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1. 发明授权

US5763461A Therapeutic phenoxyalkylheterocycles 失效
标题翻译：治疗苯氧基烷基杂环
公开(公告)号：US5763461A
公开(公告)日：1998-06-09
申请号：US822995
申请日：1997-03-21
申请人： David J. Aldous , Thomas R. Bailey , Guy Dominic Diana , Gee-Hong Kuo , Theodore J. Nitz
发明人： David J. Aldous , Thomas R. Bailey , Guy Dominic Diana , Gee-Hong Kuo , Theodore J. Nitz
IPC分类号： C07D401/12 , C07D403/12 , C07D405/12 , C07D413/12 , C07D471/04 , A61K31/44 , A61K31/415 , A61K31/47 , A61K31/505 , C07D213/16 , C07D239/26 , C07D401/10 , C07D403/10
CPC分类号： C07D401/12 , C07D403/12 , C07D405/12 , C07D413/12 , C07D471/04
摘要： Compounds of the formula ##STR1## wherein Pyr is chosen from the group consisting of pyridyl, pyrazyl, pyrimidyl, quinolyl, indolyl and 7-azaindolyl or any of these substituted with one or two substitutents chosen from alkyl, alkoxy, hydroxy, halo, cyano, nitro, hydroxyalkyl, alkoxyalkyl, alkanoyl, fluoroalkyl or the N-oxide of any of these; Y is an alkylene bridge of 3-9 carbon atoms; R.sub.1 and R.sub.2 are each independently chosen from hydrogen, halo, alkyl, alkenyl, amino, alkylthio, hydroxy, hydroxyalkyl, alkoxyalkyl, alkylthioalkyl, alkylsulfinylaikyl, alkylsulfonylalkyl, alkoxy, nitro, carboxy, alkoxycarbonyl, dialkylaminoalkyl, alkylaminoalkyl, aminoalkyl, difluoromethyl, trifluoromethyl or cyano; R.sub.3 is alkoxycarbonyl, alkyltetrazolyl, phenyl or heterocyclyl chosen from benzoxazolyl, benzathiazolyl, thiadiazolyl, imidazolyl, dihydroimidazolyl, oxazolyl, thiazolyl, oxadiazolyl, pyrazolyl, isoxazolyl, isothiazolyl, furyl, triazolyl, thiophenyl, pyridyl, pyrimidinyl, pyrazlnyl, pyridazinyl or a substituted phenyl or substituted heterocyclyl wherein the substitution is with alkyl, alkoxyalkyl, cycloalkyl, halo alkyl, hydroxyalkyl, alkoxy, hydroxy, furyl, or thienyl or fluoroalkyl, the N-oxide thereof, or a pharmaceutically acceptable acid addition salt thereof is an effective antipicornaviral agents.
摘要翻译：下式的化合物其中Pyr选自吡啶基，吡唑基，嘧啶基，喹啉基，吲哚基和7-氮杂吲哚基，或者被一个或两个选自烷基，烷氧基，羟基，卤代的取代基取代的那些氰基，硝基，羟基烷基，烷氧基烷基，烷酰基，氟代烷基或其中任何一种的N-氧化物; Y是3-9个碳原子的亚烷基桥; R 1和R 2各自独立地选自氢，卤素，烷基，烯基，氨基，烷硫基，羟基，羟基烷基，烷氧基烷基，烷硫基烷基，烷基亚磺酰基烷基，烷基磺酰基烷基，烷氧基，硝基，羧基，烷氧基羰基，二烷基氨基烷基，烷基氨基烷基，氨基烷基，二氟甲基，三氟甲基或氰基; R3是烷氧基羰基，烷基四唑基，苯基或选自苯并恶唑基，苯并噻唑基，噻二唑基，咪唑基，二氢咪唑基，恶唑基，噻唑基，恶二唑基，吡唑基，异唑基，异噻唑基，呋喃基，三唑基，噻吩基，吡啶基，嘧啶基，吡嗪基，哒嗪基或取代苯基或取代的杂环基，其中取代为烷基，烷氧基烷基，环烷基，卤代烷基，羟基烷基，烷氧基，羟基，呋喃基或噻吩基或氟代烷基，其N-氧化物或其药学上可接受的酸加成盐是有效的抗虫病毒药剂。

2. 发明授权

US5750527A Thiadiazoles and their use as antipicornaviral agents 失效
标题翻译：噻二唑及其作为止痛药物的用途
公开(公告)号：US5750527A
公开(公告)日：1998-05-12
申请号：US863388
申请日：1997-05-27
申请人： David J. Aldous , Thomas R. Bailey , Guy Dominic Diana , Theodore J. Nitz
发明人： David J. Aldous , Thomas R. Bailey , Guy Dominic Diana , Theodore J. Nitz
IPC分类号： C07D285/12 , A61K31/41 , A61K31/42 , A61K31/425 , A61K31/433 , A61K31/44 , A61K31/495 , A61K31/505 , A61P31/12 , A61P31/14 , C07D285/06 , C07D285/08 , C07D285/10 , C07D285/13 , C07D417/12 , A61K31/50
CPC分类号： C07D417/12
摘要： Described herein are compound of the formula: ##STR1## wherein: Thi is thiadiazolyl or substituted thiadiazolyl; Y is alkylene bridge of 3-9 carbon atoms; R.sub.1 and R.sub.2 are each independently chosen from hydrogen, halo, alkyl, alkenyl, amino, alkylthio, hydroxy, hydroxyalkyl, alkoxyalkyl, alkylthioalkyl, alkylsulfinyl alkyl, alkylsulfonylalkyl, alkoxy, nitro, carboxy, alkoxycarbonyl, dialkylaminoalkyl, alkylaminoalkyl, aminoalkyl, difluoromethyl, trifluoromethyl, or cyano; R.sub.3 is a heterocyclyl chosen from pyrimidinyl, pyrazinyl, or pyridazinyl; or a pharmaceutically acceptable salt thereof which are effective antipicornaviral agents.
摘要翻译：本文描述的是下式的化合物：其中：Thi是噻二唑基或取代的噻二唑基; Y是3-9个碳原子的亚烷基桥; R 1和R 2各自独立地选自氢，卤素，烷基，烯基，氨基，烷硫基，羟基，羟基烷基，烷氧基烷基，烷硫基烷基，烷基亚磺酰基烷基，烷基磺酰基烷基，烷氧基，硝基，羧基，烷氧基羰基，二烷基氨基烷基，烷基氨基烷基，氨基烷基，二氟甲基，，或氰基; R3是选自嘧啶基，吡嗪基或哒嗪基的杂环基; 或其药学上可接受的盐是有效的抗虫病毒药剂。

3. 发明授权

US5821257A Thiadiazoles and their uses as antipicornaviral agents 失效
标题翻译：噻二唑及其作为止痛药物的用途
公开(公告)号：US5821257A
公开(公告)日：1998-10-13
申请号：US52178
申请日：1998-03-31
申请人： David J. Aldous , Thomas R. Bailey , Guy Dominic Diana , Theodore J. Nitz
发明人： David J. Aldous , Thomas R. Bailey , Guy Dominic Diana , Theodore J. Nitz
IPC分类号： C07D285/12 , A61K31/41 , A61K31/42 , A61K31/425 , A61K31/433 , A61K31/44 , A61K31/495 , A61K31/505 , A61P31/12 , A61P31/14 , C07D285/06 , C07D285/08 , C07D285/10 , C07D285/13 , C07D417/12
CPC分类号： C07D417/12
摘要： Compounds of the formula; ##STR1## wherein: Thi is thiadiazolyl or substituted thiadiazolyl alkoxy, fluoromethyl, difluoromethyl, trifluoromethyl, 1,1-difluoroethyl, halo, alkyl, cycloalkyl, hydroxyalkyl, or Y is alkylene bridge of 3-9 carbon atoms; R.sub.1 and R.sub.2 are each independently chosen from hydrogen, halo, alkyl, alkenyl, amino, alkylthio, hydroxy, hydroxyalkyl, alkoxyalkyl, alkylthioalkyl, alkylsulfinyl alkyl, alkylsulfonylalkyl, alkoxy, nitro, carboxy, alkoxycarbonyl, dialkylaminoalkyl, alkylaminoalkyl, aminoalkyl, difluoromethyl, trifluoromethyl, or cyano; R.sub.3 is a heterocyclyl chosen from benzoxazolyl, benzathiazolyl, thiadiazolyl, oxazolyl, thiazolyl, oxadiazolyl, isoxazolyl, isothiazolyl, or substituted heterocyclyl wherein the substitution is with alkyl, alkoxyalkyl, cycloalkyl, haloalkyl, hydroxyalkyl, alkoxy, hydroxy, furyl, thienyl, or fluoroalkyl; or a pharmaceutically acceptable salt thereof are effective antipicornaviral agents.
摘要翻译：式的化合物; 式I其中：Thi是噻二唑基或取代的噻二唑基烷氧基，氟甲基，二氟甲基，三氟甲基，1,1-二氟乙基，卤素，烷基，环烷基，羟烷基或Y是3-9个碳原子的亚烷基桥; R 1和R 2各自独立地选自氢，卤素，烷基，烯基，氨基，烷硫基，羟基，羟基烷基，烷氧基烷基，烷硫基烷基，烷基亚磺酰基烷基，烷基磺酰基烷基，烷氧基，硝基，羧基，烷氧基羰基，二烷基氨基烷基，烷基氨基烷基，氨基烷基，二氟甲基，，或氰基; R3是选自苯并恶唑基，苯并噻唑基，噻二唑基，恶唑基，噻唑基，恶二唑基，异恶唑基，异噻唑基或取代的杂环基的杂环基，其中取代为烷基，烷氧基烷基，环烷基，卤代烷基，羟烷基，烷氧基，羟基，呋喃基，噻吩基或氟代烷基 ; 或其药学上可接受的盐是有效的抗虫病毒药剂。

4. 发明授权

US5650419A Thiadiazoles and their use as antipicornaviral agents 失效
标题翻译：噻二唑及其作为止痛药物的用途
公开(公告)号：US5650419A
公开(公告)日：1997-07-22
申请号：US706108
申请日：1996-08-30
申请人： David J. Aldous , Thomas R. Bailey , Guy Dominic Diana , Theodore J. Nitz
发明人： David J. Aldous , Thomas R. Bailey , Guy Dominic Diana , Theodore J. Nitz
IPC分类号： C07D285/12 , A61K31/41 , A61K31/42 , A61K31/425 , A61K31/433 , A61K31/44 , A61K31/495 , A61K31/505 , A61P31/12 , A61P31/14 , C07D285/06 , C07D285/08 , C07D285/10 , C07D285/13 , C07D417/12
CPC分类号： C07D417/12
摘要： Described herein are compounds of the formula; ##STR1## wherein: Thi is a unsubstituted or substituted thiadiazolyl;Y is an alkylene bridge of 3-9 carbon atoms;R.sub.1 and R.sub.2 are each independently chosen from hydrogen, halo, alkyl, alkenyl, amino, alkylthio, hydroxy, hydroxyalkyl, alkoxyalkyl, alkylthioalkyl, alkylsulfinylalkyl, alkylsulfonylalkyl, alkoxy, nitro, carboxy, alkoxylcarbonyl, dialkylaminoalkyl, alkylaminoalkyl, aminoalkyl, difluoromethyl, trifluoromethyl or cyano;R.sub.3 is alkoxycarbonyl, substituted or unsubstituted phenyl, alkyltetrazolyl or a substituted or unsubstituted imidazolyl, dihydroimidazolyl, pyrazolyl, furyl, thiazolyl or thienyl or a pharmaceutically acceptable salt thereof are effective antipicornaviral agents.
摘要翻译：本文描述的是式的化合物; 式I其中：Thi是未取代或取代的噻二唑基; Y是3-9个碳原子的亚烷基桥; R 1和R 2各自独立地选自氢，卤素，烷基，烯基，氨基，烷硫基，羟基，羟基烷基，烷氧基烷基，烷硫基烷基，烷基亚磺酰基烷基，烷基磺酰基烷基，烷氧基，硝基，羧基，烷氧基羰基，二烷基氨基烷基，烷基氨基烷基，氨基烷基，二氟甲基，氰基; R3是烷氧基羰基，取代或未取代的苯基，烷基四唑基或取代或未取代的咪唑基，二氢咪唑基，吡唑基，呋喃基，噻唑基或噻吩基或其药学上可接受的盐是有效的抗虫病毒剂。

5. 发明授权

US5846986A Therapeutic phenoxyalkylazoles and phenoxyalkylazines 失效
公开(公告)号：US5846986A
公开(公告)日：1998-12-08
申请号：US978233
申请日：1997-11-25
申请人： David J. Aldous , Thomas R. Bailey , Guy Dominic Diana , Theodore J. Nitz , Gee-Hong Kuo
发明人： David J. Aldous , Thomas R. Bailey , Guy Dominic Diana , Theodore J. Nitz , Gee-Hong Kuo
IPC分类号： C07D257/04 , C07D271/06 , C07D277/24 , C07D403/12 , C07D405/12 , C07D413/12 , C07D417/12 , C07D521/00 , A61K31/41
CPC分类号： C07D257/04 , C07D231/12 , C07D233/56 , C07D249/08 , C07D271/06 , C07D277/24 , C07D403/12 , C07D405/12 , C07D413/12 , C07D417/12
摘要： Compounds of the formula ##STR1## wherein Azo is alkyltetrazolyl or is chosen from the group consisting of oxadiazolyl, imidazolyl, pyrazolyl, triazolyl, oxazolyl, triazinyl, thiazolyl, isothiazolyl or any of these substituted with a member of the group consisting of alkyl, alkylthio, alkoxy, hydroxy, halo, cyano, nitro, hydroxyalkyl, alkoxyalkyl, alkoxycarbonyl, alkanoyl, fluoroalkyl or the N-oxide of any of the preceding; Y is an alkylene bridge of 3-9 carbon atoms; R.sub.1 and R.sub.2 are each individually chosen from hydrogen, halo, alkyl, alkenyl, amino, alkylthio, hydroxy, hydroxyalkyl, alkoxyalkyl, alkylthioalkyl, alkylsulfinylalkyl, alkylsulfonylalkyl, alkoxy, nitro, carboxy, alkoxycarbonyl, dialkylaminoalkyl, alkylaminoalkyl, aminoalkyl, difluoromethyl, trifluoromethyl or cyano; R.sub.3 is alkoxycarbonyl, alkyltetrazolyl, phenyl or a heterocycle chosen from benzoxazolyl, benzathiazolyl, thiadiazolyl, imidazolyl, dihydroimidazolyl, oxazolyl, thiazolyl, oxadiazolyl, pyrazolyl, isoxazolyl, isothiazolyl, furyl, triazolyl, tetrazolyl, thiophenyl, pyridyl, pyrimidinyl, pyrazinyl, pyridazinyl or substituted phenylor substituted heterocyclyl wherein the substitution is with alkyl, alkoxyalkyl, cycloalkyl, haloalkyl, hydroxyalkyl, alkoxy, hydroxy, furyl, thienyl or fluoroalkyl; the N-oxide thereof; or a pharmaceutically acceptable acid addition salt thereof is an effective antipicornaviral agents.

6. 发明授权

US5721261A Therapeutic phenoxyalkylazoles and phenoxyalkylazines 失效
标题翻译：治疗性苯氧基烷基唑和苯氧基烷基嗪
公开(公告)号：US5721261A
公开(公告)日：1998-02-24
申请号：US693530
申请日：1996-08-02
申请人： David J. Aldous , Thomas R. Bailey , Guy Dominic Diana , Theodore J. Nitz , Gee-Hong Kuo
发明人： David J. Aldous , Thomas R. Bailey , Guy Dominic Diana , Theodore J. Nitz , Gee-Hong Kuo
IPC分类号： C07D257/04 , C07D271/06 , C07D277/24 , C07D403/12 , C07D405/12 , C07D413/12 , C07D417/12 , C07D521/00 , A61K31/41
CPC分类号： C07D257/04 , C07D231/12 , C07D233/56 , C07D249/08 , C07D271/06 , C07D277/24 , C07D403/12 , C07D405/12 , C07D413/12 , C07D417/12
摘要： Compounds of the formula ##STR1## wherein Azo is alkyltetrazolyl or is chosen from the group consisting of oxadiazolyl, imidazolyl, pyrazolyl, triazolyl, oxazolyl, triazinyl, thiazolyl, isothiazolyl or any of these substituted with a member of the group consisting of alkyl, alkylthio, alkoxy, hydroxy, halo, cyano, nitro, hydroxyalkyl, alkoxyalkyl, alkoxycarbonyl, alkanoyl, fluoroalkyl or the N-oxide of any of the preceding; Y is an alkylene bridge of 3-9 carbon atoms; R.sub.1 and R.sub.2 are each individually chosen from hydrogen, halo, alkyl, alkenyl, amino, alkylthio, hydroxy, hydroxyalkyl, alkoxyalkyl, alkylthioalkyl, alkylsulfinylalkyl, alkylsulfonylalkyl, alkoxy, nitro, carboxy, alkoxycarbonyl, dialkylaminoalkyl, alkylaminoalkyl, aminoalkyl, difluoromethyl, trifluoromethyl or cyano; R.sub.3 is alkoxycarbonyl, alkyltetrazolyl, phenyl or a heterocycle chosen from benzoxazolyl, benzathiazolyl, thiadiazolyl, imidazolyl, dihydroimidazolyl, oxazolyl, thiazolyl, oxadiazolyl, pyrazolyl, isoxazolyl, isothiazolyl, furyl, triazolyl, tetrazolyl, thiophenyl, pyridyl, pyrimidinyl, pyrazinyl, pyridazinyl or substituted phenylor substituted heterocyclyl wherein the substitution is with alkyl, alkoxyalkyl, cycloalkyl, haloalkyl, hydroxyalkyl, alkoxy, hydroxy, furyl, thienyl or fluoroalkyl; the N-oxide thereof; or a pharmaceutically acceptable acid addition salt thereof is an effective antipicornaviral agents.
摘要翻译：式I的化合物，其中偶氮是烷基四唑基或选自恶二唑基，咪唑基，吡唑基，三唑基，恶唑基，三嗪基，噻唑基，异噻唑基或其中任何一个被烷基取代的基团，烷硫基，烷氧基，羟基，卤素，氰基，硝基，羟基烷基，烷氧基烷基，烷氧基羰基，烷酰基，氟代烷基或任何前述的N-氧化物; Y是3-9个碳原子的亚烷基桥; R 1和R 2各自独立地选自氢，卤素，烷基，烯基，氨基，烷硫基，羟基，羟基烷基，烷氧基烷基，烷硫基烷基，烷基亚磺酰基烷基，烷基磺酰基烷基，烷氧基，硝基，羧基，烷氧基羰基，二烷基氨基烷基，烷基氨基烷基，氨基烷基，二氟甲基，三氟甲基或氰基; R3是烷氧基羰基，烷基四唑基，苯基或选自苯并恶唑基，苯并噻唑基，噻二唑基，咪唑基，二氢咪唑基，恶唑基，噻唑基，恶二唑基，吡唑基，异恶唑基，异噻唑基，呋喃基，三唑基，四唑基，噻吩基，吡啶基，嘧啶基，吡嗪基，哒嗪基或取代的苯基或取代的杂环基，其中取代为烷基，烷氧基烷基，环烷基，卤代烷基，羟基烷基，烷氧基，羟基，呋喃基，噻吩基或氟代烷基; 其N-氧化物; 或其药学上可接受的酸加成盐是有效的抗虫病毒药剂。

7. 发明授权

US5665763A Therapeutic phenoxyalkylpyridazines and intermediates therefor 失效
标题翻译：治疗性苯氧基烷基哒嗪及其中间体
公开(公告)号：US5665763A
公开(公告)日：1997-09-09
申请号：US706109
申请日：1996-08-30
申请人： David J. Aldous , Thomas R. Bailey , Guy Dominic Diana , Theodore J. Nitz
发明人： David J. Aldous , Thomas R. Bailey , Guy Dominic Diana , Theodore J. Nitz
IPC分类号： C07D237/08 , C07D307/42 , C07D403/12 , C07D405/04 , C07D405/12 , C07D407/04 , C07D413/12 , C07D413/14 , A61K31/34 , A61K31/38 , C07D409/12
CPC分类号： C07D307/42 , C07D237/08 , C07D403/12 , C07D405/04 , C07D405/12 , C07D407/04 , C07D413/12 , C07D413/14
摘要： Compounds of the formula ##STR1## wherein: R.sub.1, R.sub.2, R.sub.3 and R.sub.4 are as defined in the specification,Y is alkylene of 3 to 9 carbon atoms,R.sub.5 is alkoxycarbonyl, alkyltetrazolyl, phenyl or a heterocycle chosen from benzoxazolyl, benzathiazolyl, thiadiazolyl, imidazolyl, dihydroimidazolyl, oxazolyl, thiazolyl, oxadiazolyl, pyrazolyl, oxazolinyl, isoxazolyl, isothiazolyl, furyl, triazolyl, thiophenyl, pyridyl, pyrimidinyl, pyrazinyl, pyridazinyl or any of the above substituted with alkyl, alkoxyalkyl, cycloalkyl, halo alkyl, hydroxyalkyl, alkoxy, hydroxy, halo, furyl, thienyl, fluoroalkyl;or a pharmaceutically acceptable acid addition salts thereof; N-oxides thereof, are useful as antipirconaviral agents.
摘要翻译：其中：R1，R2，R3和R4如说明书中所定义，Y是3至9个碳原子的亚烷基，R 5是烷氧基羰基，烷基四唑基，苯基或选自苯并恶唑基的杂环，苯并噻唑基，噻二唑基，咪唑基，二氢咪唑基，恶唑基，噻唑基，恶二唑基，吡唑基，恶唑啉基，异恶唑基，异噻唑基，呋喃基，三唑基，噻吩基，吡啶基，嘧啶基，吡嗪基，哒嗪基或任何上述被烷基，烷氧基烷基，环烷基，，羟基烷基，烷氧基，羟基，卤素，呋喃基，噻吩基，氟代烷基; 或其药学上可接受的酸加成盐; 其N-氧化物可用作抗血管病毒药物。

8. 发明授权

US4096280A Arylenedioxy-bis-diketones 失效
标题翻译：亚芳基二氧基双二酮
公开(公告)号：US4096280A
公开(公告)日：1978-06-20
申请号：US761944
申请日：1977-01-24
申请人： Guy Dominic Diana , Philip Michael Carabateas
发明人： Guy Dominic Diana , Philip Michael Carabateas
IPC分类号： A61K31/12 , A61P31/12 , C07C45/00 , C07C45/68 , C07C49/16 , C07C49/175 , C07C67/00 , C07C49/84 , A01N9/24
CPC分类号： C07C45/68 , C07C45/71 , C07C49/255
摘要： Phenylenedioxy-bis-dikeones having the formula ##STR1## useful as antiviral agents, are prepared by etherification of dihydric phenols and alkylation of beta-dikeones.
摘要翻译：可用作抗病毒剂的具有式“IMAGE”的亚苯基二氧基双二酮通过二元酚的醚化和β-二酮的烷基化来制备。

9. 发明授权

US5643929A 1,2,4-oxidiazolyl-phenoxyalkylisoxazoles and their use as antiviral agents 失效
标题翻译： 1,2,4-氧化噻吩基 - 苯氧基烷基异恶唑及其作为抗病毒剂的用途
公开(公告)号：US5643929A
公开(公告)日：1997-07-01
申请号：US444795
申请日：1995-05-19
申请人： Guy Dominic Diana , Theodore John Nitz
发明人： Guy Dominic Diana , Theodore John Nitz
IPC分类号： A61K31/42 , A61K31/422 , A61K31/4245 , A61P31/12 , C07D413/12 , C07D413/14 , A01K31/41
CPC分类号： C07D413/10 , C07D413/12 , C07D413/14
摘要： Compounds of the formula ##STR1## wherein: R.sub.1 is alkyl, alkoxy, hydroxy, cycloalkyl, hydroxyalkyl, alkoxyalkyl, hydroxyalkoxy, alkylthioalkyl, alkylsulfinylalkyl, alkylsulfonylalkyl, aminoalkyl, alkylaminoalkyl, dialkylaminoalkyl, alkoxycarbonyl, carboxy, or cyanomethyl;Y is alkylene of 3 to 9 carbon atoms,R.sub.2 and R.sub.3 independently are hydrogen, alkyl, alkoxy, halo, cyano, trifluoromethyl and nitro;R.sub.4 is alkoxy, hydroxy, halomethyl, dihalomethyl, trihalomethyl, dihaloethyl, cycloalkyl, heterocyclyl, alkoxycarbonyl, hydroxyalkyl, alkoxyalkyl, alkanecarbonyloxyalkyl, cyano, halo, thioalkyl, alkylthioalkyl, alkylthio, thio, 2,2,2-trifluoro-ethyl, (4-methylphenyl)sulfonyloxymethyl, N=Q or CON=Q, where N=Q is amino, alkylamino or dialkylamino;R.sub.5 is hydrogen or halo or alkyl.
摘要翻译：其中：R1是烷基，烷氧基，羟基，环烷基，羟基烷基，烷氧基烷基，羟基烷氧基，烷基硫代烷基，烷基亚磺酰基烷基，烷基磺酰基烷基，氨基烷基，烷基氨基烷基，二烷基氨基烷基，烷氧基羰基，羧基或氰基甲基。 Y是3至9个碳原子的亚烷基，R2和R3独立地是氢，烷基，烷氧基，卤素，氰基，三氟甲基和硝基; R4是烷氧基，羟基，卤代甲基，二卤代甲基，三卤代甲基，二卤代乙基，环烷基，杂环基，烷氧基羰基，羟基烷基，烷氧基烷基，烷基羰氧基烷基，氰基，卤素，硫代烷基，烷基硫代烷基，烷硫基，硫代，2,2,2-三氟乙基，（4 - 甲基苯基）磺酰氧基甲基，N = Q或CON = Q，其中N = Q是氨基，烷基氨基或二烷基氨基; R5是氢或卤素或烷基。

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