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1. 发明申请

WO2004091549A3 PROCESS FOR MAKING ALPHA-SUBSTITUTED HYDROXAMIC ACIDS 审中-公开
标题翻译：制备ALPHA取代的羟基酸的方法
公开(公告)号：WO2004091549A3
公开(公告)日：2006-02-23
申请号：PCT/US2004009407
申请日：2004-03-25
申请人： PHARMACIA CORP , BABIAK KEVIN A , BOEHM TERRI L , COLSON PIERRE-JEAN , FARID PAYMAN N , GALLAGHER DONALD J , HUBER CHRISTIAN H , LINDERMAN RUSSELL J , LIU CHIN , MAR EDUARDO K , NEWAZ MURAD , PIPPEL DANIEL J , PRZYBYLA CLAIRE A , ROBB CHRISTOPHER N , STAHL GLENN L , TOPGI RAVINDRA S , WEISENBURGER GERALD A , YONAN EDWARD E
发明人： BABIAK KEVIN A , BOEHM TERRI L , COLSON PIERRE-JEAN , FARID PAYMAN N , GALLAGHER DONALD J , HUBER CHRISTIAN H , LINDERMAN RUSSELL J , LIU CHIN , MAR EDUARDO K , NEWAZ MURAD , PIPPEL DANIEL J , PRZYBYLA CLAIRE A , ROBB CHRISTOPHER N , STAHL GLENN L , TOPGI RAVINDRA S , WEISENBURGER GERALD A , YONAN EDWARD E
IPC分类号： A61K20060101 , C07D401/12 , C07D405/12 , C07D409/12
CPC分类号： C07D335/02 , C07D211/54 , C07D309/08 , C07D401/04 , C07D401/06 , C07D401/14 , C07D405/06 , C07D405/12 , C07D405/14 , C07D409/06 , C07D409/14 , C07D413/04 , C07D417/12 , C07D417/14
摘要： This invention is directed generally to a process for making a-substituted hydroxamic acids (including salts thereof) generally corresponding in structure to formula (I) wherein n, Z, Z
摘要翻译：本发明一般涉及在通式（I）结构中对应于其中n，Z，Z

2. 发明申请

WO2002098220A3 PESTICIDAL ACTIVITY OF FUNCTIONALIZED ALKENES 审中-公开
公开(公告)号：WO2002098220A3
公开(公告)日：2002-12-12
申请号：PCT/US2002/018068
申请日：2002-06-06
申请人： NORTH CAROLINA STATE UNIVERSITY , LINDERMAN, Russell, J. , ROE, R., Michael , THOMPSON, Deborah, M. , VANDERHEREHEN, Matthew
发明人： LINDERMAN, Russell, J. , ROE, R., Michael , THOMPSON, Deborah, M. , VANDERHEREHEN, Matthew
IPC分类号： A01N37/10
摘要： The present invention provides non-peptide organic compounds that have a structure analogous to or reminiscent of the TMOF structure and have pesticidal activity. Thus the present invention concerns pesticidal compounds that inhibit digestion in pests by terminating or otherwise blocking synthesis of digestive enzymes by activating a TMOF receptor (collectively referred to herein as "pesticidal compounds"). The pesticidal compounds and other compounds of the present invention are usefully employed in the control of pests, particularly insect pests such as mosquitoes, which ingest blood.

3. 发明申请

WO0141543A3 PESTICIDAL ACTIVITY OF FUNCTIONALIZED ALKENES 审中-公开
标题翻译：功能性碱的杀虫活性
公开(公告)号：WO0141543A3
公开(公告)日：2002-01-10
申请号：PCT/US0031558
申请日：2000-11-16
申请人： UNIV NORTH CAROLINA STATE , LINDERMAN RUSSELL J
发明人： LINDERMAN RUSSELL J
IPC分类号： A01N37/10 , A01N37/18 , A01N37/38 , C07C57/26 , C07C57/42 , C07C57/60 , C07C59/64 , C07C69/608 , C07C69/618 , G01N33/50 , G01B3/00 , G01B5/00 , G01N31/00 , G06F19/00
CPC分类号： G01N33/5082 , A01N37/10 , A01N37/18 , A01N37/38 , C07C57/26 , C07C57/42 , C07C57/60 , C07C59/64 , C07C69/608 , C07C69/618 , C07C2601/14 , Y10S514/875 , Y10S514/951
摘要： The present invention provides non-peptide organic compounds that have a structure analogous to or reminiscent of the TMOF structure and have pesticidal activity. Thus the present invention concerns pesticidal compounds that inhibit digestion in pests by terminating or otherwise blocking synthesis of digestive enzymes by activating a TMOF receptor (collectively referred to herein as "pesticidal compounds"). The pesticidal compounds and other compounds of the present invention are usefully employed in the control of pests, particularly insect pests such as mosquitoes, which ingest blood.
摘要翻译：本发明提供了具有与TMOF结构类似或令人想起的具有杀虫活性的结构的非肽有机化合物。因此，本发明涉及通过终止或以其它方式阻断消化酶的合成来抑制害虫消化的农药化合物，其通过激活TMOF受体（本文统称为“杀虫化合物”）。本发明的杀虫化合物和其他化合物有效地用于控制害虫，特别是摄入血液的昆虫害虫如蚊子。

4. 发明申请

WO2003051118A1 PESTICIDAL ACTIVITY OF FUNCTIONALIZED CYCLOPROPANES 审中-公开
标题翻译：功能化环糊精的杀虫活性
公开(公告)号：WO2003051118A1
公开(公告)日：2003-06-26
申请号：PCT/US2002/039755
申请日：2002-12-12
申请人： NORTH CAROLINA STATE UNIVERSITY , LINDERMAN, Russell, J.
发明人： LINDERMAN, Russell, J.
IPC分类号： A01N37/10
CPC分类号： C07C57/46 , A01N37/10 , A01N37/18 , C07C51/09 , C07C51/353 , C07C51/36 , C07C51/38 , C07C53/132 , C07C53/134 , C07C57/26 , C07C57/42 , C07C2601/02 , C07C2601/14
摘要： The present invention provides functionalized cyclopropane compounds that have pesticidal and/or TMOF activity. The pesticidal compounds and other compounds of the present invention are usefully employed in the control of pests, particularly insect pests such as mosquitoes, which ingest blood.
摘要翻译：本发明提供具有杀虫和/或TMOF活性的官能化环丙烷化合物。本发明的杀虫化合物和其他化合物有效地用于控制害虫，特别是摄入血液的昆虫害虫如蚊子。

5. 发明申请

WO2004091549A2 PROCESS FOR MAKING ALPHA-SUBSTITUTED HYDROXAMIC ACIDS 审中-公开
标题翻译：制备ALPHA取代的羟基酸的方法
公开(公告)号：WO2004091549A2
公开(公告)日：2004-10-28
申请号：PCT/US2004/009407
申请日：2004-03-25
申请人： PHARMACIA CORPORATION , BABIAK, Kevin, A. , BOEHM, Terri, L. , COLSON, Pierre-Jean , FARID, Payman, N. , GALLAGHER, Donald, J. , HUBER, Christian, H. , LINDERMAN, Russell, J. , LIU, Chin , MAR, Eduardo, K. , NEWAZ, Murad , PIPPEL, Daniel, J. , PRZYBYLA, Claire, A. , ROBB, Christopher, N. , STAHL, Glenn, L. , TOPGI, Ravindra, S. , WEISENBURGER, Gerald, A. , YONAN, Edward, E.
发明人： BABIAK, Kevin, A. , BOEHM, Terri, L. , COLSON, Pierre-Jean , FARID, Payman, N. , GALLAGHER, Donald, J. , HUBER, Christian, H. , LINDERMAN, Russell, J. , LIU, Chin , MAR, Eduardo, K. , NEWAZ, Murad , PIPPEL, Daniel, J. , PRZYBYLA, Claire, A. , ROBB, Christopher, N. , STAHL, Glenn, L. , TOPGI, Ravindra, S. , WEISENBURGER, Gerald, A. , YONAN, Edward, E.
IPC分类号： A61K
CPC分类号： C07D335/02 , C07D211/54 , C07D309/08 , C07D401/04 , C07D401/06 , C07D401/14 , C07D405/06 , C07D405/12 , C07D405/14 , C07D409/06 , C07D409/14 , C07D413/04 , C07D417/12 , C07D417/14
摘要： This invention is directed generally to a process for making α-substituted hydroxamic acids (including salts thereof) generally corresponding in structure to formula (I) wherein n, Z, Z 3 , A, R, E, and Y are as defined in this patent. This invention also is directed to compounds that may, for example, be used as intermediates in such a process, as well as processes for making such compounds.
摘要翻译：本发明一般涉及在通式（I）的结构中对应的α-取代的异羟肟酸（包括其盐）的制备方法，其中n，Z，Z 3，A，R，E和Y定义如上在这个专利。本发明还涉及可以例如在这种方法中用作中间体的化合物以及制备这些化合物的方法。

6. 发明申请

WO0141543A8 PESTICIDAL ACTIVITY OF FUNCTIONALIZED ALKENES 审中-公开
标题翻译：功能性碱的杀虫活性
公开(公告)号：WO0141543A8
公开(公告)日：2002-12-27
申请号：PCT/US0031558
申请日：2000-11-16
申请人： UNIV NORTH CAROLINA STATE , LINDERMAN RUSSELL J
发明人： LINDERMAN RUSSELL J
IPC分类号： A01N37/10 , A01N37/18 , A01N37/38 , C07C57/26 , C07C57/42 , C07C57/60 , C07C59/64 , C07C69/608 , C07C69/618 , G01N33/50
CPC分类号： G01N33/5082 , A01N37/10 , A01N37/18 , A01N37/38 , C07C57/26 , C07C57/42 , C07C57/60 , C07C59/64 , C07C69/608 , C07C69/618 , C07C2601/14 , Y10S514/875 , Y10S514/951
摘要： The present invention provides non-peptide organic compounds that have a structure analogous to or reminiscent of the TMOF structure and have pesticidal activity. Particular pesticidal compounds/non-peptide TMOF analogs of the present invention have formula (I) wherein: X is selected from the group consisting of -CHCH-, -CH2CH2-, and -CC-; Z is selected from the group consisting of -OH, -NH2 and -OR6 wherein R6 is loweralkyl; n and m are each at last (I) and together total an integer from 2, 3 or 4 to 6, 8, 10 or 12; and R1, R2, R3, R4 and R5 are each independently selected from the group consisting of -H, -OH, halo, loweralkyl, and loweralkoxy; subject to the proviso that: a pair of R1 and R2, R2 and R3, or R3 and R4 on the phenyl ring may together represent -CR7=CR8-CR9=CR10-, to form with the phenyl ring illustrated above a naphthyl ring system, wherein R7, R8, R9 and R10 are each independently selected from the group consisting of -H, -OH, halo, loweralkyl, and loweralkoxy. Thus the present invention concerns pesticidal compounds that inhibit digestion in pests by terminating or otherwise blocking synthesis of digestive enzymes by activating a TMOF receptor (collectively referred to herein as "pesticidal compounds"). The pesticidal compounds and other compounds of the present invention are usefully employed in the control of pests, particularly insect pests such as mosquitoes, which ingest blood.
摘要翻译：本发明提供了具有与TMOF结构类似或令人想起的具有杀虫活性的结构的非肽有机化合物。本发明的特定杀虫化合物/非肽TMOF类似物具有式（I），其中：X选自-CHCH - ， - CH 2 CH 2 - 和-CC-; Z选自-OH，-NH 2和-OR 6，其中R 6是低级烷基; n和m各自为最后（I），并且总共为2,3或4至6,8,10或12的整数; 并且R 1，R 2，R 3，R 4和R 5各自独立地选自-H，-OH，卤素，低级烷基和低级烷氧基; 条件是：苯环上的一对R 1和R 2，R 2和R 3或R 3和R 4可以一起表示-CR 7 = CR 8 -CR 9 = CR 10 - ，与上述苯环形成萘基环系其中R 7，R 8，R 9和R 10各自独立地选自-H，-OH，卤素，低级烷基和低级烷氧基。因此，本发明涉及通过终止或以其它方式阻断消化酶的合成来抑制害虫消化的农药化合物，其通过激活TMOF受体（本文统称为“杀虫化合物”）。本发明的杀虫化合物和其他化合物有效地用于控制害虫，特别是摄入血液的昆虫害虫如蚊子。

7. 发明申请

WO2002098220A2 PESTICIDAL ACTIVITY OF FUNCTIONALIZED ALKENES 审中-公开
标题翻译：功能化杀虫剂的杀虫活性
公开(公告)号：WO2002098220A2
公开(公告)日：2002-12-12
申请号：PCT/US2002/018068
申请日：2002-06-06
申请人： NORTH CAROLINA STATE UNIVERSITY , LINDERMAN, Russell, J. , ROE, R., Michael , THOMPSON, Deborah, M. , VANDERHEREHEN, Matthew
发明人： LINDERMAN, Russell, J. , ROE, R., Michael , THOMPSON, Deborah, M. , VANDERHEREHEN, Matthew
IPC分类号： A01N
CPC分类号： C07C69/618 , A01N37/10 , A01N37/18 , A01N37/38 , C07C57/26 , C07C57/42 , C07C57/60 , C07C59/64 , C07C69/608 , C07C403/20 , C07C2601/14 , G01N33/5082 , Y10S424/10 , Y10S514/875 , Y10S514/919 , Y10S514/951
摘要： The present invention provides non-peptide organic compounds that have a structure analogous to or reminiscent of the TMOF structure and have pesticidal activity. Thus the present invention concerns pesticidal compounds that inhibit digestion in pests by terminating or otherwise blocking synthesis of digestive enzymes by activating a TMOF receptor (collectively referred to herein as "pesticidal compounds"). The pesticidal compounds and other compounds of the present invention are usefully employed in the control of pests, particularly insect pests such as mosquitoes, which ingest blood.
摘要翻译：本发明提供具有与TMOF结构类似或令人想起TMOF结构并具有杀虫活性的非肽有机化合物。因此，本发明涉及通过终止或以其他方式阻断通过活化TMOF受体（本文统称为“杀虫化合物”）阻断消化酶的合成来抑制害虫消化的杀虫化合物。本发明的杀虫化合物和其它化合物可用于防治有害生物，特别是摄食血液的昆虫害虫如蚊子。

8. 发明申请

WO0063233A3 PEPTIDES AND THE USE THEREOF TO CONTROL PESTS 审中-公开
标题翻译：肽及其用于控制PESTS的用途
公开(公告)号：WO0063233A3
公开(公告)日：2001-01-11
申请号：PCT/US0010235
申请日：2000-04-18
申请人： UNIV FLORIDA , UNIV NORTH CAROLINA STATE , BOROVSKY DOV , LINDERMAN RUSSELL J
发明人： BOROVSKY DOV , LINDERMAN RUSSELL J
IPC分类号： A01N37/46 , A01N63/02 , C07K5/065 , C07K5/072 , C07K5/083 , C07K5/087 , C07K5/093 , C07K7/06 , C12N15/12 , C12N1/16 , C12N5/10 , C12N15/63
CPC分类号： C07K7/06 , A01N37/46 , A01N63/02 , C07K5/06078 , C07K5/06113 , C07K5/0806 , C07K5/0812 , C07K5/0819 , Y10S514/875 , Y10S514/919
摘要： The subject invention pertains to novel pest control compounds. Specifically exemplified herein are peptides having 2 to 5 amino acids. The subject peptides are useful against a variety of pests, including pests of agricultural crops.
摘要翻译：本发明涉及新颖的有害生物防治化合物。具体示例为具有2-5个氨基酸的肽。本发明的肽可用于各种害虫，包括农作物的害虫。

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