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1. 发明授权

US4719207A CNS active substituted azetidinone compounds 失效
标题翻译： CNS活性取代的氮杂环丁酮化合物
公开(公告)号：US4719207A
公开(公告)日：1988-01-12
申请号：US747018
申请日：1985-06-20
申请人： Toshinari Tamura , Makoto Yoshida , Shin-ichi Tsukamoto , Hidenori Iwamoto , Minoru Yamamoto , Soichi Kagami
发明人： Toshinari Tamura , Makoto Yoshida , Shin-ichi Tsukamoto , Hidenori Iwamoto , Minoru Yamamoto , Soichi Kagami
IPC分类号： C07D205/08 , C07D205/085 , C07F7/10 , C07K5/097 , A61K31/415 , C07D403/12 , C07D403/14
CPC分类号： C07K5/0821 , C07D205/08 , C07D205/085 , C07F7/10
摘要： Substituted azetidinone compounds are provided which have the formula: ##STR1## wherein one of R.sup.1 and R.sup.2 represents a substituted lower alkyl group, an azido group, an amino group, a lower acylamino group, a mercapto group or a lower alkylthio group and the other represents a hydrogen group, or, both represent hydrogen atoms or lower alkyl groups; R.sup.3 represents a hydrogen atom or a group shown by formula: ##STR2## (wherein X represents ##STR3## (wherein R.sup.5 represents a hydrogen atom or a lower alkyl group) and Y represents a hydroxy group, a lower alkoxy group, an amino group, a mono- or di-lower alkylamino group); R.sup.4 represents a hydrogen atom, a substituted or unsubstituted lower alkyl group or a group shown by formula: --CH.sub.2 CO--A (wherein A represents an amino group or a group shown by formula: ##STR4## (wherein X and Y are as defined above), provided that when R.sup.1 and R.sup.2 are both hydrogen atoms, at least R.sup.4 represents a group other than a hydrogen atom and provided that either R.sup.3 or R.sup.4 represents a group other than a hydrogen atom. The compounds have strong CNS action.
摘要翻译：提供具有下式的取代的氮杂环丁酮化合物：其中R 1和R 2之一表示取代的低级烷基，叠氮基，氨基，低级酰氨基，巯基或低级烷硫基另一个表示氢基团，或者都表示氢原子或低级烷基; R3表示氢原子或由下式表示的基团：其中X表示（其中R5表示氢原子或低级烷基），Y表示羟基，低级烷氧基，氨基，一或二低级烷基氨基）; R 4表示氢原子，取代或未取代的低级烷基或由式-CH 2 CO-A（其中A表示氨基或由下式表示的基团：其中X和Y如上所定义）），条件是当R 1和R 2均为氢原子时，至少R 4表示氢原子以外的基团，只要R 3或R 4表示除氢原子以外的基团，则该化合物具有强CNS作用。

2. 发明授权

US4636567A 4-substituted-2-azetidinone compound 失效
标题翻译： 4-取代-2-氮杂环丁酮化合物
公开(公告)号：US4636567A
公开(公告)日：1987-01-13
申请号：US785169
申请日：1985-10-07
申请人： Toshinari Tamura , Hidenori Iwamoto , Makoto Yoshida , Minoru Yamamoto
发明人： Toshinari Tamura , Hidenori Iwamoto , Makoto Yoshida , Minoru Yamamoto
IPC分类号： C07D403/14 , C07D205/08 , C07D403/12 , C07K5/078 , C07K5/097
CPC分类号： C07D403/12 , C07D205/08 , C07K5/06147
摘要： A novel-4-substituted-2-azetidinone compound shown by the general formula ##STR1## and salts thereof. The compounds of this invention have a strong CNS activity and are useful for improving a disturbance of consciousness in schizophrenia, a head injury, etc., or improving hypobulia, memory loss, etc.

3. 发明授权

US4610821A 4-substituted-2-azetidinone compound, process of producing the compounds, and medicaments containing the compounds 失效
标题翻译： 4-取代-2-氮杂环丁酮化合物，制备该化合物的方法和含有这些化合物的药物
公开(公告)号：US4610821A
公开(公告)日：1986-09-09
申请号：US785168
申请日：1985-10-07
申请人： Toshinari Tamura , Hidenori Iwamoto , Makoto Yoshida , Minoru Yamamoto
发明人： Toshinari Tamura , Hidenori Iwamoto , Makoto Yoshida , Minoru Yamamoto
IPC分类号： C07D403/14 , C07D205/08 , C07D403/12 , C07K5/078 , C07K5/097 , C07D413/12
CPC分类号： C07D403/12 , C07D205/08 , C07K5/06147
摘要： A novel 4-substituted-2-azetidinone compound shown by the general formula ##STR1## and salts thereof. The compounds of this invention have a strong CNS activity and are useful for improving a disturbance of consciousness in shizophrenia, a head injury, etc., or improving hypobulia, memory loss, etc.

4. 发明授权

US4564609A 4-Substituted-2-azetidinone compound, process of producing the compounds, and medicaments containing the compounds 失效
标题翻译： 4-取代-2-氮杂环丁酮化合物，制备该化合物的方法和含有这些化合物的药物
公开(公告)号：US4564609A
公开(公告)日：1986-01-14
申请号：US592866
申请日：1984-03-23
申请人： Toshinari Tamura , Hidenori Iwamoto , Makoto Yoshida , Minoru Yamamoto
发明人： Toshinari Tamura , Hidenori Iwamoto , Makoto Yoshida , Minoru Yamamoto
IPC分类号： C07D403/14 , C07D205/08 , C07D403/12 , C07K5/078 , C07K5/097 , A61K37/00
CPC分类号： C07D403/12 , C07D205/08 , C07K5/06147
摘要： A novel 4-substituted-2-azetidinone compound shown by the general formula ##STR1## and salts thereof. The compounds of this invention have a strong CNS activity and are useful for improving a disturbance of consciousness in schizophrenia, a head injury, etc., or improving hypobulia, memory loss, etc.
摘要翻译：由通式表示的新型4-取代-2-氮杂环丁酮化合物及其盐。本发明化合物具有较强的CNS活性，可用于改善精神分裂症意识障碍，头部损伤等，或改善低血压，记忆力丧失等。

5. 发明授权

US4740586A Crystalline form III of N.sup..alpha. -[[(S)-4-oxo-2-azetidinyl]-carbonyl]- L 失效
标题翻译： Nα - [[（S）-4-氧代-2-氮杂环丁烷基] - 羰基] -L-组氨酰基-L-脯氨酰胺的结晶形式III
公开(公告)号：US4740586A
公开(公告)日：1988-04-26
申请号：US937608
申请日：1986-12-03
申请人： Toshinari Tamura , Hideya Matsuda , Makoto Yoshida
发明人： Toshinari Tamura , Hideya Matsuda , Makoto Yoshida
IPC分类号： C07K1/14 , A61K38/00 , A61P25/28 , C07D403/14 , C07K5/08 , C07K5/097 , C07D205/08
CPC分类号： C07D403/14 , C07K5/0821
摘要： A novel crystal form of N.sup..alpha. -[[(S)-4-oxo-2-azetidinyl]-carbonyl]-L-histidyl-L-prolinamide is provided and a process for preparing such crystals. The crystals provided by the present invention are the dihydrate form of the compound which exhibits a specific X-ray powder diffraction pattern, infared absorption spectrum and thermogravimetry-differential scanning calorimetry. The compound in its novel crystal form is useful in the treatment of consciousness disturbances and memory disorders.
摘要翻译：提供了Nα - [[（S）-4-氧代-2-氮杂环丁烷基] - 羰基] -L-组氨酰基-L-脯氨酰胺的新型晶体形式及其制备方法。本发明提供的晶体是化合物的二水合物形式，其表现出特定的X射线粉末衍射图，Infared吸收光谱和热重量分析 - 差示扫描量热法。其新型晶体形式的化合物可用于治疗意识障碍和记忆障碍。

6. 发明授权

US09930215B2 Image forming control apparatus, method of generating correction data, and storage medium 有权
公开(公告)号：US09930215B2
公开(公告)日：2018-03-27
申请号：US15270221
申请日：2016-09-20
申请人： Makoto Yoshida
发明人： Makoto Yoshida
IPC分类号： H04N1/407 , G06K15/02 , H04N1/405
CPC分类号： H04N1/4078 , G06K15/026 , G06K15/1835 , G06K15/1881 , H04N1/405
摘要： An image forming control apparatus for controlling an image forming apparatus to form an image on a recording medium includes a memory to store a target property data of original gradation values of image data of a target image to be formed on the recording medium; and circuitry to acquire actual property data of the target image actually formed on the recording medium, convert the original gradation values to another gradation values, generate a primary correction data based on the original gradation values and the another gradation values, generate a secondary correction data to supplement the generated primary correction data, compare the primary correction data and the secondary correction data, and generate gradation correction data used for correcting the original gradation values existing in a specific range of the original gradation values based on a comparison result of the primary correction data and the secondary correction data.

7. 发明授权

US09223281B2 Image processing apparatus, image forming system, and computer-readable recording medium having gloss control 有权
标题翻译：图像处理装置，图像形成系统和具有光泽控制的计算机可读记录介质
公开(公告)号：US09223281B2
公开(公告)日：2015-12-29
申请号：US14576409
申请日：2014-12-19
申请人： Makoto Yoshida , Hiroaki Suzuki
发明人： Makoto Yoshida , Hiroaki Suzuki
IPC分类号： G03G15/20 , G03G15/00
CPC分类号： G03G15/6585 , G03G2215/00805
摘要： An image processing apparatus includes a storage unit that stores therein a type of surface effect and predetermined glossiness in association with each other, a determining unit that determines, as first glossiness, the glossiness associated with the surface effect specified by the gloss control plane data, a measurement control unit that performs control to measure second glossiness indicating actual glossiness of a printed matter that is a recording medium on which printing has been performed by a printing apparatus, a generation unit that produces, from the gloss control plane data, gloss plane data for additional printing in which a density value is set in accordance with an amount of a transparent color material necessary for achieving the first glossiness on the basis of a difference in value between the first glossiness and the second glossiness, and an output unit that outputs the gloss plane data for additional printing.
摘要翻译：图像处理装置包括存储单元，其中存储有相关联的表面效果和预定光泽度的类型;确定单元，其确定与由光泽度控制平面数据指定的表面效果相关联的光泽度作为第一光泽度，测量控制单元，其执行控制以测量指示作为其上由打印设备执行打印的记录介质的打印物的实际光泽度的第二光泽度;生成单元，其从光泽度控制面数据生成光泽平面数据用于根据第一光泽度和第二光泽度之间的值的差异来实现根据第一光泽度所需的透明色材料的量设定浓度值的另外的印刷;以及输出单元，光泽平面数据进行额外打印。

8. 发明授权

US09157344B2 Solenoid valve and valve opening-closing timing control device 有权
标题翻译：电磁阀和开阀定时控制装置
公开(公告)号：US09157344B2
公开(公告)日：2015-10-13
申请号：US14239654
申请日：2012-06-18
申请人： Kenji Fujiwaki , Masaki Kobayashi , Makoto Yoshida , Kenji Ikeda
发明人： Kenji Fujiwaki , Masaki Kobayashi , Makoto Yoshida , Kenji Ikeda
IPC分类号： F01L1/34 , F01L1/344 , F15B13/04 , F16K3/26 , F16K31/06 , F15B13/00
CPC分类号： F01L1/3442 , F01L2001/3443 , F01L2001/34456 , F01L2001/34463 , F15B13/0402 , F15B2013/004 , F16K3/26 , F16K31/06 , Y10T137/8671
摘要： A valve opening-closing timing control device includes a solenoid valve having a solenoid mechanism provided with a spool having an oil path groove formed in an outer face thereof, and a sleeve for housing the spool to reciprocate and slide. A wall surface of the sleeve has a first port communicating with a first hydraulic oil supply section, a second port communicating with a second hydraulic oil supply section, and a third port communicating with the side of a hydraulic oil supply source. The spool is driven and set to a first position for supplying hydraulic oil from the hydraulic oil supply source to the first port, a second position for supplying the hydraulic oil from the hydraulic oil supply source to the second port, and a third position outside an area between the first and second positions to prevent supply of hydraulic oil from the first and second ports.
摘要翻译：一种阀开闭正时控制装置，包括具有螺线管机构的电磁阀，该螺线管机构设置有在其外表面形成有油路槽的阀芯，以及用于容纳阀芯往复运动的滑套的套筒。套筒的壁面具有与第一液压供油部连通的第一端口，与第二液压供油部连通的第二端口和与液压油供给源侧连通的第三端口。阀芯被驱动并设置在第一位置，用于将液压油从液压油供应源供应到第一端口;第二位置，用于将液压油从液压油供应源供应到第二端口;以及第三位置，在第一和第二位置之间的区域，以防止从第一和第二端口供应液压油。

9. 发明授权

US09028912B2 Method of manufacturing optical fiber base material and apparatus therefor 有权
标题翻译：制造光纤基材的方法及其设备
公开(公告)号：US09028912B2
公开(公告)日：2015-05-12
申请号：US11730061
申请日：2007-03-29
申请人： Makoto Yoshida
发明人： Makoto Yoshida
IPC分类号： C23C16/26 , C03B37/014
CPC分类号： C03B37/0142 , C03B2207/42 , C03B2207/50 , C03B2207/60
摘要： In a method of manufacturing an optical fiber base material including depositing soot generated by flame hydrolysis, the fluctuation band of the surface temperature of a burner fixing section including a burner holder and its fixture for burners for compounding the optical fiber base material is kept equal to or less than 80 degree C.The temperature can be controlled by a heat shield plate arranged between a burner flame and a burner fixing section and a temperature control mechanism that heats or cools the burner fixing section. Thereby the relative position between the burner and the soot deposition is stabilized, so that the manufacturing method being capable of manufacturing an optical fiber base material having a stable refractive index and the apparatus therefor can be provided.
摘要翻译：在制造包括通过火焰水解产生的烟灰的光纤基材的方法中，包括燃烧器支架的燃烧器固定部的表面温度的波动带及其用于配合光纤基材的燃烧器的固定器保持等于或小于80℃。温度可以通过布置在燃烧器火焰和燃烧器固定部分之间的隔热板和加热或冷却燃烧器固定部分的温度控制机构来控制。因此，燃烧器和烟灰沉积之间的相对位置是稳定的，从而可以提供能够制造具有稳定的折射率的光纤基材的制造方法及其装置。

10. 发明授权

US08740522B2 Shaping machine system and computer program for controlling a shaping device 有权
标题翻译：整形机系统和计算机程序，用于控制整形装置
公开(公告)号：US08740522B2
公开(公告)日：2014-06-03
申请号：US13457355
申请日：2012-04-26
申请人： Akihiro Suyama , Ryo Sato , Yoshimitsu Asahina , Makoto Yoshida
发明人： Akihiro Suyama , Ryo Sato , Yoshimitsu Asahina , Makoto Yoshida
IPC分类号： G05B19/402
CPC分类号： G05B19/402 , G05B19/40937 , G05B2219/36358 , G05B2219/50125 , G05B2219/50132 , G05B2219/50351 , Y02P90/265 , Y10T29/5124 , Y10T409/30868 , Y10T409/309464 , Y10T483/115
摘要： A shaping machine system including a shaping device and a computer is provided. The shaping device includes at least one jig mount body configured for mounting a jig; a shaping tool support body configured for supporting a shaping tool; a first drive device configured for rotating the shaping tool; and a second drive device configured for driving the shaping tool support body or the at least one jig mount body or changing a posture of the shaping tool relative to the workpiece. The computer is configured for controlling the first and second drive devices according to predetermined shaping data. The computer includes a jig position measuring unit configured for measuring a position of the jig; a position error detecting unit configured for detecting a position error of the jig, and a shaping data correcting unit configured for correcting the predetermined shaping data according to a jig position error.
摘要翻译：提供了一种包括成形装置和计算机的成形机系统。成形装置包括至少一个构造成用于安装夹具的夹具安装体; 成形工具支撑体，其构造成用于支撑成形工具; 构造成旋转成形工具的第一驱动装置; 以及构造成用于驱动成形工具支撑体或至少一个夹具安装体或改变成形工具相对于工件的姿势的第二驱动装置。计算机被配置为根据预定的成形数据来控制第一和第二驱动装置。该计算机包括夹具位置测量单元，其被配置为测量夹具的位置; 位置误差检测单元，被配置为检测夹具的位置误差;以及整形数据校正单元，被配置为根据夹具位置误差校正预定的成形数据。

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