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1. 发明授权

US5256679A Substituted guanidine derivatives, their preparation and use 失效
标题翻译：取代的胍衍生物，其制备和用途
公开(公告)号：US5256679A
公开(公告)日：1993-10-26
申请号：US745245
申请日：1991-08-14
申请人： Isao Minamida , Yasuyuki Kando , Hitoshi Ishizuka , Tetsuo Okauchi , Hideki Uneme
发明人： Isao Minamida , Yasuyuki Kando , Hitoshi Ishizuka , Tetsuo Okauchi , Hideki Uneme
IPC分类号： A01N51/00 , A01N43/40 , A01N43/78 , A01N43/84 , A01N47/44 , C07C255/58 , C07C277/08 , C07C279/34 , C07C335/40 , C07D205/10 , C07D207/40 , C07D207/404 , C07D207/44 , C07D207/448 , C07D209/48 , C07D211/88 , C07D213/16 , C07D213/36 , C07D213/61 , C07D213/69 , C07D213/75 , C07D241/12 , C07D277/12 , C07D277/20 , C07D277/28 , C07D277/32 , C07D277/34 , C07D277/38 , C07D277/48 , C07D417/12 , C07D213/26 , C07D277/30
CPC分类号： C07D207/404 , A01N51/00 , C07C255/58 , C07C335/40 , C07D205/10 , C07D207/448 , C07D209/48 , C07D211/88 , C07D213/61 , C07D213/69 , C07D241/12 , C07D277/32 , C07D277/34 , C07D417/12
摘要： Novel substituted nitroguanidine derivatives and salts thereof having the following formula: ##STR1## wherein R.sup.1 is a substituted or unsubstituted heterocyclic group; R.sup.2 is a group attached through a sulfur atom, a group attached through a phosphorus atom, cyano, --CO--OR.sup.6 wherein R.sup.6 is a substituted or unsubstituted hydrocarbon group or a substituted or unsubstituted heterocyclic group, or --CO--NR.sup.7 R.sup.8 wherein R.sup.7 and R.sup.8, which are the same or different, are each independently hydrogen, a substituted or unsubstituted hydrocarbon group or a substituted or unsubstituted heterocyclic group, or R.sup.7 and R.sup.8, taken together with the nitrogen atom to which they are attached are a cyclic amino group; R.sup.3 is hydrogen, a substituted or unsubstituted hydrocarbon group (except for one substituted with an oxo group at the binding site), a group attached through a sulfur atom, a group attached through a phosphorus atom, cyano, --CO--R.sup.9 wherein R.sup.9 is hydrogen, a substituted or unsubstituted hydrocarbon group or a substituted or unsubstituted heterocyclic group, --CO--OR.sup.10 wherein R.sup.10 is a substituted or unsubstituted hydrocarbon group or a substituted or unsubstituted heterocyclic group, or --CO--NR.sup.11 R.sup.12 wherein R.sup.11 and R.sup.12, which are the same or different, are each independently hydrogen, a substituted or unsubstituted hydrocarbon group or a substituted or unsubstituted heterocyclic group, or R.sup.11 and R.sup.12, taken together with the nitrogen atom to which they are attached are a cyclic amino group; and R.sup.4 is hydrogen or a lower alkyl group; which have unexpectedly potent pesticidal activity and very low toxicity.

2. 发明授权

US4612374A Tris-azetidinedione derivative 1,3,5-triazin-2,4,6-triones 失效
标题翻译：三 - 氮杂二酮衍生物1,3,5-三嗪-2,4,6-三嗪
公开(公告)号：US4612374A
公开(公告)日：1986-09-16
申请号：US811855
申请日：1985-12-20
申请人： Shenghong A. Dai
发明人： Shenghong A. Dai
IPC分类号： C07D205/10 , C07D205/12 , C07D403/14 , C08G18/32 , C08G18/50 , C08G18/71 , C08G18/78
CPC分类号： C07D403/14 , C07D205/10 , C07D205/12 , C08G18/3225 , C08G18/3228 , C08G18/5024 , C08G18/714 , C08G18/7881
摘要： Novel isocyanato-azetidinedione compounds are provided which have the formula ##STR1## wherein R and R.sub.1 can independently selected from hydrogen and hydrocarbyl or can be joined together and along with the carbon to which they are attached represent a cycloalkane residue having 4 to 6 ring carbon atoms, y is an integer from 1 to 7 and X is a hydrocarbon radical having a valency of y plus one.The monoisocyanate compounds are used as intermediates to provide further novel azetidinedione containing derivatives in the form of azetidinedione-isocyanurates (II) and azetidinedione-urethanes (III).All three classes of compounds can be employed as acid scavenging agents for stablizing various kinds of halogenated polymer systems. Notably, (I) and (III) form highly useful polyamide-polyureas and polyamide-polyurethanes respectively by reaction with organic polyamines.
摘要翻译：提供具有下式的新型异氰酸根合 - 氮杂二酮化合物：其中R和R 1可以独立地选自氢和烃基，或者可以连接在一起，并与它们所连接的碳一起代表具有4-6个环的环烷烃残基碳原子，y为1〜7的整数，X为化合价y为1的烃基。单异氰酸酯化合物用作中间体以提供含氮杂二酮 - 异氰脲酸酯（II）和氮杂二酮 - 氨基甲酸酯（III）形式的另外新的含有氮杂环丁二酮的衍生物。所有三类化合物都可以用作稳定各种卤化聚合物体系的酸清除剂。值得注意的是，（I）和（III）分别通过与有机多胺反应形成高度有用的聚酰胺 - 聚脲和聚酰胺 - 聚氨酯。

3. 发明授权

US4465842A Preparation of N-benzylimides 失效
标题翻译： N-苄基酰亚胺的制备
公开(公告)号：US4465842A
公开(公告)日：1984-08-14
申请号：US378223
申请日：1982-05-14
申请人： Michel Desbois , Michel Reppelin
发明人： Michel Desbois , Michel Reppelin
IPC分类号： C07D205/10 , C07D207/40 , C07D207/404 , C07D209/48 , C07D211/88 , C07D207/12
CPC分类号： C07D207/404 , C07D205/10 , C07D209/48 , C07D211/88
摘要： The N-benzylimides having the structural formula: ##STR1## wherein Ar comprises a benzene radical and R.sub.1 is an aliphatic or aromatic hydrocarbon, are prepared in good yield by reacting a compound having the structural formula:ArH (II)with a compound having the structural formula: ##STR2## in the presence of hydrofluoric acid.
摘要翻译：具有以下结构式的N-苄基酰亚胺：其中Ar包含苯基，R 1是脂族或芳族烃，通过使具有结构式：ArH（II）的化合物与化合物，其结构式为：（III）在氢氟酸存在下。

4. 发明授权

US4288366A Method of preparation of 5,6-dehydropenicillins 失效
标题翻译： 5,6-脱水青霉素的制备方法
公开(公告)号：US4288366A
公开(公告)日：1981-09-08
申请号：US58945
申请日：1979-07-19
申请人： Luciano Re , Alberto Brant , Luciano Bassignani
发明人： Luciano Re , Alberto Brant , Luciano Bassignani
IPC分类号： C07D499/46 , A61K31/397 , A61K31/43 , A61P31/04 , C07D205/08 , C07D205/095 , C07D205/10 , C07D499/00 , C07D499/06 , C07D499/21 , C07D499/44 , C07D499/60
CPC分类号： C07D499/00 , C07D205/095 , C07D205/10
摘要： A method is disclosed for the preparation of a class of dehydropenicillins by irradiating substituted 4-acylmethylthio-2-azetidinones and subsequently subjecting the as-obtained product to cyclization. Processing conditions and analytical data are reported.
摘要翻译：公开了通过照射取代的4-酰基甲硫基-2-氮杂环丁酮并随后使得到的产物环化来制备一类脱水青霉素的方法。报告处理条件和分析数据。

5. 发明授权

US4171302A Process for producing N-substituted amides 失效
标题翻译：制备N-取代酰胺的方法
公开(公告)号：US4171302A
公开(公告)日：1979-10-16
申请号：US853501
申请日：1977-11-21
申请人： Jean Abblard , Michel Baudoin
发明人： Jean Abblard , Michel Baudoin
IPC分类号： C07D207/40 , C07D207/404 , C07D207/44 , C07D207/448 , C07D207/452 , C07D205/10
CPC分类号： C07D207/404 , C07D207/448 , C07D207/452
摘要： A process of preparing a N-substituted imide as disclosed, which is carried out in accordance with the equation: ##STR1## wherein R is an alkyl radical containing 1 to 8 carbon atoms, or an aryl radical having 1 or 2 phenyl rings bearing up to 5 substituents selected from the group consisting of 1 to 3 atoms of halogen, 1 to 2 nitro, amino, or hydroxy groups, 1 to 4 alkyl radicals, and 1 to 2 alkoxy or alkylthiol radicals each containing 1 to 4 carbon atoms, or a hexyl radical, optionally substituted;R' is a single bond or a hydrocarbon chain containing from 1 to 4 carbon atoms, in which two contiguous carbons may belong to a phenyl ring, said hydrocarbon chain being saturated or unsaturated and optionally substituted andR" is a hydrogen atom, an alkaline metal atom, an ammonium atom or a lower alkyl having 1 to 4 carbon atoms, wherein the cyclization of the amic acid, R--NH--CO--R'--COOR" is carried out in the presence of a mixed catalyst which results from the association of the formula, A B, in which A is a strong inorganic or organic acid and B is a Lewis base.
摘要翻译：所公开的制备N-取代的酰亚胺的方法，其按照以下方程式进行：其中R是含有1至8个碳原子的烷基或具有1或2个苯环的芳基，至5个选自1至3个卤素原子，1至2个硝基，氨基或羟基，1至4个烷基和1至2个各自含有1至4个碳原子的烷氧基或烷基硫醇基团的取代基，或己基，任选取代; R'是单键或含有1至4个碳原子的烃链，其中两个连续的碳可以属于苯环，所述烃链是饱和或不饱和的且任选被取代，R“是氢原子，碱金属原子，铵原子或具有1至4个碳原子的低级烷基，其中酰胺酸R-NH-CO-R'-COOR“的环化在混合催化剂存在下进行，结果由式AB的结合，其中A是强无机或有机酸，B是路易斯碱。

6. 发明授权

US2955113A omega-(1-alkyl-piperidyl-4)-omega-acyl-hydrazine derivatives 失效
公开(公告)号：US2955113A
公开(公告)日：1960-10-04
申请号：US82218959
申请日：1959-06-23
申请人： SANDOZ LTD
发明人： ERNST JUCKER , ERWIN RISSI , RUDOLF SUESS , ARNOLD VOGEL , EBCRHARD WOLFF
IPC分类号： C07D205/10 , C07D401/12 , C07D403/12
CPC分类号： C07D401/12 , C07D205/10 , C07D403/12

7. 发明申请

US20220380311A1 METHOD FOR PRODUCING AROMATIC HETEROCYCLIC RING-SUBSTITUTED DIFLUOROACETIC ACID DERIVATIVE 有权
公开(公告)号：US20220380311A1
公开(公告)日：2022-12-01
申请号：US17813499
申请日：2022-07-19
申请人： AGC Inc.
发明人： Yoshitaka NOMURA , Eiichiro ANRAKU
IPC分类号： C07D213/24 , C07D215/16 , C07D241/44 , C07D237/30 , C07D277/64 , C07D205/10
摘要： A method for producing an aromatic heterocycle-substituted difluoroacetic acid derivative having a partial structure represented by the formula (III), by reacting an N-oxido aromatic heterocyclic compound having a partial structure represented by the formula (I) with tetrafluoroethylene in the presence of a compound represented by the formula (II): R—YH, in a solvent selected from an aromatic hydrocarbon solvent, an ester solvent and an ether solvent:

8. 发明授权

US5705522A Compounds having anti-inflammatory and anti-viral activity, compositions of these, alone and in combination with reverse transcriptase inhibitors 失效
标题翻译：具有抗炎和抗病毒活性的化合物，它们的组合物，单独和与逆转录酶抑制剂组合
公开(公告)号：US5705522A
公开(公告)日：1998-01-06
申请号：US600525
申请日：1996-02-13
申请人： Farid Hamedi-Sangsari , Fabienne Nugier , Thierry Vallet , Jacques Grange , Jorge Vila
发明人： Farid Hamedi-Sangsari , Fabienne Nugier , Thierry Vallet , Jacques Grange , Jorge Vila
IPC分类号： A61K31/00 , A61K31/195 , A61K31/197 , A61K31/40 , A61K31/401 , A61K31/4015 , A61P29/00 , A61P31/00 , A61P31/12 , C07C259/06 , C07D207/46 , A01N43/36 , C07C209/28 , C07D205/10 , C12P21/02
CPC分类号： C07C259/06 , C07D207/46
摘要： A new family of compounds having anti-inflammatory, anti-viral, and brocho-dilating activity having the following linear and cyclic formulas: ##STR1## and compositions of these, which alone, and in combination with reverse transcriptase inhibitors thereby resulting in an additive or synergistic effect, are useful in inhibiting or suppressing viruses including those exhibiting retroviral replication, or in treating viruses including a retrovirus such as HIV in a human cell population and methods of using these compositions, compounds, and salts thereof.
摘要翻译：一种新的具有抗炎，抗病毒和展开扩张活性的化合物，具有以下线性和环状配方：单独的这些化合物（其为单体形式）和它们的组合物并且与逆转录酶抑制剂组合，从而产生添加剂或协同效应，可用于抑制或抑制包括显示逆转录病毒复制的病毒，或在人细胞群体中治疗包括逆转录病毒例如HIV的病毒以及使用这些病毒的方法组合物，化合物及其盐。

9. 发明授权

US4803266A 3-Oxoalkylidene-2-azetidinone derivatives 失效
标题翻译： 3-氧代亚烷基-2-氮杂环丁酮衍生物
公开(公告)号：US4803266A
公开(公告)日：1989-02-07
申请号：US104152
申请日：1987-10-05
申请人： Yutaka Kawashima , Masakazu Satoh , Yuichi Hatada , Fumiko Hazato , Yoshimoto Nakashima , Kaoru Sota
发明人： Yutaka Kawashima , Masakazu Satoh , Yuichi Hatada , Fumiko Hazato , Yoshimoto Nakashima , Kaoru Sota
IPC分类号： C07D205/08 , A61K31/395 , A61K31/397 , A61P7/02 , C07D205/10 , C07D405/04
CPC分类号： C07D205/10
摘要： 2-Azetidione derivatives represented by the following formula ##STR1## wherein X is a hydrogen atom, a halogen atom, a lower alkyl group, a lower alkoxy group, a hydroxyl group or a cyano group, l is 1 or 2, R.sup.1 is a lower alkyl group, a cycloalkyl group, a 1-naphthylmethyl group, an optionally substituted phenethyl group, an optionally substituted phenyl group, an optionally substituted benzyl group or a bis(alkoxycarbonyl)ethyl group, and R.sup.2 is a lower alkyl group, a lower alkoxy group, an amino group, an adamantyl group, a lower alkoxycarbonylmethyl group or an optionally substituted phenyl group, are disclosed. These compounds are useful as blood platelet aggregation inhibiting agents.

10. 发明授权

US3505295A Polyimide molding powders 失效
标题翻译：聚酰亚胺模塑粉
公开(公告)号：US3505295A
公开(公告)日：1970-04-07
申请号：US3505295D
申请日：1967-02-13
申请人： PHILIPS CORP
发明人： GRUNSTEID WALTER EDMUND , JANSSEN PETRUS JOHANNES
IPC分类号： C07D205/10 , C07D209/48 , C07D487/04 , C08G73/10 , C08G20/32
CPC分类号： C07D487/04 , C07D205/10 , C07D209/48 , C08G73/1007

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