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31. 发明公开

EP0068591A2 Novel sulfonamide derivatives 失效
标题翻译：磺酰胺衍。
公开(公告)号：EP0068591A2
公开(公告)日：1983-01-05
申请号：EP82200797.7
申请日：1982-06-28
申请人： THE PROCTER & GAMBLE COMPANY
发明人： Buckwalter, Brian Lee , Lahann, Thomas Robert
IPC分类号： C07C143/822 , C07C143/75 , C07C143/79 , A61K7/155 , A61K31/18
CPC分类号： A61Q9/04 , A61K8/46 , A61K8/466 , A61K2800/75 , A61Q17/00
摘要： A compound, or pharmaceutically acceptable salt thereof, having the formula:
wherein X is
wherein R is C 3 -C 12 alkyl or aralkyl, branched or unbranched, unsubstituted aryl, haloaryl, or C 3 -C 22 alkenyl, branched or unbranched: wherein R, is H, OH or OCH 3 , and wherein R 2 is OH or H, at least one of R, and R 2 being OH or OCH 3 . These sulfonamides have analgesic and anti-irritant activity when administered to humans and lower animals.

32. 发明授权

US4713489A Preparation of N-substituted arylsulfonamides 失效
标题翻译： N-取代芳基磺酰胺的制备
公开(公告)号：US4713489A
公开(公告)日：1987-12-15
申请号：US820876
申请日：1986-01-16
申请人： Gail H. Birum , Richard F. Jansen
发明人： Gail H. Birum , Richard F. Jansen
IPC分类号： C07C311/15 , C07C143/79
CPC分类号： C07C311/15
摘要： N-substituted arylsulfonamides which comprises the steps of (a) reacting an aryl hydrocarbon with chlorosulfonic acid to form a crude chlorosulfonation reaction product, (b) adding said crude reaction product to a mixture comprising an aliphatic amine, an alkali or alkaline earth metal hydroxide and water to form an amidation reaction mixture, (c) maintaining the temperature of the amidation reaction mixture at between about 50.degree. C. and 100.degree. C. and the pH at above about 7 with stirring for a period of time of up to about 2 hours, and optionally (d) separating the resulting N-substituted arylsulfonamide from the amidation reaction product.
摘要翻译： N-取代的芳基磺酰胺，其包括以下步骤：（a）使芳基烃与氯磺酸反应以形成粗氯磺化反应产物，（b）将所述粗反应产物加入到包含脂族胺，碱金属或碱土金属氢氧化物和水以形成酰胺化反应混合物，（c）将酰胺化反应混合物的温度保持在约50℃至100℃，pH高于约7，同时搅拌一段时间至多约 2小时，任选地（d）从酰胺化反应产物中分离得到的N-取代的芳基磺酰胺。

33. 发明授权

US4435394A 3-Sulfonamido-benzophenonimine derivatives useful for treating virus infections 失效
标题翻译：用于治疗病毒感染的3-磺酰氨基 - 二苯甲酮亚胺衍生物
公开(公告)号：US4435394A
公开(公告)日：1984-03-06
申请号：US332099
申请日：1981-12-17
申请人： Masaru Ogata , Kosaburo Sato
发明人： Masaru Ogata , Kosaburo Sato
IPC分类号： C07D295/26 , C07C143/79 , A61K31/18 , C07C143/75
CPC分类号： C07D295/26 , Y10S514/849 , Y10S514/889
摘要： 3-Sulfonamido-benzophenonimine derivatives useful for prophylactically or therapeutically treating patients suffering from viral infections are provided from 3-sulfonamido-benzophenones.
摘要翻译：可用于预防性或治疗性治疗病毒感染患者的3-磺酰氨基 - 二苯甲酮亚胺衍生物由3-磺酰氨基 - 二苯甲酮提供。

34. 发明授权

US4281189A Sulfonamide intermediates for adrenergic blocking agents 失效
标题翻译：磺酰胺中间体用于肾上腺素能阻断剂
公开(公告)号：US4281189A
公开(公告)日：1981-07-28
申请号：US180259
申请日：1980-08-22
申请人： Jefferson W. Tilley
发明人： Jefferson W. Tilley
IPC分类号： A61K31/495 , C07D295/00 , C07D295/067 , C07D295/092 , C07D295/15 , C07D303/22 , C07D317/20 , C07D317/22 , C07D317/24 , C07D317/26 , C07D317/28 , C07D317/30 , C07D317/34 , C07C143/75 , C07C143/79
CPC分类号： C07D295/067 , A61K31/495 , C07D295/00 , C07D295/088 , C07D295/15 , C07D303/22 , C07D317/20 , C07D317/22 , C07D317/24 , C07D317/26 , C07D317/28 , C07D317/30 , C07D317/34
摘要： There are disclosed compounds of the formula ##STR1## wherein R.sub.1 is selected from the group consisting of lower alkyl; R.sub.8 is selected from the group consisting of --O--(CH.sub.2).sub.n --wherein n is 2 to 20, ##STR2## and ##STR3## and R.sub.6 is selected from the group consisting of hydrogen or lower alkoxy, and ##STR4## wherein R.sub.1 is selected from the group consisting of lower alkyl; R.sub.8 is selected from the group consisting of --O--(CH.sub.2).sub.n --wherein n is 2 to 20, ##STR5## and ##STR6## and R.sub.6 is selected from the group consisting of hydrogen or lower alkoxy and racemates thereof.There are also disclosed processes and intermediates utilized to produce the end products.The end products have utility as agents exhibiting both .alpha. and selective .beta. adrenergic blocking action.
摘要翻译：公开了式IMA的化合物，其中R 1选自低级烷基; R 8选自-O-（CH 2）n - ，其中n为2-20，和，R 6选自氢或低级烷氧基，其中R 1 选自低级烷基; R 8选自-O-（CH 2）n - ，其中n为2至20，且其中R 6选自氢或其低级烷氧基和外消旋体。还公开了用于生产最终产品的方法和中间体。最终产品具有作为显示α和选择性β肾上腺素能阻断作用的药剂的效用。

35. 发明授权

US4278577A Bis(sulfonamide) stabilizers for synthetic polymers 失效
标题翻译：用于合成聚合物的双（磺酰胺）稳定剂
公开(公告)号：US4278577A
公开(公告)日：1981-07-14
申请号：US171620
申请日：1980-07-23
申请人： John Song
发明人： John Song
IPC分类号： C08K5/43 , C08L91/00 , C07C143/79
CPC分类号： C08K5/43
摘要： Bis(sulfonamides) containing one or more hindered phenol groups are disclosed, as is their use as thermal stabilizers for polymers. Further stabilization results from combinations thereof with a thiodipropionate ester and a divalent metal salt of a carboxylic acid.
摘要翻译：公开了含有一个或多个受阻酚基团的双（磺酰胺），它们用作聚合物的热稳定剂。进一步的稳定化来自与硫代二丙酸酯和羧酸的二价金属盐的组合。

36. 发明授权

US4239699A Sulfonamidophenols, metal complexes thereof, and solutions containing such compounds for use in extraction of metal values 失效
标题翻译：磺酰胺苯酚，其金属络合物，以及含有用于提取金属价值的化合物的溶液
公开(公告)号：US4239699A
公开(公告)日：1980-12-16
申请号：US909224
申请日：1978-05-24
申请人： Kenneth D. MacKay
发明人： Kenneth D. MacKay
IPC分类号： C01G3/00 , C01G9/00 , C01G53/00 , C22B3/34 , C07C143/78 , B01D11/04 , C07C143/79
CPC分类号： C01G9/003 , C01G3/003 , C01G53/003 , C22B3/0031 , Y02P10/234
摘要： Certain sulfonamidophenols, metal complexes thereof and solutions of said compounds in essentially water-immiscible, liquid hydrocarbon solvents are disclosed. The sulfonamidophenols have the structural formula: ##STR1## wherein R.sub.1, R.sub.2, R.sub.3 and R.sub.4 are as defined in the specification and claims hereof. Particular metal values are recovered from their aqueous solutions by using sulfonamidophenols dissolved in essentially water-immiscible liquid hydrocarbon solvents. The extraction process involves contacting the metal value containing aqueous solution with the solution of sulfonamidophenol in essentially water-immiscible liquid hydrocarbon solvent and stripping the metal values from the loaded organic phase.
摘要翻译：公开了某些磺酰胺苯酚，其金属络合物和所述化合物在基本上与水不混溶的液体烃溶剂中的溶液。磺酰胺苯酚具有结构式：其中R 1，R 2，R 3和R 4如本说明书和权利要求书中所定义。通过使用溶解在基本上与水不混溶的液体烃溶剂中的磺酰胺酚从其水溶液中回收特定的金属值。提取过程包括使含金属含量的水溶液与基本上与水不混溶的液体烃溶剂中的磺酰胺基苯溶液接触并从负载的有机相中汽提金属值。

37. 发明授权

US4160807A Sulfonamido oximes, metal complexes thereof, and solutions containing such compounds for use in extraction of metal values 失效
标题翻译：磺胺肟，其金属络合物和含有这些化合物的溶液用于提取金属价值
公开(公告)号：US4160807A
公开(公告)日：1979-07-10
申请号：US90922678
申请日：1978-05-24
申请人： HENKEL CORP
发明人： VIRNIG MICHAEL J , MACKAY KENNETH D
IPC分类号： C01G3/00 , C01G9/00 , C01G51/00 , C01G53/00 , C22B3/34 , C07C143/78 , B01D11/04 , C07C143/79
CPC分类号： C22B3/0031 , C01G3/003 , C01G9/003 , C01G51/003 , C01G53/003 , Y02P10/234
摘要： Certain sulfonamido oximes, metal complexes thereof and solutions of said compounds in essentially water-immiscible, liquid hydrocarbon solvents are disclosed. The sulfonamido oximes have the general structural formula: wherein A, R1, R2 and R3 are as defined in the specification and claims hereof. Particular metal values are recovered from their aqueous solutions by using sulfonamido oximes dissolved in essentially water-immiscible liquid hydrocarbon solvents. The extraction process involves contacting the metal value containing aqueous solution with the solution of the sulfonamido oxime in essentially water-immiscible liquid hydrocarbon solvent and stripping the mertal values from the loaded organic phase.
摘要翻译：公开了某些磺酰胺肟，其金属络合物和所述化合物在基本上与水不混溶的液体烃溶剂中的溶液。亚磺酰氨基肟具有以下通式结构式：其中A，R 1，R 2和R 3如本说明书和权利要求中所定义。通过使用溶解在基本上与水不混溶的液体烃溶剂中的磺酰胺肟，从其水溶液中回收特定的金属值。提取过程包括将含金属含量的水溶液与磺酰胺肟的溶液在基本上与水不混溶的液体烃溶剂中接触并从负载的有机相中汽提出来的值。

38. 发明授权

US4160783A 4-Dedimethylamino-4-arylsulfonamido-5a,6-anhydrotetracyclines 失效
标题翻译： 4-二甲基氨基-4-芳基磺酰胺基-5a，6-脱水四环素
公开(公告)号：US4160783A
公开(公告)日：1979-07-10
申请号：US855496
申请日：1977-11-28
申请人： Marica Cakara , Slobodan Djokic , Zrinka Tamburasev
发明人： Marica Cakara , Slobodan Djokic , Zrinka Tamburasev
IPC分类号： A61K31/18 , A61K31/65 , C07C311/15 , C07C143/79
CPC分类号： A61K31/18 , A61K31/65 , C07C311/15
摘要： Novel 4-dedimethylamino-4-arylsulfonamido-5a,6-anhydrotetracyclines of the general formula I ##STR1## wherein R stands for C.sub.1 -C.sub.3 -alkyl, halogen or --NHCOR.sup.1, R.sup.1 being C.sub.1 -C.sub.3 -alkyl.
摘要翻译：通式Ⅰ的新型4-脱二甲基氨基-4-芳基亚磺酰基-5a，6-脱水四环素其中R代表C 1 -C 3烷基，卤素或-NHCOR 1，R 1是C 1 -C 3烷基。

39. 发明授权

US4157257A Benzenesulfonamide derivatives 失效
标题翻译：苯磺酰胺衍生物
公开(公告)号：US4157257A
公开(公告)日：1979-06-05
申请号：US837911
申请日：1977-09-29
申请人： Tetsuo Takematsu , Makoto Konnai , Hiroyoshi Omokawa
发明人： Tetsuo Takematsu , Makoto Konnai , Hiroyoshi Omokawa
IPC分类号： A01N41/06 , C07C311/15 , A01N9/14 , C07C143/79 , C07C143/82
CPC分类号： C07C255/00 , A01N41/06
摘要： A compound of the general formula ##STR1## wherein R.sub.0 represents an alkyl group optionally having a substituent selected from the class consisting of a cyano group, lower alkoxy groups and di-(lower alkyl)amino groups, a lower alkenyl group, or a lower alkynyl group; R.sub.1, R.sub.2 and R.sub.3, independently from each other, represent a hydrogen atom, a halogen atom, a lower alkyl group, or a lower alkoxy group; R.sub.4, R.sub.5, R.sub.6, R.sub.7 and R.sub.8, independently from each other, represent a hydrogen atom, a halogen atom, a lower alkyl group, or a lower alkoxy group; Y represents a group of the formula ##STR2## or a group of the formula ##STR3## in which one of R.sub.9 and R.sub.10 is a lower alkyl group and the other is a hydrogen atom or a lower alkyl group; with the proviso that when Y is the group ##STR4## and R.sub.0 represents an unsubstituted alkyl group, R.sub.4, R.sub.5, R.sub.6, R.sub.7 and R.sub.8 do not represent hydrogen atoms at the same time. The compounds of formula (I) are produced by the reaction of the corresponding benzenesulfonamide derivatives with the corresponding benzyl or benzoyl halides; the reaction of the corresponding benzenesulfonyl halides with the corresponding benzylamines or benzoyl amides; or by the alkylation, alkenylation or alkynylation of the corresponding compounds of formula (I) in which R.sub.0 is hydrogen. The compounds of formula (I) have superior selective herbicidal effects, and are useful as active ingredients of herbicides, especially those for application to aquatic rice paddies.
摘要翻译：通式（I）的化合物，其中R 0表示任选具有选自氰基，低级烷氧基和二 - （低级烷基）氨基的取代基的烷基，低级烯基，或低级炔基; R 1，R 2和R 3彼此独立地表示氢原子，卤素原子，低级烷基或低级烷氧基; R4，R5，R6，R7和R8彼此独立地表示氢原子，卤素原子，低级烷基或低级烷氧基; Y表示式为“IMAGE”的基团或其中R9和R10中的一个为低级烷基且另一个为氢原子或低级烷基的式“IMAGE”的基团; 条件是当Y为基团时，R 0表示未取代的烷基，R 4，R 5，R 6，R 7和R 8不同时表示氢原子。式（I）化合物通过相应的苯磺酰胺衍生物与相应的苄基或苯甲酰基卤化物的反应产生; 相应的苯磺酰卤与相应的苄胺或苯甲酰胺的反应; 或通过其中R 0是氢的相应的式（I）化合物的烷基化，烯基化或炔基化。式（I）的化合物具有优异的选择性除草效果，并且可用作除草剂的活性成分，特别是用于水稻的施用。

40. 发明授权

US4035421A N-(3,4,-dichlorophenyl)-2-phenylethenesulfonamide 失效
标题翻译： N-（3,4， - 二氯苯基）-2-苯基亚磺酰胺
公开(公告)号：US4035421A
公开(公告)日：1977-07-12
申请号：US668612
申请日：1976-03-19
申请人： Harry R. Snyder, Jr.
发明人： Harry R. Snyder, Jr.
IPC分类号： C07C311/15 , C07C143/79 , A61K31/18
CPC分类号： C07C311/15
摘要： Antibacterially active N-(3,4-dichlorophenyl)-2-phenylethenesulfonamide.
摘要翻译：抗菌活性N-（3,4-二氯苯基）-2-苯基亚磺酰胺。

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