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21. 发明申请

WO2006097489A1 BIPHENYL-N-(4-PYRIDYL) METHYLSUFONAMIDES 审中-公开
标题翻译：二苯基-N-（4-吡啶基）甲基磺酰胺
公开(公告)号：WO2006097489A1
公开(公告)日：2006-09-21
申请号：PCT/EP2006/060753
申请日：2006-03-15
申请人： BASF AKTIENGESELLSCHAFT , GRAMMENOS, Wassilios , RHEINHEIMER, Joachim , LOHMANN, Jan Klaas , GROTE, Thomas , PUHL, Michael , KORADIN, Christopher , BAUMANN, Ernst , VON DEYN, Wolfgang , LANGEWALD, Jürgen , GÖTZ, Norbert , CULBERTSON, Deborah L. , ANSPAUGH, Douglas D. , OLOUMI-SADEGHI, Hassan , COTTER, Henry Van Tuyl , KUHN, David G.
发明人： GRAMMENOS, Wassilios , RHEINHEIMER, Joachim , LOHMANN, Jan Klaas , GROTE, Thomas , PUHL, Michael , KORADIN, Christopher , BAUMANN, Ernst , VON DEYN, Wolfgang , LANGEWALD, Jürgen , GÖTZ, Norbert , CULBERTSON, Deborah L. , ANSPAUGH, Douglas D. , OLOUMI-SADEGHI, Hassan , COTTER, Henry Van Tuyl , KUHN, David G.
IPC分类号： A01N43/40 , C07D213/42
CPC分类号： A01N43/40 , C07D213/42
摘要： Biphenylsulfonamides of the formula I and the N-oxides and the agriculturally acceptable salts and the veterinarily acceptable salts of the compounds I, a process for preparing these compounds, compositions comprising them, their use for controlling phytopathogenic harmful fungi and harmful arthropodes, a method for combating arthropodal pests, a method for protecting crops from attack or infestation of arthropodal pests, a method for protecting seed and non-living materials from infestation by arthropodal pests, a method for protecting non-living materials from attack or infestation by arthropodal pests and seed comprising the compounds I.
摘要翻译：式I的联苯磺酰胺和N-氧化物和农业上可接受的盐和化合物I的兽医学可接受的盐，制备这些化合物的方法，包含它们的组合物，其用于控制植物病原性有害真菌和有害的节肢动物的方法，防治节肢动物害虫，防止作物受到节肢动物害虫侵袭或侵袭的方法，防止种子和非生物材料免受节肢动物害虫侵害的方法，保护非生物材料免遭节肢动物害虫和种子侵袭的方法包括化合物I.

22. 发明申请

WO2005054208A1 VERFAHREN ZUR HERSTELLUNG VON 3-PHENYL(THIO)URACILEN UND 3-PHENYLDITHIOURACILEN 审中-公开
标题翻译：用于生产3-苯基（硫）的尿嘧啶和3- phenyldithiouracils
公开(公告)号：WO2005054208A1
公开(公告)日：2005-06-16
申请号：PCT/EP2004/013615
申请日：2004-12-01
申请人： BASF Aktiengesellschaft , HAMPRECHT, Gerhard , PUHL, Michael , WOLF, Bernd , KEIL, Michael , REINHARD, Robert , SEITZ, Werner , MAYER, Guido
发明人： HAMPRECHT, Gerhard , PUHL, Michael , WOLF, Bernd , KEIL, Michael , REINHARD, Robert , SEITZ, Werner , MAYER, Guido
IPC分类号： C07D239/56
CPC分类号： C07D239/54 , C07D239/56
摘要： Beschrieben wird ein Verfahren zur Herstellung von 3-Phenyl(thio)uracilen oder 3-Phenyldithiouracilen der Formel I, bei dem ein Phenyliso(thio)cyanat der Formel II mit einem Enamin der Formel III umgesetzt und gegebenenfalls in einem weiteren Schritt das erhaltene 3-Phenyl(thio)uracil oder 3-Phenyldithiouracil der Formel I mit R1=R1a, wenn R1 für Wasserstoff steht, mit einem Aminierungsmittel der Formel IV zu 3-Phenyl(thio)uracilen oder 3-Phenyldithiouracilen der Formel I mit R1=Amino umgesetzt wird: worin die Variablen R1, R1a, R2, R3, R4, X1, X2, X3, Ar, A und L1 die in Anspruch 1 genannten Bedeutungen aufweisen.
摘要翻译：制备3-苯基（硫）的方法将被描述的尿嘧啶或式3-phenyldithiouracils I，其中苯基异（硫）与下式的烯胺使式II的氰酸反应III和在进一步的步骤任选获得的3- 苯基（硫代）尿嘧啶或式3-Phenyldithiouracil我与R 1 = R 1A，其中R 1是氢，与式Ⅳ的胺化剂，得到3-苯基（硫代）尿嘧啶或式的3- phenyldithiouracils我与R1 =氨基进行反应：其中变量R 1中，R 1a，R 2，R3，R4，X1，X2，X3中，Ar，A和L 1如权利要求1具有定义。

23. 发明申请

WO2005035486A1 2-CYANOBENZENESULFONAMIDES FOR COMBATING ANIMAL PESTS 审中-公开
标题翻译：用于组合动物疫苗的2-氰基苯甲醚
公开(公告)号：WO2005035486A1
公开(公告)日：2005-04-21
申请号：PCT/EP2004/011004
申请日：2004-10-01
申请人： BASF AKTIENGESELLSCHAFT , VON DEYN, Wolfgang , BAUMANN, Ernst , HOFMANN, Michael , KORDES, Markus , PUHL, Michael , SCHMIDT, Thomas , TEDESCHI, Livio , RACK, Michael , BUCCI, Toni , CULBERTSON, Deborah, L. , COTTER, Henry, Van Tuyl , OLOUMI-SADEGHI, Hassan
发明人： VON DEYN, Wolfgang , BAUMANN, Ernst , HOFMANN, Michael , KORDES, Markus , PUHL, Michael , SCHMIDT, Thomas , TEDESCHI, Livio , RACK, Michael , BUCCI, Toni , CULBERTSON, Deborah, L. , COTTER, Henry, Van Tuyl , OLOUMI-SADEGHI, Hassan
IPC分类号： C07C311/16
CPC分类号： A01N41/06 , C07C311/16 , C07C311/17 , C07C311/18 , C07C311/19 , C07C311/20 , C07C311/29 , C07C311/48 , C07C317/28 , C07C323/49 , C07C2601/02 , C07C2601/04 , C07C2601/08 , C07C2601/14
摘要： The invention relates to 2-cyanobenzenesulfonamide compounds of the formula (I) where the variables R 1 to R 5 are as defined in claim 1 and/or to their agriculturally useful salts. Moreover, the present invention relates to the use of compounds (I) and/or their salts for combating animal pests; agricultural compositions comprising such an amount of at least one compound of the general formula (I) and/or at least one agriculturally useful salt of I and at least one inert liquid and/or solid agronomically acceptable carrier that it has a pesticidal action and, if desired, at least one surfactant; and a method of combating animal pests which comprises contacting the animal pests, their habit, breeding ground, food supply, plant, seed, soil, area, material or environment in which the animal pests are growing or may grow, or the materials, plants, seads, soils, surfaces or spaces to be protected from animal attack or infestation with a pesticidally effective amount of at least one 2-cyanobenzenesulfonamide compound of the general formula I and/or at least one agriculturally acceptable salt thereof.
摘要翻译：本发明涉及式（I）的2-氰基苯磺酰胺化合物，其中变量R 1至R 5如权利要求1所定义，和/或其农业上有用的盐。此外，本发明涉及化合物（I）和/或其盐对抗动物害虫的用途; 包含这种量的至少一种通式（I）的化合物和/或至少一种农业上可用的I盐和至少一种惰性液体和/或其农业上可接受的载体的农药组合物，其具有杀虫作用，如果需要，至少一种表面活性剂; 以及一种对抗动物害虫的方法，包括使动物有害生物，其习惯，繁殖地，食物供应，植物，种子，土壤，区域，动物害虫生长或可能生长的区域，材料或环境，或材料，植物，防护物，表面或空间，以防止动物攻击或侵袭与杀虫有效量的至少一种通式I的2-氰基苯磺酰胺化合物和/或其至少一种农业上可接受的盐。

24. 发明申请

WO2004080170A2 AMINO SUBSTITUTED BENZO(HETERO)CYCLIC DERIVATIVES 审中-公开
标题翻译：氨基取代的苯甲（环）环化合物
公开(公告)号：WO2004080170A2
公开(公告)日：2004-09-23
申请号：PCT/EP2004/001677
申请日：2004-02-20
申请人： BASF AKTIENGESELLSCHAFT , STEINER, Gerd , SCHMIDT, Thomas , KORDES, Markus , VON DEYN, Wolfgang , HOFMANN, Michael , BAUMANN, Ernest , PUHL, Michael , HEFFERNAN, Gavin , CULBERTSON, Deborah, L. , TREACY, Michael, F.
发明人： STEINER, Gerd , SCHMIDT, Thomas , KORDES, Markus , VON DEYN, Wolfgang , HOFMANN, Michael , BAUMANN, Ernest , PUHL, Michael , HEFFERNAN, Gavin , CULBERTSON, Deborah, L. , TREACY, Michael, F.
IPC分类号： A01N
CPC分类号： A01N43/72 , A01N43/60
摘要： Use of compounds Formula (I), A = a 5- to 7-membered ring which may contain 1-3 heteroatoms and which may be saturated or partially or completely unsaturated; R 1 = OH, SH, NH 2 , CN, NO 2 , halogen, C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl; C 1 -C 6 - alkoxy, C 1 -C 6 -haloalkoxy, C 1 -C 6 -alkylthio, C 1 -C 6 -haloalkylthio, C 2 -C 6 -alkenyl, C 2 -C 6 -alkenyloxy, C 2 -C 6 -alkenylthio, C 2 -C 6 -alkynyl, C 2 -C 6 alkynyloxy, C 2 -C 6 -alkynylthio, C 1 -C 6 -alkylsulfonyl, C 1 -C6-alkylsulfoxyl, C 2 -C 6 -alkenylsulfonyl, C 2 -C 6 -alkynylsulfoxyl, C 1 -C 6 -alkylcarbonyl, C 1 -C 6 - alkoxycarbonyl, C 1 -C 6 -alkylcarbonyloxy; R 2 = C 1 -C 6 -alkyl or a mono- or bicyclic 5- to 10-membered aromatic ringsystem which may contain 1 to 4 heteroatoms and which is either bonded directly or through an O, S, C 1 -C 6 -alkylene or C 1 -C 6 -alkyleneoxy linkage to A or fused to A and which may be substituted; R 3 , R 4 = H, C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, C 1 -C 6 -alkylamino, C 1 -C 6 -alkoxy, C 3 -C 6 - cycloalkyl, or R 3 and R 4 together with the nitrogen atom to which they are attached form a saturated or partially saturated mono- or bicyclic 5- to 10-membered ring system con-taining 1 to 3 heteroatoms or a 5-membered hetaryl containing 1 to 4 nitro-gen atoms, wherein the carbon and/or nitrogen atoms in the ring systems may be substituted or phenyl or benzyl which may be substituted; or R 3 and R 4 together form the chains -(CH 2 ) 2 N + (O-)(CH 2 ) 2 - or -(CH 2 ) 3 N + (O - )(CH 2 ) 2 - ; m = 0 to 4; n is 0 to 4; and the enantiomers, diastereomers, cis/trans isomers or salts thereof for combatting insects, arachnids or nematodes, methods for the control of these pests and of protecting growing plants attack or infestation by these pests by applying a pesticidally effective amount of a compound of formula (I), processes for preparing them, and compositions comprising them.
摘要翻译：化合物式（I）的用途，A =可含有1-3个杂原子并且可以是饱和或部分或完全不饱和的5-至7-元环; R 1 = OH，SH，NH 2，CN，NO 2，卤素，C 1 -C 6烷基，C 1 -C 6 - 卤代烷基; C 1 -C 6烷氧基，C 1 -C 6 - 卤代烷氧基，C 1 -C 6 - 烷硫基，C 1 -C 6卤代烷硫基，C 2 -C 6 - 烯基，C 2 -C 6 - 烯氧基，C 2 -C 6 - 烯硫基，C 2 -C 6炔基， C 1 -C 6烷氧羰基，C 1 -C 6烷氧基羰基，C 1 -C 6烷氧基羰基，C 1 -C 6烷氧羰基，C 1 -C 6烷氧羰基， R 2 = C 1 -C 6 - 烷基或可以含有1至4个杂原子并且直接键合或通过O，S，C 1 -C 6亚烷基或通过C 1 -C 6 - 烷基取代的单 - 或双环5-至10-元芳环体系与A或与A稠合的C1-C6-亚烷基氧键，并且其可以被取代; R 3，R 4 = H，C 1 -C 6烷基，C 1 -C 6卤代烷基，C 1 -C 6烷基氨基，C 1 -C 6 - 烷氧基，C 3 -C 6环烷基或R 3和 R 4与它们所连接的氮原子一起形成饱和或部分饱和的单环或双环的5-至10-元环系统，其含有1至3个杂原子或含有1至4个硝基的5元杂芳基 - 原子，其中环系中的碳原子和/或氮原子可以被取代，或可被取代的苯基或苄基; 或者R 3和R 4一起形成链 - （CH 2）2 N +（O - ）（CH 2）2 - 或 - （CH 2）3 N +（O - ）（CH 2）2 < - >; m = 0〜4; n为0〜4; 以及用于防治昆虫，蜘蛛或线虫的对映异构体，非对映异构体，顺式/反式异构体或其盐，用于控制这些害虫的方法以及通过施用杀虫有效量的这种化合物来保护这些害虫的生长植物侵袭或侵染（I），其制备方法和包含它们的组合物。

25. 发明申请

WO2003097589A1 VERFAHREN ZUR HERSTELLUNG VON SULFAMIDSÄUREHALOGENIDEN 审中-公开
标题翻译：用于生产氨基磺酸卤化物
公开(公告)号：WO2003097589A1
公开(公告)日：2003-11-27
申请号：PCT/EP2003/005126
申请日：2003-05-15
申请人： BASF AKTIENGESELLSCHAFT , HAMPRECHT, Gerhard , PUHL, Michael , REINHARD, Robert , SAGASSER, Ingo , SCHMIDT, Thomas , GÖTZ, Norbert , ZIERKE, Thomas
发明人： HAMPRECHT, Gerhard , PUHL, Michael , REINHARD, Robert , SAGASSER, Ingo , SCHMIDT, Thomas , GÖTZ, Norbert , ZIERKE, Thomas
IPC分类号： C07C307/02
CPC分类号： C07D295/26 , C07C303/34 , C07C307/00 , C07C2601/14 , C07D207/48 , C07D211/96 , C07D239/46
摘要： Die vorliegende Erfindung betrifft ein Verfahren zur Herstellung von Sulfamidsäurehalogeniden primärer oder sekundärer Amine, umfassend die folgenden Schritte: i) Umsetzung eines primären oder sekundären Amins A1 mit wenigstens äquimolaren Mengen S03 oder einer S03Quelle in Gegenwart von wenigstens äquimolaren Mengen eines tertiären Amins A2, jeweils bezogen auf das Amin A1, und ii) Umsetzung der in Schritt i) erhaltenen Reaktionsmischung mit wenigstens der stöchiometrisch erforderlichen Menge eines Phosphorhalogenids; Die Erfindung betrifft weiterhin ein Verfahren zur Herstellung von Sulfonsäurediamiden, umfassend die Herstellung von Sulfamidsäurehalogeniden mittels Durchführung der Schritte i) and ii) und anschliessende Umsetzung des erhaltenen Sulfamidsäurehalogenids mit Ammoniak. Die Erfindung betrifft weiterhin den Einsatz dieses Verfahrens zur Herstellung von Herbizid-Wirkstoffen mit Sulfodiamid-Struktur. Die Erfindung betrifft auch neue Sulfamidsäurechloride.
摘要翻译：本发明涉及一种用于制备包括以下步骤伯或仲胺的氨基磺酸卤化物：基于在每种情况下I）的伯或仲胺A1与至少等摩尔量的叔胺A2的存在至少等摩尔量的S03或S03Quelle的反应，在胺A1，和ii）在步骤i）的反应混合物与至少一个磷卤化物的化学计量所需量而得到的混合物进行反应; 本发明还涉及一种用于Sulfonsäurediamiden的制备通过执行我的步骤包括氨基磺酸卤化物的制备）和ii），而与氨的获得Sulfamidsäurehalogenids的随后的反应。本发明还涉及使用这种方法的用于具有Sulfodiamid结构除草活性化合物的制备。本发明还涉及新的Sulfamidsäurechloride。

26. 发明申请

WO2010100189A1 3-ARYLQUINAZOLIN-4-ONE COMPOUNDS FOR COMBATING INVERTEBRATE PESTS 审中-公开
标题翻译： 3-ARYLQUINAZOLIN-4-ONE化合物，用于混合反相胶束
公开(公告)号：WO2010100189A1
公开(公告)日：2010-09-10
申请号：PCT/EP2010/052693
申请日：2010-03-03
申请人： BASF SE , GROSS, Steffen , KÖRBER, Karsten , VON DEYN, Wolfgang , KAISER, Florian , DESHMUKH, Prashant , DICKHAUT, Joachim , BANDUR, Nina, Gertrud , NARINE, Arun , POHLMAN, Matthias , PUHL, Michael , THOMPSON, Sarah , EBUENGA, Cecille , ANSPAUGH, Douglas, D. , CULBERTSON, Deborah, L.
发明人： GROSS, Steffen , KÖRBER, Karsten , VON DEYN, Wolfgang , KAISER, Florian , DESHMUKH, Prashant , DICKHAUT, Joachim , BANDUR, Nina, Gertrud , NARINE, Arun , POHLMAN, Matthias , PUHL, Michael , THOMPSON, Sarah , EBUENGA, Cecille , ANSPAUGH, Douglas, D. , CULBERTSON, Deborah, L.
IPC分类号： C07D239/88 , C07D401/04 , C07D403/04 , A01N43/54
CPC分类号： C07D239/88 , C07D401/04 , C07D403/04
摘要： The present invention relates to the 3-arylquinazolin-4-one compounds of the formula (I) and the salts thereof, formula (I) wherein n is O, 1 or 2; X is O, S or N-R 4 ; Y 1 is N or CH; Y 2 is N or C-R 5 ; R 1 is C 1 -C 10 -alkyl, C 1 -C 10 -haloalkyl, C 2 -C 10 -alkenyl, C 2 -C 10 -haloalkenyl, C 2 -C 10 -alkynyl, C 2 -C 10 -haloalkynyl, C 3 -C 12 -cycloalkyl, C 5 -C 12 -cycloalkenyl, C 3 -C 12 -cycloalkyl-C 1 -C 4 -alkyl, C 5 -C 12 -cycloalkenyl-C 1 -C 4 -alkyl, where the cycloalkyl radical and the cycloalkenyl radical in the last four mentioned radicals are unsubstituted, partially or fully halogenated and/or carry 1, 2, 3, 4, or 5 C 1 -C 4 -alkyl radicals; R 2 is hydrogen, halogen, CN, C(Z)NH 2 , C 1 -C 4 -alkyl or C 1 -C 4 -haloalkyl, wherein Z is O, S or NR 6 ; and the variables k, R, R 3 , R 4 , R 5 and R 6 are as defined in the claims. The invention also relates to the use of novel compounds of formula (I) for combating invertebrate pests and to a method for controlling invertebrate pests. The invention also relates to a plant propagation material and to an agricultural composition comprising a 3-arylquinazolin-4-one compound of formula (I).
摘要翻译：本发明涉及式（I）的3-芳基喹唑啉-4-酮化合物及其盐，式（I）其中n为O，1或2; X为O，S或N-R4; Y1是N或CH; Y2是N或C-R5; R 1是C 1 -C 10 - 烷基，C 1 -C 10 - 卤代烷基，C 2 -C 10 - 烯基，C 2 -C 10 - 卤代烯基，C 2 -C 10 - 炔基，C 2 -C 10 - 卤代炔基，C 3 -C 12环烷基，C 5 -C 12 - 环烯基， C 3 -C 12 - 环烷基-C 1 -C 4 - 烷基，C 5 -C 12 - 环烯基-C 1 -C 4 - 烷基，其中最后四个所述基团中的环烷基和环烯基是未取代的，部分或全部卤化的和/或携带1 ，2,3,4或5个C 1 -C 4 - 烷基; R 2是氢，卤素，CN，C（Z）NH 2，C 1 -C 4烷基或C 1 -C 4卤代烷基，其中Z是O，S或NR 6; 变量k，R，R3，R4，R5和R6如权利要求中所定义。本发明还涉及式（I）的新型化合物用于防治无脊椎动物害虫以及控制无脊椎动物害虫的方法。本发明还涉及植物繁殖材料和包含式（I）的3-芳基喹唑啉-4-酮化合物的农业组合物。

27. 发明申请

WO2009141274A1 SUBSTITUTED PYRIDIN-4 -YL-METHYL SULFONAMIDES AS FUNGICIDES 审中-公开
标题翻译：取代的吡啶-4-基甲基磺酰胺作为杀真菌剂
公开(公告)号：WO2009141274A1
公开(公告)日：2009-11-26
申请号：PCT/EP2009/055899
申请日：2009-05-15
申请人： BASF SE , GRAMMENOS, Wassilios , GLÄTTLI, Alice , LOHMANN, Jan Klaas , PUHL, Michael , MÜLLER, Bernd , VRETTOU, Marianna
发明人： GRAMMENOS, Wassilios , GLÄTTLI, Alice , LOHMANN, Jan Klaas , PUHL, Michael , MÜLLER, Bernd , VRETTOU, Marianna
IPC分类号： C07D401/12 , C07D405/12 , C07D409/12 , C07D413/12 , C07D417/12 , A01N43/40 , A01N43/78
CPC分类号： C07D409/12 , C07D401/12 , C07D405/12 , C07D413/12 , C07D417/12
摘要： The present invention relates to pyridin-4-ylmethyl sulfonamides of formula I wherein R a , n, R, A and Het are as defined in the claims, to the N-oxides, and salts thereof and their use for combating harmful fungi, and also to compositions and seed comprising at least one such compound. The invention also relates to a process and intermediates for preparing these compounds.
摘要翻译：本发明涉及式I的吡啶-4-基甲基磺酰胺，其中Ra，n，R，A和Het如权利要求中所定义，与N-氧化物及其盐及其用于对抗有害真菌的用途包含至少一种这样的化合物的组合物和种子。本发明还涉及制备这些化合物的方法和中间体。

28. 发明申请

WO2009101082A9 SUBSTITUTED SULFONIC ACID AMIDE COMPOUNDS 审中-公开
公开(公告)号：WO2009101082A9
公开(公告)日：2009-08-20
申请号：PCT/EP2009/051509
申请日：2009-02-10
申请人： BASF SE , Dietz, Jochen , Grammenos, Wassilios , Müller, Bernd , Lohmann, Jan Klaas , Renner, Jens , Ulmschneider, Sarah , Vrettou, Marianna , Puhl, Michael
发明人： Dietz, Jochen , Grammenos, Wassilios , Müller, Bernd , Lohmann, Jan Klaas , Renner, Jens , Ulmschneider, Sarah , Vrettou, Marianna , Puhl, Michael
IPC分类号： C07D231/12 , C07D233/61 , C07D249/08 , C07D261/08 , C07D263/32 , C07D271/06 , C07D275/02 , C07D277/28 , C07D285/12 , C07D401/12 , C07D409/12 , C07D409/14 , C07D417/12 , C07D417/14 , A01N43/50
摘要： The present invention relates to the use of substituted sulfonic acid amide compounds of formula I, wherein R a , n, Het, A, Y and D are as defined in the claims and the N-oxides and the salts thereof for combating phytopathogenic harmful fungi, and and to compositions and seeds comprising at least one such compound. The invention also relates to to novel substituted sulfonic acid amide compounds and processes for preparing these compounds.

29. 发明申请

WO2007054558A3 RESORCINE DERIVATIVES AND THEIR USE AS PESTICIDES 审中-公开
公开(公告)号：WO2007054558A3
公开(公告)日：2007-05-18
申请号：PCT/EP2006/068329
申请日：2006-11-10
申请人： BASF AKTIENGESELLSCHAFT , PUHL, Michael , KORDES, Markus , POHLMAN, Matthias , GÖTZ, Norbert , RACK, Michael , LANGEWALD, Jürgen , SCHNEIDER, Felix , ANSPAUGH, Douglas D. , CULBERTSON, Deborah L. , OLOUMI-SADEGHI, Hassan , KUHN, David G.
发明人： PUHL, Michael , KORDES, Markus , POHLMAN, Matthias , GÖTZ, Norbert , RACK, Michael , LANGEWALD, Jürgen , SCHNEIDER, Felix , ANSPAUGH, Douglas D. , CULBERTSON, Deborah L. , OLOUMI-SADEGHI, Hassan , KUHN, David G.
IPC分类号： C07C43/29 , C07D213/16 , C07D213/26 , C07D277/22 , A01N29/10
摘要： This invention relates to resorcine derivatives of formula (I) wherein R 1 is phenyl or a 5- to 6-membered heteroaromatic ring which may contain 1 to 3 heteroatoms selected from oxygen, nitrogen and sulfur, wherein phenyl or the heteroaromatic ring may be fused to a ring selected from phenyl and a 5- to 6-membered saturated, partially unsaturated or aromatic heterocyclic ring which may contain 1 to 3 heteroatoms selected from oxygen, nitrogen and sulfur, wherein phenyl or the 5- to 6-membered heteroaromatic ring or the respective fused ring systems may be unsubstituted or substituted by any combination of 1 to 6 optionally substituted groups R 3 , wherein R 3 is halogen, cyano, nitro, hydroxy, mercapto, amino, alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, haloalkyl, haloalkenyl, haloalkynyl, halocycloalkyl, halocycloalkenyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy, haloalkenyloxy, haloalkynyloxy, alkylthio, alkenylthio, alkynylthio, haloalkylthio, haloalkenylthio, haloalkynylthio, alkylamino, alkenylamino, alkynylamino, dialkylamino, dialkenylamino, dialkynylamino, alkyl-alkenylamino, alkyl-alkynylamino, alkenyl- alkynylamino, trialkylsilyl, or phenyl or a 5-to 7-membered saturated or partially unsaturated heterocyclic ring which may contain 1 to 3 heteroatoms selected from oxygen, sulfur and nitrogen or a 5- to 6-membered heteraromatic ring system which may contain 1 to 4 heteroatoms selected from oxygen, nitrogen and sulfur, which phenyl and which heteroaromatic ring may be bonded via an oxygen or a sulfur atom, or -C(=G)R a , -C(=G)OR a , -C(=G)NR a 2 , -C(=G)[N=SR a 2 ], -C(=NOR a )R a , -C(=NOR a )NR a 2 , -C(=NNR a 2 )R a , -OC(=G)-OC(=G)OR a , N=SR a 2 , -NR a C(=G)R a , -N[C(=G)R a ] 2 , - NR a C(=G)OR a , -C(=G)NR a -NR a 2 , -C(=G)NR a -NR a [C(=G)R a ], -NR a -C(=G)NR a 2 , -NR a -NR a C(=G)R a , -NR a -N[C(=G)R a ] 2 , -N[(C=G)R a ]-NR a 2 , -NR a -NR a [(C=G)GR a ], -NR a [(C=G)NR a 2 , -NR a [C=NR a ]R a , -NR a (C=NR a )NR a 2 , -O-NR a 2 , -O-NR a (C=G)R a , - SO 2 NR a 2 , -NR a SO 2 R a , -S(=O)R a , -S(=O) 2 R a , -SO 2 OR a , or -OSO 2 R a , wherein G is oxygen or sulfur and Ra is as defined in the description, R 2 is hydrogen, halogen, cyano, alkyl, haloalkyl, alkenyl, haloalkenyl, alkynyl, haloalkynyl, alkoxy, or haloalkoxy, x is 2, 3, 4, 5, 6, or 7, or the diastereomers, enantiomers, salts or N-oxides thereof, with the proviso that R 1 is not 5-chloro-2,2,-dimethyl-2,3-dihydrobenzo[b]furan-7-yl when R 2 is hydrogen and x is 3 or 4, processes and intermediates for the preparation of compounds I, use of compounds I for combating insects, acarids, or nematodes, and a method for treating, controlling, preventing or protecting animals against infestation or infection by parasites using compounds I.

30. 发明申请

WO2007054558A2 RESORCINE DERIVATIVES AND THEIR USE AS PESTICIDES 审中-公开
标题翻译： RESORCINE衍生物及其作为杀虫剂的用途
公开(公告)号：WO2007054558A2
公开(公告)日：2007-05-18
申请号：PCT/EP2006068329
申请日：2006-11-10
申请人： BASF AG , PUHL MICHAEL , KORDES MARKUS , POHLMAN MATTHIAS , GOETZ NORBERT , RACK MICHAEL , LANGEWALD JUERGEN , SCHNEIDER FELIX , ANSPAUGH DOUGLAS D , CULBERTSON DEBORAH L , OLOUMI-SADEGHI HASSAN , KUHN DAVID G
发明人： PUHL MICHAEL , KORDES MARKUS , POHLMAN MATTHIAS , GOETZ NORBERT , RACK MICHAEL , LANGEWALD JUERGEN , SCHNEIDER FELIX , ANSPAUGH DOUGLAS D , CULBERTSON DEBORAH L , OLOUMI-SADEGHI HASSAN , KUHN DAVID G
CPC分类号： C07D213/64 , C07D277/34 , C07D307/80
摘要： This invention relates to resorcine derivatives of formula (I) wherein R 1 is phenyl or a 5- to 6-membered heteroaromatic ring which may contain 1 to 3 heteroatoms selected from oxygen, nitrogen and sulfur, wherein phenyl or the heteroaromatic ring may be fused to a ring selected from phenyl and a 5- to 6-membered saturated, partially unsaturated or aromatic heterocyclic ring which may contain 1 to 3 heteroatoms selected from oxygen, nitrogen and sulfur, wherein phenyl or the 5- to 6-membered heteroaromatic ring or the respective fused ring systems may be unsubstituted or substituted by any combination of 1 to 6 optionally substituted groups R 3 , wherein R 3 is halogen, cyano, nitro, hydroxy, mercapto, amino, alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, haloalkyl, haloalkenyl, haloalkynyl, halocycloalkyl, halocycloalkenyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy, haloalkenyloxy, haloalkynyloxy, alkylthio, alkenylthio, alkynylthio, haloalkylthio, haloalkenylthio, haloalkynylthio, alkylamino, alkenylamino, alkynylamino, dialkylamino, dialkenylamino, dialkynylamino, alkyl-alkenylamino, alkyl-alkynylamino, alkenyl- alkynylamino, trialkylsilyl, or phenyl or a 5-to 7-membered saturated or partially unsaturated heterocyclic ring which may contain 1 to 3 heteroatoms selected from oxygen, sulfur and nitrogen or a 5- to 6-membered heteraromatic ring system which may contain 1 to 4 heteroatoms selected from oxygen, nitrogen and sulfur, which phenyl and which heteroaromatic ring may be bonded via an oxygen or a sulfur atom, or -C(=G)Ra, -C(=G)ORa, -C(=G)NRa2, -C(=G)[N=SRa2], -C(=NORa)Ra, -C(=NORa)NRa2, -C(=NNRa2)Ra , -OC(=G)-OC(=G)ORa, N=SRa2, -NRaC(=G)Ra, -N[C(=G)Ra]2, - NRaC(=G)ORa, -C(=G)NRa-NRa2, -C(=G)NRa-NRa [C(=G)Ra], -NRa-C(=G)NRa2, -NRa-NRaC(=G)Ra, -NRa-N[C(=G)Ra]2, -N[(C=G)Ra]-NRa2, -NRa-NRa[(C=G)GRa], -NRa[(C=G)NRa2, -NRa[C=NRa]Ra, -NRa(C=NRa)NRa2, -O-NRa2, -O-NRa(C=G)Ra, - SO2NRa2, -NRaSO2Ra, -S(=O)Ra, -S(=O)2Ra, -SO2ORa, or -OSO2Ra, wherein G is oxygen or sulfur and Ra is as defined in the description, R 2 is hydrogen, halogen, cyano, alkyl, haloalkyl, alkenyl, haloalkenyl, alkynyl, haloalkynyl, alkoxy, or haloalkoxy, x is 2, 3, 4, 5, 6, or 7, or the diastereomers, enantiomers, salts or N-oxides thereof, with the proviso that R 1 is not 5-chloro-2,2,-dimethyl-2,3-dihydrobenzo[b]furan-7-yl when R 2 is hydrogen and x is 3 or 4, processes and intermediates for the preparation of compounds I, use of compounds I for combating insects, acarids, or nematodes, and a method for treating, controlling, preventing or protecting animals against infestation or infection by parasites using compounds I.
摘要翻译：本发明涉及其中R 1为苯基或可含有1-3个选自氧，氮和硫的杂原子的5至6元杂芳环的式（I）的间苯二酚衍生物，其中苯基或杂芳环可以与选自苯基和5-至6-元饱和，部分不饱和或芳族杂环的环稠合，所述杂环可以含有1-3个选自氧，氮和硫的杂原子，其中苯基或5- 至6元杂芳环或相应的稠环体系可以是未取代的或被1至6个任选取代的基团R 3 3的任何组合取代，其中R 3是卤素，氰基，硝基，羟基，巯基，氨基，烷基，烯基，炔基，环烷基，环烯基，卤代烷基，卤代烯基，卤代炔基，卤代环烷基，卤代环烯基，烷氧基，烯氧基，炔氧基，卤代烷氧基，卤代烯氧基，卤代炔氧基，烷硫基，烯硫基，炔硫基，卤代烷硫基， H 烯基氨基，炔基氨基，二烷基氨基，二链烷基氨基，二炔基氨基，烷基 - 链烯基氨基，烷基 - 炔基氨基，烯基 - 炔基氨基，三烷基甲硅烷基或苯基或5至7元饱和或部分不饱和的杂环，至3个选自氧，硫和氮的杂原子或5至6元杂芳环体系，其可以含有1至4个选自氧，氮和硫的杂原子，该苯基和杂芳环可以通过氧或硫原子或-C（= G）R a，-C（= G）OR a，-C（= G）NR a 2，-C（= G）[N = SR a 2] （= NORa）NRa2，-C（= NNRa2）Ra，-OC（= G）-OC（= G）ORa，N = SRa2，-NRaC（= G）Ra，-N [C（= G）Ra] 2，-NR a C（= G）OR a，-C（= G）NR a -NR a 2，-C（= G）NR a -NR a [C（= G）R a] -NRaC（= G）Ra，-NRa-N [C（= G）Ra] 2，-N [（C = G）Ra] -NRa2，-NRa-NRa [（C = G） [（C = G）NRa2，-NRa [C = NRa] Ra，-NRa（C = NRa）NRa2，-O-NRa2，-O-NRa（C = G）Ra，-SO2NRa2，-NRaSO2Ra，-S （= O）R a，-S（= O）2 R a，-SO 2 OR a或-O SO 2 R a，其中G是氧或硫，Ra如说明书中所定义，R 2是氢，卤素，氰基，烷基，卤代烷基，烯基，卤代烯基，炔基，卤代炔基，烷氧基或卤代烷氧基， x是2,3,4,5,6或7，或其非对映异构体，对映异构体，盐或N-氧化物，条件是R 1不是5-氯-2,2 ，当R 2是氢并且x是3或4时，制备化合物I的方法和中间体，使用化合物I，其中R 1，R 2，R 3，用于防治昆虫，螨虫或线虫，以及用化合物I治疗，控制，预防或保护动物免受寄生虫侵袭或感染的方法。

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