专利快速检索-快速检索全球专利，免费商用专利数据库-IPRDB

1. 发明申请

US20110004000A1 Mitotic Kinesin Inhibitor 审中-公开
标题翻译：有丝分裂驱动蛋白抑制剂
公开(公告)号：US20110004000A1
公开(公告)日：2011-01-06
申请号：US12883338
申请日：2010-09-16
申请人： Chikara MURAKATA , Yoshinori YAMASHITA , Ryuichiro NAKAI , Kazuhito AKASAKA , Yoji INO , Kazuhiko KATO , Yushi KITAMURA
发明人： Chikara MURAKATA , Yoshinori YAMASHITA , Ryuichiro NAKAI , Kazuhito AKASAKA , Yoji INO , Kazuhiko KATO , Yushi KITAMURA
IPC分类号： C07D285/135
CPC分类号： C07D285/13 , A61K31/433 , A61K31/4439 , A61K31/506 , A61K31/5377 , C07D285/135
摘要： A mitotic kinesin Eg5 inhibitor which comprises a thiadiazoline derivative represented by the general formula (I) or a pharmacologically acceptable salt thereof as an active ingredient: [wherein R1 represents a hydrogen atom and the like, R2 represents a hydrogen atom, —C(═W)R6 (wherein W represents an oxygen atom or a sulfur atom, and R6 represents substituted or unsubstituted lower alkyl and the like) and the like, R3 represents —C(═Z)R19 (wherein Z represents an oxygen atom or a sulfur atom, and R19 represents substituted or unsubstituted lower alkyl and the like) and the like, R4 represents substituted or unsubstituted lower alkyl and the like, and R5 represents substituted or unsubstituted aryl and the like] and the like are provided.
摘要翻译：一种有丝分裂驱动蛋白Eg5抑制剂，其包含由通式（I）表示的噻二唑啉衍生物或其药理学上可接受的盐作为活性成分：[其中R 1表示氢原子等，R 2表示氢原子，-C（= W）R6（其中W表示氧原子或硫原子，R6表示取代或未取代的低级烷基等）等，R3表示-C（= Z）R19（其中Z表示氧原子或硫原子原子，R 19表示取代或未取代的低级烷基等）等，R 4表示取代或未取代的低级烷基等，R 5表示取代或未取代的芳基等〕等。

2. 发明申请

US20100197696A1 PESTICIDAL HETEROCYCLIC DIHALOALLYL COMPOUNDS 审中-公开
标题翻译：杀虫剂杂环二氢化合物
公开(公告)号：US20100197696A1
公开(公告)日：2010-08-05
申请号：US12756596
申请日：2010-04-08
申请人： Roger Graham Hall , Stephan Trah , Werner Zambach , Juraj Tuleja
发明人： Roger Graham Hall , Stephan Trah , Werner Zambach , Juraj Tuleja
IPC分类号： A01N43/824 , C07D285/13 , C07D271/10 , C07D249/12 , C07D257/04 , C07D237/14 , C07D239/36 , C07D241/18 , A01N43/653 , A01N43/713 , A01N43/58 , A01N43/60 , A01N43/54
CPC分类号： C07D271/113 , C07D233/72 , C07D237/14 , C07D239/36 , C07D241/18 , C07D249/12 , C07D273/04 , C07D285/13
摘要： The invention relates to compounds of formula wherein Het, A1, A2, A3, A4, D, W, T, Q, Y, X1, X2, R1, R2, R3, R4, k and m are as defined hereinabove, and, where applicable, to possible E/Z isomers, mixtures of E/Z isomers and/or tautomers thereof, in each case in free form or in salt form, to a process for the preparation of and to the use of those compounds, E/Z isomers, mixtures of E/Z isomers and/or tautomers, to pesticidal compositions in which the active ingredient has been selected from those compounds, E/Z isomers, mixtures of E/Z isomers and/or tautomers, in each case in free form or in agrochemically usable salt form, to a process for the preparation of and to the use of those compositions, to plant propagation material treated with those compositions, to a method of controlling pests, to intermediates and, where applicable, to possible E/Z isomers, mixtures of E/Z isomers and/or tautomers thereof, in each case in free form or in salt form, for the preparation of those compounds, E/Z isomers, mixtures of E/Z isomers and/or tautomers, and to a process for the preparation of and to the use of those intermediates and, where applicable, possible E/Z isomers, mixtures of E/Z isomers and/or tautomers thereof.
摘要翻译：本发明涉及下式的化合物，其中Het，A1，A2，A3，A4，D，W，T，Q，Y，X1，X2，R1，R2，R3，R4，k和m如上所定义，在适用的情况下，可能的E / Z异构体，E / Z异构体和/或其互变异构体的混合物，在每种情况下为游离形式或盐形式，用于制备和使用这些化合物的方法E / Z异构体，E / Z异构体和/或互变异构体的混合物，其中活性成分选自那些化合物，E / Z异构体，E / Z异构体和/或互变异构体的混合物，在每种情况下为游离形式或农业化学上可用的盐形式，涉及制备和使用这些组合物，用这些组合物处理的繁殖材料的方法，控制害虫的方法，中间体和适用时可能的E / Z异构体，E / Z异构体和/或其互变异构体的混合物，在每种情况下为游离形式或盐形式，用于制备这些化合物 ds，E / Z异构体，E / Z异构体和/或互变异构体的混合物，以及制备和使用那些中间体的方法，以及在适用时可能的E / Z异构体，E / Z异构体的混合物和/或其互变异构体。

3. 发明申请

US20080255196A1 Pesticide Thiazolyloxy Substituted Phenylamidine Derivatives 有权
标题翻译：农药噻唑氧基取代的苯脒衍生物
公开(公告)号：US20080255196A1
公开(公告)日：2008-10-16
申请号：US12063670
申请日：2006-09-12
申请人： Klaus Kunz , Jorg Greul , Oliver Guth , Benoit Hartmann , Kerstin Ilg , Wahed Ahmed Moradi , Thomas Seitz , Peter Dahmen , Arnd Voerste , Ulrike Wachendorff-Neumann , Ralf Dunkel , Ronald Ebbert , Eva-Maria Franken , Olga Malsam
发明人： Klaus Kunz , Jorg Greul , Oliver Guth , Benoit Hartmann , Kerstin Ilg , Wahed Ahmed Moradi , Thomas Seitz , Peter Dahmen , Arnd Voerste , Ulrike Wachendorff-Neumann , Ralf Dunkel , Ronald Ebbert , Eva-Maria Franken , Olga Malsam
IPC分类号： A01N43/78 , C07D277/34 , C07D285/08 , A01N43/836 , A01P3/00 , A01P7/04 , C07D401/12
CPC分类号： A01N43/78 , A01N43/82 , C07D277/34 , C07D277/56 , C07D277/68 , C07D285/08 , C07D285/125 , C07D285/13 , C07D417/12
摘要： The present invention relates to aryloxy substituted phenylamidine derivatives of formula (I) wherein the substituents are as in the description, their process of preparation, their use as fungicide or insecticide active agents, particularly in the form of fungicide or insecticide compositions, and methods for the control of phytopathogenic fungi or damaging insects, notably of plants, using these compounds or compositions (I).
摘要翻译：本发明涉及式（I）的芳氧基取代的苯基脒衍生物，其中取代基如说明书，其制备方法，它们作为杀真菌剂或杀虫剂活性剂的用途，特别是杀真菌剂或杀虫剂组合物的形式，以及用于使用这些化合物或组合物（I）控制植物病原真菌或损害昆虫，特别是植物的昆虫。

4. 发明授权

US06893650B1 N2-phenylamidine derivatives 有权
标题翻译： N2-苯基脒衍生物
公开(公告)号：US06893650B1
公开(公告)日：2005-05-17
申请号：US09890775
申请日：2000-02-04
申请人： Mark David Charles , Wilfried Franke , David Eric Green , Thomas Lawley Hough , Dale Robert Mitchell , Donald James Simpson , John Frederick Atherall
发明人： Mark David Charles , Wilfried Franke , David Eric Green , Thomas Lawley Hough , Dale Robert Mitchell , Donald James Simpson , John Frederick Atherall
IPC分类号： C07D249/08 , A01N25/02 , A01N37/52 , A01N41/10 , A01N43/06 , A01N43/18 , A01N43/40 , A01N43/54 , A01N43/74 , A01N43/76 , A01N43/80 , A01N43/82 , A01N43/836 , A01N43/84 , A01N43/88 , A01N43/90 , A01N47/42 , A01P3/00 , C07C233/37 , C07C251/04 , C07C257/12 , C07C257/14 , C07C317/40 , C07C323/20 , C07C323/41 , C07D207/325 , C07D207/50 , C07D209/48 , C07D213/64 , C07D213/68 , C07D215/22 , C07D237/14 , C07D237/16 , C07D239/34 , C07D239/46 , C07D239/88 , C07D241/24 , C07D251/30 , C07D251/34 , C07D257/04 , C07D261/08 , C07D261/14 , C07D263/38 , C07D263/46 , C07D263/58 , C07D271/06 , C07D271/10 , C07D273/00 , C07D277/20 , C07D277/34 , C07D277/68 , C07D285/00 , C07D285/08 , C07D285/10 , C07D285/12 , C07D285/13 , C07D295/12 , C07D295/125 , C07D307/12 , C07D307/81 , C07D307/83 , C07D311/22 , C07D311/56 , C07D317/64 , C07D333/16 , C07D333/20 , C07D333/28 , C07D333/54 , C07D333/58 , C07D333/64 , C07D487/04 , C07D495/04 , C07F7/08 , A61K31/155 , C07D237/00 , C07D261/20 , C07D233/37
CPC分类号： C07D209/48 , A01N37/52 , A01N43/06 , A01N43/40 , A01N43/54 , A01N43/74 , A01N43/82 , A01N43/90 , A01N47/42 , C07C257/12 , C07C257/14 , C07D207/50 , C07D239/88 , C07D251/34 , C07D261/08 , C07D263/38 , C07D263/46 , C07D263/58 , C07D271/06 , C07D271/10 , C07D285/08 , C07D285/13 , C07D295/125 , C07D311/22 , C07D333/54 , C07D487/04 , C07D495/04 , C07F7/0812
摘要： The invention provides fungicidal compounds of formula (I) and salts thereof wherein: R1 is alkyl, alkenyl, alkynyl, carbocyclyl or heterocyclyl, each of which may be substituted, or hydrogen; R2 and R3, which may be the same or different, are any group defined for R1; cyano; acyl; —ORa or —SRa, where Ra is alkyl, alkenyl, alkynyl, carbocyclyl or heterocyclyl, each of which may be substituted; or R2 and R3, or R2 and R1, together with their interconnecting atoms may form a ring, which may be substituted; R4 is alkyl, alkenyl, alkynyl, carbocyclyl or heterocyclyl, each of which may be substituted; hydroxy; mercapto; azido; nitro; halogen; cyano; acyl; optionally substituted amino; cyanato; thiocyanato; —SF5; —ORa; —SRa or —Si(Ra)3; m is 0 to 3; when present R5, which may be the same or different to any other R5, is any group defined for R4; R6 is optionally substituted carbo- or heterocylclyl; and A is a defined linking group, or —A—R6 and R5 together with benzene ring M form an optionally substituted fused ring system.
摘要翻译：本发明提供式（I）的杀真菌化合物及其盐，其中：R 1是烷基，烯基，炔基，碳环基或杂环基，其各自可以被取代，或氢; R 2和R 3可以相同或不同，为R 1定义的任何基团; 氰基酰基; 其中R a是烷基，烯基，炔基，碳环基或杂环基，其各自可以被取代;或者其中R a，或R 2和R 3，或R 2和R 1以及它们的互连原子可以形成环，其可以被取代; R 4是烷基，烯基，炔基，碳环基或杂环基，其各自可以被取代; 羟基; 巯基叠氮硝基卤素; 氰基酰基; 任选取代的氨基; 青色硫氰酸 -SF 5; -OR ^{a ; -SR ^{a或-Si（R a a）3 3; m为0〜3; 当存在R 5可以与任何其它R 5相同或不同时，R 5为限定的任何基团。 R 6是任选取代的碳 - 或杂环基; 并且A是限定的连接基团，或者-A-R 6和R 5和苯环M一起形成任选取代的稠环体系。}}

5. 发明申请

US20040192704A1 Non-nucleoside reverse transcriptase inhibitors 有权
标题翻译：非核苷逆转录酶抑制剂
公开(公告)号：US20040192704A1
公开(公告)日：2004-09-30
申请号：US10807766
申请日：2004-03-23
申请人： Roche Palo Alto LLC
发明人： James Patrick Dunn , Steven Swallow , Zachary Kevin Sweeney
IPC分类号： A61K031/506 , A61K031/497 , A61K031/4709 , A61K031/517 , A61K031/4439 , A61K031/4196 , C07D43/02
CPC分类号： C07D271/113 , C07D249/12 , C07D285/13
摘要： This invention relates to novel heterocyclic compounds of formula I wherein R1nullR4, X1 and X2 are as defined in the summary and pharmaceutically acceptable salts and solvates thereof, methods to inhibit or modulate Human Immunodeficiency Virus (HIV) reverse transcriptase with compounds of formula I, pharmaceutical compositions containing of formula I admixed with at least one solvent, carrier or excipient and processes to prepare compounds of formula I. The compounds are useful for treating disorders in which HIV and genetically related viruses are implicated 1
摘要翻译：本发明涉及式I的新型杂环化合物，其中R 1 -R 4，X 1和X 2如其概述及其药学上可接受的盐和溶剂化物所定义，抑制或调节人的方法具有式I化合物的免疫缺陷病毒（HIV）逆转录酶，含有式I的药物组合物与至少一种溶剂，载体或赋形剂混合，以及制备式I化合物的方法。该化合物可用于治疗HIV和遗传性疾病涉及相关病毒

6. 发明授权

US5985797A Herbicidal compositions based on N-isopropyl-N-(4-fluorophenyl) (5-trifluoromethyl-1,3,4-thiadiazol-2-yloxy)acetamide 失效
标题翻译：基于N-异丙基-N-（4-氟苯基）（5-三氟甲基-1,3,4-噻二唑-2-基氧基）乙酰胺的除草组合物
公开(公告)号：US5985797A
公开(公告)日：1999-11-16
申请号：US85881
申请日：1998-05-27
申请人： Peter Dahmen , Dieter Feucht
发明人： Peter Dahmen , Dieter Feucht
IPC分类号： A01N43/82 , C07D285/12 , C07D285/13 , A01N43/36 , A01N43/40 , A01N43/50
CPC分类号： C07D285/13 , A01N43/82
摘要： The present invention relates to novel synergistic herbicidal combinations of N-isopropyl-N-(4-fluorophenyl)(5-trifluoromethyl-1,3,4-thiadiazol-2-yloxy)acetamide with fenoxaprop-ethyl and/or clodinafop-propargyl.
摘要翻译：本发明涉及N-异丙基-N-（4-氟苯基）（5-三氟甲基-1,3,4-噻二唑-2-基氧基）乙酰胺与二烯丙基和/或氯二膦酰炔丙基的新型协同除草组合。

7. 发明授权

US5550140A Oxa(thia)diazol- and triazol-ones(thiones) having a miticide and insecticide activity 失效
公开(公告)号：US5550140A
公开(公告)日：1996-08-27
申请号：US391240
申请日：1995-02-21
申请人： Franco Bettarini , Luigi Capuzzi , Piero La Porta , Sergio Massimini , Vincenzo Caprioli
发明人： Franco Bettarini , Luigi Capuzzi , Piero La Porta , Sergio Massimini , Vincenzo Caprioli
IPC分类号： A01N43/653 , A01N43/82 , A01N43/824 , C07D249/12 , C07D271/10 , C07D271/113 , C07D285/12 , C07D285/125 , C07D285/13 , A61K31/41
CPC分类号： C07D271/113 , A01N43/653 , A01N43/82 , C07D249/12 , C07D285/13
摘要： A description follows of oxa(thia)diazol- and triazol-ones(thiones), with aiticide and insecticide activity, having the general formula ##STR1## wherein: Y=0, S; Z=0, S, NCH.sub.3, one of the two substituents P and Q is an ortho-substituted phenyl and the other a substituted benzyl.

8. 发明授权

US5418246A Oxa(thia)diazol- and triazol-ones(thiones) having a miticide and insecticide activity 失效
标题翻译：具有杀螨剂和杀虫剂活性的牛（thia）二唑和三唑（thiones）
公开(公告)号：US5418246A
公开(公告)日：1995-05-23
申请号：US945135
申请日：1992-09-15
申请人： Franco Bettarini , Luigi Capuzzi , Piero La Porta , Sergio Massimini , Vincenzo Caprioli
发明人： Franco Bettarini , Luigi Capuzzi , Piero La Porta , Sergio Massimini , Vincenzo Caprioli
IPC分类号： A01N43/653 , A01N43/82 , A01N43/824 , C07D249/12 , C07D271/10 , C07D271/113 , C07D285/12 , C07D285/125 , C07D285/13
CPC分类号： C07D271/113 , A01N43/653 , A01N43/82 , C07D249/12 , C07D285/13
摘要： A description follows of oxa(thia)diazol- and triazol-ones(thiones), with aiticide and insecticide activity, having the general formula ##STR1## wherein: Y=0, S; Z=0, S, NCH.sub.3, one of the two substituents P and Q is an ortho-substituted phenyl and the other a substituted benzyl.
摘要翻译：以下描述具有杀螨剂和杀虫活性的具有通式（I）的氧杂（噻吩）二唑和三唑（thiones）（thiones），其中：Y = 0，S; Z = 0，S，NCH 3，两个取代基P和Q中的一个是邻位取代的苯基，另一个是取代的苄基。

9. 发明授权

US5250551A New (hetero)aryl substituted diazole derivatives, the method of preparing them and application thereof in therapeutics 失效
标题翻译：新的（杂）芳基取代的二唑衍生物，其制备方法及其在治疗中的应用
公开(公告)号：US5250551A
公开(公告)日：1993-10-05
申请号：US816819
申请日：1992-01-03
申请人： Rene L. Milcent , Luc Lebreton , Fathi Mazouz , Claude Burstein , Salah Gueddari
发明人： Rene L. Milcent , Luc Lebreton , Fathi Mazouz , Claude Burstein , Salah Gueddari
IPC分类号： C07D257/04 , C07D271/10 , C07D271/113 , C07D285/12 , C07D285/125 , C07D285/13 , C07D401/04 , C07D403/06 , A61K31/41
CPC分类号： C07D257/04 , C07D271/113 , C07D285/125 , C07D285/13 , C07D401/04 , C07D403/06
摘要： Compounds for therapeutic use of formula: ##STR1## where the chain--W--V--N--represents--N.dbd.N--N--, --N--N.dbd.N--,--O--CO--N--,--O--CS--N--, --S--CO--N--or--S--CS--N--; Ar is an aryl group; and A is a vinyl group or an alkylene chain terminated by CN, methoxy, ethoxy, OH, halogen or NH.sub.2 which may possibly be substituted.
摘要翻译：用于治疗用途的化合物：其中链-WVN-表示-N = NN-，-NN = N - ， - O-CO-N - ， - O-CS-N-，-S -CO-N-或-S-CS-N-; Ar是芳基; 并且A是乙烯基或被CN，甲氧基，乙氧基，OH，卤素或可能被取代的NH 2封端的亚烷基链。

10. 发明授权

US5236939A Substituted 1,3,4-oxa(thia)diazolinones process for their preparation and their use of combating endoparasites 失效
标题翻译：取代1,3,4-氧杂（噻吩）二唑啉酮的制备方法及其对抗内寄生虫
公开(公告)号：US5236939A
公开(公告)日：1993-08-17
申请号：US778023
申请日：1991-10-17
申请人： Gerhard Bonse , Nikolaus Muller , Achim Harder
发明人： Gerhard Bonse , Nikolaus Muller , Achim Harder
IPC分类号： A01N43/824 , C07D271/10 , C07D271/113 , C07D285/12 , C07D285/125 , C07D285/13
CPC分类号： C07D271/113 , C07D285/125 , C07D285/13
摘要： Substituted 1,3,4 -oxa- diazolinones of the formula (I) ##STR1## in which X represents O andY represents O or S,are disclosed as useful to combat endoparasites.
摘要翻译：公开了其中X代表O且Y代表O或S的式（I）的取代的1,3,4-恶二唑啉酮用于对抗内寄生虫。

你已经成功收藏专利！

检索式保存成功!

IPRDB

热门服务

关于我们

友情链接

联系方式