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41. 发明申请

US20100029668A1 NOVEL PYRIDAZINE DERIVATIVES 审中-公开
标题翻译：新的吡咯烷酮衍生物
公开(公告)号：US20100029668A1
公开(公告)日：2010-02-04
申请号：US12374052
申请日：2007-07-16
申请人： Stephan Trah , Clemens Lamberth , Sebastian Volker Wendeborn
发明人： Stephan Trah , Clemens Lamberth , Sebastian Volker Wendeborn
IPC分类号： A01N43/58 , C07D405/04 , A01P3/00
CPC分类号： C07D401/14 , A01N43/58 , C07D403/14 , C07D405/14 , C07D407/14 , C07D409/14 , C07D417/14
摘要： The present invention relates to novel pyridazine derivatives of formula (I) as active ingredients which have microbiocidal activity, in particular fungicidal activity: wherein R1 is hydrogen, C1-C6alkyl, C1-C6haloalkyl or C3-C6cycloalkyl; R2 is an optionally substituted heteroaryl; R3 is an optionally substituted heteroaryl; and R4 is hydrogen, halogen, C1-C6alkyl, C1-C6haloalkyl, C1-C6alkoxy, C1-C6haloalkoxy, hydroxy or cyano; or an agrochemically usable salt form thereof.
摘要翻译：本发明涉及具有杀微生物活性，特别是杀真菌活性的活性成分的式（I）的新哒嗪衍生物，其中R1是氢，C1-C6烷基，C1-C6卤代烷基或C3-C6环烷基; R2是任选取代的杂芳基; R3是任选取代的杂芳基; R4是氢，卤素，C1-C6烷基，C1-C6卤代烷基，C1-C6烷氧基，C1-C6卤代烷氧基，羟基或氰基; 或其农业化学上可用的盐形式。

42. 发明授权

US06989394B2 Tetrahydropyridines 失效
公开(公告)号：US06989394B2
公开(公告)日：2006-01-24
申请号：US10651688
申请日：2003-08-29
申请人： Stephan Trah
发明人： Stephan Trah
IPC分类号： A01N43/40 , C07D401/10
CPC分类号： C07D401/10 , A01N43/40 , A01N43/58 , A01N43/713 , A01N47/20 , C07D211/70 , C07D211/94
摘要： Compounds of formula are described, wherein R1 and R2 are for example, independently of each other, halogen, C1-C6-alkyl, C3-C6-cycloalkyl, halogen-C1-C6-alkyl, halogen-C3-C6-cycloalkyl, C2-C4-alkenyl, C2-C4-alkinyl, halogen-C2-C4-alkenyl and halogen-C2-C4-alkinyl; R3 is hydrogen, OH, halogen, C1-C6-alkoxy, or —O—C(═O)—C1-C6-alkyl; R4 is for example phenyl, benzyl, phenoxy or benzyloxy, which is substituted by substituents selected from the group consisting of halogen, cyano, NO2, C1-C6-alkyl, C3-C8-cycloalkyl, C3-C8-cyclalkyl-C1-C6-alkyl, halogen-C1-C6-alkyl, C1-C6-alkoxy, C3-C8-cycloalkoxy, C3-C8-cycloalkoxy-C1-C6-alkyl, C3-C8-cycloalkoxy-C1-C6-alkoxy, halogen-C1-C6-alkoxy, C2-C4-alkenyl, C2-C4-alkinyl, halogen-C2-C4-alkenyl, halogen-C2-C4-alkinyl, C2-C6-alkenyloxy, C2-C6-alkinyloxy, halogen-C2-C6-alkenyloxy, halogen-C2-C6-alkinyloxy, —NR6—C(═O)—O—C1-C6-alkyl, —NR6—C(═O)—O-halogen-C1-C6-alkyl, —C(R7)═N—W—R8, phenyl, benzyl, phenoxy, benzyloxy, heterocycyl and heterocyclyoxy; the two R5 independently of one another, are hydrogen or C1-C6-alkyl; R6 is hydrogen, C1-C6-alkyl or benzyl; R7 is for example halogen or C1-C6-alkyl; R8 is for example hydrogen or C1-C6-alkyl; m is 0, 1, 2, 3, 4 or 5; n is 0, 1, 2, 3, 4 or 5; p is 0, 1 or 2; q is 0 or 1; W is O or NH or N—C1-C6-alkyl; a method of producing and the use of these compounds, pesticides whose active ingredient is selected from these compounds or from an agrochemically employable salt thereof, a method of producing and the use of these compositions, plant propagating material that has been treated with these compositions and a method of controlling pests.

43. 发明授权

US06953811B2 N-substituted tetrahydropyridines and their use as pesticides 失效
标题翻译： N-取代四氢吡啶类及其作为农药的用途
公开(公告)号：US06953811B2
公开(公告)日：2005-10-11
申请号：US10470790
申请日：2002-02-04
申请人： Stephan Trah , Josef Ehrenfreund , Peter Maienfisch , André Jeanguenat , Saleem Farooq
发明人： Stephan Trah , Josef Ehrenfreund , Peter Maienfisch , André Jeanguenat , Saleem Farooq
IPC分类号： A01N43/40 , C07D211/70 , C07D211/94 , C07D401/06
CPC分类号： C07D401/06 , C07D211/70 , C07D211/94
摘要： A description is given of compounds of the formula in which R1 and R2 independently of one another are halogen, C1-C6alkyl, halo-C1-C6alkyl, C1-C6alkoxy, halo-C1-C6alkoxy, or SF5, R3 is hydrogen, OH, halogen, C1-C6alkoxy or —O—C(═O)—C1-C6alkyl, R4 is for example hydrogen, halogen, C1-C6alkyl, halo-C1-C6alkyl, C1-C6alkoxy, halo-C1-C6alkoxy or SCN; R5 and R6 independently of one another are for example hydrogen, C1-C12alkyl, halo-C1-C12alkyl, C2-C12alkenyl, halo-C2-C12alkenyl or C2-C12alkynyl; and q is 0 or 1; and, where appropriate, E/Z isomers, E/Z isomer mixtures and/or tautomers, each in free form or in salt form; a process for the preparation of these compounds and their use, pesticide compositions whose active ingredient is selected from these compounds, or an agrochemically useable salt thereof, a process for preparing these compositions, and their use, plant propagation material treated with these compositions, and a method of combating pests.
摘要翻译：给出下式的化合物，其中R 1和R 2彼此独立地是卤素，C 1 -C 3 C 6 -C 6烷基，卤代C 1 -C 6烷基，C 1 -C 6烷基，C 1 -C 6烷基，C 1 -C 6烷基，烷氧基，卤代-C 1 -C 6烷氧基或SF 5，R 3是氢，OH，卤素，C 1 -C 6烷氧基或-OC（-O）-C 1 -C 6 -C 6烷基 R 4是例如氢，卤素，C 1 -C 6烷基，卤代C 1 -C 4烷基， C 1 -C 6烷基，C 1 -C 6烷氧基，卤代C 1 -C 6烷基，C 1 -C 6烷氧基，C 1 -C 6烷基，烷氧基或SCN; R 5和R 6彼此独立地是例如氢，C 1 -C 12 - 烷基，卤代 C 1 -C 12烷基，C 2 -C 12链烯基，卤代-C 2烷基，C 1 -C 12烷基，C 2 -C 12 - C 12 -C 12链烯基或C 2 -C 12 - 炔基; q为0或1; 和/或互变异构体，各自为游离形式或盐形式的E / Z异构体，E / Z异构体混合物和/或互变异构体; 制备这些化合物及其用途的方法，其活性成分选自这些化合物的农药组合物或其农业上可用的盐，这些组合物的制备方法及其用途，用这些组合物处理的植物繁殖材料，以及一种防治害虫的方法。

44. 发明授权

US5977182A O-benzyl oxime ether derivatives and their use as pesticides 失效
标题翻译： O-苄基肟醚衍生物及其作为农药的用途
公开(公告)号：US5977182A
公开(公告)日：1999-11-02
申请号：US836176
申请日：1997-05-01
申请人： Rene Zurfluh , Hugo Ziegler , Stephan Trah
发明人： Rene Zurfluh , Hugo Ziegler , Stephan Trah
IPC分类号： A01C1/08 , A01N35/10 , A01N37/34 , A01N37/50 , A01N37/52 , A01N55/10 , C07C251/38 , C07C251/48 , C07C251/52 , C07C251/54 , C07C251/60 , C07C255/62 , C07C255/64 , C07C257/06 , C07C257/14 , C07C257/22 , C07C317/32 , C07C323/47 , C07C327/40 , C07C327/58 , C07D213/76 , C07D277/10 , C07D277/12 , C07D277/28 , C07D295/185 , C07D295/30 , C07D521/00 , A01N33/24 , A01N43/40
CPC分类号： C07D295/185 , A01N37/50 , A01N37/52 , C07C251/38 , C07C251/48 , C07C255/64 , C07C257/06 , C07C257/14 , C07C257/22 , C07D295/30 , C07C2101/02
摘要： Compounds of formula (I), wherein Y is hydrogen, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy, OH, CN, NO.sub.2, Si(CH.sub.3).sub.3, CF.sub.3 or halogen, and T is a group (a) or (b), and wherein the remaining substituents have the following definitions: X is O, S or NR.sub.13 ; A is O or NR.sub.4 ; R.sub.1 is hydrogen, C.sub.1 -C.sub.4 alkyl, halo-C.sub.1 -C.sub.4 alkyl, cyclopropyl, C.sub.1 -C.sub.4 alkoxymethyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 alkylthio or cyano; R.sub.2 is hydrogen, C.sub.1 -C.sub.6 alkyl, C.sub.3 -C.sub.6 cycloalkyl, cyano unsubstituted or substituted C.sub.1 -C.sub.6 alkoxycarbonyl, unsubstituted or substituted di(C.sub.1 -C.sub.6 alkyl)aminocarbonyl, unsubstituted or substituted C.sub.1 -C.sub.6 alkyl-S(O).sub.q, unsubstituted or substituted aryl-S(O).sub.q, unsubstituted or substituted heteroaryl, unsubstituted or substituted heterocyclyl, unsubstituted or substituted heterocyclylcarbonyl or unsubstituted or substituted phenyl; and R.sub.3 is hydrogen, unsubstituted or substituted alkyl, unsubstituted or substituted C.sub.3 -C.sub.6 cycloalkyl, unsubstituted or substituted phenyl or unsubstituted or substituted pyridyl; and wherein the remaining substituents are as defined herein, are pesticidal active ingredients. They can be used in pest control, especially as microbicides, insecticides and acaricides in agriculture, in horticulture and in the hygiene sector. ##STR1##
摘要翻译： PCT No.PCT / EP95 / 04357 Sec。 371日期1997年5月1日 102（e）日期1997年5月1日PCT提交1995年11月6日PCT公布。公开号WO96 / 16026 日期：5月30日，式（I）的化合物，其中Y为氢，C1-C4烷基，C1-C4烷氧基，OH，CN，NO2，Si（CH3）3，CF3或卤素，T为（a）或 b），其中其余取代基具有以下定义：X是O，S或NR 13; A为O或NR4; R 1是氢，C 1 -C 4烷基，卤代C 1 -C 4烷基，环丙基，C 1 -C 4烷氧基甲基，C 1 -C 4烷氧基，C 1 -C 4烷硫基或氰基; 未取代或取代的二（C 1 -C 6烷基）氨基羰基，未取代或取代的C 1 -C 6烷基-S（O）q，未取代或取代的芳基-S（O）q，C 1 -C 6烷基，C 3 -C 6环烷基，氰基未取代或取代的C 1 -C 6烷氧基羰基，（O）q，未取代或取代的杂芳基，未取代或取代的杂环基，未取代或取代的杂环基羰基或未取代或取代的苯基; 未取代或取代的烷基，未取代或取代的C 3 -C 6环烷基，未取代或取代的苯基或未取代或取代的吡啶基; 并且其中剩余的取代基如本文所定义，是杀虫活性成分。它们可用于病虫害防治，特别是作为农业，园艺和卫生领域的杀菌剂，杀虫剂和杀螨剂。

45. 发明授权

US5786374A Benzisoxazole derivatives and pesticidal compositions containing them 失效
标题翻译：苯并异恶唑衍生物和含有它们的杀虫组合物
公开(公告)号：US5786374A
公开(公告)日：1998-07-28
申请号：US836072
申请日：1997-05-01
申请人： Saleem Farooq , Stephan Trah , Rene Zurfluh
发明人： Saleem Farooq , Stephan Trah , Rene Zurfluh
IPC分类号： A01N43/80 , A01N55/00 , C07D261/20 , C07D413/02 , A61K31/42 , C07D263/56
CPC分类号： C07D261/20 , A01N43/80
摘要： The present invention relates to benzisoxazole compounds, pesticidal compositions containing them, and their preparations thereof.
摘要翻译： PCT No.PCT / EP95 / 04154 Sec。 371日期1997年5月1日 102（e）日期1997年5月1日PCT提交1995年10月23日PCT公布。公开号WO96 / 14305 日期1996年5月17日本发明涉及苯并异恶唑化合物，含有它们的杀虫组合物及其制备方法。

46. 发明授权

US5612338A Pyrazolyl acrylic acid derivatives, intermediates thereto, and in their use as microbicides 失效
标题翻译：吡唑基丙烯酸衍生物，其中间体及其作为杀微生物剂的用途
公开(公告)号：US5612338A
公开(公告)日：1997-03-18
申请号：US495532
申请日：1995-07-28
申请人： Stephan Trah
发明人： Stephan Trah
IPC分类号： C07D231/20 , A01N43/54 , A01N43/56 , A01N43/64 , A01N43/66 , C07D231/18 , C07D401/12 , C07D403/12
CPC分类号： C07D401/12 , A01N43/56 , A01N43/66 , C07D231/18 , C07D403/12
摘要： Compounds of the formula ##STR1## wherein R.sub.1 is hydrogen or methyl,R.sub.2 is hydrogen, halogen, OCH.sub.3, SCH.sub.3 or CN,R.sub.3, R.sub.4, R.sub.5 are each independently of one another hydrogen, halogen, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.2 -C.sub.5 alkoxycarbonyl, C.sub.1 -C.sub.5 alkanoyl, C.sub.1 -C.sub.4 haloalkyl, C.sub.1 -C.sub.4 haloalkoxy, CN, NO.sub.2, or wherein two of those substituents are adjacent to each other and together are a methylenedioxy or difluoromethylenedioxy radical,K, L, M are each independently of one another CH or N (=nitrogen atom), but at least one of these three substituents is N, andY is oxygen or sulfur,are effective microbicides for controlling fungal diseases. They can be used for plant protection by themselves or as formulated compositions.
摘要翻译： PCT No.PCT / EP94 / 00103 Sec。 371日期：1995年7月28日 102（e）日期1995年7月28日PCT 1994年1月17日PCT PCT。公开号WO94 / 17060 PCT 日期：1994年8月4日化学式其中R 1为氢或甲基，R 2为氢，卤素，OCH 3，SCH 3或CN，R 3，R 4，R 5各自独立地为氢，卤素，C 1 -C 4烷基， C 1 -C 4烷氧基，C 2 -C 5烷氧基羰基，C 1 -C 5烷酰基，C 1 -C 4卤代烷基，C 1 -C 4卤代烷氧基，CN，NO 2，或其中两个取代基彼此相邻并且一起是亚甲二氧基或二氟亚甲二氧基，K，L，M 各自独立地是CH或N（=氮原子），但这三个取代基中的至少一个是N，Y是氧或硫，是用于控制真菌疾病的有效的杀微生物剂。它们可以自己或作为配制的组合物用于植物保护。

47. 发明授权

US5606095A 2-aminooxymethylenephenylacetic acid derivatives 失效
标题翻译： 2-氨氧基亚甲基苯乙酸衍生物
公开(公告)号：US5606095A
公开(公告)日：1997-02-25
申请号：US462259
申请日：1995-06-05
申请人： Albert Pfiffner , Stephan Trah , Hugo Ziegler
发明人： Albert Pfiffner , Stephan Trah , Hugo Ziegler
IPC分类号： C07C239/08 , C07C239/20 , C07C255/57 , C07C323/23 , C07F9/38 , C07F9/40 , C07C229/00
CPC分类号： C07C239/20
摘要： 2-Aminooxymethylenephenylacetic acid ester derivatives of the formula ##STR1## wherein Z.sub.1 and Z.sub.2 are hydrogen, halogen, hydroxy, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy, C.sub.1 -C.sub.4 haloalkyl, C.sub.1 -C.sub.4 haloalkoxy, C.sub.1 -C.sub.4 alkylcarbonyl, phenoxy, nitro or cyano, or Z.sub.1 and Z.sub.2, together with the linking phenyl radical, are naphthalene or hydrogenated naphthalene, and R.sub.3 is hydrogen or C.sub.1 -C.sub.12 alkyl. The compounds of this invention may be used as the free base or as a protic acid salt and are important intermediates for the manufacture of microbicides for plant protection.
摘要翻译：式（I）的2-氨氧基亚甲基苯基乙酸酯衍生物其中Z 1和Z 2是氢，卤素，羟基，C 1 -C 4烷基，C 1 -C 4烷氧基，C 1 -C 4卤代烷基，C 1 -C 4卤代烷氧基，C 1 -C 4烷基羰基，苯氧基，硝基或氰基或Z 1和Z 2与连接的苯基一起是萘或氢化萘，并且R 3是氢或C 1 -C 12烷基。本发明的化合物可以用作游离碱或质子酸盐，并且是制备用于植物保护的杀微生物剂的重要中间体。

48. 发明授权

US5554735A Azo oxime ethers and their use as fungicides 失效
标题翻译：偶氮肟醚及其用作杀真菌剂
公开(公告)号：US5554735A
公开(公告)日：1996-09-10
申请号：US295775
申请日：1994-08-26
申请人： Hugo Ziegler , Stephan Trah
发明人： Hugo Ziegler , Stephan Trah
IPC分类号： C07D251/22 , A01N37/52 , A01N43/40 , C07C259/20 , C07C311/38 , C07C323/48 , C07D209/08 , C07D209/88 , C07D213/76 , C07D213/77 , C07D215/38 , C07D215/40 , C07D215/42 , C07D217/02 , C07D231/38 , C07D231/56 , C07D235/30 , C07D237/20 , C07D239/42 , C07D241/20 , C07D253/06 , C07D257/02 , C07D261/14 , C07D275/02 , C07D277/20 , C07D277/50 , C07D277/82 , C07D285/06 , C07D285/12 , C07D285/135 , C07D285/18 , C07D295/12 , C07D311/80 , C07D317/66 , C07D319/16 , C07D319/18 , C07D333/38 , C07D471/04 , C07D521/00 , C07C245/02 , A01N33/26 , C07C245/04 , C07C251/12
CPC分类号： C07D213/77 , A01N37/52 , A01N43/40 , C07C259/20 , C07C311/38 , C07D319/18 , C07C2101/02
摘要： Azo oxime ethers of formula (I), in which X is CH or N, R.sub.1 is hydrogen, C.sub.1 -C.sub.3 alkyl, trifluoromethyl or cylclopopy and R.sub.2 is aryl or heteroaryl, have an activity against phytopathogenic fungi. They can be used in the form of formulaions as crop protection products, seed-dressing products and wood preservatives.
摘要翻译：式（I）的偶氮肟醚，其中X为CH或N，R 1为氢，C 1 -C 3烷基，三氟甲基或环丙基，R2为芳基或杂芳基，具有抗植物病原性真菌的活性。它们可以作为作物保护产品，拌种产品和木材防腐剂的形式使用。

49. 发明授权

US08658801B2 Pesticides containing a bicyclic bisamide structure 失效
标题翻译：含有双环双酰胺结构的农药
公开(公告)号：US08658801B2
公开(公告)日：2014-02-25
申请号：US12278807
申请日：2007-02-14
申请人： Olivier Loiseleur , Patricia Durieux , Stephan Trah , Andrew Edmunds , André Jeanguenat , André Stoller , David John Hughes
发明人： Olivier Loiseleur , Patricia Durieux , Stephan Trah , Andrew Edmunds , André Jeanguenat , André Stoller , David John Hughes
IPC分类号： C07D401/14
CPC分类号： C07D401/14 , A01N43/56 , A01N43/60 , A01N43/78 , A01N43/82 , A01N43/86 , C07D409/14 , C07D413/14 , C07D417/14
摘要： Compounds of formula (I), wherein the substituents are as defined in claim 1, and the agrochemically acceptable salts and all stereoisomers and tautomeric forms of the compounds of formula I can be used as agrochemical active ingredients and can be prepared in a manner known per se.
摘要翻译：式（I）的化合物，其中取代基如权利要求1中所定义，以及式I化合物的农业化学上可接受的盐和所有立体异构体和互变异构形式可用作农业化学活性成分，并且可以以已知的方式制备 se。

50. 发明授权

US08658644B2 Pyridazine derivatives, processes for their preparation and their use as fungicides 失效
标题翻译：哒嗪衍生物，其制备方法及其作为杀真菌剂的用途
公开(公告)号：US08658644B2
公开(公告)日：2014-02-25
申请号：US13576945
申请日：2011-02-01
申请人： Stephan Trah , Clemens Lamberth
发明人： Stephan Trah , Clemens Lamberth
IPC分类号： C07D237/08 , C07D237/12 , C07D237/14 , A61K31/50
CPC分类号： C07D237/12 , A01N43/58 , C07D237/14 , C07D307/58 , C07D307/60
摘要： The present invention relates to novel pyridazine derivatives of formula (I) wherein R1 is methyl or ethyl; R2 is H or chloro; R3 is fluoro or chloro; R4 is fluoro or methoxy; and R5 is chloro or methoxy or an agrochemically usable salt from thereof, as active ingredients which have microbiodidal activity, in particular fungicidal activity.
摘要翻译：本发明涉及式（I）的新的哒嗪衍生物，其中R 1是甲基或乙基; R2是H或氯; R3是氟或氯; R4是氟或甲氧基; R5为氯或甲氧基或其农药可用盐，作为具有微生物活性的活性成分，特别是杀真菌活性。

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