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1. 发明申请

WO2006097279A8 AMIDRAZONE COMPOUNDS FOR COMBATING ANIMAL PESTS 审中-公开
标题翻译：用于组合动物疫苗的咪唑啉酮化合物
公开(公告)号：WO2006097279A8
公开(公告)日：2007-05-18
申请号：PCT/EP2006002331
申请日：2006-03-14
申请人： BASF AG , KORADIN CHRISTOPHER , DEYN WOLFGANG VON , RACK MICHAEL , KUHN DAVID G , CULBERTSON DEBORAH L , ANSPAUGH DOUGLAS , OLOUMI-SADEGHI HASSAN
发明人： KORADIN CHRISTOPHER , VON DEYN WOLFGANG , RACK MICHAEL , KUHN DAVID G , CULBERTSON DEBORAH L , ANSPAUGH DOUGLAS , OLOUMI-SADEGHI HASSAN
IPC分类号： A01N37/52 , A01P5/00 , A01P7/00 , A01P7/04 , C07C259/20
CPC分类号： C07C259/20 , A01N37/52 , C07C2601/02
摘要： The present invention relates to new amidrazone compounds which are useful for combating animal pests, in particular insects, arachnids and nematodes. The invention also relates to a method for combating insects, nematodes and arachnids. The amidrazone compounds are of the general formula (I) including the tautomers of I and the salts thereof; wherein X and Y are hydrogen or together form a chemical bond; Ar is an aromatic radical selected from phenyl and a 5- or 6-membered heteroaryl having 1 , 2, 3 or 4 heteroatoms as ring members, which are selected, independently of one another, from O, N and S, and where the aromatic radical may have 1 , 2, 3, 4 or 5 substituents R a ; R 1 is selected from the group consisiting of C 1 -C 1O -alkyl, C 1 -C 4 -alkoxy-C 1 -C 4 -alkyl, cyano-C 1 -C 4 -alkyl, hydroxy-C 1- C 4 -alkyl, C 1 -C 10 -haloalkyl, tri-(C 1 -C 4 -alkyl)-silyl-C 1 - C 4 -alkyl, C 2 -C 10 -alkenyl, C 2 -C 10 -haloalkenyl, C 2 -C 10 -alkynyl, C 2 -C 10 -haloalkynyl, C 3 -C 10 -cycloalkyl, phenyl, heteroaryl, C 3 -C 10 -cycloalkyl-C 1 C 4 -alkyl, phenyl-C 1 -C 4 - alkyl and heteroaryl-C 1 C 4 alkyl, wherein C 3 -C 10 -cycloalkyl, heteroaryl and phenyl in the last six mentioned radicals may be unsubstituted or carry 1 , 2, 3, 4 or 5 substituents R b as defined above; R 2 is selected from the group consisiting of C 1- C 1 0-alkyl, c 1- c 4 -alkoxy- C 1- C 4 -alkyl, C 1- C 10 -haloalkyl, C 2 -C 10 -alkenyl, C 2 -C 10 -haloalkenyl, C 2 -C 10 -alkynyl, C 2 -C 10 - haloalkynyl,c 3 -C 10 -cycloalkyl, phenyl, heteroaryl, C 3 -C 10 -cycloalkyl-C 1- C 4 -alkyl, phenyl-C 1 -C 4 -alkyl and heteroaryI-C 1- C 4 -alkyl, wherein C 3 -C 10 -cycloalkyl, heteroaryl and phenyl in the last six mentioned radicals may be unsubstituted or carry 1 , 2, 3, 4 or 5 substituents R b as defined above.
摘要翻译：本发明涉及可用于对抗动物害虫，特别是昆虫，蜘蛛和线虫的新的氨基腙化合物。本发明还涉及一种防治昆虫，线虫和蜘蛛的方法。氨基腙化合物具有通式（I），其包括I的互变异构体及其盐; 其中X和Y是氢或一起形成化学键; Ar是选自苯基和具有1,2,3或4个杂原子作为环成员的5-或6-元杂芳基的芳族基团，其彼此独立地选自O，N和S，并且其中芳族基团可以具有1,2,3,4或5个取代基R a， R 1选自C 1 -C 10 - 烷基，C 1 -C 1 - 烷基， C 1 -C 4烷基，C 1 -C 4烷基，C 1 -C 4烷基，氰基-C 1 -C 4烷基， C 1 -C 6烷基，羟基-C 1 -C 4 - 亚烷基，C 1 -C 10 - 烷基，卤代烷基，三 - （C 1 -C 4 - 烷基） - 甲硅烷基-C 1 -C 4 - 烷基，C 2 -C 10 - 烯基，C 2 -C 10 - 卤代烯基，C 1 -C 10 - C 2 -C 10 - 炔基，C 2 -C 10 - 卤代炔基，C 3 - C 10 - 环烷基，苯基，杂芳基，C 3 -C 10 - 环烷基-C 1 -C C 1-4烷基，苯基-C 1 -C 4 - 烷基和杂芳基-C 1 -C 4烷基，其中C 3 -C 10 - 环烷基，杂芳基和苯基在后面六个提及的基团中可以是未取代的或携带1,2,3,4或4个 5个取代基R b如上所定义; R 2选自C 1 -C 1-4烷基，C 1 -C 4烷基， C 1-4烷基，C 1 -C 10烷基，C 1 -C 4烷基，C 1〜亚烷基，C 2 -C 10 - 烯基，C 2 -C 10 - 卤代烯基，C C 2 -C 10 - 炔基，C 2 -C 10 - 卤代炔基，C 3 - C 1 -C 10 - 环烷基，苯基，杂芳基，C 3 -C 10 - 环烷基-C 1 - C 1 -C 4 - 烷基，苯基-C 1 -C 4 - 烷基和杂芳基C 1 -C 其中C 3 -C 10 - 环烷基，最后六个所述基团中的杂芳基和苯基可以是未取代的或携带1， 2,3,4或5个如上定义的取代基R b。

2. 发明申请

WO02034711A1 BIARYL COMPOUNDS AS SERINE PROTEASE INHIBITORS 审中-公开
标题翻译： BIARYL化合物作为丝氨酸蛋白酶抑制剂
公开(公告)号：WO02034711A1
公开(公告)日：2002-05-02
申请号：PCT/US2001/032582
申请日：2001-10-22
IPC分类号： A61K31/192 , A61K31/341 , A61K31/381 , A61K31/426 , A61K31/4418 , C07C229/38 , C07C233/54 , C07C235/84 , C07C251/48 , C07C255/57 , C07C255/58 , C07C257/18 , C07C259/18 , C07C259/20 , C07C271/22 , C07C271/64 , C07C309/65 , C07D207/32 , C07D207/337 , C07D209/08 , C07D213/40 , C07D213/56 , C07D213/74 , C07D213/75 , C07D213/78 , C07D213/79 , C07D213/80 , C07D213/81 , C07D213/82 , C07D231/56 , C07D233/54 , C07D235/10 , C07D235/14 , C07D235/30 , C07D235/32 , C07D239/14 , C07D239/42 , C07D239/48 , C07D277/30 , C07D277/82 , C07D307/54 , C07D311/80 , C07D317/46 , C07D317/68 , C07D333/24 , C07D333/38 , C07D521/00 , A61K31/155 , A61K31/24 , A61K31/255 , A61K31/27 , A61K31/34 , A61K31/38 , A61K31/40 , A61K31/415 , A61K31/425 , A61K31/44 , A61K31/495 , A61K31/505 , A61K31/535 , A61K31/55 , A61K31/69 , C07C63/04 , C07C257/00 , C07C317/22 , C07D207/08 , C07D207/30 , C07D211/70 , C07D239/02 , C07D265/30 , C07D277/62 , C07D307/02 , C07D311/78 , C07D317/44 , C07D333/22
CPC分类号： C07D249/08 , A61K31/192 , A61K31/341 , A61K31/381 , A61K31/426 , A61K31/4418 , C07C229/38 , C07C233/54 , C07C235/84 , C07C251/48 , C07C255/57 , C07C255/58 , C07C257/18 , C07C259/18 , C07C259/20 , C07C271/22 , C07C271/64 , C07C309/65 , C07C2601/02 , C07C2601/04 , C07C2601/08 , C07C2601/14 , C07C2601/18 , C07D207/337 , C07D209/08 , C07D213/40 , C07D213/56 , C07D213/74 , C07D213/75 , C07D213/78 , C07D213/79 , C07D213/80 , C07D213/81 , C07D213/82 , C07D231/12 , C07D231/56 , C07D233/56 , C07D233/64 , C07D235/14 , C07D235/30 , C07D235/32 , C07D239/14 , C07D239/42 , C07D239/48 , C07D277/30 , C07D277/82 , C07D307/54 , C07D311/80 , C07D317/46 , C07D317/68 , C07D333/24 , C07D333/38
摘要： Compounds of formula (I) are useful as inhibitors of trypsin like serine protease enzymes such as thrombin, factor VIIa, factor Xa, TF/FVIIa, and trypsin. These compounds could be useful to treat and/or prevent clotting disorders, and as anticoagulating agents.
摘要翻译：式（I）化合物可用作胰蛋白酶样丝氨酸蛋白酶如凝血酶，因子VIIa，因子Xa，TF / FVIIa和胰蛋白酶的抑制剂。这些化合物可用于治疗和/或预防凝血障碍，以及作为抗凝剂。

3. 发明申请

WO1998004520A1 FUNGICIDES 审中-公开
标题翻译：杀菌剂
公开(公告)号：WO1998004520A1
公开(公告)日：1998-02-05
申请号：PCT/GB1997001729
申请日：1997-06-27
申请人： ZENECA LIMITED , ASPINALL, Ian, Henry , WORTHINGTON, Paul, Anthony , TSERIOTIS, George
发明人： ZENECA LIMITED
IPC分类号： C07C259/20
CPC分类号： A01N37/52 , C07C259/20
摘要： A fungicidal compound of formula (I): or a stereoisomer thereof, wherein A is CH or N, B is OCH3 or NHCH3, E is -NR -C(CH3)=N- or -N=C(CH3)-NR -, R is H, C1-4 alkyl, C2-4 alkenyl, C2-4 alkynyl or optionally substituted benzyl, R is H, C1-4 alkyl, halo(C1-4)alkyl, C3-6 cycloalkyl, C2-4 alkenyl or C2-4 alkynyl, and R is optionally substituted aryl or optionally substituted heterocyclyl.
摘要翻译：式（I）的杀真菌化合物或其立体异构体，其中A为CH或N，B为OCH 3或NHCH 3，E为-NR 1 -C（CH 3）= N-或-N = C（CH 3） -NR 1 - ，R 1是H，C 1-4烷基，C 2-4烯基，C 2-4炔基或任选取代的苄基，R 2是H，C 1-4烷基，卤代（C 1-4 ）烷基，C 3-6环烷基，C 2-4烯基或C 2-4炔基，R 3是任选取代的芳基或任选取代的杂环基。

4. 发明申请

WO2006097279A1 AMIDRAZONE COMPOUNDS FOR COMBATING ANIMAL PESTS 审中-公开
标题翻译：用于组合动物疫苗的咪唑烷化合物
公开(公告)号：WO2006097279A1
公开(公告)日：2006-09-21
申请号：PCT/EP2006/002331
申请日：2006-03-14
申请人： BASF AKTIENGESELLSCHAFT , KORADIN, Christopher , VON DEYN, Wolfgang , RACK, Michael , KUHN, David, G. , CULBERTSON, Deborah, L. , ANSPAUGH, Douglas , OLOUMI-SADEGHI, Hassan
发明人： KORADIN, Christopher , VON DEYN, Wolfgang , RACK, Michael , KUHN, David, G. , CULBERTSON, Deborah, L. , ANSPAUGH, Douglas , OLOUMI-SADEGHI, Hassan
IPC分类号： A01N37/52 , C07C259/20 , A01P7/00 , A01P5/00 , A01P7/04
CPC分类号： C07C259/20 , A01N37/52 , C07C2601/02
摘要： The present invention relates to new amidrazone compounds which are useful for combating animal pests, in particular insects, arachnids and nematodes. The invention also relates to a method for combating insects, nematodes and arachnids. The amidrazone compounds are of the general formula (I) including the tautomers of I and the salts thereof; wherein X and Y are hydrogen or together form a chemical bond; Ar is an aromatic radical selected from phenyl and a 5- or 6-membered heteroaryl having 1 , 2, 3 or 4 heteroatoms as ring members, which are selected, independently of one another, from O, N and S, and where the aromatic radical may have 1 , 2, 3, 4 or 5 substituents R a ; R 1 is selected from the group consisiting of C 1 -C 1O -alkyl, C 1 -C 4 -alkoxy-C 1 -C 4 -alkyl, cyano-C 1 -C 4 -alkyl, hydroxy-C 1- C 4 -alkyl, C 1 -C 10 -haloalkyl, tri-(C 1 -C 4 -alkyl)-silyl-C 1 - C 4 -alkyl, C 2 -C 10 -alkenyl, C 2 -C 10 -haloalkenyl, C 2 -C 10 -alkynyl, C 2 -C 10 -haloalkynyl, C 3 -C 10 -cycloalkyl, phenyl, heteroaryl, C 3 -C 10 -cycloalkyl-C 1 C 4 -alkyl, phenyl-C 1 -C 4 - alkyl and heteroaryl-C 1 C 4 alkyl, wherein C 3 -C 10 -cycloalkyl, heteroaryl and phenyl in the last six mentioned radicals may be unsubstituted or carry 1 , 2, 3, 4 or 5 substituents R b as defined above; R 2 is selected from the group consisiting of C 1- C 1 0-alkyl, c 1- c 4 -alkoxy- C 1- C 4 -alkyl, C 1- C 10 -haloalkyl, C 2 -C 10 -alkenyl, C 2 -C 10 -haloalkenyl, C 2 -C 10 -alkynyl, C 2 -C 10 - haloalkynyl,c 3 -C 10 -cycloalkyl, phenyl, heteroaryl, C 3 -C 10 -cycloalkyl-C 1- C 4 -alkyl, phenyl-C 1 -C 4 -alkyl and heteroaryI-C 1- C 4 -alkyl, wherein C 3 -C 10 -cycloalkyl, heteroaryl and phenyl in the last six mentioned radicals may be unsubstituted or carry 1 , 2, 3, 4 or 5 substituents R b as defined above.
摘要翻译：本发明涉及可用于对抗动物害虫，特别是昆虫，蜘蛛和线虫的新的氨基腙化合物。本发明还涉及一种防治昆虫，线虫和蜘蛛的方法。氨基腙化合物具有通式（I），其包括I的互变异构体及其盐; 其中X和Y是氢或一起形成化学键; Ar是选自苯基和具有1,2,3或4个杂原子作为环成员的5-或6-元杂芳基的芳族基团，其彼此独立地选自O，N和S，并且其中芳族基团可以具有1,2,3,4或5个取代基R a， R 1选自C 1 -C 10 - 烷基，C 1 -C 1 - 烷基， C 1 -C 4烷基，C 1 -C 4烷基，C 1 -C 4烷基，氰基-C 1 -C 4烷基， C 1 -C 6烷基，羟基-C 1 -C 4 - 亚烷基，C 1 -C 10 - 烷基，卤代烷基，三 - （C 1 -C 4 - 烷基） - 甲硅烷基-C 1 -C 4 - 烷基，C 2 -C 10 - 烯基，C 2 -C 10 - 卤代烯基，C 1 -C 10 - C 2 -C 10 - 炔基，C 2 -C 10 - 卤代炔基，C 3 - C 10 - 环烷基，苯基，杂芳基，C 3 -C 10 - 环烷基-C 1 -C C 1-4烷基，苯基-C 1 -C 4 - 烷基和杂芳基-C 1 -C 4烷基，其中C 3 -C 10 - 环烷基，杂芳基和苯基在后面六个提及的基团中可以是未取代的或携带1,2,3,4或4个 5个取代基R b如上所定义; R 2选自C 1 -C 1-4烷基，C 1 -C 4烷基， C 1-4烷基，C 1 -C 10烷基，C 1 -C 4烷基，C 1〜亚烷基，C 2 -C 10 - 烯基，C 2 -C 10 - 卤代烯基，C C 2 -C 10 - 炔基，C 2 -C 10 - 卤代炔基，C 3 - C 1 -C 10 - 环烷基，苯基，杂芳基，C 3 -C 10 - 环烷基-C 1 - C 1 -C 4 - 烷基，苯基-C 1 -C 4 - 烷基和杂芳基C 1 -C 其中C 3 -C 10 - 环烷基，最后六个所述基团中的杂芳基和苯基可以是未取代的或携带1， 2,3,4或5个如上定义的取代基R b。

5. 发明申请

WO1993016986A1 AZO OXIME ETHERS AND THEIR USE AS FUNGICIDES 审中-公开
标题翻译： AZO OXIME ETHERS及其作为防腐剂使用
公开(公告)号：WO1993016986A1
公开(公告)日：1993-09-02
申请号：PCT/EP1993000373
申请日：1993-02-17
申请人： CIBA-GEIGY AG , ZIEGLER, Hugo , TRAH, Stephan
发明人： CIBA-GEIGY AG
IPC分类号： C07C259/20
CPC分类号： C07D213/77 , A01N37/52 , A01N43/40 , C07C259/20 , C07C311/38 , C07C2601/02 , C07D319/18
摘要： Azo oxime ethers of general formula (I), in which X is CH or N, R1 is hydrogen, C1-C3alkyl, trifluoromethyl or cylclopropyl and R2 is aryl or heteroaryl, have an activity against phytopathogenic fungi. They can be used in the form of formulations as crop protection products, seed-dressing products and wood preservatives.
摘要翻译：通式（I）的偶氮肟醚，其中X为CH或N，R 1为氢，C 1 -C 3烷基，三氟甲基或环丙基，R 2为芳基或杂芳基，具有抗植物病原性真菌的活性。它们可以以制剂形式用作作物保护产品，拌种产品和木材防腐剂。

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