR18 or N; Y1, Y2, Y3, and Y4 are independently CR19 or N; Q is O or S; n is 1 or 2; p is 1 or 2, providing that when n is 2, p is 1. R1 is phenyl, pyridyl, imidazolyl, or pyrazolyl; wherein the phenyl, pyridyl, imidazolyl and pyrazolyl are each optionally substituted by 1 to 3 substituents independently selected from C1-C4 alkyl, C1-C4 haloalkyl, halogen, cyano, hydroxy and amino; R2, R3, R4, R5, R6, R7, R10, R11, R12, R13, R16, R17, R18,R19 and R30 each independently are hydrogen, halogen, cyano, C1-C4alkyl, or C1-C4haloalkyl; R8, R14 and R15 each independently are hydrogen or C1-C4alkyl; and R9 is phenyl, benzyl or group (a): wherein the phenyl, benzyl and group (a) are each optionally substituted with 1 to 3 substituents independently selected from C1-C4 alkyl, C1-C4 haloalkyl, halogen, cyano, hydroxy and amino; or a salt or a N-oxide thereof.
摘要翻译：本发明涉及具有杀微生物活性，特别是杀真菌活性的式I杂环化合物以及使用式（I）化合物控制微生物的方法：其中A是xC（R 10 R 11）-C（= O） - ，xC（R 12 R 13）-C（= S） - ，xOC（= O） - ，xOC（= S） - ，xN（R 14）-C（= O），xC（R 16 R 17）-SO 2 - 或XN = C（R 30） - ，在每种情况下，x表示连接至R 1的键; T是CR18或N; Y1，Y2，Y3和Y4独立地为CR19或N; Q是O或S; n是1或2; p是1或2，条件是当n是2时，p是1。其中所述苯基，吡啶基，咪唑基和吡唑基各自任选被1至3个独立地选自C 1 -C 4烷基，C 1 -C 4卤代烷基，卤素，氰基，羟基和氨基的取代基取代; R2，R3，R4，R5，R6，R7，R10，R11，R12，R13，R16，R17，R18，R19和R30各自独立地为氢，卤素，氰基，C1-4烷基或C1-4卤代烷基; R8，R14和R15各自独立地为氢或C1-C4烷基; （a）：其中苯基，苄基和基团（a）各自任选被1至3个取代基取代，所述取代基独立地选自C 1 -C 4烷基，C 1 -C 4卤代烷基，卤素，氰基，羟基和氨基; 或其盐或N-氧化物。

3. 发明申请

WO2011018415A2 MICROBIOCIDAL HETEROCYCLES 审中-公开
标题翻译：微生物杂交
公开(公告)号：WO2011018415A2
公开(公告)日：2011-02-17
申请号：PCT/EP2010/061464
申请日：2010-08-06
申请人： SYNGENTA PARTICIPATIONS AG , SULZER, Sarah , LAMBERTH, Clemens , QUARANTA, Laura , RESPONDEK, Mathias, Stephan
发明人： SULZER, Sarah , LAMBERTH, Clemens , QUARANTA, Laura , RESPONDEK, Mathias, Stephan
CPC分类号： C07D401/14 , C07D231/12 , C07D401/04 , C07D401/06 , C07D401/12
摘要： The present invention relates to heterocyclic compounds of formula I which have microbiocidal activity, in particular fungicidal activity as well as methods of using the compounds of formula (I) to control microbes: wherein A is x-C(R 10 R 11 )-C(=O)-, x-C(R 12 R 13 )-C(=S)-, x-O-C(=O)-, x-O-C(=S)-, x-N(R 14 )-C(=O)-, x-N(R 15 )-C(=S)-,x-C(R 16 R 17 )-SO 2 - or X-N=C(R 30 )-,, in each case x indicates the bond that is connected to R 1 ; T is CR 18 or N; Y 1 , Y 2 , Y 3 , and Y 4 are independently CR 19 or N; Q is O or S; n is 1 or 2; p is 1 or 2, providing that when n is 2, p is 1. R 1 is phenyl, pyridyl, imidazolyl, or pyrazolyl; wherein the phenyl, pyridyl, imidazolyl and pyrazolyl are each optionally substituted by 1 to 3 substituents independently selected from C 1 -C 4 alkyl, C 1 -C 4 haloalkyl, halogen, cyano, hydroxy and amino; R 2 , R 3 , R 4 , R 5 , R 6 , R 7 , R 10 , R 11 , R 12 , R 13 , R 16 , R 17 , R 18 ,R 19 and R 30 each independently are hydrogen, halogen, cyano, C 1 -C 4 alkyl, or C 1 -C 4 haloalkyl; R 8 , R 14 and R 15 each independently are hydrogen or C 1 -C 4 alkyl; and R 9 is phenyl, benzyl or group (a): wherein the phenyl, benzyl and group (a) are each optionally substituted with 1 to 3 substituents independently selected from C 1 -C 4 alkyl, C 1 -C 4 haloalkyl, halogen, cyano, hydroxy and amino; or a salt or a N-oxide thereof.
摘要翻译：本发明涉及具有杀微生物活性，特别是杀真菌活性的式I的杂环化合物以及使用式（I）化合物来控制微生物的方法：其中A是xC（R10R11）-C（= O） - ，xC（R12R13）-C（= S） - ，xOC（= O） - ，xOC（= S） - ，xN（R14）-C（= O） - ，xN（R15）-C（= S），xC（R16R17）-SO2-或XN = C（R30） - ，在各种情况下，x表示与R1连接的键; T为CR18或N; Y1，Y2，Y3和Y4独立地为CR19或N; Q是O或S; n为1或2; p为1或2，条件是当n为2时，p为1. R1为苯基，吡啶基，咪唑基或吡唑基; 其中苯基，吡啶基，咪唑基和吡唑基各自任选被1至3个独立地选自C 1 -C 4烷基，C 1 -C 4卤代烷基，卤素，氰基，羟基和氨基的取代基取代; R2，R3，R4，R5，R6，R7，R10，R11，R12，R13，R16，R17，R18，R19和R30各自独立地为氢，卤素，氰基，C1-C4烷基或C1-C4卤代烷基; R8，R14和R15各自独立地为氢或C1-C4烷基; 并且R 9为苯基，苄基或基团（a）：其中苯基，苄基和基团（a）各自任选被1至3个独立地选自C 1 -C 4烷基，C 1 -C 4卤代烷基，卤素，氰基，羟基和氨基; 或其盐或N-氧化物。

4. 发明申请

WO2009090038A1 FUNGICIDAL COMPOSITIONS 审中-公开
标题翻译：杀真菌剂
公开(公告)号：WO2009090038A1
公开(公告)日：2009-07-23
申请号：PCT/EP2009/000165
申请日：2009-01-14
申请人： SYNGENTA PARTICIPATIONS AG , GODWIN, Jeremy, R. , TRAH, Stephan , LAMBERTH, Clemens , DUMEUNIER, Raphael , WENDEBORN, Sebastian, Volker , GRASSO, Valeria
发明人： GODWIN, Jeremy, R. , TRAH, Stephan , LAMBERTH, Clemens , DUMEUNIER, Raphael , WENDEBORN, Sebastian, Volker , GRASSO, Valeria
IPC分类号： A01N43/58 , A01P3/00
CPC分类号： A01N43/58 , A01N37/34 , A01N43/54 , A01N43/653 , A01N47/14 , A01N51/00 , A01N2300/00
摘要： A fungicidal composition suitable for control of diseases caused by phytopathogens comprising (A) a compound of formula (I), wherein R 1 is methyl, ethyl or isopropyl; R 2 is 2-chloro-6-fluoro-phenyl, 2,4,6-trifluorophenyl or 2,6-difluoro-4-methoxy-phenyl; R 3 is chloro, fluoro or methoxy; and (B) a compound selected, for example, from the group consisting of (B1) a strobilurin fungicide, (B2) an azole fungicide, (B3) a morpholine fungicide, and (B4) an anilinopyrimidine fungicide.
摘要翻译：一种适于控制由植物病原体引起的疾病的杀真菌组合物，其包含（A）式（I）化合物，其中R 1为甲基，乙基或异丙基; R2是2-氯-6-氟 - 苯基，2,4,6-三氟苯基或2,6-二氟-4-甲氧基 - 苯基; R3是氯，氟或甲氧基; 和（B）选自例如（B1）嗜球果伞素杀真菌剂，（B2）唑类杀真菌剂，（B3）吗啉杀真菌剂和（B4）苯胺基嘧啶杀真菌剂的组合的化合物。

5. 发明申请

WO2008009405A3 NOVEL PYRIDAZINE DERIVATIVES 审中-公开
标题翻译：新的吡咯烷酮衍生物
公开(公告)号：WO2008009405A3
公开(公告)日：2008-03-27
申请号：PCT/EP2007006303
申请日：2007-07-16
申请人： SYNGENTA PARTICIPATIONS AG , TRAH STEPHAN , LAMBERTH CLEMENS , WENDEBORN SEBASTIAN VOLKER
发明人： TRAH STEPHAN , LAMBERTH CLEMENS , WENDEBORN SEBASTIAN VOLKER
IPC分类号： C07D401/14 , A01N43/58 , C07D403/14 , C07D405/14 , C07D407/14 , C07D409/14 , C07D417/14
CPC分类号： C07D401/14 , A01N43/58 , C07D403/14 , C07D405/14 , C07D407/14 , C07D409/14 , C07D417/14
摘要： The present invention relates to novel pyridazine derivatives of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity: wherein R 1 is hydrogen, C 1 -C 6 alkyl, C 1 -C 6 haloalkyl or C 3 -C 6 cycloalkyl; R 2 is an optionally substituted hereroaryl; R 3 is an optionally substituted heteroaryl; and R 4 is hydrogen, halogen, C 1 -C 6 alkyl, C 1 -C 6 haloalkyl, C 1 -C 6 alkoxy, C 1 -C 6 haloalkoxy, hydroxy or cyano; or an agrochemically usable salt form thereof.
摘要翻译：本发明涉及式（I）的新颖哒嗪衍生物作为具有杀微生物活性，特别是杀真菌活性的活性成分：其中R 1是氢，C 1 -C C 1 -C 6烷基，C 1 -C 6卤代烷基或C 3 -C 6烷基，C 1 -C 6烷基，C 1 -C 6 - 环烷基; R 2是任选取代的二芳基; R 3是任选取代的杂芳基; R 4是氢，卤素，C 1 -C 6烷基，C 1 -C 3烷基，C 1 -C 6烷基， 6个卤代烷基，C 1 -C 6烷氧基，C 1 -C 6卤代烷氧基，羟基（C 1 -C 6）或氰基; 或其农业化学上可用的盐形式。

6. 发明申请

WO2006100038A1 TRIAZOLOPYRIMIDINE DERIVATIVES USEFUL AS FUNGICIDES 审中-公开
标题翻译：三唑并嘧啶衍生物有效用作杀真菌剂
公开(公告)号：WO2006100038A1
公开(公告)日：2006-09-28
申请号：PCT/EP2006/002591
申请日：2006-03-21
申请人： SYNGENTA PARTICIPATIONS AG , SYNGENTA LIMITED , WENDEBORN, Sebastian , LAMBERTH, Clemens , NEBEL, Kurt , CROWLEY, Patrick, Jelf
发明人： WENDEBORN, Sebastian , LAMBERTH, Clemens , NEBEL, Kurt , CROWLEY, Patrick, Jelf
IPC分类号： C07D487/04 , C07D519/00 , A01N43/90 , A01P3/00
CPC分类号： A01N43/90 , C07D487/04
摘要： The present invention relates to novel triazolopyrimidine derivatives of formula I as active ingredients which have microbiocidal activity, in particular fungicidal activity wherein the substituents are as defined in claim 1.
摘要翻译：本发明涉及式I的新型三唑并嘧啶衍生物作为活性成分，其具有杀微生物活性，特别是杀真菌活性，其中取代基如权利要求1所定义。

7. 发明申请

WO2006100037A1 TRIAZOLOPYRIMIDINE DERIVATIVES USEFUL AS MICROBIOCIDES 审中-公开
标题翻译：三氮唑嘧啶衍生物作为微生物有用
公开(公告)号：WO2006100037A1
公开(公告)日：2006-09-28
申请号：PCT/EP2006/002590
申请日：2006-03-21
申请人： SYNGENTA PARTICIPATIONS AG , SYNGENTA LIMITED , LAMBERTH, Clemens , WENDEBORN, Sebastian , NEBEL, Kurt , CROWLEY, Patrick, Jelf
发明人： LAMBERTH, Clemens , WENDEBORN, Sebastian , NEBEL, Kurt , CROWLEY, Patrick, Jelf
IPC分类号： C07D487/04 , C07D519/00 , A01N43/90
CPC分类号： C07D487/04 , A01N43/90
摘要： The present invention relates to novel triazolopyrimidine derivatives of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity: wherein the substituents are as defined in Claim 1.
摘要翻译：本发明涉及具有杀微生物活性，特别是杀真菌活性的作为活性成分的式（I）的新型三唑并嘧啶衍生物，其中取代基如权利要求1所定义。

8. 发明申请

WO2006087222A1 PROCESS FOR THE PRODUCTION OF NITROBENZOLES 审中-公开
标题翻译：生产硝基苯酚的方法
公开(公告)号：WO2006087222A1
公开(公告)日：2006-08-24
申请号：PCT/EP2006/001507
申请日：2006-02-20
申请人： SYNGENTA PARTICIPATIONS AG , WALTER, Harald , CORSI, Camilla , EHRENFREUND, Josef , LAMBERTH, Clemens , SCHNEIDER, Hermann , TOBLER, Hans
发明人： WALTER, Harald , CORSI, Camilla , EHRENFREUND, Josef , LAMBERTH, Clemens , SCHNEIDER, Hermann , TOBLER, Hans
IPC分类号： C07C201/12 , C07C205/06 , C07C205/19 , C07C309/65 , A01N33/18
CPC分类号： C07C201/12 , C07C303/28 , C07C309/65 , C07C2601/02 , C07C205/06 , C07C205/11 , C07C205/19 , C07C205/45
摘要： The present invention relates to a process for the preparation of compounds of formula (I) wherein the substituents are as defined in claim 1 , by a) reaction of a compound of formula (II) wherein the substituents are as defined in claim 1 , with a reducing agent to form a compound of formula (III) wherein the substituents are as defined in claim 1 , and b) reaction of that compound either b1 ) with triphenylphosphine dibromide or triphenylphosphine dichloride or b2) with RSO2CI, wherein R is Ci-C4alkyl, CrC4fluoroalkyl, benzyl, phenyl, nitrophenyl, halophenyl or CrC6alkylphenyl, in the presence of a base, to form a compound of formula (IV) wherein the substituents are as defined in claim 1 ; and c) conversion of that compound in the presence of a base into a compound of formula (I); and also to novel nitrobenzene intermediates for use in that process.
摘要翻译：本发明涉及一种制备式（I）化合物的方法，其中取代基如权利要求1所定义，通过a）将式（Ⅱ）化合物（其中取代基如权利要求1所定义）与还原剂形成式（III）的化合物，其中取代基如权利要求1所定义，和b）该化合物b1）与三苯基膦二溴化物或三苯基膦二氯化物或b2）与RSO2Cl的反应，其中R是C 1 -C 4烷基，C 1 -C 4氟烷基，苄基，苯基，硝基苯基，卤代苯基或C 1 -C 6烷基苯基，以形成式（IV）的化合物，其中取代基如权利要求1所定义; 和c）将所述化合物在碱存在下转化为式（I）的化合物; 以及用于该方法的新型硝基苯中间体。

9. 发明申请

WO2006005612A1 PROCESS FOR THE PREPARATION OF 4,4-DIFLUORO-3-OXOBUTANOIC ACID ESTERS 审中-公开
标题翻译：制备4,4-二氟-3-氧代戊酸的方法
公开(公告)号：WO2006005612A1
公开(公告)日：2006-01-19
申请号：PCT/EP2005/007635
申请日：2005-07-13
申请人： SYNGENTA PARTICIPATIONS AG , WALTER, Harald , CORSI, Camilla , EHRENFREUND, Josef , LAMBERTH, Clemens , TOBLER, Hans
发明人： WALTER, Harald , CORSI, Camilla , EHRENFREUND, Josef , LAMBERTH, Clemens , TOBLER, Hans
IPC分类号： C07C67/343
CPC分类号： C07C67/343 , C07C69/716
摘要： The present invention relates to a process for the preparation of a compound of the formula (I), wherein R is C 1-12 alkyl, by the contact of a compound of the general formula (II) , wherein R 1 and R 2 are each, independently, C 1-12 alkyl; or R 1 and R 2 join together with the nitrogen atom to which they are attached to form an alicyclic amine ring containing 4 to 7 carbon atoms or a morpholine ring, with an acetic acid ester of the general formula (III) CH 3 COOR, wherein R is as defined under formula (I), in the presence of a base.
摘要翻译：本发明涉及制备式（I）化合物的方法，其中R是C 1-12烷基，通过通式（II）的化合物与其中R 1和R 2各自独立地为C 1-12烷基; 或R 1和R 2 2与它们所连接的氮原子一起形成含有4至7个碳原子的脂环族胺环或吗啉环，其中（III）CH 3 COOR的乙酸酯，其中R如式（I）所定义，在碱的存在下。

10. 发明申请

WO2005123722A1 HETEROCYCLIC CARBOXAMIDES WITH MICROBIOCIDAL ACTIVITY 审中-公开
标题翻译：具有微生物活性的杂环碳酰胺
公开(公告)号：WO2005123722A1
公开(公告)日：2005-12-29
申请号：PCT/EP2005/006688
申请日：2005-06-21
申请人： SYNGENTA PARTICIPATIONS AG , LAMBERTH, Clemens , CORSI, Camilla , EHRENFREUND, Josef , TOBLER, Hans , WALTER, Harald
发明人： LAMBERTH, Clemens , CORSI, Camilla , EHRENFREUND, Josef , TOBLER, Hans , WALTER, Harald
IPC分类号： C07D403/12
CPC分类号： C07D403/12 , C07D231/40 , C07D333/20 , C07D409/12
摘要： Compounds of the formula (I), in which the substituents are as defined in claim 1 are suitable for use as microbiocides.
摘要翻译：其中取代基如权利要求1中所定义的式（I）化合物适合用作杀微生物剂。

你已经成功收藏专利！

检索式保存成功!

IPRDB

热门服务

关于我们

友情链接

联系方式