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1. 发明授权

US07001897B2 1-methylcarbapenem derivatives 失效
标题翻译： 1-甲基碳青霉烯衍生物
公开(公告)号：US07001897B2
公开(公告)日：2006-02-21
申请号：US10439198
申请日：2003-05-15
申请人： Yoshiyuki Kobayashi , Tsuyoshi Shinozuka , Osamu Kanno
发明人： Yoshiyuki Kobayashi , Tsuyoshi Shinozuka , Osamu Kanno
IPC分类号： C07D477/20 , A61K31/454 , A61K31/421 , A61K31/426 , A61P31/04
CPC分类号： C07D477/20
摘要： A 1-methylcarbapenem compound represented by the formula (I): having antibacterial activity, pharmacologically acceptable esters or salts thereof and pharmaceutical compositions (particularly antibacterial agents) containing them as an active ingredient are described. In addition, the invention includes the use of these compounds, ester derivatives or salts for the manufacture of pharmaceutical compositions, or a method for the prevention or treatment of diseases (particularly bacterial infections) by administering a pharmacologically effective amount of the compounds, ester derivatives or salts to warm-blooded animals (particularly human beings).
摘要翻译：由式（I）表示的1-甲基碳青霉烯化合物

2. 发明申请

US20070219234A1 Thienopyridine Derivatives 审中-公开
标题翻译：噻吩并吡啶衍生物
公开(公告)号：US20070219234A1
公开(公告)日：2007-09-20
申请号：US11578492
申请日：2005-04-11
申请人： Kiyoshi Oizumi , Satoru Naito , Akira Nakao , Tsuyoshi Shinozuka , Satoshi Matsui , Kousei Shimada
发明人： Kiyoshi Oizumi , Satoru Naito , Akira Nakao , Tsuyoshi Shinozuka , Satoshi Matsui , Kousei Shimada
IPC分类号： A61K31/4365 , C07D513/04
CPC分类号： C07D495/04 , A61K31/4365 , A61K31/4545 , A61K31/4725 , A61K31/496 , A61K31/5377 , A61K31/541 , A61K31/55 , A61K31/551 , A61K31/553 , A61K31/554
摘要： [Problem to be Solved]The present invention provides a compound promoting osteogenesis. [Solution] The present invention provides a compound having the following general formula (I) wherein R1 is H or alkyl, R2 is RaS—, RaO—, RaNH—, Ra(Rb)N— or cyclic amino, and Ra and Rb are alkyl which may be substituted, cycloalkyl which may be substituted, or the like, or a pharmacologically acceptable salt thereof.
摘要翻译： [待解决的问题]本发明提供促进成骨的化合物。 [溶液]本发明提供具有以下通式（I）的化合物，其中R 1是H或烷基，R 2是R a，O （S），R a，O，R a，O，R a，或环状氨基，R a和R b都为可被取代的烷基，可被取代的环烷基等，或其药学上可接受的盐。

3. 发明申请

US20100004221A1 THIAZEPINE DERIVATIVE 审中-公开
标题翻译：噻吩衍生物
公开(公告)号：US20100004221A1
公开(公告)日：2010-01-07
申请号：US12493056
申请日：2009-06-26
申请人： Toru Hasegawa , Tsuyoshi Shinozuka
发明人： Toru Hasegawa , Tsuyoshi Shinozuka
IPC分类号： A61K31/554 , C07D513/04 , A61P3/10 , A61P3/00
CPC分类号： C07D513/04
摘要： Thiazepine derivative or a pharmacologically acceptable salt thereof having an effect of inhibiting 11β-hydroxysteroid dehydrogenase type 1 and having a formula (1): wherein in one embodiment, R1 represents a hydrogen atom, a C1-C6 alkyl group; R2 represents a C1-C6 alkyl group, a C1-C6 halogenated alkyl group, a C1-C6 hydroxyalkyl group; R1 represents a hydrogen atom or a C1-C6 alkyl group; R4 represents a C6-C10 aryl group that may be substituted with 1 to 5 group(s) independently selected from Substituent Group a or a heterocyclic group that may be substituted with 1 to 3 group(s) independently selected from Substituent Group a; Substituent Group a consists of a halogen atom, a C1-C6 alkyl group, a C6-C10 aryl group that may be substituted with 1 to 5 group(s) independently selected from Substituent Group b; Substituent Group b consists of a halogen atom, a C1-C6 alkyl group, and a C1-C6 halogenated alkyl group.
摘要翻译：具有抑制1型11β-羟类固醇脱氢酶1型并具有式（1）的作用的噻吩衍生物或其药学上可接受的盐：其中在一个实施方案中，R 1表示氢原子，C 1 -C 6烷基; R2表示C1-C6烷基，C1-C6卤代烷基，C1-C6羟烷基; R1表示氢原子或C1-C6烷基; R4表示可以被独立地选自取代基组a的1〜5个基团或可以被1〜3个独立地选自取代基组a的基团取代的杂环基团取代的C6〜C10芳基; 取代基a由卤素原子，C1-C6烷基，可以被1至5个独立地选自取代基组b的基团取代的C6-C10芳基组成; 取代基组b由卤素原子，C1-C6烷基和C1-C6卤代烷基组成。

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