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1. 发明授权

US4310533A Guanidinobenzoic acid derivatives 失效
标题翻译：胍基苯甲酸衍生物
公开(公告)号：US4310533A
公开(公告)日：1982-01-12
申请号：US182513
申请日：1980-08-29
申请人： Yoshiaki Uegai , Tsuyoshi Watanabe , Masashi Shiota , Itsuo Okumoto , Naohiro Kayama
发明人： Yoshiaki Uegai , Tsuyoshi Watanabe , Masashi Shiota , Itsuo Okumoto , Naohiro Kayama
IPC分类号： A61K31/215 , A61K31/245 , A61K31/395 , A61K31/445 , A61P7/04 , A61P43/00 , C07C279/18 , C07D295/185 , C12N9/99 , C07C101/68
CPC分类号： C07D295/185 , C07C279/18
摘要： The guanidinobenzoic acid derivatives of the general formula: ##STR1## wherein Z represents a carbon-carbon covalent bond, or a methylene, ethylene or vinylene group, R.sup.1 represents a hydrogen atom, or a straight- or branched-chain alkyl group containing from 1 to 4 carbon atoms, R.sup.2 represents a straight- or branched-chain alkyl group containing from 4 to 10 carbon atoms, or a cycloalkyl or cycloalkenyl or straight- or branched-chain alkenyl group containing from 3 to 8 carbon atoms, or a phenyl or benzyl group, or NR.sup.1 R.sup.2 represents a 4- to 8-membered heterocyclic ring, and acid addition salts thereof, have anti-plasmin and anti-trypsin activities.
摘要翻译：通式为：其中Z表示碳 - 碳共价键，或亚甲基，亚乙基或亚乙烯基的通式为（I）的胍基苯甲酸衍生物，R1表示氢原子或直链或支链烷基含有1至4个碳原子，R 2表示含有4至10个碳原子的直链或支链烷基，或含有3至8个碳原子的环烷基或环烯基或直链或支链烯基，或苯基或苄基，或NR1R2表示4至8元杂环，并且其酸加成盐具有抗纤溶酶和抗胰蛋白酶活性。

2. 发明授权

US4283418A Guanidinobenzoic acid derivatives and process for their preparation 失效
标题翻译：胍基苯甲酸衍生物及其制备方法
公开(公告)号：US4283418A
公开(公告)日：1981-08-11
申请号：US123609
申请日：1980-02-22
申请人： Setsuro Fujii , Tsuyoshi Watanabe , Masashi Shiota , Itsuo Okumoto , Naohiro Kayama
发明人： Setsuro Fujii , Tsuyoshi Watanabe , Masashi Shiota , Itsuo Okumoto , Naohiro Kayama
IPC分类号： A61K31/155 , A61K31/165 , A61K31/18 , A61K31/24 , A61K31/245 , C07C101/56
CPC分类号： A61K31/155 , A61K31/165 , A61K31/18 , A61K31/24 , A61K31/245
摘要： Guanidinobenzoic acid derivatives represented by the general formula [I] ##STR1## wherein R.sup.1, R.sup.2 and Z are as defined hereinafter, having antiplasmin and anti-trypsin activities and process for their preparation as well as a pharmaceutical composition and a method of inhibiting the activity of plasmin and trypsin is disclosed.
摘要翻译：由通式[I]表示的胍基苯甲酸衍生物其中R1，R2和Z如下文所定义，具有抗血浆素和抗胰蛋白酶活性及其制备方法以及药物组合物和方法公开了抑制纤溶酶和胰蛋白酶的活性。

3. 发明授权

US4224342A Guanidinobenzoic acid compounds and process for preparing the same 失效
标题翻译：胍基苯甲酸化合物及其制备方法
公开(公告)号：US4224342A
公开(公告)日：1980-09-23
申请号：US959276
申请日：1978-11-09
申请人： Setsuro Fujii , Tsuyoshi Watanabe , Masashi Shiota , Okumoto Itsuo , Naohiro Kayama
发明人： Setsuro Fujii , Tsuyoshi Watanabe , Masashi Shiota , Okumoto Itsuo , Naohiro Kayama
IPC分类号： A61K31/245 , A61P1/00 , A61P7/04 , C07C279/18 , A61K31/155 , C07C129/12
CPC分类号： C07C279/18 , Y02P20/55
摘要： Guanidinobenzoic acid compounds represented by the formula ##STR1## wherein R and Z are as defined hereinafter, having anti-plasmin and anti-trypsin activities and processes for preparing the same as well as a pharmaceutical composition and a method of inhibiting the activity of plasmin and a trypsin is disclosed.
摘要翻译：由下式表示的胍基苯甲酸化合物，其中R和Z如下文所定义，具有抗纤溶酶和抗胰蛋白酶活性及其制备方法以及药物组合物和抑制活性的方法的纤溶酶和胰蛋白酶。

4. 发明授权

US5876760A Granules containing pranlukast, process for producing the granules, and method of improving adhesiveness of pranlukast 失效
标题翻译：含有普鲁司特的颗粒，生产颗粒的方法，以及提高普鲁司特的粘合性的方法
公开(公告)号：US5876760A
公开(公告)日：1999-03-02
申请号：US981083
申请日：1997-12-12
申请人： Seiei Sasatani , Masashi Shiota , Yoshinori Ii
发明人： Seiei Sasatani , Masashi Shiota , Yoshinori Ii
IPC分类号： A61K9/16 , A61K31/41
CPC分类号： A61K9/1652 , A61K31/41 , A61K9/1623 , A61K9/1635 , A61K9/1641
摘要： Spray-dried granules comprising pranlukast (A) and one or more saccharide(s) (B) as essential ingredients and further comprising one or more water-soluble polymer(s) (C) and/or one or more surfactant(s) (D); a process for producing the same; and a method for improving adhesiveness of pranlukast are provided. According to the present invention, the very strong adhesiveness of pranlukast is reduced, and pranlukast-containing granules having little adhesiveness, a narrow particle size distribution, and good flow properties can be produced efficiently. The pranlukast-containing granules of the present invention cause no troubles in continuous production of capsules, tablets, and the like, and the resulting pranlukast-containing granules exhibit excellent disintegrating and dispersing properties.
摘要翻译： PCT No.PCT / JP96 / 01578 Sec。 371日期1997年12月12日 102（e）日期1997年12月12日PCT提交1996年6月11日PCT公布。公开号WO96 / 41628 日期1996年12月27日喷雾干燥的颗粒包含普兰昔斯特（A）和一种或多种糖（B）作为必需成分，并且还包含一种或多种水溶性聚合物（C）和/或一种或多种表面活性剂（D）; 其制造方法; 提供了改善普鲁司特的粘合性的方法。根据本发明，降低了普兰司特的非常强的粘合性，并且可以有效地制备具有很小粘合性，窄粒度分布和良好流动性的含普鲁酮糖的颗粒。本发明的含有泼草素的颗粒在胶囊，片剂等的连续生产中不会产生麻烦，并且所得的含有普鲁酮糖的颗粒具有优异的崩解和分散性能。

5. 发明申请

US20110135979A1 LEAD-ACID BATTERY 有权
标题翻译：铅酸蓄电池
公开(公告)号：US20110135979A1
公开(公告)日：2011-06-09
申请号：US13057886
申请日：2009-08-04
申请人： Yasuhide Nakayama , Eiji Hojo , Masashi Shiota , Shin Ohsaki , Shinichi Egami
发明人： Yasuhide Nakayama , Eiji Hojo , Masashi Shiota , Shin Ohsaki , Shinichi Egami
IPC分类号： H01M2/12 , H01M2/04
CPC分类号： H01M2/1252 , H01M2/1217
摘要： There is provided a lead-acid battery in which the joint state between a lid body and a lid body cover can be checked based on both the joint state between a protruding portion in the periphery of a second exhaust hole and a joining portion of the lid body cover, and the joint state between a protruding portion of the lid body and a joining portion of the lid body cover. The lead-acid battery comprises: a container having at least one cell chamber; a lid body 1 for covering a top opening of the container, the lid body 1 having on a top surface a recessed portion 4, the recessed portion 4 having therein an annular protruding portion 4C protruding upward and having, in an area of a bottom wall inside the protruding portion, an exhaust hole 4D for exhausting gas from the cell chamber, wherein a guide passage for guiding gas from the exhaust hole 4D to the outside is formed by joining the protruding portion 4C with a joining portion provided on the lid body cover; an annular groove 4M formed between the protruding portion and the vertical wall is covered with an outer periphery of the lid body cover 5; and the guide passage is isolated from the groove 4M.
摘要翻译：提供了一种铅酸电池，其中可以基于第二排气孔的周边的突出部分和盖的接合部分之间的接合状态来检查盖体和盖体盖之间的接合状态盖体，以及盖体的突出部与盖体罩的接合部之间的接合状态。铅酸电池包括：具有至少一个电池室的容器; 用于覆盖容器的顶部开口的盖体1，盖体1在顶表面上具有凹部4，凹部4具有向上突出的环状突出部4C，并且具有在底壁在突出部分的内部设置有用于从电池室排出气体的排气孔4D，其中，用于将气体从排气孔4D引导到外部的引导通道通过将突出部4C与设置在盖体盖上的接合部接合而形成 ; 形成在突出部与垂直壁之间的环状槽4M被盖体盖5的外周覆盖; 并且引导通道与槽4M隔离。

6. 发明授权

US08652669B2 Lead-acid battery 有权
标题翻译：铅酸蓄电池
公开(公告)号：US08652669B2
公开(公告)日：2014-02-18
申请号：US13057886
申请日：2009-08-04
申请人： Yasuhide Nakayama , Eiji Hojo , Masashi Shiota , Shin Ohsaki , Shinichi Egami
发明人： Yasuhide Nakayama , Eiji Hojo , Masashi Shiota , Shin Ohsaki , Shinichi Egami
IPC分类号： H01M2/12
CPC分类号： H01M2/1252 , H01M2/1217
摘要： A lead-acid battery comprising a container having at least one cell chamber and a lid body for covering a top opening of the container. The lid body has on a top surface a recessed portion having therein an annular portion protruding upward and having, in an area of a bottom wall inside the protruding portion, an exhaust hole for exhausting gas from the cell chamber, wherein a guide passage for guiding gas from the exhaust hole to the outside is formed by joining the protruding portion with a joining portion provided on the lid body cover. An annular groove formed between the protruding portion and the vertical wall is covered with an outer periphery of the lid body cover 5 and the guide passage is isolated from the groove.
摘要翻译：一种铅酸电池，包括具有至少一个电池室的容器和用于覆盖容器顶部开口的盖体。所述盖体在顶面上具有凹部，所述凹部具有向上突出的环状部，在所述突出部内部的底壁区域具有用于从所述电池室排出气体的排气孔，其特征在于，通过将突出部与设置在盖体盖上的接合部接合而形成从排气孔到外部的气体。形成在突出部和垂直壁之间的环形槽被盖体盖5的外周覆盖，并且引导通道与槽隔离。

7. 发明授权

US08980467B2 Storage battery 有权
标题翻译：蓄电池
公开(公告)号：US08980467B2
公开(公告)日：2015-03-17
申请号：US12988750
申请日：2009-04-24
申请人： Yasuhide Nakayama , Eiji Hojo , Hirofumi Umetani , Masashi Shiota , Shin Ohsaki , Shinichi Egami
发明人： Yasuhide Nakayama , Eiji Hojo , Hirofumi Umetani , Masashi Shiota , Shin Ohsaki , Shinichi Egami
IPC分类号： H01M2/02 , H01M2/12 , H01M2/30 , H01M2/04 , H01M2/06
CPC分类号： H01M2/305 , H01M2/043 , H01M2/06 , H01M2/1252
摘要： There is provided a storage battery, including: a container having at least one cell chamber; a lid body (2) made of synthetic resin for covering a top opening of the container, the lid body having on a top surface a recessed portion that is recessed downward, the lid body having positive and negative electrode terminals disposed close to one side of the lid body and respectively at both end portions of said one side in a longitudinal direction, wherein the positive and negative electrode terminals (4) respectively have lower portions embedded in the lid body and upper portions projecting from the lid body; and an auxiliary lid (9) for closing the recessed portion. Conventional production of the storage battery has problems, for example, in that: when embedding a portion of a terminal to a lid body by insert molding, difference in shrinkage is caused between a surface in which a terminal body is embedded and a surface on which the terminal body is exposed, which results in difficulty in fitting the lid body to the container. The present invention is intended to solve this problem, for example, by providing the lid body of the storage battery with projections (6T, 7T), each at a location at which the upper portion of each of the terminals projects, at a location proximate to the location at which the upper portion of each of the terminals 4 projects, or at each of these locations.
摘要翻译：提供一种蓄电池，包括：具有至少一个电池室的容器; 由合成树脂制成的用于覆盖容器顶部开口的盖体（2），所述盖体在顶表面上具有向下凹陷的凹陷部分，所述盖体具有靠近一侧的正极端子和负极端子所述盖体和所述一侧的长度方向的两端部，分别具有嵌入所述盖体的下部和从所述盖体突出的上部的正极端子和所述负极端子; 和用于封闭凹部的辅助盖（9）。蓄电池的常规生产具有以下问题：例如：当通过嵌件成型将端子的一部分嵌入盖体时，在嵌入端子体的表面与其上嵌入端子体的表面之间产生收缩差异端子体露出，难以将盖体装配到容器上。本发明的目的是为了解决这个问题，例如，通过将蓄电池的盖体设置在每个端子的上部突出的位置处的突起（6T，7T）处于邻近的位置到每个终端4的上部突出的位置，或者在这些位置的每一个处。

8. 发明申请

US20110039153A1 STORAGE BATTERY 有权
标题翻译：储存电池
公开(公告)号：US20110039153A1
公开(公告)日：2011-02-17
申请号：US12988750
申请日：2009-04-24
申请人： Yasuhide Nakayama , Eiji Hojo , Hirofumi Umetani , Masashi Shiota , Shin Ohsaki , Shinichi Egami
发明人： Yasuhide Nakayama , Eiji Hojo , Hirofumi Umetani , Masashi Shiota , Shin Ohsaki , Shinichi Egami
IPC分类号： H01M2/30
CPC分类号： H01M2/305 , H01M2/043 , H01M2/06 , H01M2/1252
摘要： There is provided a storage battery, including: a container having at least one cell chamber; a lid body (2) made of synthetic resin for covering a top opening of the container, the lid body having on a top surface a recessed portion that is recessed downward, the lid body having positive and negative electrode terminals disposed close to one side of the lid body and respectively at both end portions of said one side in a longitudinal direction, wherein the positive and negative electrode terminals (4) respectively have lower portions embedded in the lid body and upper portions projecting from the lid body; and an auxiliary lid (9) for closing the recessed portion. Conventional production of the storage battery has problems, for example, in that: when embedding a portion of a terminal to a lid body by insert molding, difference in shrinkage is caused between a surface in which a terminal body is embedded and a surface on which the terminal body is exposed, which results in difficulty in fitting the lid body to the container. The present invention is intended to solve this problem, for example, by providing the lid body of the storage battery with projections (6T, 7T), each at a location at which the upper portion of each of the terminals projects, at a location proximate to the location at which the upper portion of each of the terminals 4 projects, or at each of these locations.
摘要翻译：提供一种蓄电池，包括：具有至少一个电池室的容器; 由合成树脂制成的用于覆盖容器顶部开口的盖体（2），所述盖体在顶表面上具有向下凹陷的凹陷部分，所述盖体具有靠近一侧的正极端子和负极端子所述盖体和所述一侧的长度方向的两端部，分别具有嵌入所述盖体的下部和从所述盖体突出的上部的正极端子和所述负极端子; 和用于封闭凹部的辅助盖（9）。蓄电池的常规生产具有以下问题：例如：当通过嵌件成型将端子的一部分嵌入盖体时，在嵌入端子体的表面与其上嵌入端子体的表面之间产生收缩差异端子体露出，难以将盖体装配到容器上。本发明的目的是为了解决这个问题，例如，通过将蓄电池的盖体设置在每个端子的上部突出的位置处的突起（6T，7T）处于邻近的位置到每个终端4的上部突出的位置，或在这些位置的每一个处。

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