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1. 发明授权

US5201932A Carboxamides 失效
公开(公告)号：US5201932A
公开(公告)日：1993-04-13
申请号：US877365
申请日：1992-05-04
申请人： Volker Maywald , Wolfgang Freund , Gerhard Hamprecht , Thomas Kuekenhoehner , Peter Plath , Bruno Wuerzer , Karl-Otto Westphalen
发明人： Volker Maywald , Wolfgang Freund , Gerhard Hamprecht , Thomas Kuekenhoehner , Peter Plath , Bruno Wuerzer , Karl-Otto Westphalen
IPC分类号： A01N43/80 , C07D261/18 , C07D275/02 , C07D275/03
CPC分类号： C07D275/03 , A01N43/80 , C07D261/18
摘要： Carboxamides Ia, Ib, Ic and Id ##STR1## (X=O, S; R.sup.1 =H, halogen, substituted or unsubstituted alkyl, substituted or unsubstituted benzyl, alkoxy, alkylthio, haloalkoxy, haloalkylthio, substituted or unsubstituted phenyl, substituted or unsubstituted phenoxy or phenylthio, a substituted or unsubstituted 5- or 6-membered heterocyclic radical containing one or two heteroatoms, cycloalkyl-substituted alkyl, substituted or unsubstituted alkenyl which may be epoxidized, substituted or unsubstituted alkynyl, substituted or unsubstituted cycloalkyl or cycloalkenyl; R.sup.1 '=cycloalkyl-substituted alkyl, substituted or unsubstituted alkenyl which may be epoxidized, substituted or unsubstituted cycloalkenyl; R.sup.2 =CHO, 4,5-dihydrooxazol-2-yl, COYR.sup.5, CONR.sup.6 R.sup.7 ; Y=O, S; R.sup.5 =H, substituted or unsubstituted alkyl, cycloalkyl, substituted or unsubstituted alkenyl, substituted or unsubstituted cycloalkenyl, substituted or unsubstituted alkynyl, substituted or unsubstituted phenyl, a 5- or 6-membered heterocyclic radical containing up to 3 heteroatoms, benzotriazole, N-phthalimido, tetrahydrophthalimido, succinimido, maleiimido, 2,2-dimethyl-1,3-dioxolan-4-ylmethyl, 1,3-dioxolan-2-on-4-ylmethyl, and when Y.dbd.O: one equivalent of a cation from the group of the alkali or alkaline earth metals, Mn, Cu, Fe ammonium and substituted ammonium, a radical --N.dbd.CR.sup.8 R.sup.9 or --W--Z; R.sup.8, R.sup.9 .dbd.H, substituted or unsubstituted alkyl, substituted or unsubstituted haloalkyl, cycloalkyl, alkoxy, furanyl, substituted or unsubstituted phenyl; R.sup.8 +R.sup.9 =4-7-membered methylene chain; W=alkylene chain, ethoxyethylene chain, butylene, butynylene chain; Z=a molecular moiety bonded to W in the .omega.-position and is the same as that linked to W in the .alpha.-position of W; R.sup.6 .dbd.H, alkyl, cycloalkyl; R.sup.7 .dbd.H; alkyl; --C(O-alkyl).dbd.N--H or --(O--alkyl).dbd.N--alkyl; R.sup.6 +R.sup.7 =4-5-membered methylene chain; R.sup.3 .dbd.H, substituted or unsubstituted alkyl, substituted or unsubstituted cycloalkyl; R.sup.4 .dbd.H, OH, alkoxy, subsituted or unsubstituted alkyl, substituted or unsubstituted cycloalkyl, substituted or unsubstituted alkenyl, substituted or unsubstituted alkynyl, di-(C.sub.1 -C.sub.4)-alkylamino, a substituted or unsubstituted 5- or 6-membered heterocyclic radical containing one or two heteroatoms, substituted or unsubstituted phenyl, substituted or unsubstituted naphthyl; R.sub.3 +R.sub.4 =4-7-membered methylene chain which may be interrupted by O, S or N--CH.sub.3, or --(CH.sub.2).sub.3 --CO--)and their environmentally tolerated salts.The compounds Ia to Id are suitable as herbicides.

2. 发明授权

US5378680A Dicarboximides and their use as herbicides 失效
标题翻译：二酰亚胺及其作为除草剂的用途
公开(公告)号：US5378680A
公开(公告)日：1995-01-03
申请号：US931951
申请日：1992-08-19
申请人： Volker Maywald , Klaus Ditrich , Thomas Kuekenhoehner , Gerhard Hamprecht , Wolfgang Freund , Karl-Otto Westphalen , Matthias Gerber , Helmut Walter
发明人： Volker Maywald , Klaus Ditrich , Thomas Kuekenhoehner , Gerhard Hamprecht , Wolfgang Freund , Karl-Otto Westphalen , Matthias Gerber , Helmut Walter
IPC分类号： A01N43/76 , A01N43/78 , A01N43/80 , A01N43/90 , C07D498/04 , C07D499/04 , C07D513/04
CPC分类号： C07D513/04 , A01N43/90
摘要： Dicarboximides of the formulae Ia, Ib and Ic ##STR1## where X is oxygen or sulfur,R.sup.1 is hydrogen, halogen, cyano, alkyl, cycloalkyl, alkenyl, alkynyl, alkoxy, alkenyloxy, alkynyloxy, alkylthio, haloalkoxy, haloalkylthio, alkylsulfonyl, haloalkylsulfonyl, phenyl, phenylalkyl, phenoxy or phenylthio, a 5-membered or 6-membered saturated or aromatic heterocyclic radical containing one or two hetero atoms selected from the group consisting of oxygen, sulfur and nitrogen, where the stated organic radicals may be further substituted, andR.sup.2 is hydrogen, hydroxyl, alkoxy, alkyl, cycloalkyl, alkenyl, alkynyl, di-C.sub.1 -C.sub.4 - alkylamino, a 5-membered or 6-membered heterocyclic saturated or aromatic radical having one or two hetero atoms selected from the group consisting of oxygen, sulfur and nitrogen, phenyl or naphthyl, where the stated organic radicals may be further substituted,and plant-tolerated salts of the dicarboximides I, except for 3-methylisoxazole-4,5-dicarboximide and thiazole-4,5-dicarboximides in which R.sup.2 is phenyl when R.sup.1 is methyl or 2-thiazolyl,and herbicides containing these compounds.
摘要翻译：其中X是氧或硫，R 1是氢，卤素，氰基，烷基，环烷基，烯基，炔基，烷氧基，烯氧基，炔氧基，烷氧基，烷硫基，卤代烷氧基，卤代烷硫基，烷基磺酰基，卤代烷基磺酰基，苯基，苯基烷基，苯氧基或苯硫基，含有一个或两个选自氧，硫和氮的杂原子的5元或6元饱和或芳族杂环基团，所述有机基团可以被进一步取代，并且R 2是氢，羟基，烷氧基，烷基，环烷基，链烯基，炔基，二-C 1 -C 4 - 烷基氨基，5元或6元杂环饱和或芳族基，选自氧，硫和氮的两个杂原子，苯基或萘基，其中所述有机基团可以被进一步取代，以及二甲酰亚胺I的植物耐受盐，除了3-甲基异恶唑-4,5-二甲酰亚胺 de和噻唑-4,5-二羧酰亚胺，其中当R 1是甲基或2-噻唑基时，R 2是苯基，以及含有这些化合物的除草剂。

3. 发明授权

US5176739A Dicarboximides and their use as herbicides 失效
标题翻译： DICARBOXIMIDES及其作为除草剂的用途
公开(公告)号：US5176739A
公开(公告)日：1993-01-05
申请号：US718639
申请日：1991-06-21
申请人： Volker Maywald , Klaus Ditrich , Thomas Kuekenhoehner , Gerhard Hamprecht , Wolfgang Freund , Karl-Otto Westphalen , Matthias Gerber , Helmut Walter
发明人： Volker Maywald , Klaus Ditrich , Thomas Kuekenhoehner , Gerhard Hamprecht , Wolfgang Freund , Karl-Otto Westphalen , Matthias Gerber , Helmut Walter
IPC分类号： A01N43/76 , A01N43/78 , A01N43/80 , A01N43/90 , C07D498/04 , C07D499/04 , C07D513/04
CPC分类号： C07D513/04 , A01N43/90
摘要： Dicarboximides of the formulae Ia, Ib and Ic ##STR1## where X is oxygen or sulfur, R.sup.1 is hydrogen, halogen, cyano, alkyl, cycloalkyl, alkenyl, alkynyl, alkoxy, alkenyloxy, alkynyloxy, alkylthio, haloalkoxy, haloalkylthio, alkylsulfonyl, haloalkylsulfonyl, phenyl, phenylalkyl, phenoxy or phenylthio, a 5-membered or 6-membered saturated or aromatic heterocyclic radical containing one or two hetero atoms selected from the group consisting of oxygen, sulfur and nitrogen, where the stated organic radicals may be further substituted, andR.sup.2 is hydrogen, hydroxyl, alkoxy, alkyl, cycloalkyl, alkenyl, alkynyl, di-C.sub.1 -C.sub.4 -alkylamino, a 5-membered or 6-membered heterocyclic saturated or aromatic radical having one or two hetero atoms selected from the group consisting of oxygen, sulfur and nitrogen, phenyl or naphthyl, where the stated organic radicals may be further substituted,and plant-tolerated salts of the dicarboximides I, except for 3-methylisoxazole-4,5-dicarboximide and thiazole-4,5-dicarboximides in which R.sup.2 is phenyl when R.sup.1 is methyl or 2-thiazolyl,and herbicides containing these compounds.
摘要翻译：其中X是氧或硫，R 1是氢，卤素，氰基，烷基，环烷基，烯基，炔基，烷氧基，烯氧基，炔氧基，烷氧基，烷硫基，卤代烷氧基，卤代烷硫基，烷基磺酰基，卤代烷基磺酰基，苯基，苯基烷基，苯氧基或苯硫基，含有一个或两个选自氧，硫和氮的杂原子的5元或6元饱和或芳族杂环基团，所述有机基团可以被进一步取代，并且R 2是氢，羟基，烷氧基，烷基，环烷基，烯基，炔基，二-C 1 -C 4 - 烷基氨基，具有一个或多个的五元或六元杂环饱和或芳族基团选自氧，硫和氮的两个杂原子，苯基或萘基，其中所述有机基团可以被进一步取代，以及二甲酰亚胺I的植物耐受盐，除了3-甲基异恶唑-4,5-二甲酰亚胺 e和噻唑-4,5-二羧酰亚胺，当R 1为甲基或2-噻唑基时，R 2为苯基，以及含有这些化合物的除草剂。

4. 发明授权

US5080708A Isoxazole(isothiazole)-5-carboxamides 失效
标题翻译：异佛唑（异噻唑）-5-羧酰胺
公开(公告)号：US5080708A
公开(公告)日：1992-01-14
申请号：US337640
申请日：1989-04-13
申请人： Wolfgang Freund , Thomas Kuekenhoehner , Gerhard Hamprecht , Bruno Wuerzer , Karl-Otto Westphalen , Norbert Meyer , Hans Theobald
发明人： Wolfgang Freund , Thomas Kuekenhoehner , Gerhard Hamprecht , Bruno Wuerzer , Karl-Otto Westphalen , Norbert Meyer , Hans Theobald
IPC分类号： A01N43/80 , A01N43/84 , A01N55/00 , A01N57/24 , C07D261/18 , C07D275/02 , C07D275/03 , C07D413/04 , C07D413/12 , C07D417/12
CPC分类号： C07D275/03 , A01N43/80 , A01N43/84 , A01N55/00 , A01N57/24 , C07D261/18 , C07D413/04 , C07D413/12 , C07D417/12
摘要： Isoxazole(isothiazole)-5-carboxamides of the formula ##STR1## where X is oxygen or sulfur,R.sup.1 is hydrogen, substituted or unsubstituted alkyl, alkoxy, substituted or unsubstituted cycloalkyl, a 5- or 6-membered heterocyclic radical having one or two heteroatoms selected from the group consisting of oxygen, sulfur and nitrogen, and which may be substituted, or substituted or unsubstituted phenyl, orR.sup.2 is formyl, 4,5-dihydrooxazol-2-yl or a radical of the formula COYR.sup.5 or CONR.sup.6 R.sup.7, whereY is oxygen or sulfur,R.sup.5 ishydrogen, substituted or unsubstituted alkyl, substituted or unsubstituted alkenyl, haloalkenyl, substituted or unsubstituted alkynyl,cycloalkyl,cycloalkenyl,substituted or unsubstituted phenyl,a 5- or 6-membered heterocyclic radical having one or two heteroatoms selected from the group consisting of oxygen, sulfur and nitrogen,cycloalkanimino, phthalimido, succinimido, or a radical ##STR2## R.sup.3 and R.sup.4 have the meanings defined herein, or their agriculturally acceptable salts possess herbicidal activity.
摘要翻译：其中X是氧或硫，R 1是氢，取代或未取代的烷基，烷氧基，取代或未取代的环烷基，具有一个或两个的5-或6-元杂环基的异噻唑（异噻唑）-5-甲酰胺，选自氧，硫和氮的杂原子，并且其可以被取代，或取代或未取代的苯基，或R 2是甲酰基，4,5-二氢恶唑-2-基或式COYR 5或CONR 6 R 7的基团，其中 Y是氧或硫，R5是氢，取代或未取代的烷基，取代或未取代的烯基，卤代烯基，取代或未取代的炔基，环烷基，环烯基，取代或未取代的苯基，具有一个或两个杂原子的5-或6-元杂环基选自氧，硫和氮，环亚烷基亚氨基，邻苯二甲酰亚氨基，琥珀酰亚胺基或自由基，CH 2 CH（OH）CH 2（OH）等，R 3和R 4具有本文定义的含义或其农业超可接受的盐具有除草活性。

5. 发明授权

US5205854A Isoxazole(isothiazole)-5-carboxamides 失效
标题翻译：异恶唑（异噻唑）-5-甲酰胺
公开(公告)号：US5205854A
公开(公告)日：1993-04-27
申请号：US764214
申请日：1991-09-23
申请人： Wolfgang Freund , Thomas Kuekenhoehner , Gerhard Hamprecht , Bruno Wuerzer , Karl-Otto Westphalen , Norbert Meyer , Hans Theobald
发明人： Wolfgang Freund , Thomas Kuekenhoehner , Gerhard Hamprecht , Bruno Wuerzer , Karl-Otto Westphalen , Norbert Meyer , Hans Theobald
IPC分类号： A01N43/80 , A01N43/84 , A01N55/00 , A01N57/24 , C07D261/18 , C07D275/02 , C07D275/03 , C07D413/04 , C07D413/12 , C07D417/12
CPC分类号： C07D275/03 , A01N43/80 , A01N43/84 , A01N55/00 , A01N57/24 , C07D261/18 , C07D413/04 , C07D413/10 , C07D417/12
摘要： Isoxazole(isothiazole)-5-carboxamides, having herbicidal activity, of the formula ##STR1## where X is oxygen or sulfur,R.sup.1 is hydrogen, substituted or unsubstituted alkyl, alkoxy, substituted or unsubstituted cycloalkyl, a 5- or 6-membered heterocyclic radical having one or two heteroatoms selected from the group consisting of oxygen, sulfur and nitrogen, and which may be substituted, or substituted or unsubstituted phenyl, orR.sup.2 is formyl, 4,5-dihydrooxazol-2-yl or a radical of the formula COYR.sup.5 or CONR.sup.6 R.sup.7.
摘要翻译：具有除草活性的具有除草活性的异噻唑（异噻唑）-5-甲酰胺，其中X是氧或硫，R1是氢，取代或未取代的烷基，烷氧基，取代或未取代的环烷基，5-或6-元杂环具有一个或两个选自氧，硫和氮的杂原子的基团，并且其可以被取代或取代或未取代的苯基，或R 2是甲酰基，4,5-二氢恶唑-2-基或式 COYR5或CONR6R7。

6. 发明授权

US5256633A Oxazole-and thiazolecarboxyamides as herbicides 失效
标题翻译：恶唑和噻唑酰胺作为除草剂
公开(公告)号：US5256633A
公开(公告)日：1993-10-26
申请号：US870386
申请日：1992-04-17
申请人： Klaus Ditrich , Volker Maywald , Gerhard Hamprecht , Albrecht Harreus , Bruno Wuerzer , Karl-Otto Westphalen
发明人： Klaus Ditrich , Volker Maywald , Gerhard Hamprecht , Albrecht Harreus , Bruno Wuerzer , Karl-Otto Westphalen
IPC分类号： A01N43/74 , C07D263/34 , C07D277/56 , C07D417/04 , A01N43/78
CPC分类号： C07D263/34 , A01N43/74 , C07D277/56 , C07D417/04
摘要： Oxazole- and thiazolecarboxamides of the formulae Ia and Ib ##STR1## where the substituents have the following meanings: oxygen or sulfur;hydrogen; halogen; substituted or unsubstituted C.sub.1 -C.sub.6 -alkyl, benzyl, cycloalkyl, alkenyl, alkynyl, phenyl, phenoxy or phenylthio; alkoxy; alkylthio; haloalkoxy; haloalkylthio; or a substituted or unsubstituted 5- or 6-membered heterocyclic radical;formyl, 4,5-dihydrooxazol-2-yl or --COYR.sup.5 ;oxygen or sulfur;hydrogen; cycloalkyl; substituted or unsubstituted alkyl, phenyl, benzyl, alkenyl, cycloalkenyl or alkynyl; a substituted or unsubstituted 5- or 6-membered heterocyclic radical; phthalimido; tetrahydrophthalimido; succinimido; maleiimido; one equivalent of a cation; or--N.dbd.CR.sup.6 R.sup.7 ; R.sup.6, R.sup.7 hydrogen; alkyl; cycloalkyl; phenyl; furyl or together a methylene chain or 4 to 7 members;hydrogen or substituted or unsubstituted alkyl or cycloalkyl;R.sup.4 hydroxy; alkoxy; substituted or unsubstituted alkyl, cycloalkyl, alkenyl, alkynyl, phenyl or naphthyl; a substituted or unsubstituted 5- or 6-membered heterocyclic radical; or R.sup.3 and R.sup.4 together are --(CH.sub.2).sub.n --Y.sub.p --(CH.sub.2).sub.q --, where n and q are 1, 2 or 3, p is 0 or 1 and Y is oxygen, sulfur or N-methyl, or form a radical of the formula --(CH.sub.2).sub.3 --CO--, and their environmentally tolerated salts,X is formula Ib not being sulfur when R.sup.1 is 3-pyridyl, R.sup.2 is CO.sub.2 CH.sub.2 CH.sub.3 or R.sup.3 is hydrogen, and X in formula Ia X not being sulfur and R.sup.1 not being thien-2-yl when YR.sup.5 is OH, R.sup.3 is hydrogen and R.sup.4 is methyl, processes for manufacturing such compounds and herbicidal agents containing compounds of the formula Ia or Ib as active ingredients.
摘要翻译：式Ia和Ib的恶唑和噻唑甲酰胺其中取代基具有以下含义：氧或硫; 氢; 卤素; 取代或未取代的C 1 -C 6烷基，苄基，环烷基，烯基，炔基，苯基，苯氧基或苯硫基; 烷氧基烷硫基卤代烷氧基卤代烷硫基; 或取代或未取代的五元或六元杂环基; 甲酰基，4,5-二氢恶唑-2-基或-COYR 5; 氧或硫; 氢; 环烷基取代或未取代的烷基，苯基，苄基，烯基，环烯基或炔基; 取代或未取代的5或6元杂环基; 邻苯二甲酰亚氨基; 四氢邻苯二甲酰亚胺琥珀酰亚胺马来西亚一个阳离子; 或-N = CR 6 R 7; R6，R7氢; 烷基; 环烷基苯基; 呋喃基或亚甲基链或4至7个成员; 氢或取代或未取代的烷基或环烷基; R4羟基; 烷氧基取代或未取代的烷基，环烷基，烯基，炔基，苯基或萘基; 取代或未取代的5或6元杂环基; 或者R 3和R 4一起是 - （CH 2）n -Yp-（CH 2）q - ，其中n和q是1,2或3，p是0或1，Y是氧，硫或N-甲基，或形成式（CH 2）3 -CO-的基团及其环境耐受的盐，X是当R1是3-吡啶基时R2不是硫，R2是CO2CH2 CH3或R3是氢，式Ia中的X不是硫和R1不是噻吩-2-基，当YR5是OH时，R3是氢，R4是甲基，制备这种化合物的方法和除草剂，其含有式Ia或Ib的化合物作为活性成分。

7. 发明授权

US5244867A Oxazole- and thiazolecarboxamides 失效
标题翻译：恶唑和噻唑甲酰胺
公开(公告)号：US5244867A
公开(公告)日：1993-09-14
申请号：US830326
申请日：1991-12-26
申请人： Klaus Ditrich , Volker Maywald , Gerhard Hamprecht , Albrecht Harreus , Bruno Wuerzer , Karl-Otto Westphalen
发明人： Klaus Ditrich , Volker Maywald , Gerhard Hamprecht , Albrecht Harreus , Bruno Wuerzer , Karl-Otto Westphalen
IPC分类号： A01N43/74 , C07D263/34 , C07D277/56 , C07D417/04
CPC分类号： C07D263/34 , A01N43/74 , C07D277/56 , C07D417/04
摘要： Oxazole- and thiazolecarboxamides of the formulae Ia and Ib ##STR1## where the substituents have the following meanings: X oxygen or sulfur;R.sup.2 formyl, 4,5-dihydrooxazol-2-yl or --COYR.sup.5 ;Y oxygen or sulfur; andR.sup.4 is methyl and herbicidal agents containing compounds of the formulae Ia or Ib as active ingredients.
摘要翻译：式Ia和Ib的恶唑和噻唑甲酰胺其中取代基具有以下含义：X氧或硫; R2甲酰基，4,5-二氢恶唑-2-基或-COYR 5; Y氧或硫; 和R4是含有式Ia或Ib化合物的甲基和除草剂作为活性成分。

8. 发明授权

US5284821A Oxazole- and thiazolecarboxamides 失效
标题翻译：恶唑和噻唑甲酰胺
公开(公告)号：US5284821A
公开(公告)日：1994-02-08
申请号：US919457
申请日：1992-07-27
申请人： Klaus Ditrich , Volker Maywald , Gerhard Hamprecht , Albrecht Harreus , Bruno Wuerzer , Karl-Otto Westphalen
发明人： Klaus Ditrich , Volker Maywald , Gerhard Hamprecht , Albrecht Harreus , Bruno Wuerzer , Karl-Otto Westphalen
IPC分类号： A01N43/74 , C07D263/34 , C07D277/56 , C07D417/04 , A01N43/76
CPC分类号： C07D263/34 , A01N43/74 , C07D277/56 , C07D417/04
摘要： Oxazole- and thiazolecarboxamides of the formulae Ia and Ib ##STR1## where the substituents have the following meanings: X oxygen or sulfur;R.sup.1 hydrogen; halogen; substituted or unsubstituted C.sub.1 -C.sub.6 -alkyl, benzyl, cycloalkyl, alkenyl, alkynyl, phenyl, phenoxy or phenylthio; alkoxy; alkylthio; haloalkoxy; haloalkylthio; or a substituted or unsubstituted 5- or 6-membered heterocyclic radical;R.sup.2 formyl, 4,5-dihydrooxazol-2-yl or --COYR.sup.5 ;Y oxygen or sulfur;R.sup.5 hydrogen; cycloalkyl; substituted or unsubstituted alkyl, phenyl, benzyl, alkenyl, cycloalkenyl or alkynyl; a substituted or unsubstituted 5- or 6-membered heterocyclic radical; phthalimido; tetrahydrophthalimido; succinimido; maleiimido; one equivalent of a cation; or--N.dbd.CR.sup.6 R.sup.7 ; R.sup.6, R.sup.7 hydrogen; alkyl; cycloalkyl; phenyl; furyl or together a methylene chain of 4 to 7 members;R.sup.3 hydrogen or substituted or unsubstituted alkyl or cycloalkyl;R.sup.4 hydroxy; alkoxy; substituted or unsubstituted alkyl, cycloalkyl, alkenyl, alkynyl, phenyl or naphthyl; a substituted or unsubstituted 5- or 6-membered heterocyclic radical; or R.sup.3 and R.sup.4 together are --(CH.sub.2).sub.n --Y.sub.p --(CH.sub.2).sub.q --, where n and q are 1, 2 or 3, p is 0 or 1 and Y is oxygen, sulfur or N-methyl, or form a radical of the formula --(CH.sub.2).sub.3 --CO--, and their environmentally tolerated salts,X in formula Ib not being sulfur when R.sup.1 is 3-pyridyl, R.sup.2 is CO.sub.2 CH.sub.2 CH.sub.3 or R.sup.3 is hydrogen, and X in formula Ia X not being sulfur and R.sup.1 not being thien-2-yl when YR.sup.5 is OH, R.sup.3 is hydrogen and R.sup.4 is methyl, processes for manufacturing such compounds and herbicidal agents containing compounds of the formulae Ia or Ib as active ingredients.
摘要翻译：式Ia和Ib的恶唑和噻唑甲酰胺其中取代基具有以下含义：X氧或硫; R1氢; 卤素; 取代或未取代的C 1 -C 6烷基，苄基，环烷基，烯基，炔基，苯基，苯氧基或苯硫基; 烷氧基烷硫基卤代烷氧基卤代烷硫基; 或取代或未取代的五元或六元杂环基; R2甲酰基，4,5-二氢恶唑-2-基或-COYR 5; Y氧或硫; R5氢; 环烷基取代或未取代的烷基，苯基，苄基，烯基，环烯基或炔基; 取代或未取代的5或6元杂环基; 邻苯二甲酰亚氨基四氢邻苯二甲酰亚胺琥珀酰亚胺马来西亚一个阳离子; 或-N = CR 6 R 7; R6，R7氢; 烷基; 环烷基苯基; 呋喃基或一起形成4至7个成员的亚甲基链; R3氢或取代或未取代的烷基或环烷基; R4羟基烷氧基取代或未取代的烷基，环烷基，烯基，炔基，苯基或萘基; 取代或未取代的5或6元杂环基; 或者R 3和R 4一起是 - （CH 2）n -Yp-（CH 2）q - ，其中n和q是1,2或3，p是0或1，Y是氧，硫或N-甲基，或形成式（（CH2）3-CO-）及其环境耐受盐的基团，当R1为3-吡啶基时，式Ib中的X不为硫，R2为CO2CH2CH3或R3为氢，式Ia中的X为硫，并且当YR 5是OH时，R 1不是噻吩-2-基，R 3是氢，R 4是甲基，制备这种化合物的方法和含有式Ia或Ib化合物的除草剂作为活性成分。

9. 发明授权

US5399544A Isoxazole- and isothiazole-5-carboxamides 失效
标题翻译：异恶唑和异噻唑-5-甲酰胺
公开(公告)号：US5399544A
公开(公告)日：1995-03-21
申请号：US117102
申请日：1993-09-14
申请人： Volker Maywald , Peter Muenster , Hartmann Koenig , Gerhard Hamprecht , Thomas Kuekenhoehner , Wolfgang Rohr , Helmut Walter , Karl-Otto Westphalen , Matthias Gerber
发明人： Volker Maywald , Peter Muenster , Hartmann Koenig , Gerhard Hamprecht , Thomas Kuekenhoehner , Wolfgang Rohr , Helmut Walter , Karl-Otto Westphalen , Matthias Gerber
IPC分类号： A01N43/80 , C07D261/18 , C07D275/02 , C07D275/03 , C07D413/04 , C07D417/12
CPC分类号： C07D275/03 , A01N43/80 , C07D261/18
摘要： Isoxazole- and isothiazole-5-carboxamides of the formula ##STR1## where X is oxygen or sulfur, R.sup.1 is hydrogen, substituted or unsubstituted alkyl, cycloalkyl, cycloalkenyl, alkenyl (may be epoxidized at the double bond), alkynyl, alkoxy, a heterocyclic radical or phenyl, R.sup.2 is a derivative carboxylic acid function and R.sup.3 and R.sup.4 have the meanings given in the disclosure, and herbicidal agents containing compounds I.
摘要翻译： PCT No.PCT / EP92 / 00183 Sec。 371日期：1993年9月14日 102（e）1993年9月14日PCT PCT 1992年1月29日PCT公布。公开号WO92 / 16514 1991年10月1日，1992.异唑和异噻唑-5-甲酰胺，其中X为氧或硫，R 1为氢，取代或未取代的烷基，环烷基，环烯基，烯基（可在双键环氧化），炔基，烷氧基，杂环基或苯基，R2是衍生羧酸官能团，R3和R4具有本发明中给出的含义，和含有化合物I的除草剂。

10. 发明授权

US5203907A Isoxazole- and isothiazole-5-carboxamides 失效
标题翻译：异佛唑酮和异唑唑-5-羧酰胺
公开(公告)号：US5203907A
公开(公告)日：1993-04-20
申请号：US849256
申请日：1992-03-11
申请人： Volker Maywald , Peter Muenster , Hartmann Koenig , Gerhard Hamprecht , Thomas Kuekenhoehner , Helmut Walter , Karl-Otto Westphalen , Matthias Gerber
发明人： Volker Maywald , Peter Muenster , Hartmann Koenig , Gerhard Hamprecht , Thomas Kuekenhoehner , Helmut Walter , Karl-Otto Westphalen , Matthias Gerber
IPC分类号： A01N43/80 , C07D261/18 , C07D275/02 , C07D275/03 , C07D413/04 , C07D417/04 , C07F9/653 , C07F9/6539
CPC分类号： C07D275/03 , A01N43/80 , C07D261/18 , C07F9/653 , C07F9/6539
摘要： Isoxazole- and isothiazole-5-carboxamides of the formula I ##STR1## where X is oxygen or sulfur, R.sup.1 is halogen, alkylthio, haloalkoxy, haloalkylthio, cyano, formyl, alkanoyl, alkoxycarbonyl, alkylaminocarbonyl, di-(C.sub.1 -C.sub.3)-alkylaminocarbonyl, cyclopropylaminocarbonyl, methylsulfonyl, trifluoromethylsulfonyl, unsubstituted or substituted phenoxy or phenylthio; R.sup.2 is formyl, haloformyl, 4,5-dihydro-2-oxazolyl, COOR.sup.5, COSR.sup.5 or CONR.sup.6 R.sup.7, and R.sup.3 to R.sup.7 have the meanings specified in the description, are suitable as herbicides.
摘要翻译：式I的异恶唑和异噻唑-5-甲酰胺其中X是氧或硫，R1是卤素，烷硫基，卤代烷氧基，卤代烷硫基，氰基，甲酰基，烷酰基，烷氧基羰基，烷基氨基羰基，二（C1-C3）烷基氨基羰基，环丙基氨基羰基，甲基磺酰基，三氟甲基磺酰基，未取代或取代的苯氧基或苯硫基; R 2是甲酰基，卤代甲酰基，4,5-二氢-2-恶唑基，COOR 5，COSR 5或CONR 6 R 7，并且R 3至R 7具有本说明书中规定的含义，适合作为除草剂。

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