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1. 发明授权

US4438109A Tylosin derivatives 失效
标题翻译：泰乐菌素衍生物
公开(公告)号：US4438109A
公开(公告)日：1984-03-20
申请号：US285747
申请日：1981-07-22
申请人： Hamao Umezawa , Sumio Umezawa , Tsutomu Tsuchiya , Akihiro Tanaka
发明人： Hamao Umezawa , Sumio Umezawa , Tsutomu Tsuchiya , Akihiro Tanaka
IPC分类号： C07H17/08 , A61K31/70
CPC分类号： C07H17/08
摘要： Tylosin derivatives shown by the general formula ##STR1## wherein R represents a hydrogen atom or a hydroxyl group; R.sub.1 represents a halogen atom, a hydroxyl group, a tetrahydrofuranyloxy group, a tetrahydropyranyloxy group, a tetrahydrothiofuranyloxy group, a tetrahydrothiopyranyloxy group, an alkanoyloxy group, an arylcarbonyloxy group, an aralkylcarbonyloxy group, a lower alkylthiomethyloxy group, a heterocyclic thio group which may have a substituent, a mono- or di- lower alkylamino lower alkylthio group or a group of ##STR2## (wherein R.sub.4 represents a hydroxyl group or an alkanoyloxy group); R.sub.2 represents a hydrogen atom, a hydroxyl group, or an alkanoyloxy group; R.sub.3 represents a hydroxyl group or an alkanoyloxy group; and represents a single bond or a double bond, but represents a double bond when R.sub.2 is a hydrogen atom.These compounds are useful as antibiotics.
摘要翻译：由通式表示的泰乐菌素衍生物，其中R表示氢原子或羟基; R 1表示卤素原子，羟基，四氢呋喃氧基，四氢吡喃氧基，四氢噻喃氧基，四氢噻喃氧基，烷酰氧基，芳基羰基氧基，芳烷基羰基氧基，低级烷基硫代甲氧基，可具有的杂环硫基取代基，单 - 或二 - 低级烷基氨基低级烷硫基或一组（其中R 4表示羟基或烷酰氧基）。 R2表示氢原子，羟基或烷酰氧基; R3表示羟基或烷酰氧基; 并且表示单键或双键，但当R 2为氢原子时，表示双键。这些化合物可用作抗生素。

2. 发明授权

US4945081A Mycaminosyl tylonolide derivatives 失效
标题翻译：碳霉糖太乐内酯衍生物
公开(公告)号：US4945081A
公开(公告)日：1990-07-31
申请号：US232904
申请日：1988-08-16
申请人： Hamao Umezawa , Sumio Umezawa , Tsutomu Tsuchiya , Tomio Takeuchi , Akihiro Tanaka , Shuichi Sakamoto
发明人： Hamao Umezawa , Sumio Umezawa , Tsutomu Tsuchiya , Tomio Takeuchi , Akihiro Tanaka , Shuichi Sakamoto
IPC分类号： A61K31/70 , A61K31/7042 , A61K31/7048 , A61P31/04 , C07H17/08
CPC分类号： C07H17/08 , Y02P20/55
摘要： Mycaminosyl tylonolide derivatives represented by the following general formula ##STR1## (wherein R.sup.1 denotes hydroxyl group, a lower alkanoyloxy group, benzyloxy group, azido group, or amino group which may optionally be substituted with a lower alkyl or a lower alkanoyl radical; R.sup.2 stands for hydrogen atom or hydroxyl group; R.sup.3 expresses hydrogen atom or formyl group; and means a double bond or a radical represented by ##STR2## and salts thereof.

3. 发明授权

US4914192A Mycaminosyl tylonolide derivatives 失效
公开(公告)号：US4914192A
公开(公告)日：1990-04-03
申请号：US244500
申请日：1988-09-14
申请人： Hamao Umezawa , Sumio Umezawa , Tsutomu Tsuchiya , Tomio Takeuchi , Akihiro Tanaka , Shuichi Sakamoto
发明人： Hamao Umezawa , Sumio Umezawa , Tsutomu Tsuchiya , Tomio Takeuchi , Akihiro Tanaka , Shuichi Sakamoto
IPC分类号： A61K31/70 , A61K31/7042 , A61K31/7048 , A61P31/04 , C07H17/08
CPC分类号： C07H17/08 , Y02P20/55
摘要： Mycaminosyl tylonolide derivatives represented by the following general formula ##STR1## (wherein R.sup.1 denoted hydroxyl group, a lower alkanoyloxy group, benzyloxy group, azido group, or amino group which may optionally be substituted with a lower alkyl or a lower alkanoyl radical; R.sup.2 stands for hydrogen atom or hydroxyl group; R.sup.3 expresses hydrogen atom or formyl group; and means a double bond or a radical represented by ##STR2## and salts thereof.

4. 发明授权

US5101022A Mycaminosyl tylonolide derivatives 失效
标题翻译： MYCAMINOSYL TYLONOLIDE DERIVATIVES
公开(公告)号：US5101022A
公开(公告)日：1992-03-31
申请号：US650060
申请日：1991-02-04
申请人： Hamao Umezawa , Sumio Umezawa , Tsutomu Tsuchiya , Tomio Takeuchi , Akihiro Tanaka , Shuichi Sakamoto
发明人： Hamao Umezawa , Sumio Umezawa , Tsutomu Tsuchiya , Tomio Takeuchi , Akihiro Tanaka , Shuichi Sakamoto
IPC分类号： A61K31/70 , A61K31/7042 , A61K31/7048 , A61P31/04 , C07H17/08
CPC分类号： C07H17/08 , Y02P20/55
摘要： Mycaminosyl tylonolide derivatives represented by the following general formula ##STR1## (wherein R.sup.1 denotes hydroxyl group, a lower alkanoyloxy group, benzoyloxy group, azido group, or amino group which may optionally be substituted with a lower alkyl or a lower alkanoyl radical; R.sup.2 stands for hydrogen atom or hydroxyl group; R.sup.3 expresses hydrogen atom or formyl group; and means a double bond or a radical represented by ##STR2## and salts thereof.

5. 发明授权

US4794173A Mycaminosyl tylonolide derivatives 失效
标题翻译：碳霉糖太乐内酯衍生物
公开(公告)号：US4794173A
公开(公告)日：1988-12-27
申请号：US861537
申请日：1986-05-09
申请人： Hamao Umezawa , Sumio Umezawa , Tsutomu Tsuchiya , Tomio Takeuchi , Akihiro Tanaka , Shuichi Sakamoto
发明人： Hamao Umezawa , Sumio Umezawa , Tsutomu Tsuchiya , Tomio Takeuchi , Akihiro Tanaka , Shuichi Sakamoto
IPC分类号： A61K31/70 , A61K31/7042 , A61K31/7048 , A61P31/04 , C07H17/08
CPC分类号： C07H17/08 , Y02P20/55
摘要： Mycaminosyl tylonolide derivatives represented by the following general formula ##STR1## (wherein R.sup.1 denotes hydroxyl group, a lower alkanoyloxy group, benzoyloxy group, azido group, or amino group which mat optionally be substituted with a lower alkyl or a lower alkanoyl radical; R.sup.2 stands for hydrogen atom or hydroxyl group; R.sup.3 expresses hydrogen atom or formyl group; and means a double bond or a radical represented by ), and salts thereof.
摘要翻译：由以下通式表示的碳霉糖基太乐内酯衍生物（其中R 1表示羟基，低级烷酰氧基，苯甲酰氧基，叠氮基或任选被低级烷基或低级烷酰基取代的氨基）对于氢原子或羟基; R 3表示氢原子或甲酰基;并且表示双键或由...表示的基团）及其盐。

6. 发明授权

US4576931A 23-C-Substituted mycaminosyl tylonolide, pharmaceutical compositions and method of use 失效
标题翻译： 23-C-取代的碳霉糖太乐内酯，药物组合物和使用方法
公开(公告)号：US4576931A
公开(公告)日：1986-03-18
申请号：US719286
申请日：1985-04-03
申请人： Hamao Umezawa , Sumio Umezawa , Tsutomu Tsuchiya , Tomio Takeuchi , Akihiro Tanaka , Shuichi Sakamoto
发明人： Hamao Umezawa , Sumio Umezawa , Tsutomu Tsuchiya , Tomio Takeuchi , Akihiro Tanaka , Shuichi Sakamoto
IPC分类号： C07H17/08 , A61K31/78
CPC分类号： C07H17/08
摘要： Novel 23-C-substituted mycaminosyl tylonolide of the general formula (I) ##STR1## wherein R.sup.1 represents a lower alkyl group, an aryl group, a lower alkenyl group or a lower alkynyl group, R.sup.2 represents a hydrogen atom or a hydroxyl group.These compounds have excellent antibacterial activities.
摘要翻译：通式（I）的新型23-C取代的碳霉糖基太乐内酯其中R 1表示低级烷基，芳基，低级烯基或低级炔基，R 2表示氢原子或羟基。这些化合物具有优良的抗菌活性。

7. 发明授权

US4477443A Tylosin derivatives, their preparation and pharmaceutical compositions containing them 失效
标题翻译：泰乐菌素衍生物，它们的制剂和含有它们的药物组合物
公开(公告)号：US4477443A
公开(公告)日：1984-10-16
申请号：US395463
申请日：1982-07-06
申请人： Hamao Umezawa , Sumio Umezawa , Tsutomu Tsuchiya , Tomio Takeuchi , Akihiro Tanaka , Hidenori Iwamoto , Shuichi Sakamoto
发明人： Hamao Umezawa , Sumio Umezawa , Tsutomu Tsuchiya , Tomio Takeuchi , Akihiro Tanaka , Hidenori Iwamoto , Shuichi Sakamoto
IPC分类号： C07H17/08 , A61K31/71
CPC分类号： C07H17/08
摘要： Tylosin compounds of the formula ##STR1## wherein R.sub.1 represents a hydroxyl group; a halogen atom; ##STR2## group (wherein R.sub.5 is a hydrogen atom or a lower alkyl group which may be substituted by a hydroxyl group and R.sub.6 is a hydrogen atom, a lower alkyl group which may be substituted by a hydroxyl group, an aryl group, an aralkyl group, a cycloalkyl group having 3-10 carbon atoms, --CO(O).sub.m --R.sub.7 group (wherein m is 0 or 1 and R.sub.7 is a lower alkyl group, an aryl group, an aralkyl group, a furanyl group, or a pyridyl group), or --CH.sub.2 --R.sub.13 group (wherein R.sub.13 is a mono-, di-, or trifluoromethyl group)); --N(CH.sub.2).sub.n group (wherein n is an integer of 2-15) which may be substituted by an oxo group, a hydroxyl group, a lower alkyl group, or a hydroxy lower alkyl group; an imidazolyl group, a morpholino group, or a piperazino group each may be substituted by a lower alkyl group; or --OOCCH.sub.2 --R.sub.8 group (wherein R.sub.8 is ##STR3## group (wherein R.sub.9 and R.sub.10, which may be the same or different, each is a hydrogen atom or a lower alkyl group; said R.sub.9 and R.sub.10 may be combined with each other to form an alkylene group having 3-7 carbon atoms) or --S--R.sub.11 group (wherein R.sub.11 is a furanyl group or a pyridyl group)); R.sub.2 represents a hydrogen atom or a lower alkanoyl group; R.sub.3 represents a methyl group or --CH.sub.2 CHO group; R.sub.4 represents a hydrogen atom or a hydroxyl group; A represents 0.dbd., ##STR4## line represents a single bond or a double bond; and line ---- represents a single bond, a double bond, or ; however, when said R.sub.1 is a hydroxyl group, said R.sub.3 is a methyl group and R.sub.4 is a hydrogen atom, or said line ---- is ; or when said R.sub.1 is a halogen atom, said R.sub.3 is a methyl group of said line ---- is .The foregoing compounds of this invention are useful as antibiotics.
摘要翻译：式“IMAGE”的泰乐菌素化合物，其中R 1表示羟基; 卤素原子; 基（其中R5是氢原子或可被羟基取代的低级烷基，R6是氢原子，可被羟基取代的低级烷基，芳基，芳烷基基团，具有3-10个碳原子的环烷基，-CO（O）m-R7基团（其中m为0或1，R7为低级烷基，芳基，芳烷基，呋喃基或吡啶基）或-CH 2 -R 13基（其中R 13是单 - ，二 - 或三氟甲基））; -N（CH 2）n基（其中n为2-15的整数），其可被氧代基，羟基，低级烷基或羟基低级烷基取代; 咪唑基，吗啉代基或哌嗪子基各自可以被低级烷基取代; 或-OOCCH 2 -R 8基团（其中R 8为<基团）（其中R 9和R 10可以相同或不同，各自为氢原子或低级烷基;所述R 9和R 10可彼此组合形成具有3-7个碳原子的亚烷基）或-S-R11基（其中R11是呋喃基或吡啶基））; R2表示氢原子或低级烷酰基; R3表示甲基或-CH2CHO基; R4表示氢原子或羟基; A代表0 =，线代表单键或双键; 线----代表单键，双键，或; 然而，当所述R 1为羟基时，所述R 3为甲基，R 4为氢原子，或者当所述R 1为卤素原子时，所述R 3为所述线----甲基。本发明的前述化合物可用作抗生素。

8. 发明授权

US09112677B2 Communication device and cryptographic key creation method in cryptographic key sharing system 有权
标题翻译：密码密钥共享系统中的通信设备和加密密钥创建方法
公开(公告)号：US09112677B2
公开(公告)日：2015-08-18
申请号：US14110644
申请日：2012-04-06
申请人： Akihiro Tanaka , Akio Tajima
发明人： Akihiro Tanaka , Akio Tajima
IPC分类号： H04L9/00 , H04L9/08
CPC分类号： H04L9/0816 , H04L9/0838 , H04L9/0861 , H04L9/0894 , H04L2209/34
摘要： A communication device and a cryptographic key creation method are provided that enable efficient creation of cryptographic keys of which different error rates are required. A communication device (11) that performs communication with another communication device (12) through a transmission link includes a cryptographic key sharing section (1103) that share a first cryptographic key with the other communication device, an error rate control section (1115, 1105-1108) that creates second cryptographic keys with error rates according to purposes of use of the cryptographic keys from the first cryptographic key, and an accumulation section (111, 1112) that separately accumulates the plurality of second cryptographic keys with the different error rates.
摘要翻译：提供通信装置和加密密钥创建方法，其能够有效地创建需要不同错误率的密码密钥。通过传输链路与另一通信设备（12）进行通信的通信设备（11）包括：与其他通信设备共享第一密码密钥的密码密钥共享部分（1103），错误率控制部分（1115,1105） -1108），其根据来自第一密码密钥的加密密钥的目的产生具有错误率的第二加密密钥，以及累积部分（111,1112），其分别累积具有不同错误率的多个第二加密密钥。

9. 发明申请

US20120115368A1 Contact, and card adaptor and card connector having the same 有权
公开(公告)号：US20120115368A1
公开(公告)日：2012-05-10
申请号：US13351805
申请日：2012-01-17
申请人： Akihiro Tanaka , Yasuo Nakai
发明人： Akihiro Tanaka , Yasuo Nakai
IPC分类号： H01R24/28
CPC分类号： H01R12/57 , H01R12/714 , H01R12/87 , H01R13/2442 , H01R13/447 , H01R13/6583 , H01R31/06 , H01R43/16
摘要： In a contact of the present invention, a first plate spring piece portion 11c having a first fulcrum portion 11b in one side extends in a cantilevered manner from the first fulcrum portion 11b in a direction opposite to a card insertion direction so as to be elastically deformable in a thickness direction of the card. A second plate spring piece portion 11e having in one side a second fulcrum portion 11d which is the other side of the first plate spring piece portion 11c is formed in a shape where the second plate spring piece portion extends at an inclination angle from the second fulcrum portion 11d in the card insertion direction so as to be elastically deformable in the card thickness direction. The other side of the second plate spring piece portion 11e is to be contacted with the contact pad 2 of the card 1.

10. 发明授权

US08089193B2 Automotive alternator having brush device covered with surrounding wall 有权
标题翻译：具有覆盖有周围壁的刷装置的汽车交流发电机
公开(公告)号：US08089193B2
公开(公告)日：2012-01-03
申请号：US12219370
申请日：2008-07-21
申请人： Akihiro Tanaka , Hiroshi Ishida
发明人： Akihiro Tanaka , Hiroshi Ishida
IPC分类号： H01R39/38 , H02K13/00
CPC分类号： H02K5/141 , H02K2205/09
摘要： An alternator for generating electric power is mounted on an automotive vehicle. The alternator includes a housing, a stator fixed in the housing, a rotor driven by an engine of the automotive vehicle, and electric components such as a brush holder. The brush holder is mounted on a rear surface of a rear frame constituting the housing and is covered with a rear cover fixed to the rear frame. The rear cover includes a surrounding wall covering the brush device to prevent water from reaching a brush area. The surrounding wall is composed of plural partial walls having respective radiuses from a rotational axis of the rotor. The surrounding wall may be continuously made by the partial walls. Alternatively, openings for draining water may be formed in the partial walls positioned downward of the rotational axis of the rotor.
摘要翻译：用于发电的交流发电机安装在机动车辆上。交流发电机包括壳体，固定在壳体中的定子，由机动车辆的发动机驱动的转子以及诸如电刷架的电气部件。刷架安装在构成壳体的后框架的后表面上，并且被固定到后框架的后盖覆盖。后盖包括覆盖刷装置的周围壁，以防止水到达刷子区域。周围的壁由具有来自转子的旋转轴线的相应半径的多个部分壁组成。周围的壁可以由部分壁连续地制成。或者，可以在位于转子的旋转轴线的下方的部分壁中形成用于排水的开口。

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